DrugRepV Browse Page


DrugRepV browse page allows user to take a glance of the particular antiviral agent.Fields in the webpage is hylerlinked ot various external repositories like DrugBank, PubChem, Clinicaltrials.gov,and PubMed.User can explore the biological, Clinical, Chemical, and Structural details of every repurposed drug candidate.By clicking on the table header arrows, user can sort entries in ascending or descending order.


Total number of Records for NA are 3814




DrugRepV_ID Antiviral Name
Drug type
Primary Indication
Secondary Indication
Strain
Pathways
Assay
Activity
Clinical Status
References
DrugRepV_0012BHSA
NA
NA
Zika virus
GZ01, a recent Asian lineage
NA
Plaque assay
No significant effect (45 %)
NA
29033372
DrugRepV_0015Chlorogenic Acid
NA
Cancer
Zika virus
GZ01, a recent Asian lineage
NA
Plaque assay
No significant effect (10 %)
Investigational
29033372
DrugRepV_0016Tetrandrine
NA
Congestive circulatory disorder and inflammatory diseases
Zika virus
GZ01, a recent Asian lineage
NA
Plaque assay
No significant effect (0 %)
Experimental
29033372
DrugRepV_0019Delphinidin Chloride
NA
NA
Zika virus
GZ01, a recent Asian lineage
NA
Plaque assay
Increase (110 %)
NA
29033372
DrugRepV_0073Sunitinib-Erlotinib
NA
NA
Ebola virus
rVSV-GP EBOV
NA
Flow cytometry
Decrease
NA
28240606
DrugRepV_0074Sunitinib-Erlotinib
NA
NA
Ebola virus
Mouse adapted strain
NA
NA
Increase
NA
28240606
DrugRepV_0090Imukin
NA
NA
Zika virus
Puerto Rico strain PRVABC-59
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved, Investigational
28185815
DrugRepV_0091Imukin
NA
NA
Zika virus
Puerto Rico strain PRVABC-59
NA
Real-time PCR
Decrease (>2 Log viral titer (copies/ml))
Approved, Investigational
28185815
DrugRepV_0092Imukin
NA
NA
Zika virus
Puerto Rico strain PRVABC-59
NA
Plaque assay
Decrease (>90 %)
Approved, Investigational
28185815
DrugRepV_0097Ki8751
NA
NA
Zika virus
Mex2-81
NA
Immunoflourescence assay
Decrease (50 %)
NA
28099856
DrugRepV_0100GSK2656157
NA
NA
Zika virus
Mex2-81
NA
Immunoflourescence assay
No significant effect
NA
28099856
DrugRepV_0110RGFP966
NA
NA
Zika virus
Mex2-81
NA
Immunoflourescence assay
Decrease (50 %)
NA
28099856
DrugRepV_0116Methotrexate
NA
Gestational choriocarcinoma | Chorioadenoma destruens | Hydatidiform mole | Meningeal leukemia | Breast cancer | Epidermoid cancers of the head and neck | Lung cancer
Zika virus
Mex2-81
NA
Immunoflourescence assay
Decrease (50 %)
Approved
28099856
DrugRepV_0117PF-04691502
NA
Breast Cancer
Zika virus
Mex2-81
NA
Immunoflourescence assay
No significant effect
Investigational
28099856
DrugRepV_0120Navitoclax
NA
Cancer
Zika virus
Mex2-81
NA
Immunoflourescence assay
Decrease (50 %)
Investigational
28099856
DrugRepV_0123GZD824
NA
NA
Zika virus
Mex2-81
NA
Immunoflourescence assay
No significant effect (No significant effect No significant effect)
NA
28099856
DrugRepV_0124VE-822
NA
Ovarian Neoplasms, Ovarian Serous Tumor, Adult Solid Neoplasm, Advanced Solid Tumor, and Advanced Solid Neoplasm
Zika virus
Mex2-81
NA
Immunoflourescence assay
No significant effect (No significant effect No significant effect)
Investigational
28099856
DrugRepV_0125Amuvatinib
NA
Cancer
Zika virus
Mex2-81
NA
Immunoflourescence assay
No significant effect (No significant effect No significant effect)
Investigational
28099856
DrugRepV_0126NVP-BHG712
NA
NA
Zika virus
Mex2-81
NA
Immunoflourescence assay
No significant effect (No significant effect No significant effect)
NA
28099856
DrugRepV_0127WAY-600
NA
Cancer
Zika virus
Mex2-81
NA
Immunoflourescence assay
Decrease (50 %)
NA
28099856
DrugRepV_0128YM201636
NA
NA
Zika virus
Mex2-81
NA
Immunoflourescence assay
No significant effect
NA
28099856
DrugRepV_0129RGFP966
NA
NA
Zika virus
Mex2-81
NA
Immunoflourescence assay
Decrease (50 %)
NA
28099856
DrugRepV_0130QNZ
NA
NA
Zika virus
Mex2-81
NA
Immunoflourescence assay
Decrease (50 %)
NA
28099856
DrugRepV_0133STF-118804
NA
NA
Zika virus
Mex2-81
NA
Immunoflourescence assay
Decrease (50 %)
NA
28099856
DrugRepV_0144AMG-458
NA
Cancer
Zika virus
MR766
NA
Immunoflourescence assay
Decrease (60 %)
NA
28099856
DrugRepV_0145AMG-458
NA
Cancer
Zika virus
MR766
NA
Immunoflourescence assay
No significant effect (20 %)
NA
28099856
DrugRepV_0146AMG-458
NA
Cancer
Zika virus
MR766
NA
Immunoflourescence assay
No significant effect (10 %)
NA
28099856
DrugRepV_0165AMG-458
NA
Cancer
Zika virus
Mex2-81
NA
Immunoflourescence assay
Decrease (60 %)
NA
28099856
DrugRepV_0166AMG-458
NA
Cancer
Zika virus
Mex2-81
NA
Immunoflourescence assay
Decrease (70 %)
NA
28099856
DrugRepV_0167AMG-458
NA
Cancer
Zika virus
Mex2-81
NA
Immunoflourescence assay
No significant effect (30 %)
NA
28099856
DrugRepV_0205Toremifene-Clarithromycin-Posaconazole
NA
NA
Ebola virus
VLP
NA
Immunoflourescence assay
Decrease (50 %)
NA
27890675
DrugRepV_0206Toremifene-Mefloquine-Posaconazole
NA
NA
Ebola virus
VLP
NA
Immunoflourescence assay
Decrease (50 %)
NA
27890675
DrugRepV_0207Chloroquine-Maprotiline-Azithromycin
NA
Malaria and Depression
Ebola virus
VLP
NA
Immunoflourescence assay
Decrease (50 %)
Approved
27890675
DrugRepV_0213Toremifene-Clarithromycin-Posaconazole
NA
NA
Ebola virus
EBOLA/Mayinga-eGFP
NA
Immunoflourescence assay
Decrease (>90 %)
NA
27890675
DrugRepV_0214Toremifene-Mefloquine-Posaconazole
NA
NA
Ebola virus
EBOLA/Mayinga-eGFP
NA
Immunoflourescence assay
Decrease (74 %)
NA
27890675
DrugRepV_0217Alvespimycin
NA
Cancer
Ebola virus
ME718-1976/Yambuku-Ecran
NA
Real-time PCR
Decrease (3.72 ± 0.18 Ct)
Investigational
27801778
DrugRepV_0218Alvespimycin
NA
Cancer
Ebola virus
ME718-1976/Yambuku-Ecran
NA
Real-time PCR
Increase (?0.63 ± 1.39 Ct)
Investigational
27801778
DrugRepV_0231JB1a
NA
NA
Ebola virus
ME718-1976/Yambuku-Ecran
NA
Real-time PCR
Increase (?4.02 ± 0.13 Ct)
NA
27801778
DrugRepV_0232JB1a
NA
NA
Ebola virus
ME718-1976/Yambuku-Ecran
NA
Real-time PCR
Increase (?5.48 ± 0.50 Ct)
NA
27801778
DrugRepV_0239Aimspro
NA
Multiple sclerosis
Ebola virus
ME718-1976/Yambuku-Ecran
NA
Real-time PCR
Increase (?2.03 ± 0.95 Ct)
Phase II
27801778
DrugRepV_0240Aimspro
NA
Multiple sclerosis
Ebola virus
ME718-1976/Yambuku-Ecran
NA
Real-time PCR
Increase (?4.60 ± 1.15 Ct)
Phase II
27801778
DrugRepV_0241NCK-8
NA
NA
Ebola virus
ME718-1976/Yambuku-Ecran
NA
Real-time PCR
Decrease (>10 Ct)
NA
27801778
DrugRepV_0242NCK-8
NA
NA
Ebola virus
ME718-1976/Yambuku-Ecran
NA
Real-time PCR
Decrease (>10 Ct)
NA
27801778
DrugRepV_0252Alvespimycin
NA
Cancer
Ebola virus
ME718-1976/Yambuku-Ecran
NA
Real-time PCR
Decrease (0.44 ± 0.06 Ct)
Investigational
27801778
DrugRepV_0257NCK-8
NA
NA
Ebola virus
ME718-1976/Yambuku-Ecran
NA
Real-time PCR
Decrease (1.54 ± 0.44 Ct)
NA
27801778
DrugRepV_0259Alvespimycin
NA
Cancer
Ebola virus
ME718-1976/Yambuku-Ecran
NA
NA
No significant effect
Investigational
27801778
DrugRepV_0261NCK-8
NA
NA
Ebola virus
ME718-1976/Yambuku-Ecran
NA
NA
No significant effect
NA
27801778
DrugRepV_0302PIK-75
NA
NA
Influenza virus
A/Anhui/1/ 2013
Pathway
Immunoflourescence assay
Decrease (50 %)
NA
26192013
DrugRepV_0303PIK-75
NA
NA
Influenza virus
A/California/04/09
Pathway
Immunoflourescence assay
Decrease (50 %)
NA
26192013
DrugRepV_0304PIK-75
NA
NA
Influenza virus
A/Philippines/2/82-X79
Pathway
Immunoflourescence assay
Decrease (50 %)
NA
26192013
DrugRepV_0309PIK-75
NA
NA
Influenza virus
A/Mississippi/3/01 wt
Pathway
TCID50 assay
Decrease (~1 Log10 virus titer (TCID50/ml))
NA
26192013
DrugRepV_0310PIK-75
NA
NA
Influenza virus
A/Mississippi/3/01 H275Y
Pathway
TCID50 assay
Decrease (~1 Log10 virus titer (TCID50/ml))
NA
26192013
DrugRepV_0315PIK-75
NA
NA
Influenza virus
A/Mississippi/3/01 wt
Pathway
Immunoflourescence assay
Decrease (90 %)
NA
26192013
DrugRepV_0316PIK-75
NA
NA
Influenza virus
A/Mississippi/3/01 H275Y
Pathway
Immunoflourescence assay
Decrease (85 %)
NA
26192013
DrugRepV_0406Quinacrine Dihydrochloride
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Ebola virus
eGFP-EBOV
NA
Fluorescence-based assay
Decrease (50 %)
Investigational
26041706
DrugRepV_0441Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Ebola virus
eGFP-EBOV
NA
Fluorescence-based assay
Decrease (50 %)
Investigational
26041706
DrugRepV_0469Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Ebola virus
eGFP-EBOV
NA
Fluorescence-based assay
Decrease (50 %)
Investigational
26041706
DrugRepV_0498Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Ebola virus
EBOV-VLP
NA
Flow cytometry
No significant effect
Investigational
26041706
DrugRepV_0551Tilorone
NA
Acquired immunodeficiency syndrome
Ebola virus
EBOVBlaVP40
NA
Fluorescence-based assay
Decrease (50 %)
Approved
26038505
DrugRepV_0559Nitrovin
NA
NA
Ebola virus
EBOVBlaVP40
NA
Fluorescence-based assay
Decrease (50 %)
NA
26038505
DrugRepV_0564Cyclomethycaine
NA
Anesthesia
Ebola virus
EBOVBlaVP40
NA
Fluorescence-based assay
Decrease (50 %)
Withdrawn
26038505
DrugRepV_0567Azaclorzine
NA
Anginal
Ebola virus
EBOVBlaVP40
NA
Fluorescence-based assay
Decrease (50 %)
NA
26038505
DrugRepV_0712Aminoquinoline-13
NA
Malaria
Marburg virus
GP derived Pseudovirus
NA
Luciferase reporter assay
Decrease (50 %)
NA
23577127
DrugRepV_0716Aminoquinoline-13
NA
Malaria
Marburg virus
Musoke
NA
Immunoflourescence assay
Decrease (50 %)
NA
23577127
DrugRepV_0720Aminoquinoline-13
NA
Malaria
Ebola virus
GP derived Pseudovirus
NA
Luciferase reporter assay
Decrease (50 %)
NA
23577127
DrugRepV_0724Aminoquinoline-13
NA
Malaria
Ebola virus
EBOLA-eGFP
NA
Fluorescence-based assay
Decrease (50 %)
NA
23577127
DrugRepV_0772Dactinomycin
NA
Cancer
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (99.435 %)
Approved
27476412
DrugRepV_0773Methotrexate
NA
Gestational choriocarcinoma | Chorioadenoma destruens | Hydatidiform mole | Meningeal leukemia | Breast cancer | Epidermoid cancers of the head and neck | Lung cancer
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (97.715 %)
Approved
27476412
DrugRepV_0896Prilocaine Hydrochloride
NA
Anesthesia
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (53.97 %)
Approved
27476412
DrugRepV_0955Guanfacine Hydrochloride
NA
Hypertension
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (53.975 %)
Approved, Investigational
27476412
DrugRepV_0985Mestranol
NA
Contraception
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (45.56 %)
Approved
27476412
DrugRepV_0989Ursodiol
NA
Gallstone and cholestatic forms of liver diseases including primary biliary cirrhosis
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (49.78 %)
Approved
27476412
DrugRepV_0997Metaxalone
NA
Musculoskeletal pain caused by strains, sprains, and other musculoskeletal conditions
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (50.445 %)
Approved
27476412
DrugRepV_1000Beclomethasone Dipropionate
NA
Allergic rhinitis
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (51.25 %)
Approved
27476412
DrugRepV_1033Zileuton
NA
Asthma
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (54.355 %)
Approved, Withdrawn
27476412
DrugRepV_1039Tiludronate Disodium
NA
Paget disease
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (46.63 %)
Approved, Investigational, Vet approved
27476412
DrugRepV_1067Midodrine Hydrochloride
NA
Orthostatic Hypotension
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (48.235 %)
Approved
27476412
DrugRepV_1115Niacin
NA
Hyperlipidemia
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (46.67 %)
Approved, Investigational, Nutraceutical
27476412
DrugRepV_1149Rizatriptan Benzoate
NA
Migraine disorders
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (44.98 %)
Approved
27476412
DrugRepV_1205Naringenin
NA
NA
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (46.34 %)
Experimental
27476412
DrugRepV_1224Galantamine Hydrobromide
NA
Alzheimer's disease
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (50.96 %)
Approved
27476412
DrugRepV_1269Carglumic Acid
NA
Hyperammonaemia in patients with N-acetylglutamate synthase (NAGS) deficiency
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (46.855 %)
Approved
27476412
DrugRepV_1290Gentamycin Sulfate
NA
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (47.715 %)
Approved
27476412
DrugRepV_1337Phytonadione
NA
Haemorrhagic conditions in infants | Antidote for coumarin anticoagulants in hypoprothrombinaemia
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (44.655 %)
Approved, Investigational
27476412
DrugRepV_1353Tetrahydrozoline Hydrochloride
NA
Discomfort and redness of the eye due to minor eye irritations
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (43.315 %)
Approved
27476412
DrugRepV_1394Tinidazole
NA
Trichomonasis | Amebiasis | Giardiasis
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (44.3 %)
Approved
27476412
DrugRepV_1417Difluprednate
NA
Anterior uveitis
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (41.575 %)
Approved
27476412
DrugRepV_1511Acyclovir Zovirax
NA
Viral infections (Herpes simplex, Zoster and varicella zoster)
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (42.46 %)
Approved
27476412
DrugRepV_1564Desmethyl Erlotinib
NA
Cancer
Rift Valley fever virus
MP12-Luc
NA
Luciferase reporter assay
Decrease (65 %)
Approved, Investigational
26217313
DrugRepV_1615Quinacrine Hydrochloride
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Ebola virus
Recombinant, infectious Ebola virus encoding green fluorescent protein
NA
Cell based assay
Decrease (50 %)
Investigational
26834994
DrugRepV_1617Tilorone Dihydrochloride
NA
Viral infections
Ebola virus
Recombinant, infectious Ebola virus encoding green fluorescent protein
NA
Cell based assay
Decrease (50 %)
NA
26834994
DrugRepV_1623Lavendustin A
NA
NA
Influenza virus
A/Anhui/01/2013
Pathway
Transcriptomic response-DEG
Decrease
NA
24991006
DrugRepV_1628D-serine
NA
NA
Influenza virus
A/Anhui/01/2013
Pathway
Transcriptomic response-DEG
Decrease
Approved
24991006
DrugRepV_16322,2-Dipyridyl Disulfide
NA
NA
Influenza virus
A/Anhui/01/2013
Pathway
Transcriptomic response-DEG
Decrease
Experimental
24991006
DrugRepV_1635Pobilukast
NA
NA
Influenza virus
A/Anhui/01/2013
Pathway
Transcriptomic response-DEG
Decrease
NA
24991006
DrugRepV_1636PD-180970
NA
NA
Influenza virus
A/Anhui/01/2013
Pathway
Transcriptomic response-DEG
Decrease
NA
24991006
DrugRepV_1637Methylanthraniloyl guanosine triphosphate
NA
NA
Influenza virus
A/Anhui/01/2013
Pathway
Transcriptomic response-DEG
Decrease
NA
24991006
DrugRepV_1638Mastoparan
NA
NA
Influenza virus
A/Anhui/01/2013
Pathway
Transcriptomic response-DEG
Decrease
NA
24991006
DrugRepV_1639Hexadimethrine Bromide
NA
NA
Influenza virus
A/Anhui/01/2013
Pathway
Transcriptomic response-DEG
Decrease
NA
24991006
DrugRepV_1640Dideooxyforskolin
NA
NA
Influenza virus
A/Anhui/01/2013
Pathway
Transcriptomic response-DEG
Decrease
NA
24991006
DrugRepV_1641Compound 48/80
NA
NA
Influenza virus
A/Anhui/01/2013
Pathway
Transcriptomic response-DEG
Decrease
NA
24991006
DrugRepV_16423-(N-methylanthraniloyl)-2-deoxy-ATP
NA
NA
Influenza virus
A/Anhui/01/2013
Pathway
Transcriptomic response-DEG
Decrease
NA
24991006
DrugRepV_16433-Aminotriazole
NA
NA
Influenza virus
A/Anhui/01/2013
Pathway
Transcriptomic response-DEG
Decrease
NA
24991006
DrugRepV_16442/3-O-N-methyanthraniloyl-ITP-gamma-S
NA
NA
Influenza virus
A/Anhui/01/2013
Pathway
Transcriptomic response-DEG
Decrease
NA
24991006
DrugRepV_16452/3-O-N-methyanthraniloyl-GTP-gamma-S
NA
NA
Influenza virus
A/Anhui/01/2013
Pathway
Transcriptomic response-DEG
Decrease
NA
24991006
DrugRepV_16462-(or3)-O-(N-methylanthranioyl)ATP
NA
NA
Influenza virus
A/Anhui/01/2013
Pathway
Transcriptomic response-DEG
Decrease
NA
24991006
DrugRepV_16472-Aminopurine
NA
NA
Influenza virus
A/Anhui/01/2013
Pathway
Transcriptomic response-DEG
Decrease
NA
24991006
DrugRepV_16481-cyclopropyl-3
NA
NA
Influenza virus
A/Anhui/01/2013
Pathway
Transcriptomic response-DEG
Decrease
NA
24991006
DrugRepV_1649Emricasan
NA
Antiapoptotic and anti-inflammatory
Zika virus
MR766
NA
Cell viability assay
Decrease (98.7 %)
Investigational
27571349
DrugRepV_1652Ensulizole
NA
Sunburn
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Approved
27571349
DrugRepV_1654Isoliquirtigenin
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Experimental
27571349
DrugRepV_1658Vidofludimus
NA
Crohn disease; Inflammatory bowel diseases and Rheumatoid arthritis
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Investigational
27571349
DrugRepV_1659SB-366791
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1660Emodin
NA
Polycystic Kidney
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Investigational
27571349
DrugRepV_1661Diphenyl isophthalate
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1662Benzoylpas
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1663Fenobam
NA
Fragile X Syndrome
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Investigational
27571349
DrugRepV_1665Drometrizole
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1666PHA-690509
NA
Cancer
Zika virus
MR766
NA
Cell viability assay
Decrease (81.9 %)
NA
27571349
DrugRepV_1670Cinanserin
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_16715-Nitro-2-(3-phenylpropylamino)benzoic Acid
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1672Veliflapon
NA
Myocardial infarction (Heart attack)
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Phase III
27571349
DrugRepV_1676Naringenin
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Experimental
27571349
DrugRepV_1678Fanetizole
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1681CAY10505
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1682Hesperetin
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Experimental
27571349
DrugRepV_1687Piraxostat
NA
NA
Zika virus
MR766
NA
Cell viability assay
Decrease (34.7 %)
NA
27571349
DrugRepV_1688Albendazole oxide
NA
Parasitic infections
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Experimental
27571349
DrugRepV_1689Tyrphostin AG 494
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1693RITA
NA
Cancer
Zika virus
MR766
NA
Cell viability assay
Decrease (81.7 %)
NA
27571349
DrugRepV_1695BF-170-hydrochloride
NA
NA
Zika virus
MR766
NA
Cell viability assay
Decrease (65.8 %)
NA
27571349
DrugRepV_1697Tribromsalan
NA
Bacterial infections
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1698Pifexole
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1699Formononetin
NA
Postmenopausal Osteopenia
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Investigational
27571349
DrugRepV_1701Tranilast
NA
Bronchial asthma | Keloid and hypertrophic scar | Allergic disorders such as asthma, allergic rhinitis | Atopic dermatitis
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Investigational
27571349
DrugRepV_1702Benzylparaben
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Approved, Experimental
27571349
DrugRepV_17032-Ethoxylethyl-p-methoxycinnamate
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1705Nemorubicin
NA
NA
Zika virus
MR766
NA
Cell viability assay
Decrease
NA
27571349
DrugRepV_1706Rutaecarpine
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1707MPEP
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_17085,7-Dihydroxyflavone
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_17112 Amino-6-nitrobenzothiazole
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1713Enfenamic Acid
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1714Fenaminosulf
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1715AS-252424
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1716Phenserine
NA
Alzheimer's disease
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Investigational
27571349
DrugRepV_1718Alizarin
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1720Emricasan
NA
Antiapoptotic and anti-inflammatory
Zika virus
MR766
NA
Cell viability assay
Decrease
Investigational
27571349
DrugRepV_1723Ensulizole
NA
Sunburn
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Approved
27571349
DrugRepV_1725Isoliquirtigenin
NA
NA
Zika virus
MR766
NA
Cell viability assay
Decrease (36.3 %)
Experimental
27571349
DrugRepV_1729Vidofludimus
NA
Crohn disease; Inflammatory bowel diseases and Rheumatoid arthritis
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Investigational
27571349
DrugRepV_1730SB-366791
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1731Emodin
NA
Polycystic Kidney
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Investigational
27571349
DrugRepV_1732Diphenyl isophthalate
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1733Benzoylpas
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1734Fenobam
NA
Fragile X Syndrome
Zika virus
MR766
NA
Cell viability assay
Decrease (60.5 %)
Investigational
27571349
DrugRepV_1736Drometrizole
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1737PHA-690509
NA
Cancer
Zika virus
MR766
NA
Cell viability assay
Decrease
NA
27571349
DrugRepV_1741Cinanserin
NA
NA
Zika virus
MR766
NA
Cell viability assay
Decrease (56.9 %)
NA
27571349
DrugRepV_17425-Nitro-2-(3-phenylpropylamino)benzoic Acid
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1743Veliflapon
NA
Myocardial infarction (Heart attack)
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Phase III
27571349
DrugRepV_1747Naringenin
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Experimental
27571349
DrugRepV_1749Fanetizole
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1752CAY10505
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1753Hesperetin
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Experimental
27571349
DrugRepV_1758Piraxostat
NA
NA
Zika virus
MR766
NA
Cell viability assay
Decrease (60.3 %)
NA
27571349
DrugRepV_1759Albendazole oxide
NA
Parasitic infections
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Experimental
27571349
DrugRepV_1760Tyrphostin AG 494
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (45.6 %)
NA
27571349
DrugRepV_1764RITA
NA
Cancer
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1766BF-170-hydrochloride
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1768Tribromsalan
NA
Bacterial infections
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1769Pifexole
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1770Formononetin
NA
Postmenopausal Osteopenia
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Investigational
27571349
DrugRepV_1772Tranilast
NA
Bronchial asthma | Keloid and hypertrophic scar | Allergic disorders such as asthma, allergic rhinitis | Atopic dermatitis
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Investigational
27571349
DrugRepV_1773Benzylparaben
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Approved, Experimental
27571349
DrugRepV_17742-Ethoxylethyl-p-methoxycinnamate
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1776Nemorubicin
NA
NA
Zika virus
MR766
NA
Cell viability assay
Decrease
NA
27571349
DrugRepV_1777Rutaecarpine
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1778MPEP
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_17795,7-Dihydroxyflavone
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_17822 Amino-6-nitrobenzothiazole
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1784Enfenamic Acid
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1785Fenaminosulf
NA
NA
Zika virus
MR766
NA
Cell viability assay
Decrease (36.7 %)
NA
27571349
DrugRepV_1786AS-252424
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1787Phenserine
NA
Alzheimer's disease
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Investigational
27571349
DrugRepV_1789Alizarin
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1791Emricasan
NA
Antiapoptotic and anti-inflammatory
Zika virus
MR766
NA
Cell viability assay
Decrease (54.4 %)
Investigational
27571349
DrugRepV_1794Ensulizole
NA
Sunburn
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Approved
27571349
DrugRepV_1796Isoliquirtigenin
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect
Experimental
27571349
DrugRepV_1800Vidofludimus
NA
Crohn disease; Inflammatory bowel diseases and Rheumatoid arthritis
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Investigational
27571349
DrugRepV_1801SB-366791
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect
NA
27571349
DrugRepV_1802Emodin
NA
Polycystic Kidney
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Investigational
27571349
DrugRepV_1803Diphenyl isophthalate
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1804Benzoylpas
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1805Fenobam
NA
Fragile X Syndrome
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Investigational
27571349
DrugRepV_1807Drometrizole
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1808PHA-690509
NA
Cancer
Zika virus
MR766
NA
Cell viability assay
No significant effect
NA
27571349
DrugRepV_1812Cinanserin
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_18135-Nitro-2-(3-phenylpropylamino)benzoic Acid
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1814Veliflapon
NA
Myocardial infarction (Heart attack)
Zika virus
MR766
NA
Cell viability assay
No significant effect
Phase III
27571349
DrugRepV_1818Naringenin
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect
Experimental
27571349
DrugRepV_1820Fanetizole
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1823CAY10505
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1824Hesperetin
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect
Experimental
27571349
DrugRepV_1829Piraxostat
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect
NA
27571349
DrugRepV_1830Albendazole oxide
NA
Parasitic infections
Zika virus
MR766
NA
Cell viability assay
No significant effect
Experimental
27571349
DrugRepV_1831Tyrphostin AG 494
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect
NA
27571349
DrugRepV_1835RITA
NA
Cancer
Zika virus
MR766
NA
Cell viability assay
No significant effect
NA
27571349
DrugRepV_1837BF-170-hydrochloride
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect
NA
27571349
DrugRepV_1839Tribromsalan
NA
Bacterial infections
Zika virus
MR766
NA
Cell viability assay
No significant effect
NA
27571349
DrugRepV_1840Pifexole
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect
NA
27571349
DrugRepV_1841Formononetin
NA
Postmenopausal Osteopenia
Zika virus
MR766
NA
Cell viability assay
No significant effect
Investigational
27571349
DrugRepV_1843Tranilast
NA
Bronchial asthma | Keloid and hypertrophic scar | Allergic disorders such as asthma, allergic rhinitis | Atopic dermatitis
Zika virus
MR766
NA
Cell viability assay
No significant effect
Investigational
27571349
DrugRepV_1844Benzylparaben
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
Approved, Experimental
27571349
DrugRepV_18452-Ethoxylethyl-p-methoxycinnamate
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1847Nemorubicin
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect
NA
27571349
DrugRepV_1848Rutaecarpine
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect
NA
27571349
DrugRepV_1849MPEP
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_18505,7-Dihydroxyflavone
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect
NA
27571349
DrugRepV_18532 Amino-6-nitrobenzothiazole
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1855Enfenamic Acid
NA
NA
Zika virus
MR766
NA
Cell viability assay
Decrease (58.5 %)
NA
27571349
DrugRepV_1856Fenaminosulf
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect
NA
27571349
DrugRepV_1857AS-252424
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1858Phenserine
NA
Alzheimer's disease
Zika virus
MR766
NA
Cell viability assay
No significant effect
Investigational
27571349
DrugRepV_1860Alizarin
NA
NA
Zika virus
MR766
NA
Cell viability assay
No significant effect (0 %)
NA
27571349
DrugRepV_1862Emricasan
NA
Antiapoptotic and anti-inflammatory
Zika virus
MR766 (1947 Ugandan strain)
NA
Cell viability assay
Decrease (50 %)
Investigational
27571349
DrugRepV_1863Emricasan
NA
Antiapoptotic and anti-inflammatory
Zika virus
FSS13025 (2010 Cambodian strain)
NA
Cell viability assay
Decrease (50 %)
Investigational
27571349
DrugRepV_1864Emricasan
NA
Antiapoptotic and anti-inflammatory
Zika virus
PRVABC-59 (2015 Puerto Rican strain)
NA
Cell viability assay
Decrease (50 %)
Investigational
27571349
DrugRepV_1865Emricasan
NA
Antiapoptotic and anti-inflammatory
Zika virus
NA
NA
Cell viability assay
Decrease (50 %)
Investigational
27571349
DrugRepV_1866Emricasan
NA
Antiapoptotic and anti-inflammatory
Zika virus
NA
NA
Cell viability assay
Decrease (50 %)
Investigational
27571349
DrugRepV_1867Emricasan
NA
Antiapoptotic and anti-inflammatory
Zika virus
NA
NA
Cell viability assay
Decrease (50 %)
Investigational
27571349
DrugRepV_1870PHA-690509
NA
Cancer
Zika virus
NA
NA
Cell viability assay
Decrease (50 %)
NA
27571349
DrugRepV_1871PHA-690509
NA
Cancer
Zika virus
NA
NA
Cell viability assay
Decrease (50 %)
NA
27571349
DrugRepV_1872PHA-690509
NA
Cancer
Zika virus
MR766 (1947 Ugandan strain)
NA
Western blot
Decrease (Decrease Band intensity)
NA
27571349
DrugRepV_1873PHA-690509
NA
Cancer
Zika virus
FSS13025 (2010 Cambodian strain)
NA
Western blot
Decrease (Decrease Band intensity)
NA
27571349
DrugRepV_1874PHA-690509
NA
Cancer
Zika virus
PRVABC-59 (2015 Puerto Rican strain)
NA
Western blot
Decrease (Decrease Band intensity)
NA
27571349
DrugRepV_1875PHA-690509
NA
Cancer
Zika virus
MR766 (1947 Ugandan strain)
NA
Western blot
Decrease (Decrease Band intensity)
NA
27571349
DrugRepV_1876PHA-690509
NA
Cancer
Zika virus
FSS13025 (2010 Cambodian strain)
NA
Western blot
Decrease (Decrease Band intensity)
NA
27571349
DrugRepV_1877PHA-690509
NA
Cancer
Zika virus
PRVABC-59 (2015 Puerto Rican strain)
NA
Western blot
Decrease (Decrease Band intensity)
NA
27571349
DrugRepV_1880PHA-690509
NA
Cancer
Zika virus
PRVABC-59 (2015 Puerto Rican strain)
NA
Enzyme-linked immunosorbent assay
Decrease
NA
27571349
DrugRepV_1882PHA-690509
NA
Cancer
Zika virus
PRVABC-59 (2015 Puerto Rican strain)
NA
Plaque assay
Decrease (50 %)
NA
27571349
DrugRepV_1885PHA-690509
NA
Cancer
Zika virus
FSS13026
NA
Real-time PCR
Decrease (50 %)
NA
27571349
DrugRepV_1887PHA-690509
NA
Cancer
Zika virus
FSS13026
NA
Real-time PCR
Decrease
NA
27571349
DrugRepV_1890PHA-690509
NA
Cancer
Zika virus
PRVABC-59 (2015 Puerto Rican strain)
NA
Western blot
Decrease (Decrease Band intensity)
NA
27571349
DrugRepV_1891PHA-690509
NA
Cancer
Zika virus
PRVABC-59 (2015 Puerto Rican strain)
NA
Western blot
Decrease (Decrease Band intensity)
NA
27571349
DrugRepV_1893SNS-032
NA
Cancer
Zika virus
FSS13026
NA
NA
Decrease (50 %)
Investigational
27571349
DrugRepV_1895AT7519
NA
Cancer
Zika virus
FSS13026
NA
NA
Decrease (50 %)
NA
27571349
DrugRepV_1897RGB-286147
NA
NA
Zika virus
FSS13026
NA
NA
Decrease (50 %)
NA
27571349
DrugRepV_1899Alvocidib
NA
Cancer
Zika virus
FSS13026
NA
NA
Decrease (50 %)
Experimental
27571349
DrugRepV_1900PHA-690509
NA
Cancer
Zika virus
FSS13026
NA
Western blot
Decrease (Decrease Band intensity)
NA
27571349
DrugRepV_1901Alvocidib
NA
Cancer
Zika virus
FSS13026
NA
Western blot
Decrease (Decrease Band intensity)
Experimental
27571349
DrugRepV_1905PHA-690509
NA
Cancer
Zika virus
PRVABC-59 (2015 Puerto Rican strain)
NA
Western blot
Decrease (Decrease Band intensity)
NA
27571349
DrugRepV_1906Alvocidib
NA
Cancer
Zika virus
PRVABC-59 (2015 Puerto Rican strain)
NA
Western blot
Decrease (Decrease Band intensity)
Experimental
27571349
DrugRepV_1965Fenretinide-Butylated Hydroxyanisole
NA
NA
Influenza virus
Strain A/PR8/ 34
Pathway
Plaque assay
No significant effect
Investigational
25313218
DrugRepV_2029Levonordefrin
NA
Dental disorders
Ebola virus
Zaire strain-pEBOV
NA
Firefly luciferase assay
Decrease (50 %)
Approved
26585243
DrugRepV_2070Phenothrin
NA
NA
Lassa virus
LASVpv
NA
Luciferase reporter assay
Decrease (50 %)
Experimental
29899092
DrugRepV_2079Tiotidine
NA
NA
Ebola virus
HIV/EBOV
NA
Luciferase reporter assay
No significant decrease (50 %)
NA
29981374
DrugRepV_2080Tiotidine
NA
NA
Marburg virus
HIV/MARV
NA
Luciferase reporter assay
No significant decrease (50 %)
NA
29981374
DrugRepV_2081Impentamine
NA
NA
Ebola virus
HIV/EBOV
NA
Luciferase reporter assay
No significant decrease (50 %)
NA
29981374
DrugRepV_2082Impentamine
NA
NA
Marburg virus
HIV/MARV
NA
Luciferase reporter assay
No significant decrease (50 %)
NA
29981374
DrugRepV_2085Nordiphenhydramine
NA
NA
Ebola virus
HIV/EBOV
NA
Luciferase reporter assay
Decrease (50 %)
NA
29981374
DrugRepV_2086Nordiphenhydramine
NA
NA
Marburg virus
HIV/MARV
NA
Luciferase reporter assay
Decrease (50 %)
NA
29981374
DrugRepV_21322-C-Methylcytidine
NA
Hepatitis C virus
Zika virus
MR766
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Experimental
27163257
DrugRepV_21332-C-Methylcytidine
NA
Hepatitis C virus
Zika virus
MR766
NA
Virus yield reduction assay
Decrease (50 %)
Experimental
27163257
DrugRepV_21347-deaza-2-C-methyl-D-adenosine
NA
Viral infection
Zika virus
MR766
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
27163257
DrugRepV_21357-deaza-2-C-methyl-D-adenosine
NA
Viral infection
Zika virus
MR766
NA
Virus yield reduction assay
Decrease (50 %)
NA
27163257
DrugRepV_21367-deaza-2-C-methyl-D-adenosine
NA
Viral infection
Zika virus
MR766
NA
Plaque assay
Decrease (50 %)
NA
27163257
DrugRepV_21377-deaza-2-C-methyl-D-adenosine
NA
Viral infection
Zika virus
MR766
NA
Immunoflourescence assay
Decrease (50 %)
NA
27163257
DrugRepV_21387-deaza-2-C-methyl-D-adenosine
NA
Viral infection
Zika virus
MR766
NA
Survival assay
Increase
NA
27163257
DrugRepV_21397-deaza-2-C-methyl-D-adenosine
NA
Viral infection
Zika virus
MR766
NA
Real-time PCR
Decrease
NA
27163257
DrugRepV_2140BCX4430 Dihydrochloride
NA
Ebola virus
Zika virus
Puerto Rican strain PRVABC-59
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Phase I
27838352
DrugRepV_2141BCX4430 Dihydrochloride
NA
Ebola virus
Zika virus
Puerto Rican strain PRVABC-59
NA
Virus yield reduction assay
Decrease (90 %)
Phase I
27838352
DrugRepV_2142BCX4430 Dihydrochloride
NA
Ebola virus
Zika virus
Puerto Rican strain PRVABC-59
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Phase I
27838352
DrugRepV_2143BCX4430 Dihydrochloride
NA
Ebola virus
Zika virus
Puerto Rican strain PRVABC-59
NA
Virus yield reduction assay
Decrease (90 %)
Phase I
27838352
DrugRepV_2144BCX4430 Dihydrochloride
NA
Ebola virus
Zika virus
Puerto Rican strain PRVABC-59
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Phase I
27838352
DrugRepV_2145BCX4430 Dihydrochloride
NA
Ebola virus
Zika virus
Puerto Rican strain PRVABC-59
NA
Virus yield reduction assay
Decrease (90 %)
Phase I
27838352
DrugRepV_2146BCX4430 Dihydrochloride
NA
Ebola virus
Zika virus
Malaysian P 6-740
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Phase I
27838352
DrugRepV_2147BCX4430 Dihydrochloride
NA
Ebola virus
Zika virus
Malaysian P 6-740
NA
Virus yield reduction assay
Decrease (90 %)
Phase I
27838352
DrugRepV_2148BCX4430 Dihydrochloride
NA
Ebola virus
Zika virus
Malaysian P 6-740
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Phase I
27838352
DrugRepV_2149BCX4430 Dihydrochloride
NA
Ebola virus
Zika virus
Malaysian P 6-740
NA
Virus yield reduction assay
Decrease (90 %)
Phase I
27838352
DrugRepV_2150BCX4430 Dihydrochloride
NA
Ebola virus
Zika virus
Ugandan MR-766
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Phase I
27838352
DrugRepV_2151BCX4430 Dihydrochloride
NA
Ebola virus
Zika virus
Ugandan MR-766
NA
Virus yield reduction assay
Decrease (90 %)
Phase I
27838352
DrugRepV_2152BCX4430 Dihydrochloride
NA
Ebola virus
Zika virus
Ugandan MR-766
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Phase I
27838352
DrugRepV_2153BCX4430 Dihydrochloride
NA
Ebola virus
Zika virus
Ugandan MR-766
NA
Virus yield reduction assay
Decrease (90 %)
Phase I
27838352
DrugRepV_2154BCX4430 Dihydrochloride
NA
Ebola virus
Zika virus
Ugandan MR-766
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Phase I
27838352
DrugRepV_2155BCX4430 Dihydrochloride
NA
Ebola virus
Zika virus
Ugandan MR-766
NA
Virus yield reduction assay
Decrease (90 %)
Phase I
27838352
DrugRepV_2177Avobenzone
NA
Sunburn
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (16.643533 %)
Approved
27742486
DrugRepV_2215Fudosteine
NA
Bronchial asthma | Chronic bronchitis | Pulmonary emphysema | Bronchiectasis | Pulmonary tuberculosis | Pneumoconiosis | Atypical mycobacterial disease
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (7.62256156 %)
NA
27742486
DrugRepV_2220Tylosin tartrate
NA
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (7.36358127 %)
Vet Approved
27742486
DrugRepV_2235Arbidol Hydrochloride
NA
Influenza
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (6.59070859 %)
NA
27742486
DrugRepV_2241Novobiocin Sodium
NA
Staphylococci infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (6.24445866 %)
Approved, Investigational, Vet approved
27742486
DrugRepV_2244Azacyclonol
NA
Psychosis
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (6.14203789 %)
NA
27742486
DrugRepV_2261Azasetron Hydrochloride
NA
Nausea and vomiting induced by cancer chemotherapy
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (5.49334625 %)
NA
27742486
DrugRepV_2280OSI-420
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (4.78127734 %)
NA
27742486
DrugRepV_2294Daidzein
NA
Dietary supplement
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (4.45147852 %)
Experimental
27742486
DrugRepV_2296Adenine Hydrochloride
NA
Nutritional supplement
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (4.42334798 %)
Approved
27742486
DrugRepV_2323Geniposide
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (3.7860683 %)
NA
27742486
DrugRepV_2329Chloroxine
NA
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (3.67704383 %)
Approved
27742486
DrugRepV_2337Adiphenine Hydrochloride
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (3.4400476 %)
NA
27742486
DrugRepV_2357Mecarbinate
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (3.00956049 %)
NA
27742486
DrugRepV_2370Cytidine
NA
Biopolar Depression
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (2.69043453 %)
Experimental
27742486
DrugRepV_2381Niacin
NA
Hyperlipidemia
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (2.44049164 %)
Approved, Investigational, Nutraceutical
27742486
DrugRepV_2388Albendazole oxide
NA
Parasitic infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (2.36721682 %)
Experimental
27742486
DrugRepV_2392Geniposidic Acid
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (2.33842957 %)
NA
27742486
DrugRepV_2399Paeoniflorin
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (2.22636429 %)
NA
27742486
DrugRepV_2407Adenine
NA
Nutritional supplement
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (2.12499687 %)
Approved
27742486
DrugRepV_2415Adenine Sulfate
NA
Nutritional supplement
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (1.95953472 %)
Approved
27742486
DrugRepV_2465Sodium Butyrate
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (0.80232337 %)
NA
27742486
DrugRepV_2471Azelnidipine
NA
Hypertension
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (0.64469838 %)
Approved
27742486
DrugRepV_2477Mestranol
NA
Contraception
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (0.44756785 %)
Approved
27742486
DrugRepV_2488Aspartame
NA
Diet supplement and sugar substitute
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (0.28008959 %)
Approved
27742486
DrugRepV_2494Curcumin
NA
Depressive disorder
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (0.21930657 %)
Approved
27742486
DrugRepV_2515Talc
NA
Rashes
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-0.1085991 %)
Approved
27742486
DrugRepV_2521Pregnenolone
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-0.2797662 %)
Approved, Experimental
27742486
DrugRepV_2533Pimobendan
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-0.5850328 %)
Vet approved
27742486
DrugRepV_2538Alibendol
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-0.6238122 %)
NA
27742486
DrugRepV_2539Vicriviroc Malate
NA
AIDS
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-0.6325066 %)
Investigational
27742486
DrugRepV_2542Sodium orthovanadate
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-0.6967088 %)
NA
27742486
DrugRepV_2545Irsogladine
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-0.8011514 %)
Investigational
27742486
DrugRepV_2563Detomidine Hydrochloride
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-1.086047 %)
Approved, Vet Approved
27742486
DrugRepV_2564Hydroxyflutamide
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-1.1400626 %)
NA
27742486
DrugRepV_2570Ursodiol
NA
Gallstone and cholestatic forms of liver diseases including primary biliary cirrhosis
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-1.242893 %)
Approved
27742486
DrugRepV_2596Methacycline Hydrochloride
NA
Acute bacterial exacerbations of chronic bronchitis
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-1.5238499 %)
Approved, Investigational
27742486
DrugRepV_26102-Methoxyestradiol
NA
Cancer
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-1.7014075 %)
Investigational
27742486
DrugRepV_2619Nafamostat Mesylate
NA
Blood vessel coagulation | Hemorrhagic lesions
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-1.7795584 %)
Investigational
27742486
DrugRepV_2623Liranaftate
NA
Fungal infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-1.8068752 %)
NA
27742486
DrugRepV_2625NAD
NA
Parkinson's disease | Chronic fatigue syndrome | Alzheimer's disease | Cardiovascular disease
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-1.8213385 %)
Approved
27742486
DrugRepV_2633Zileuton
NA
Asthma
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-1.9379253 %)
Approved, Withdrawn
27742486
DrugRepV_2650Bepotastine besilate
NA
Allergic rhinitis and uriticaria/puritus
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-2.1704391 %)
Approved
27742486
DrugRepV_2668Moguisteine
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-2.4037393 %)
NA
27742486
DrugRepV_268310-DAB
NA
Cancer
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-2.5981982 %)
NA
27742486
DrugRepV_2692Dextrose
NA
Hypoglycemia
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-2.8688015 %)
Approved
27742486
DrugRepV_2709Arecoline
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-3.0469253 %)
Experimental
27742486
DrugRepV_2746Gabexate Mesylate
NA
Cancer | Ischemia-reperfusion injury | Pancreatitis
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-3.7539063 %)
Investigational
27742486
DrugRepV_2751Marbofloxacin
NA
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-3.8874309 %)
Vet approved
27742486
DrugRepV_2763Taurine
NA
Nutritional supplementation
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-4.1985759 %)
Approved
27742486
DrugRepV_2780BIBR 953
NA
Hypertension
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-4.5344416 %)
Approved
27742486
DrugRepV_2811Cefoselis Sulfate
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-5.3205301 %)
NA
27742486
DrugRepV_2813Rizatriptan Benzoate
NA
Migraine disorders
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-5.3908172 %)
Approved
27742486
DrugRepV_28142-Thiouracil
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-5.4015713 %)
NA
27742486
DrugRepV_2818Suplatast tosylate
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-5.4609451 %)
NA
27742486
DrugRepV_2831Xylazine Hydrochloride
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-5.9275587 %)
Approved, Vet Approved
27742486
DrugRepV_2843Danofloxacin Mesylate
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-6.3487008 %)
Experimental, Vet approved
27742486
DrugRepV_2856Amidopyrine
NA
Pain
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-6.8828073 %)
NA
27742486
DrugRepV_2861Ubenimex
NA
Acute myelocytic leukemia
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-7.1327673 %)
Approved
27742486
DrugRepV_2878Betapar
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-8.1507562 %)
NA
27742486
DrugRepV_2889Malotilate
NA
Liver disease
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-8.5901104 %)
NA
27742486
DrugRepV_2891PMSF
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-8.6777643 %)
NA
27742486
DrugRepV_2907Tranilast
NA
Bronchial asthma | Keloid and hypertrophic scar | Allergic disorders such as asthma, allergic rhinitis | Atopic dermatitis
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-9.5539143 %)
Investigational
27742486
DrugRepV_2913Noradrenaline Bitartrate Monohydrate
NA
NA
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-9.8741533 %)
NA
27742486
DrugRepV_2961Doxycycline-Ribavirin
NA
NA
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
Enzyme-linked immunosorbent assay
Decrease (50 %)
Approved
25970853
DrugRepV_2964Doxycycline-Ribavirin
NA
NA
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
Enzyme-linked immunosorbent assay
Decrease (95 %)
Approved
25970853
DrugRepV_2967Doxycycline-Ribavirin
NA
NA
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
Plaque assay
Decrease (91 %)
Approved
25970853
DrugRepV_2970Doxycycline-Ribavirin
NA
NA
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
Plaque assay
Decrease (92 %)
Approved
25970853
DrugRepV_2973Doxycycline-Ribavirin
NA
NA
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
Plaque assay
Decrease (91 %)
Approved
25970853
DrugRepV_2976Doxycycline-Ribavirin
NA
NA
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
MTT assay
Decrease (88.2 %)
Approved
25970853
DrugRepV_2977Apigenin
NA
NA
Chikungunya virus
CHIKV replicon
NA
EGFP assay
Decrease (50 %)
Experimental
22205980
DrugRepV_2979Naringenin
NA
NA
Chikungunya virus
CHIKV replicon
NA
EGFP assay
Decrease (50 %)
Experimental
22205980
DrugRepV_2980Silybin
NA
NA
Chikungunya virus
CHIKV replicon
NA
EGFP assay
Decrease (50 %)
Experimental, Investigational
22205980
DrugRepV_29846-Azauridine
NA
Cancer
Chikungunya virus
CHIKV replicon
NA
EGFP assay
Decrease (50 %)
NA
22205980
DrugRepV_29853-NH2-3-deoxyadenosine
NA
NA
Chikungunya virus
CHIKV replicon
NA
EGFP assay
Decrease (50 %)
NA
22205980
DrugRepV_2986Apigenin
NA
NA
Chikungunya virus
CHIKV replicon
NA
Rluc assay
Decrease (50 %)
Experimental
22205980
DrugRepV_2988Naringenin
NA
NA
Chikungunya virus
CHIKV replicon
NA
Rluc assay
Decrease (50 %)
Experimental
22205980
DrugRepV_2989Silybin
NA
NA
Chikungunya virus
CHIKV replicon
NA
Rluc assay
Decrease (50 %)
Experimental, Investigational
22205980
DrugRepV_29936-Azauridine
NA
Cancer
Chikungunya virus
CHIKV replicon
NA
Rluc assay
Decrease (50 %)
NA
22205980
DrugRepV_29943-NH2-3-deoxyadenosine
NA
NA
Chikungunya virus
CHIKV replicon
NA
Rluc assay
Decrease (50 %)
NA
22205980
DrugRepV_2999Sulfonyl Amidine
NA
NA
Chikungunya virus
NA
NA
Plaque assay
Decrease (10 %)
NA
25643977
DrugRepV_3000Sulfonyl Amidine
NA
NA
Chikungunya virus
NA
NA
Plaque assay
Decrease (40 %)
NA
25643977
DrugRepV_3011Curcumin
NA
Cancer, mucositis, chronic schizophrenia and mild cognitive impairment
Zika virus
HD78788
NA
Plaque assay
Decrease (75 %)
Approved
28343845
DrugRepV_3012Curcumin
NA
Cancer, mucositis, chronic schizophrenia and mild cognitive impairment
Zika virus
HD78788
NA
Real-time PCR
Decrease
Approved
28343845
DrugRepV_3013Curcumin
NA
Cancer, mucositis, chronic schizophrenia and mild cognitive impairment
Zika virus
HD78788
NA
Real-time PCR
Decrease (0.8 log)
Approved
28343845
DrugRepV_3014Curcumin
NA
Cancer, mucositis, chronic schizophrenia and mild cognitive impairment
Chikungunya virus
La Reunion strain, 06-049 AM258994
NA
Real-time PCR
Decrease (1 log)
Approved
28343845
DrugRepV_3015Curcumin
NA
Cancer, mucositis, chronic schizophrenia and mild cognitive impairment
Zika virus
HD78788
NA
Real-time PCR
Decrease (1 log)
Approved
28343845
DrugRepV_3016Curcumin
NA
Cancer, mucositis, chronic schizophrenia and mild cognitive impairment
Zika virus
HD78788
NA
Real-time PCR
Decrease (1 log)
Approved
28343845
DrugRepV_3017Curcumin
NA
Cancer, mucositis, chronic schizophrenia and mild cognitive impairment
Chikungunya virus
La Reunion strain, 06-049 AM258994
NA
Real-time PCR
Decrease (0.7 log)
Approved
28343845
DrugRepV_3018Curcumin
NA
Cancer, mucositis, chronic schizophrenia and mild cognitive impairment
Chikungunya virus
La Reunion strain, 06-049 AM258994
NA
Real-time PCR
Decrease (0.8 log)
Approved
28343845
DrugRepV_3019Curcumin
NA
Cancer, mucositis, chronic schizophrenia and mild cognitive impairment
Chikungunya virus
La Reunion strain, 06-049 AM258994
NA
Real-time PCR
Decrease (0.5 log)
Approved
28343845
DrugRepV_3020Demethoxycurcumin
NA
NA
Zika virus
HD78788
NA
Plaque assay
Decrease
Phase II
28343845
DrugRepV_3022EF-24
NA
NA
Zika virus
HD78788
NA
Plaque assay
Decrease
NA
28343845
DrugRepV_3023FLLL31
NA
NA
Zika virus
HD78788
NA
Plaque assay
Decrease
NA
28343845
DrugRepV_3024Demethoxycurcumin
NA
NA
Chikungunya virus
La Reunion strain, 06-049 AM258994
NA
Plaque assay
Decrease
Phase II
28343845
DrugRepV_3026EF-24
NA
NA
Chikungunya virus
La Reunion strain, 06-049 AM258994
NA
Plaque assay
Decrease
NA
28343845
DrugRepV_3027FLLL31
NA
NA
Chikungunya virus
La Reunion strain, 06-049 AM258994
NA
Plaque assay
Decrease
NA
28343845
DrugRepV_3028Demethoxycurcumin
NA
NA
Zika virus
HD78788
NA
Plaque assay
Decrease (50 %)
Phase II
28343845
DrugRepV_3030EF-24
NA
NA
Zika virus
HD78788
NA
Plaque assay
Decrease (50 %)
NA
28343845
DrugRepV_3031FLLL31
NA
NA
Zika virus
HD78788
NA
Plaque assay
Decrease (50 %)
NA
28343845
DrugRepV_3032Curcumin
NA
Cancer, mucositis, chronic schizophrenia and mild cognitive impairment
Zika virus
HD78788
NA
Plaque assay
Decrease (50 %)
Approved
28343845
DrugRepV_3033Demethoxycurcumin
NA
NA
Chikungunya virus
La Reunion strain, 06-049 AM258994
NA
Plaque assay
Decrease (50 %)
Phase II
28343845
DrugRepV_3035EF-24
NA
NA
Chikungunya virus
La Reunion strain, 06-049 AM258994
NA
Plaque assay
Decrease (50 %)
NA
28343845
DrugRepV_3036FLLL31
NA
NA
Chikungunya virus
La Reunion strain, 06-049 AM258994
NA
Plaque assay
Decrease (50 %)
NA
28343845
DrugRepV_3037Curcumin
NA
Cancer, mucositis, chronic schizophrenia and mild cognitive impairment
Chikungunya virus
La Reunion strain, 06-049 AM258994
NA
Plaque assay
Decrease (50 %)
Approved
28343845
DrugRepV_3038Berberine
NA
Parasitic and fungal infection
Chikungunya virus
LR2006 OPY1
NA
Luciferase reporter assay
Decrease (50 %)
Approved
26752081
DrugRepV_3039Abamectin
NA
Helmintic infection
Chikungunya virus
LR2006 OPY1
NA
Luciferase reporter assay
Decrease (50 %)
Terminated
26752081
DrugRepV_3043Berberine
NA
Parasitic and fungal infection
Chikungunya virus
LR2006 OPY1
NA
Luciferase reporter assay
Decrease (50 %)
Approved
26752081
DrugRepV_3044Abamectin
NA
Helmintic infection
Chikungunya virus
LR2006 OPY1
NA
Luciferase reporter assay
Decrease (50 %)
Terminated
26752081
DrugRepV_3048Abamectin
NA
Helmintic infection
Chikungunya virus
CHIKV-Rluc
NA
Luciferase reporter assay
Decrease (100 %)
Terminated
26752081
DrugRepV_3050Berberine
NA
Parasitic and fungal infection
Chikungunya virus
CHIKV-Rluc
NA
Luciferase reporter assay
Decrease (87 %)
Approved
26752081
DrugRepV_3061Abamectin
NA
Helmintic infection
Chikungunya virus
CHIKV-Rluc
NA
Renilla luciferase assay
No significant effect (No significant effect %)
Terminated
26752081
DrugRepV_3063Berberine
NA
Parasitic and fungal infection
Chikungunya virus
CHIKV-Rluc
NA
Renilla luciferase assay
No significant effect (No significant effect %)
Approved
26752081
DrugRepV_3066Abamectin
NA
Helmintic infection
Chikungunya virus
CHIKV-Rluc
NA
Northern blot
Decrease
Terminated
26752081
DrugRepV_3068Abamectin
NA
Helmintic infection
Chikungunya virus
CHIKV-Rluc
NA
Western blot
Decrease
Terminated
26752081
DrugRepV_3069Abamectin
NA
Helmintic infection
Chikungunya virus
CHIKV-Rluc
NA
Western blot
Decrease
Terminated
26752081
DrugRepV_3072Abamectin
NA
Helmintic infection
Chikungunya virus
CHIKV-Rluc
NA
Western blot
Decrease
Terminated
26752081
DrugRepV_3073Abamectin
NA
Helmintic infection
Chikungunya virus
CHIKV-Rluc
NA
Western blot
Decrease
Terminated
26752081
DrugRepV_3076Abamectin
NA
Helmintic infection
Chikungunya virus
CHIKV-Rluc
NA
Plaque assay
Decrease (3.5 Log)
Terminated
26752081
DrugRepV_3077Berberine
NA
Parasitic and fungal infection
Chikungunya virus
CHIKV-Rluc
NA
Plaque assay
Decrease (5.2 Log)
Approved
26752081
DrugRepV_3082Abamectin
NA
Helmintic infection
Chikungunya virus
NA
NA
Plaque assay
Decrease (2 Log)
Terminated
26752081
DrugRepV_3083Berberine
NA
Parasitic and fungal infection
Chikungunya virus
NA
NA
Plaque assay
Decrease (3.3 Log)
Approved
26752081
DrugRepV_3085Abamectin
NA
Helmintic infection
Chikungunya virus
NA
NA
Plaque assay
Decrease (0.3 Log)
Terminated
26752081
DrugRepV_3086Berberine
NA
Parasitic and fungal infection
Chikungunya virus
NA
NA
Plaque assay
Decrease (1.2 Log)
Approved
26752081
DrugRepV_3089Dipterocarpol
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (100 %)
NA
23275491
DrugRepV_3091Aloe-emodin
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (99.89 %)
NA
23275491
DrugRepV_3092Retrorsine
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (99.84 %)
NA
23275491
DrugRepV_3094Harringtonine
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (99.76 %)
NA
23275491
DrugRepV_3096Tunicamycin B
NA
Bacterial infections
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (99.7 %)
Experimental
23275491
DrugRepV_3097Corydaline
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (99.69 %)
NA
23275491
DrugRepV_3100Usnic Acid
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (99.54 %)
NA
23275491
DrugRepV_3101Rhapontin
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (99.53 %)
NA
23275491
DrugRepV_3103Ferutinin
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (99.43 %)
NA
23275491
DrugRepV_3104Diacetoxyscirpenol
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (99.27 %)
NA
23275491
DrugRepV_3107Acivicin
NA
Cancer
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (99.07 %)
Phase I
23275491
DrugRepV_3109Jervine
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (98.35 %)
NA
23275491
DrugRepV_3110Hypocrellin B
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (98.08 %)
NA
23275491
DrugRepV_3111Valinomycin
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (97.79 %)
Experimental
23275491
DrugRepV_3112Hypocrellin A
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (97.64 %)
NA
23275491
DrugRepV_3114E-64
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (95.94 %)
NA
23275491
DrugRepV_3115Magnolol
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (95.74 %)
NA
23275491
DrugRepV_3117Nonactin
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (95.31 %)
NA
23275491
DrugRepV_3119Ochratoxin A
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (94.95 %)
NA
23275491
DrugRepV_3121Parthenolide
NA
Allergic Contact Dermatitis
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (93.95 %)
Approved, Investigational
23275491
DrugRepV_3124Rottlerin
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (92.81 %)
NA
23275491
DrugRepV_3125Grayanotoxin III
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (91.39 %)
NA
23275491
DrugRepV_3126Gossypol
NA
Non-small Cell Lung Cancer
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (90.89 %)
Investigational
23275491
DrugRepV_3127Sanguinarine
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (90.83 %)
NA
23275491
DrugRepV_3130Cyclopiazonic Acid
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (79.93 %)
NA
23275491
DrugRepV_3131Harmine Hydrochloride
NA
NA
Chikungunya virus
CHIKV-0708
NA
Immunoflourescence assay
Decrease (73.68 %)
NA
23275491
DrugRepV_3132Harringtonine
NA
NA
Chikungunya virus
CHIKV-0708
NA
Plaque assay
Decrease (50 %)
NA
23275491
DrugRepV_3133Hypocrellin A
NA
NA
Chikungunya virus
CHIKV-0708
NA
Plaque assay
Decrease (50 %)
NA
23275491
DrugRepV_3134Rottlerin
NA
NA
Chikungunya virus
CHIKV-0708
NA
Plaque assay
Decrease (50 %)
NA
23275491
DrugRepV_3136Harringtonine
NA
NA
Chikungunya virus
CHIKV-122508
NA
Plaque assay
Decrease (4.3 Log)
NA
23275491
DrugRepV_3137Harringtonine
NA
NA
Chikungunya virus
CHIKV-0708
NA
Plaque assay
Decrease (2.3 Log)
NA
23275491
DrugRepV_3140Harringtonine
NA
NA
Chikungunya virus
CHIKV-0708
NA
Plaque assay
Decrease (3 Log)
NA
23275491
DrugRepV_3141Harringtonine
NA
NA
Chikungunya virus
CHIKV-122508
NA
Plaque assay
Decrease (3.5 Log)
NA
23275491
DrugRepV_3142Harringtonine
NA
NA
Chikungunya virus
CHIKV-0708
NA
Plaque assay
Decrease (2.8 Log)
NA
23275491
DrugRepV_3143Harringtonine
NA
NA
Chikungunya virus
CHIKV-0708
NA
Plaque assay
Decrease (7.8 Log)
NA
23275491
DrugRepV_3144Harringtonine
NA
NA
Chikungunya virus
CHIKV-0708
NA
Plaque assay
Decrease (6.4 Log)
NA
23275491
DrugRepV_3145Harringtonine
NA
NA
Chikungunya virus
CHIKV-0708
NA
Real-time PCR
Decrease (6 (Complete inhibition) Log)
NA
23275491
DrugRepV_3146Harringtonine
NA
NA
Chikungunya virus
CHIKV-0708
NA
Real-time PCR
Decrease (2 Log)
NA
23275491
DrugRepV_3147Harringtonine
NA
NA
Chikungunya virus
CHIKV-0708
NA
Real-time PCR
Decrease (2 Log)
NA
23275491
DrugRepV_3148Harringtonine
NA
NA
Chikungunya virus
CHIKV-122508
NA
Real-time PCR
Decrease (2.4 Log)
NA
23275491
DrugRepV_3149Harringtonine
NA
NA
Chikungunya virus
CHIKV-122508
NA
Real-time PCR
Decrease (3 Log)
NA
23275491
DrugRepV_3150Harringtonine
NA
NA
Chikungunya virus
CHIKV-0708
NA
Western blot
Decrease
NA
23275491
DrugRepV_3151Harringtonine
NA
NA
Chikungunya virus
CHIKV-122508
NA
Western blot
Decrease
NA
23275491
DrugRepV_3152Harringtonine
NA
NA
Chikungunya virus
CHIKV-0708
NA
Western blot
Decrease
NA
23275491
DrugRepV_3153Harringtonine
NA
NA
Chikungunya virus
CHIKV-0708
NA
Western blot
Decrease
NA
23275491
DrugRepV_3154Harringtonine
NA
NA
Chikungunya virus
CHIKV-122508
NA
Western blot
Decrease
NA
23275491
DrugRepV_3155Harringtonine
NA
NA
Chikungunya virus
CHIKV-122508
NA
Western blot
Decrease
NA
23275491
DrugRepV_31576-Azauridine
NA
Cancer
Chikungunya virus
Ross C347
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
14670584
DrugRepV_3160Fucoidan
NA
NA
Chikungunya virus
Ross C347
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
14670584
DrugRepV_31656-Azauridine
NA
Cancer
Chikungunya virus
Ross C347
NA
Cytopathic effect (CPE) assay
Decrease (1.8 Log)
NA
14670584
DrugRepV_31696-Azauridine
NA
Cancer
Chikungunya virus
Ross C347
NA
Cytopathic effect (CPE) assay
Decrease (99 %)
NA
14670584
DrugRepV_3172IFN-alpha2b-Ribavirin
NA
NA
Chikungunya virus
Ross C347
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
14670584
DrugRepV_3181Arbidol
NA
Viral infection
Influenza virus
A/Aichi/2/68
Pathway
Plaque assay
Decrease (50 %)
Investigational
22028179
DrugRepV_3182Arbidol
NA
Viral infection
Influenza virus
B/Beijing/184/93
Pathway
Plaque assay
Decrease (50 %)
Investigational
22028179
DrugRepV_3183Arbidol
NA
Viral infection
Influenza virus
A/Mem Bel
Pathway
Plaque assay
Decrease (50 %)
Investigational
22028179
DrugRepV_3184Arbidol
NA
Viral infection
Influenza virus
A/Queensland/6/72
Pathway
Plaque assay
Decrease (50 %)
Investigational
22028179
DrugRepV_3185Arbidol
NA
Viral infection
Influenza virus
A/Sydney/5/ 97
Pathway
Plaque assay
Decrease (50 %)
Investigational
22028179
DrugRepV_3186Arbidol
NA
Viral infection
Influenza virus
A/Moscow/16/98
Pathway
Plaque assay
Decrease (50 %)
Investigational
22028179
DrugRepV_3187Arbidol
NA
Viral infection
Influenza virus
A/PR/8/34
Pathway
Plaque assay
Decrease (50 %)
Investigational
22028179
DrugRepV_3188Arbidol
NA
Viral infection
Influenza virus
A/Moscow/17/98
Pathway
Plaque assay
Decrease (50 %)
Investigational
22028179
DrugRepV_3191Arbidol
NA
Viral infection
Influenza virus
A/Aichi/2/68
Pathway
Plaque assay
Decrease (Decrease (0.5-1.0) log)
Investigational
22028179
DrugRepV_3194Arbidol
NA
Viral infection
Influenza virus
A/Aichi/2/68
Pathway
Quantal assay
Decrease (1.5 log)
Investigational
22028179
DrugRepV_3197Arbidol
NA
Viral infection
Influenza virus
A/Aichi/2/68
Pathway
Plaque assay
Decrease (2.5 log)
Investigational
22028179
DrugRepV_3198Arbidol
NA
Viral infection
Influenza virus
A/Aichi/2/68
Pathway
Plaque assay
Decrease (3.73 log)
Investigational
22028179
DrugRepV_3199Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226VT
NA
Plaque assay
No significant effect (No significant reduction log)
Investigational
26384169
DrugRepV_3200Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226VT
NA
Flow cytometry
Decrease (90 %)
Investigational
26384169
DrugRepV_3201Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226AS
NA
Plaque assay
Decrease (3 Log)
Investigational
26384169
DrugRepV_3202Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226VT
NA
Plaque assay
Decrease (2 Log)
Investigational
26384169
DrugRepV_3203Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226AS
NA
Plaque assay
Decrease (50 %)
Investigational
26384169
DrugRepV_3204Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226VT
NA
Plaque assay
Decrease (50 %)
Investigational
26384169
DrugRepV_3205Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226VT
NA
Western blot
Decrease (Capsid protein Protein expression)
Investigational
26384169
DrugRepV_3206Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226VT
NA
Western blot
Decrease (E1 protein Protein expression)
Investigational
26384169
DrugRepV_3207Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226VT
NA
Western blot
Decrease (pE2 protein Protein expression)
Investigational
26384169
DrugRepV_3208Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226VT
NA
Western blot
Decrease (E2 protein Protein expression)
Investigational
26384169
DrugRepV_3209Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226VT
NA
Western blot
Decrease (nsP2 protein Protein expression)
Investigational
26384169
DrugRepV_3210Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226VT
NA
Western blot
Decrease (nsP3 protein Protein expression)
Investigational
26384169
DrugRepV_3211Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226VT
NA
Real-time PCR
Decrease (2 Log)
Investigational
26384169
DrugRepV_3212Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226AS
NA
Real-time PCR
Decrease (2 Log)
Investigational
26384169
DrugRepV_3213Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226VT
NA
Cell viability assay
Decrease (25 %)
Investigational
26384169
DrugRepV_3214Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226VT
NA
Cell viability assay
Decrease (65 %)
Investigational
26384169
DrugRepV_3215Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226VT
NA
Cell viability assay
Decrease (65 %)
Investigational
26384169
DrugRepV_3216Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226VT
NA
Plaque assay
Decrease (1 Log)
Investigational
26384169
DrugRepV_3217Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226VT
NA
Plaque assay
Decrease (2 Log)
Investigational
26384169
DrugRepV_3218Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226VT
NA
Plaque assay
Decrease (1.8 Log)
Investigational
26384169
DrugRepV_3219Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226AS
NA
Plaque assay
No significant effect (No significant reduction Log)
Investigational
26384169
DrugRepV_3220Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226AS
NA
Plaque assay
Decrease (1 Log)
Investigational
26384169
DrugRepV_3221Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226AS
NA
Plaque assay
Decrease (0.9 Log)
Investigational
26384169
DrugRepV_3222Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226AS
NA
Plaque assay
Decrease (No significant reduction Log)
Investigational
26384169
DrugRepV_3223Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226AS
NA
Plaque assay
Decrease (1.2 Log)
Investigational
26384169
DrugRepV_3224Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226AS
NA
Plaque assay
Decrease (1.2 Log)
Investigational
26384169
DrugRepV_3225Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226VS
NA
Western blot
Decrease (pE2 protein expression Protein expression)
Investigational
26384169
DrugRepV_3226Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226VS
NA
Western blot
Decrease (E2 protein expresion Protein expression)
Investigational
26384169
DrugRepV_3227Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226AS
NA
Western blot
Decrease (pE2 protein expression Protein expression)
Investigational
26384169
DrugRepV_3228Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226AS
NA
Western blot
Decrease (E2 protein expresion Protein expression)
Investigational
26384169
DrugRepV_3229Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226VS
NA
Plaque assay
Decrease (1.3 Log)
Investigational
26384169
DrugRepV_3230Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226AS
NA
Plaque assay
Decrease (2.5 Log)
Investigational
26384169
DrugRepV_3231Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226AS
NA
Plaque assay
Decrease (2 Log)
Investigational
26384169
DrugRepV_3232Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226AS
NA
Real-time PCR
Decrease (2 Log)
Investigational
26384169
DrugRepV_3233Andrographolide
NA
Ulcerative colitis and Upper respiratory tract infection
Chikungunya virus
E1:226AS
NA
Plaque assay
Decrease (50 %)
Investigational
26384169
DrugRepV_3240T-1105
NA
Zika virus
Chikungunya virus
Indian Ocean strain 899
NA
Colorimetric method
Decrease (50 %)
NA
24951535
DrugRepV_3241T-1105
NA
Zika virus
Chikungunya virus
Indian Ocean strain 899
NA
Colorimetric method
Decrease (50 %)
NA
24951535
DrugRepV_3248T-1105
NA
Zika virus
Chikungunya virus
Indian Ocean strain 899
NA
Plaque assay
Decrease (50 %)
NA
24951535
DrugRepV_3249T-1105
NA
Zika virus
Chikungunya virus
Indian Ocean strain 899
NA
Real-time PCR
Decrease (50 %)
NA
24951535
DrugRepV_3250T-1105
NA
Zika virus
Chikungunya virus
LR2006 OPY1
NA
Real-time PCR
Decrease (50 %)
NA
24951535
DrugRepV_3251T-1105
NA
Zika virus
Chikungunya virus
Venturini (Italy 2008)
NA
Real-time PCR
Decrease (50 %)
NA
24951535
DrugRepV_3252T-1105
NA
Zika virus
Chikungunya virus
Bianchi (Italy 2008)
NA
Real-time PCR
Decrease (50 %)
NA
24951535
DrugRepV_3253T-1105
NA
Zika virus
Chikungunya virus
Congo 95 (2011)
NA
Real-time PCR
Decrease (50 %)
NA
24951535
DrugRepV_3264T-1105
NA
Zika virus
Chikungunya virus
Favipiravir_res C1-CHIKV 899
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
24951535
DrugRepV_3265T-1105
NA
Zika virus
Chikungunya virus
Favipiravir_res C2-CHIKV 899
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
24951535
DrugRepV_3266T-1105
NA
Zika virus
Chikungunya virus
Favipiravir_res C3-CHIKV 899
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
24951535
DrugRepV_3270T-1105
NA
Zika virus
Chikungunya virus
Favipiravir_res_p7 C1-CHIKV 899
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
24951535
DrugRepV_3271T-1105
NA
Zika virus
Chikungunya virus
Favipiravir_res_p7 C2-CHIKV 899
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
24951535
DrugRepV_3272T-1105
NA
Zika virus
Chikungunya virus
Favipiravir_res_p7 C3-CHIKV 899
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
24951535
DrugRepV_32735-Tetradecyloxy-2-furoic Acid
NA
NA
Chikungunya virus
NA
NA
Flow cytometry
Decrease (50 %)
NA
27177310
DrugRepV_3275Cerulenin
NA
Fungal infection
Chikungunya virus
NA
NA
Flow cytometry
Decrease (50 %)
Approved
27177310
DrugRepV_3277AnnH18
NA
NA
Chikungunya virus
NA
NA
Flow cytometry
Decrease (50 %)
NA
27177310
DrugRepV_3278AnnH14
NA
NA
Chikungunya virus
NA
NA
Flow cytometry
Decrease (50 %)
NA
27177310
DrugRepV_3279KH-CB19
NA
NA
Chikungunya virus
NA
NA
Flow cytometry
Decrease (50 %)
NA
27177310
DrugRepV_3280Anacardic Acid
NA
NA
Chikungunya virus
NA
NA
Flow cytometry
Decrease (50 %)
NA
27177310
DrugRepV_3281TAE684
NA
NA
Chikungunya virus
NA
NA
Flow cytometry
Decrease (50 %)
NA
27177310
DrugRepV_32846-Hydroxyflavone
NA
Anxiety-like disorders
Chikungunya virus
NA
NA
Flow cytometry
Decrease (50 %)
NA
27177310
DrugRepV_3287Alsterpaullone
NA
NA
Chikungunya virus
NA
NA
Flow cytometry
Decrease (50 %)
Experimental
27177310
DrugRepV_3290Tivozanib
NA
Solid Tumors, Glioblastoma, Ovarian Cancer, Prostate Cancer, and Stage IV Disease
Chikungunya virus
NA
NA
Flow cytometry
Decrease (50 %)
Investigational
27177310
DrugRepV_3292Linifanib
NA
NA
Chikungunya virus
NA
NA
Flow cytometry
Decrease (50 %)
NA
27177310
DrugRepV_32935-Tetradecyloxy-2-furoic Acid
NA
NA
Influenza virus
NA
Pathway
Flow cytometry
Decrease (100 %)
NA
27177310
DrugRepV_3294Cerulenin
NA
Fungal infection
Influenza virus
NA
Pathway
Flow cytometry
Decrease (100 %)
Approved
27177310
DrugRepV_3297TIvozanib
NA
Solid Tumors, Glioblastoma, Ovarian Cancer, Prostate Cancer, and Stage IV Disease
Influenza virus
NA
Pathway
Flow cytometry
Decrease (100 %)
Investigational
27177310
DrugRepV_3298Anacardic Acid
NA
NA
Chikungunya virus
NA
NA
Flow cytometry
Decrease (75 %)
NA
27177310
DrugRepV_3300Cerulenin
NA
Fungal infection
Chikungunya virus
NA
NA
Flow cytometry
Decrease (75 %)
Approved
27177310
DrugRepV_3302TIvozanib
NA
Solid Tumors, Glioblastoma, Ovarian Cancer, Prostate Cancer, and Stage IV Disease
Chikungunya virus
NA
NA
Flow cytometry
Decrease (90 %)
Investigational
27177310
DrugRepV_3303Cerulenin
NA
Fungal infection
Chikungunya virus
NA
NA
Real-time PCR
Decrease (100 %)
Approved
27177310
DrugRepV_33045-Tetradecyloxy-2-furoic Acid
NA
NA
Chikungunya virus
NA
NA
Real-time PCR
Decrease (100 %)
NA
27177310
DrugRepV_3306TIvozanib
NA
Solid Tumors, Glioblastoma, Ovarian Cancer, Prostate Cancer, and Stage IV Disease
Chikungunya virus
NA
NA
Real-time PCR
Decrease (50 %)
Investigational
27177310
DrugRepV_3307Cerulenin
NA
Fungal infection
Chikungunya virus
NA
NA
Real-time PCR
Decrease (100 %)
Approved
27177310
DrugRepV_33085-Tetradecyloxy-2-furoic Acid
NA
NA
Chikungunya virus
NA
NA
Real-time PCR
Decrease (100 %)
NA
27177310
DrugRepV_3310TIvozanib
NA
Solid Tumors, Glioblastoma, Ovarian Cancer, Prostate Cancer, and Stage IV Disease
Chikungunya virus
NA
NA
Real-time PCR
Decrease (80 %)
Investigational
27177310
DrugRepV_3311TIvozanib
NA
Solid Tumors, Glioblastoma, Ovarian Cancer, Prostate Cancer, and Stage IV Disease
Chikungunya virus
C21
NA
Survival assay
NA
Investigational
27177310
DrugRepV_3312TIvozanib
NA
Solid Tumors, Glioblastoma, Ovarian Cancer, Prostate Cancer, and Stage IV Disease
Chikungunya virus
C21
NA
Plaque assay
No significant reduction (0.9 Log)
Investigational
27177310
DrugRepV_3313TIvozanib
NA
Solid Tumors, Glioblastoma, Ovarian Cancer, Prostate Cancer, and Stage IV Disease
Chikungunya virus
C21
NA
Plaque assay
Decrease (1.2 Log)
Investigational
27177310
DrugRepV_3314TIvozanib
NA
Solid Tumors, Glioblastoma, Ovarian Cancer, Prostate Cancer, and Stage IV Disease
Chikungunya virus
C21
NA
Plaque assay
No significant reduction (0.8 Log)
Investigational
27177310
DrugRepV_33165-Tetradecyloxy-2-furoic Acid
NA
NA
Chikungunya virus
C21
NA
Plaque assay
No significant reduction (0.2 Log)
NA
27177310
DrugRepV_3350Trametinib-Oseltamivir
NA
NA
Influenza virus
WSN/H1N1
Pathway
Plaque assay
Decrease (95 %)
Approved
29990517
DrugRepV_3352Trametinib-Oseltamivir
NA
NA
Influenza virus
WSN/H1N1
Pathway
Plaque assay
Decrease (3.5 Log)
Approved
29990517
DrugRepV_3376Mycophenolic Acid-Betaferon
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
CPE inhibition assay
Decrease (50 %)
NA
24096239
DrugRepV_3382Betaferon
NA
Multiple sclerosis
Middle East respiratory syndrome coronavirus
NA
NA
CPE inhibition assay
Decrease (50 %)
Approved
24096239
DrugRepV_3407SSYA10-001
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
Plaque assay
Decrease (50 %)
NA
24841268
DrugRepV_3408SSYA10-001
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Plaque assay
Decrease (50 %)
NA
24841268
DrugRepV_3409Dapivirine
NA
Acquired immunodeficiency syndrome
Influenza virus
A/California/07/2009 (H1N1)
Pathway
Plaque assay
Decrease (50 %)
Investigational
28778830
DrugRepV_3413Dapivirine
NA
Acquired immunodeficiency syndrome
Influenza virus
B/Bris/60/2008 (Victoria)
Pathway
Plaque assay
Decrease (50 %)
Investigational
28778830
DrugRepV_3416Dapivirine
NA
Acquired immunodeficiency syndrome
Influenza virus
A/California/7/2009 (H1N1)
Pathway
Plaque assay
Decrease (2.1 Log)
Investigational
28778830
DrugRepV_3417Dapivirine
NA
Acquired immunodeficiency syndrome
Influenza virus
A/California/7/2009 (H1N1)
Pathway
Plaque assay
Decrease (2.9 Log)
Investigational
28778830
DrugRepV_3420Dapivirine
NA
Acquired immunodeficiency syndrome
Influenza virus
A/WSN/1933 (H1N1)
Pathway
Plaque assay
Decrease (1.7 Log)
Investigational
28778830
DrugRepV_3422Dapivirine
NA
Acquired immunodeficiency syndrome
Influenza virus
A/DM/528/2009 (H1N1)
Pathway
Plaque assay
Decrease (50 %)
Investigational
28778830
DrugRepV_3423Dapivirine
NA
Acquired immunodeficiency syndrome
Influenza virus
A/Texas/4/2009 (H1N1)
Pathway
Plaque assay
Decrease (50 %)
Investigational
28778830
DrugRepV_3424Dapivirine
NA
Acquired immunodeficiency syndrome
Influenza virus
A/North Carolina/39/2009 (H1N1)
Pathway
Plaque assay
Decrease (50 %)
Investigational
28778830
DrugRepV_3425Dapivirine
NA
Acquired immunodeficiency syndrome
Influenza virus
A/Washington/29/2009 (H1N1)
Pathway
Plaque assay
Decrease (50 %)
Investigational
28778830
DrugRepV_3426Dapivirine
NA
Acquired immunodeficiency syndrome
Influenza virus
A/WSN/1933 (H1N1)
Pathway
Plaque assay
Decrease (50 %)
Investigational
28778830
DrugRepV_3427Dapivirine
NA
Acquired immunodeficiency syndrome
Influenza virus
A/California/07/2009 (H1N1)
Pathway
Plaque assay
Decrease (50 %)
Investigational
28778830
DrugRepV_3428Dapivirine
NA
Acquired immunodeficiency syndrome
Influenza virus
A/DM/524/2009 (H1N1)
Pathway
Plaque assay
Decrease (50 %)
Investigational
28778830
DrugRepV_3429Dapivirine
NA
Acquired immunodeficiency syndrome
Influenza virus
A/Switzerland/9715293/2013 (H3N2)
Pathway
Plaque assay
Decrease (50 %)
Investigational
28778830
DrugRepV_3430Dapivirine
NA
Acquired immunodeficiency syndrome
Influenza virus
A/Switzerland/9715293/2013 X-247 (H3N2)
Pathway
Plaque assay
Decrease (50 %)
Investigational
28778830
DrugRepV_3431Dapivirine
NA
Acquired immunodeficiency syndrome
Influenza virus
A/Hongkong/4801/2014 (H3N2)
Pathway
Cytopathic effect (CPE) assay
Decrease (50 %)
Investigational
28778830
DrugRepV_3432Dapivirine
NA
Acquired immunodeficiency syndrome
Influenza virus
A/California/2/2014 (H3N2)
Pathway
Plaque assay
Decrease (50 %)
Investigational
28778830
DrugRepV_3433Dapivirine
NA
Acquired immunodeficiency syndrome
Influenza virus
A/Udorn/1972 (H3N2)
Pathway
Plaque assay
Decrease (50 %)
Investigational
28778830
DrugRepV_3434Dapivirine
NA
Acquired immunodeficiency syndrome
Influenza virus
A/Soloman Islands/3/2006 (H1N1)
Pathway
Plaque assay
Decrease (50 %)
Investigational
28778830
DrugRepV_3435Dapivirine
NA
Acquired immunodeficiency syndrome
Influenza virus
B/Wisconsin/1/2010 (Yamagata)
Pathway
Plaque assay
Decrease (50 %)
Investigational
28778830
DrugRepV_3436Dapivirine
NA
Acquired immunodeficiency syndrome
Influenza virus
B/Bris/60/2008 (Victoria)
Pathway
Plaque assay
Decrease (50 %)
Investigational
28778830
DrugRepV_3439Saliphenylhalamide
NA
NA
Influenza virus
PR8-GFP
Pathway
GFP assay
Decrease (50 %)
NA
22910914
DrugRepV_3442NVP-AUY922
NA
NA
Influenza virus
PR8-GFP
Pathway
GFP assay
Decrease (50 %)
NA
22910914
DrugRepV_3443Alvespimycin
NA
Cancer
Influenza virus
PR8-GFP
Pathway
GFP assay
Decrease (50 %)
Investigational
22910914
DrugRepV_3444Tanespimycin
NA
Cancer
Influenza virus
PR8-GFP
Pathway
GFP assay
Decrease (50 %)
Investigational
22910914
DrugRepV_3447Saliphenylhalamide
NA
NA
Influenza virus
PR8-GFP
Pathway
GFP assay
Decrease (50 %)
NA
22910914
DrugRepV_3450NVP-AUY922
NA
NA
Influenza virus
PR8-GFP
Pathway
GFP assay
Decrease (50 %)
NA
22910914
DrugRepV_3451Alvespimycin
NA
Cancer
Influenza virus
PR8-GFP
Pathway
GFP assay
Decrease (50 %)
Investigational
22910914
DrugRepV_3452Tanespimycin
NA
Cancer
Influenza virus
PR8-GFP
Pathway
GFP assay
Decrease (50 %)
Investigational
22910914
DrugRepV_3470Pyrrolopyridinamine PPA-7
NA
NA
Influenza virus
CA/09 (H1N1)
Pathway
Immunoflourescence assay
Decrease (50 %)
NA
27586275
DrugRepV_3471Aminothiadiazole ATD-1
NA
NA
Influenza virus
CA/09 (H1N1)
Pathway
Immunoflourescence assay
Decrease (50 %)
NA
27586275
DrugRepV_3472Dihydrofuropyridine carboxamide HPC-2
NA
NA
Influenza virus
CA/09 (H1N1)
Pathway
Immunoflourescence assay
Decrease (50 %)
NA
27586275
DrugRepV_3473Pyrrolopyridinamine PPA-7
NA
NA
Influenza virus
PE/09 (H3N2)
Pathway
Immunoflourescence assay
Decrease (50 %)
NA
27586275
DrugRepV_3474Aminothiadiazole ATD-1
NA
NA
Influenza virus
PE/09 (H3N2)
Pathway
Immunoflourescence assay
Decrease (50 %)
NA
27586275
DrugRepV_3475Dihydrofuropyridine carboxamide HPC-2
NA
NA
Influenza virus
PE/09 (H3N2)
Pathway
Immunoflourescence assay
Decrease (50 %)
NA
27586275
DrugRepV_3476Pyrrolopyridinamine PPA-7
NA
NA
Influenza virus
B/Florida/04/2006 (B/FL/06)
Pathway
Immunoflourescence assay
Decrease (50 %)
NA
27586275
DrugRepV_3477Aminothiadiazole ATD-1
NA
NA
Influenza virus
B/Florida/04/2006 (B/FL/06)
Pathway
Immunoflourescence assay
Decrease (50 %)
NA
27586275
DrugRepV_3478Dihydrofuropyridine carboxamide HPC-2
NA
NA
Influenza virus
B/Florida/04/2006 (B/FL/06)
Pathway
Immunoflourescence assay
Decrease (50 %)
NA
27586275
DrugRepV_3479Pyrrolopyridinamine PPA-1
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3480Pyrrolopyridinamine PPA-2
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3481Pyrrolopyridinamine PPA-3
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3482Pyrrolopyridinamine PPA-4
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3483Pyrrolopyridinamine PPA-5
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3484Pyrrolopyridinamine PPA-6
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3485Pyrrolopyridinamine PPA-7
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3486Pyrrolopyridinamine PPA-8
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3487Pyrrolopyridinamine PPA-9
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3488Pyrrolopyridinamine PPA-10
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3489Pyrrolopyridinamine PPA-11
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3490Pyrrolopyridinamine PPA-12
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3491Pyrrolopyridinamine PPA-1
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3492Pyrrolopyridinamine PPA-2
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3493Pyrrolopyridinamine PPA-3
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3494Pyrrolopyridinamine PPA-4
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3495Pyrrolopyridinamine PPA-5
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3496Pyrrolopyridinamine PPA-6
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3497Pyrrolopyridinamine PPA-7
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3498Pyrrolopyridinamine PPA-8
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3499Pyrrolopyridinamine PPA-9
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3500Pyrrolopyridinamine PPA-10
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3501Pyrrolopyridinamine PPA-11
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3502Pyrrolopyridinamine PPA-12
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3503Aminothiadiazole ATD-1
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3504Aminothiadiazole ATD-2
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3505Aminothiadiazole ATD-1
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3506Aminothiadiazole ATD-2
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3507Dihydrofuropyridine carboxamide HPC-1
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3508Dihydrofuropyridine carboxamide HPC-2
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3509Dihydrofuropyridine carboxamide HPC-3
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3510Dihydrofuropyridine carboxamide HPC-1
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3511Dihydrofuropyridine carboxamide HPC-2
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3512Dihydrofuropyridine carboxamide HPC-3
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3513Imidazopyridinamine IPA-1
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3514Imidazopyridinamine IPA-1
NA
NA
Influenza virus
A/Puerto Rico/8/1934 virus (NS1-GFP virus)
Pathway
PR8GFP Assay
Decrease (50 %)
NA
27586275
DrugRepV_3578AY9944
NA
NA
Ebola virus
EBOV trVLP
NA
Luciferase reporter assay
Decrease (50 %)
NA
30149038
DrugRepV_3581GBR-12783
NA
Psychosis
Ebola virus
EBOV trVLP
NA
Luciferase reporter assay
Decrease (50 %)
NA
30149038
DrugRepV_3582Tabimorelin
NA
NA
Ebola virus
EBOV trVLP
NA
Luciferase reporter assay
Decrease (50 %)
NA
30149038
DrugRepV_3584Camylofine
NA
NA
Ebola virus
EBOV trVLP
NA
Luciferase reporter assay
Decrease (50 %)
NA
30149038
DrugRepV_3587ML9
NA
NA
Ebola virus
EBOV trVLP
NA
Luciferase reporter assay
Decrease (50 %)
NA
30149038
DrugRepV_3593Iminodyn 17
NA
NA
Ebola virus
EBOV trVLP
NA
Luciferase reporter assay
Decrease (50 %)
NA
30149038
DrugRepV_3594Nobiletin
NA
NA
Ebola virus
EBOV trVLP
NA
Luciferase reporter assay
Decrease (50 %)
NA
30149038
DrugRepV_3596N-Acetyl-L-leucyl- L- leucyl-L- methional
NA
NA
Ebola virus
EBOV trVLP
NA
Luciferase reporter assay
Decrease (50 %)
NA
30149038
DrugRepV_3597Calpeptin
NA
NA
Ebola virus
EBOV trVLP
NA
Luciferase reporter assay
Decrease (50 %)
NA
30149038
DrugRepV_3599Gentian Violet
NA
Bacterial infection | Fungal infections (mouth (thrush) and skin)
Nipah virus
NA
NA
Taqman PCR
Decrease (50 %)
Approved
19889218
DrugRepV_3600Gliotoxin
NA
NA
Nipah virus
NA
NA
Taqman PCR
Decrease (50 %)
NA
19889218
DrugRepV_3602Gentian Violet
NA
Bacterial infection | Fungal infections (mouth (thrush) and skin)
Hendra virus
NA
NA
Taqman PCR
Decrease (50 %)
Approved
19889218
DrugRepV_3603Gliotoxin
NA
NA
Hendra virus
NA
NA
Taqman PCR
Decrease (50 %)
NA
19889218
DrugRepV_3605Gentian Violet
NA
Bacterial infection | Fungal infections (mouth (thrush) and skin)
Nipah virus
NA
NA
Taqman PCR
Decrease (50 %)
Approved
19889218
DrugRepV_3606Gliotoxin
NA
NA
Nipah virus
NA
NA
Taqman PCR
Decrease (50 %)
NA
19889218
DrugRepV_3608Gentian Violet
NA
Bacterial infection | Fungal infections (mouth (thrush) and skin)
Hendra virus
NA
NA
Taqman PCR
Decrease (50 %)
Approved
19889218
DrugRepV_3609Gliotoxin
NA
NA
Hendra virus
NA
NA
Taqman PCR
Decrease (50 %)
NA
19889218
DrugRepV_3610Gliotoxin
NA
NA
Influenza virus
A/ swine/Rachaburi/2000 (H1N1)
Pathway
Taqman PCR
Decrease (50 %)
NA
19889218
DrugRepV_3611C-c3 Ado
NA
NA
Nipah virus
NA
NA
RT-PCR
Decrease
NA
16641448
DrugRepV_36125 Noraristeromycin
NA
NA
Nipah virus
NA
NA
RT-PCR
Decrease
NA
16641448
DrugRepV_3613DHCaA
NA
NA
Nipah virus
NA
NA
RT-PCR
Decrease
NA
16641448
DrugRepV_3615EICAR
NA
NA
Nipah virus
NA
NA
RT-PCR
Decrease
NA
16641448
DrugRepV_3616Pyrazofurin
NA
NA
Nipah virus
NA
NA
RT-PCR
Decrease
NA
16641448
DrugRepV_3617Carbodine
NA
NA
Nipah virus
NA
NA
RT-PCR
Decrease
NA
16641448
DrugRepV_36186-Azauridine
NA
Cancer
Nipah virus
NA
NA
RT-PCR
Decrease
NA
16641448
DrugRepV_3619Poly(I)-poly(C12U)
NA
NA
Nipah virus
NA
NA
RT-PCR
Decrease
NA
16641448
DrugRepV_36216-Azauridine
NA
Cancer
Nipah virus
NA
NA
RT-PCR
Decrease
NA
16641448
DrugRepV_3627Cyanovirin-N
NA
NA
Ebola virus
Zaire
NA
Luciferase assay
Decrease (50 %)
NA
15073681
DrugRepV_3628Cyanovirin-N
NA
NA
Marburg virus
NA
NA
Luciferase assay
Decrease (50 %)
NA
15073681
DrugRepV_3629Cyanovirin-N
NA
NA
Ebola virus
Zaire
NA
Luciferase assay
Decrease (50 %)
NA
15073681
DrugRepV_3630N-methyl-5,7-dinitro-N-propylquinolin-8-amine
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (90 %)
NA
21270170
DrugRepV_36312-[3-(4-chlorophenyl)-1-(3-methoxyphenyl)-3-oxopropyl]propanedinitrile
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (90 %)
NA
21270170
DrugRepV_3632(19S)-19-ethyl-19-hydroxy-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2(11),3,9,15(20)-pentaene-14,18-dione
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (90 %)
NA
21270170
DrugRepV_36332-[(1E)-2-(5-nitrofuran-2-yl)ethenyl]-3-[3-(trifluoromethyl)phenyl]-3,4-dihydroquinazolin-4-one
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (90 %)
NA
21270170
DrugRepV_3634N-(3,4-dichlorophenyl)-5-nitrofuran-2-carboxamide
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (90 %)
NA
21270170
DrugRepV_36357-[(furan-2-yl)methyl]-3-[3-(1H-imidazol-1-yl)propyl]-5,6-diphenyl-3H,4H,7H-pyrrolo[2,3-d]pyrimidin-4-imine
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (90 %)
NA
21270170
DrugRepV_36362-phenyl-4-(1,1,2,2-tetrafluoroethyl)-3H-1,5-benzodiazepine
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (90 %)
NA
21270170
DrugRepV_3637N,N-bis(4-methylphenyl)pyridin-3-amine
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (90 %)
NA
21270170
DrugRepV_3638N-methyl-5,7-dinitro-N-propylquinolin-8-amine
NA
NA
Ebola virus
Zaire
NA
Luciferase assay
Decrease (50 %)
NA
21270170
DrugRepV_36392-[3-(4-chlorophenyl)-1-(3-methoxyphenyl)-3-oxopropyl]propanedinitrile
NA
NA
Ebola virus
Zaire
NA
Luciferase assay
Decrease (50 %)
NA
21270170
DrugRepV_3640(19S)-19-ethyl-19-hydroxy-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2(11),3,9,15(20)-pentaene-14,18-dione
NA
NA
Ebola virus
Zaire
NA
Luciferase assay
Decrease (50 %)
NA
21270170
DrugRepV_36412-[(1E)-2-(5-nitrofuran-2-yl)ethenyl]-3-[3-(trifluoromethyl)phenyl]-3,4-dihydroquinazolin-4-one
NA
NA
Ebola virus
Zaire
NA
Luciferase assay
Decrease (50 %)
NA
21270170
DrugRepV_3642N-(3,4-dichlorophenyl)-5-nitrofuran-2-carboxamide
NA
NA
Ebola virus
Zaire
NA
Luciferase assay
Decrease (50 %)
NA
21270170
DrugRepV_36437-[(furan-2-yl)methyl]-3-[3-(1H-imidazol-1-yl)propyl]-5,6-diphenyl-3H,4H,7H-pyrrolo[2,3-d]pyrimidin-4-imine
NA
NA
Ebola virus
Zaire
NA
Luciferase assay
Decrease (50 %)
NA
21270170
DrugRepV_36442-phenyl-4-(1,1,2,2-tetrafluoroethyl)-3H-1,5-benzodiazepine
NA
NA
Ebola virus
Zaire
NA
Luciferase assay
Decrease (50 %)
NA
21270170
DrugRepV_3645N,N-bis(4-methylphenyl)pyridin-3-amine
NA
NA
Ebola virus
Zaire
NA
Luciferase assay
Decrease (50 %)
NA
21270170
DrugRepV_36462-phenyl-4-(1,1,2,2-tetrafluoroethyl)-3H-1,5-benzodiazepine
NA
NA
Ebola virus
Zaire
NA
Luciferase assay
Decrease (50 %)
NA
21270170
DrugRepV_36472-phenyl-4-(1,1,2,2-tetrafluoroethyl)-3H-1,5-benzodiazepine
NA
NA
Marburg virus
NA
NA
Luciferase assay
Decrease (50 %)
NA
21270170
DrugRepV_36482-phenyl-4-(1,1,2,2-tetrafluoroethyl)-3H-1,5-benzodiazepine
NA
NA
Rift Valley fever virus
MP12
NA
Luciferase assay
Decrease (50 %)
NA
21270170
DrugRepV_36492-phenyl-4-(1,1,2,2-tetrafluoroethyl)-3H-1,5-benzodiazepine
NA
NA
Influenza virus
California/07/2009
Pathway
Luciferase assay
Decrease (50 %)
NA
21270170
DrugRepV_36502-phenyl-4-(1,1,2,2-tetrafluoroethyl)-3H-1,5-benzodiazepine
NA
NA
Influenza virus
Brisbane/10/2007
Pathway
Luciferase assay
Decrease (50 %)
NA
21270170
DrugRepV_36512-phenyl-4-(1,1,2,2-tetrafluoroethyl)-3H-1,5-benzodiazepine
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
Luciferase assay
Decrease (50 %)
NA
21270170
DrugRepV_36522-phenyl-4-(1,1,2,2-tetrafluoroethyl)-3H-1,5-benzodiazepine
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (90 %)
NA
21270170
DrugRepV_36532-methyl-4-phenyl-1H-naphtho[2,3-b][1,4]diazepine hydrochloride
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (90 %)
NA
21270170
DrugRepV_36542-(4-chlorophenyl)-7,8-dimethyl-4-(trifluoromethyl)-3H-1,5-benzodiazepine
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (90 %)
NA
21270170
DrugRepV_36552-(1,1,2,2,2-pentafluoroethyl)-4-phenyl-3H-1,5-benzodiazepine
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (90 %)
NA
21270170
DrugRepV_36567,8-dichloro-2-(1,1,2,2,2-pentafluoroethyl)-4-phenyl-3H-1,5-benzodiazepine
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (90 %)
NA
21270170
DrugRepV_36572-[4-(trifluoromethyl)-3H-1,5-benzodiazepin-2-yl]phenol
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (90 %)
NA
21270170
DrugRepV_36582-(4-methylphenyl)-4-(trifluoromethyl)-3H-1,5-benzodiazepine
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (90 %)
NA
21270170
DrugRepV_36594-methoxy-2-[4-(trifluoromethyl)-3H-1,5-benzodiazepin-2-yl]phenol
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (90 %)
NA
21270170
DrugRepV_36602-[4-(thiophen-2-yl)-3H-1,5-benzodiazepin-2-yl]phenol
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (90 %)
NA
21270170
DrugRepV_36614-chloro-2-[4-(furan-2-yl)-3H-1,5-benzodiazepin-2-yl]phenol
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (90 %)
NA
21270170
DrugRepV_36624-methoxy-2-[4-(thiophen-2-yl)-3H-1,5-benzodiazepin-2-yl]phenol
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (90 %)
NA
21270170
DrugRepV_36632-[4-(furan-2-yl)-3H-1,5-benzodiazepin-2-yl]phenol
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (90 %)
NA
21270170
DrugRepV_36642-[4-(3-nitrophenyl)-3H-1,5-benzodiazepin-2-yl]phenol
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (90 %)
NA
21270170
DrugRepV_36652-phenyl-4-(1,1,2,2-tetrafluoroethyl)-3H-1,5-benzodiazepine
NA
NA
Marburg virus
Lake Victoria
NA
Luciferase reporter assay
Decrease (90 %)
NA
21270170
DrugRepV_36662-phenyl-4-(1,1,2,2-tetrafluoroethyl)-3H-1,5-benzodiazepine
NA
NA
Marburg virus
Lake Victoria
NA
Luciferase reporter assay
Decrease (50 %)
NA
21270170
DrugRepV_36672-phenyl-4-(1,1,2,2-tetrafluoroethyl)-3H-1,5-benzodiazepine
NA
NA
Marburg virus
Lake Victoria
NA
Luciferase reporter assay
Decrease (100 %)
NA
21270170
DrugRepV_36682-phenyl-4-(1,1,2,2-tetrafluoroethyl)-3H-1,5-benzodiazepine
NA
NA
Marburg virus
Lake Victoria
NA
Luciferase reporter assay
Decrease (98 %)
NA
21270170
DrugRepV_36692-phenyl-4-(1,1,2,2-tetrafluoroethyl)-3H-1,5-benzodiazepine
NA
NA
Lassa virus
NA
NA
Luciferase reporter assay
Decrease (40 %)
NA
21270170
DrugRepV_36702-phenyl-4-(1,1,2,2-tetrafluoroethyl)-3H-1,5-benzodiazepine
NA
NA
Influenza virus
Goose/Qinghai/59/05
Pathway
Luciferase reporter assay
Decrease (15 %)
NA
21270170
DrugRepV_36712,6-bis[(3-tert-butyl-2-hydroxy-5-methylphenyl)methyl]-4-methylphenol
NA
NA
Ebola virus
NA
NA
RT-PCR
Decrease (100 %)
NA
22027648
DrugRepV_3672NSC 62914
NA
NA
Ebola virus
NA
NA
RT-PCR
Decrease
NA
22027648
DrugRepV_3673NSC 62914
NA
NA
Ebola virus
NA
NA
RT-PCR
Decrease (50 %)
NA
22027648
DrugRepV_3674Trolox
NA
NA
Ebola virus
Zaire
NA
RT-PCR
Decrease (45 %)
NA
22027648
DrugRepV_3675Trolox
NA
NA
Marburg virus
NA
NA
RT-PCR
Decrease (70 %)
NA
22027648
DrugRepV_3676NSC 62914
NA
NA
Marburg virus
Ci67
NA
RT-PCR
Decrease (98 %)
NA
22027648
DrugRepV_3677NSC 62914
NA
NA
Lassa virus
Josiah
NA
RT-PCR
Decrease (98 %)
NA
22027648
DrugRepV_3678NSC 62914
NA
NA
Rift Valley fever virus
MP12
NA
RT-PCR
Decrease (97 %)
NA
22027648
DrugRepV_3679NSC 62914
NA
NA
Ebola virus
NA
NA
NA
Decrease
NA
22027648
DrugRepV_3680NSC 62914
NA
NA
Marburg virus
NA
NA
NA
Decrease
NA
22027648
DrugRepV_3681N3,N12-bis[2-(morpholin-4-yl)ethyl]-6,15-diazatetracyclo[8.8.0.02,7.011,16]octadeca-1(10),2,4,6,8,11(16),12,14,17-nonaene-3,12-diamine tetrahydrochloride
NA
NA
Ebola virus
Zaire-95
NA
NA
Decrease (50 %)
NA
23012625
DrugRepV_3682N5,N14-bis[2-(morpholin-4-yl)ethyl]-3,12-bis({[2-(morpholin-4-yl)ethyl]amino})-6,15-diazatetracyclo[8.8.0.02,7.011,16]octadeca-1(10),2,4,6,8,11(16),12,14,17-nonaene-5,14-dicarboxamide; hexakis(trifluoroacet
NA
NA
Ebola virus
Zaire-95
NA
NA
Decrease (50 %)
NA
23012625
DrugRepV_3683N3,N12-bis[2-(morpholin-4-yl)ethyl]-6,15-diazatetracyclo[8.8.0.02,7.011,16]octadeca-1(10),2,4,6,8,11(16),12,14,17-nonaene-3,12-diamine
NA
NA
Ebola virus
Zaire-95
NA
NA
Decrease (50 %)
NA
23012625
DrugRepV_3684N3,N12-bis[2-(morpholin-4-yl)ethyl]-6,15-diazatetracyclo[8.8.0.02,7.011,16]octadeca-1(10),2,4,6,8,11(16),12,14,17-nonaene-3,12-diamine tetrahydrochloride
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
23012625
DrugRepV_3685N3,N12-bis[2-(morpholin-4-yl)ethyl]-6,15-diazatetracyclo[8.8.0.02,7.011,16]octadeca-1(10),2,4,6,8,11(16),12,14,17-nonaene-3,12-diamine
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
23012625
DrugRepV_3686BCX4430
NA
Ebola virus
Marburg virus
Musoke
NA
RT-PCR
Decrease (50 %)
Investigational
24590073
DrugRepV_3687BCX4430
NA
Ebola virus
Marburg virus
Ci67
NA
RT-PCR
Decrease (50 %)
Investigational
24590073
DrugRepV_3688BCX4430
NA
Ebola virus
Marburg virus
Angola
NA
RT-PCR
Decrease (50 %)
Investigational
24590073
DrugRepV_3689BCX4430
NA
Ebola virus
Ebola virus
Kikwit
NA
RT-PCR
Decrease (50 %)
Investigational
24590073
DrugRepV_3690BCX4430
NA
Ebola virus
Chikungunya virus
AF 15561
NA
RT-PCR
Decrease (50 %)
Investigational
24590073
DrugRepV_3691BCX4430
NA
Ebola virus
Rift Valley fever virus
ZH5018
NA
RT-PCR
Decrease (50 %)
Investigational
24590073
DrugRepV_3692BCX4430
NA
Ebola virus
Lassa virus
Josiah
NA
RT-PCR
Decrease (50 %)
Investigational
24590073
DrugRepV_3693BCX4430
NA
Ebola virus
Nipah virus
Malaysia
NA
RT-PCR
Decrease (50 %)
Investigational
24590073
DrugRepV_3694BCX4430
NA
Ebola virus
Middle East respiratory syndrome coronavirus
Jordan N3
NA
RT-PCR
Decrease (50 %)
Investigational
24590073
DrugRepV_3695BCX4430
NA
Ebola virus
Severe acute respiratory syndrome coronavirus
Urbani
NA
RT-PCR
Decrease (50 %)
Investigational
24590073
DrugRepV_3696BCX4430
NA
Ebola virus
Influenza virus
pH1N1
Pathway
RT-PCR
Decrease (50 %)
Investigational
24590073
DrugRepV_36986-Azauridine
NA
Cancer
Marburg virus
NA
NA
Luciferase assay
Decrease (50 %)
NA
24713118
DrugRepV_36992-C-Methylcytidine
NA
Hepatitis C virus
Marburg virus
NA
NA
Luciferase assay
Decrease (50 %)
Experimental
24713118
DrugRepV_37016-Azauridine
NA
Cancer
Ebola virus
NA
NA
Luciferase assay
Decrease (50 %)
NA
24713118
DrugRepV_37022-C-Methylcytidine
NA
Hepatitis C virus
Ebola virus
NA
NA
Luciferase assay
Decrease (50 %)
Experimental
24713118
DrugRepV_37046-Azauridine
NA
Cancer
Marburg virus
NA
NA
NA
Decrease (98 %)
NA
24713118
DrugRepV_37086-Azauridine
NA
Cancer
Ebola virus
NA
NA
NA
Decrease (99 %)
NA
24713118
DrugRepV_3711C795-0925
NA
NA
Rift Valley fever virus
ZH548/MP-12
NA
RT-PCR
Decrease (50 %)
NA
25144302
DrugRepV_3712D011-2120
NA
NA
Rift Valley fever virus
ZH548/MP-12
NA
RT-PCR
Decrease (50 %)
NA
25144302
DrugRepV_3713F694-1532
NA
NA
Rift Valley fever virus
ZH548/MP-12
NA
RT-PCR
Decrease (50 %)
NA
25144302
DrugRepV_3714G202-0362
NA
NA
Rift Valley fever virus
ZH548/MP-12
NA
RT-PCR
Decrease (50 %)
NA
25144302
DrugRepV_3715C795-0925
NA
NA
Ebola virus
Zaire
NA
RT-PCR
Decrease (50 %)
NA
25144302
DrugRepV_3716D011-2120
NA
NA
Ebola virus
Zaire
NA
RT-PCR
Decrease (50 %)
NA
25144302
DrugRepV_3717F694-1532
NA
NA
Ebola virus
Zaire
NA
RT-PCR
Decrease (50 %)
NA
25144302
DrugRepV_3718G202-0362
NA
NA
Ebola virus
Zaire
NA
RT-PCR
Decrease (50 %)
NA
25144302
DrugRepV_3719C795-0925
NA
NA
Marburg virus
Ci67
NA
RT-PCR
Decrease (50 %)
NA
25144302
DrugRepV_3720D011-2120
NA
NA
Marburg virus
Ci67
NA
RT-PCR
Decrease (50 %)
NA
25144302
DrugRepV_3721F694-1532
NA
NA
Marburg virus
Ci67
NA
RT-PCR
Decrease (50 %)
NA
25144302
DrugRepV_3722G202-0362
NA
NA
Marburg virus
Ci67
NA
RT-PCR
Decrease (50 %)
NA
25144302
DrugRepV_3723C795-0925
NA
NA
Lassa virus
Josiah
NA
RT-PCR
Decrease (50 %)
NA
25144302
DrugRepV_3724D011-2120
NA
NA
Lassa virus
Josiah
NA
RT-PCR
Decrease (50 %)
NA
25144302
DrugRepV_3725F694-1532
NA
NA
Lassa virus
Josiah
NA
RT-PCR
Decrease (50 %)
NA
25144302
DrugRepV_3727AZD8055
NA
Cancer
Lassa virus
NA
NA
NA
Decrease
Investigational
25986249
DrugRepV_3728TWS119
NA
NA
Lassa virus
NA
NA
NA
Decrease
NA
25986249
DrugRepV_3729SU 4312
NA
NA
Lassa virus
NA
NA
NA
Decrease
NA
25986249
DrugRepV_3730Falnidamol dihydrochloride
NA
Solid Tumor
Lassa virus
NA
NA
NA
Decrease
Investigational
25986249
DrugRepV_3731Ki 8751
NA
NA
Lassa virus
NA
NA
NA
Decrease
NA
25986249
DrugRepV_373210-DEBC hydrochloride
NA
NA
Lassa virus
NA
NA
NA
Decrease
NA
25986249
DrugRepV_3738Falnidamol dihydrochloride
NA
Solid Tumor
Lassa virus
NA
NA
RT-PCR
Decrease (50 %)
Investigational
25986249
DrugRepV_3739Falnidamol dihydrochloride
NA
Solid Tumor
Ebola virus
NA
NA
RT-PCR
Decrease (50 %)
Investigational
25986249
DrugRepV_3740Falnidamol dihydrochloride
NA
Solid Tumor
Marburg virus
NA
NA
RT-PCR
Decrease (50 %)
Investigational
25986249
DrugRepV_3742Falnidamol
NA
Solid Tumor
Lassa virus
NA
NA
RT-PCR
Decrease (50 %)
Investigational
25986249
DrugRepV_3744Falnidamol
NA
Solid Tumor
Ebola virus
NA
NA
RT-PCR
Decrease (50 %)
Investigational
25986249
DrugRepV_3745Falnidamol
NA
Solid Tumor
Ebola virus
1976
NA
Firefly luciferase assay
Decrease (50 %)
Investigational
25986249
DrugRepV_3746Falnidamol
NA
Solid Tumor
Ebola virus
2014
NA
Firefly luciferase assay
Decrease (50 %)
Investigational
25986249
DrugRepV_3747Falnidamol
NA
Solid Tumor
Lassa virus
NA
NA
Firefly luciferase assay
Decrease (50 %)
Investigational
25986249
DrugRepV_3751MLS000078751
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3752MLS000394177
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3753MLS000534476
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3754MLS000554255
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3755MLS000555232
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3756MLS000730532
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3757MLS000733230
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3758MLS000762907
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3759MLS001101371
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3760MLS000078751
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3761MLS000394177
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3762MLS000534476
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3763MLS000554255
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3764MLS000555232
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3765MLS000730532
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3766MLS000733230
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3767MLS000762907
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3768MLS001101371
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3769MLS001239325
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3770MLS001239325
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3771MLS001030162
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3772MLS001030162
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3773MLS000666802
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3774MLS000666802
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3775MLS000999960
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3776MLS000999960
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3777MLS001173370
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3778MLS001173370
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3779MLS001174896
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3780MLS001174896
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3781MLS001196083
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3782MLS001196083
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3783MLS001239358
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3784MLS001239358
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3785MLS001177927
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3786MLS001177927
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3787MLS001209453
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3788MLS001209453
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3789MLS000580080
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3790MLS000580080
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3791MLS000106706
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3792MLS000106706
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3793MLS001175455
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3794MLS001175455
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3795MLS000772389
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3796MLS000772389
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3797MLS000042810
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3798MLS000042810
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3799MLS001162808
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3800MLS001162808
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3801MLS000684231
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3802MLS000684231
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3803MLS000556387
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3804MLS000556387
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3805MLS001179278
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3806MLS001179278
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3807MLS000567464
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3808MLS000567464
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3809MLS000583959
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3810MLS000583959
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3811MLS001018888
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3812MLS001018888
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3813MLS001047402
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3814MLS001047402
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3815MLS001029946
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3816MLS001029946
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3817MLS000332573
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3818MLS000332573
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3819MLS000936259
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3820MLS000936259
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3821MLS000718690
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3822MLS000718690
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3823MLS000880330
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3824MLS000880330
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3825MLS001207131
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3826MLS001207131
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3827MLS000673118
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3828MLS000673118
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3829MLS000689481
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3830MLS000689481
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3831MLS001179272
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3832MLS001179272
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3833MLS002702500
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3834MLS002702500
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3835MLS001180408
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3836MLS000737975
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3837MLS001237534
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3838MLS000336293
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3839MLS000780111
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3840MLS001179997
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3841MLS000418057
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3842MLS000936795
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3843MLS000092187
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3844MLS000391391
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3845MLS000569139
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3846MLS001045935
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3847MLS001181479
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3848MLS000391984
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3849MLS000063146
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3850MLS000768081
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3851MLS000091920
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3852MLS001150589
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3853MLS000736237
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3855Enclomiphene
NA
Male hypogonadism
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
Investigational
27490565
DrugRepV_3856Zuclomiphene
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27490565
DrugRepV_3858Enclomiphene
NA
Male hypogonadism
Ebola virus
Mayinga
NA
Renilla luciferase assay
Decrease (100 %)
Investigational
27490565
DrugRepV_3859Zuclomiphene
NA
NA
Ebola virus
Mayinga
NA
Renilla luciferase assay
Decrease (100 %)
NA
27490565
DrugRepV_3867BCX4430
NA
Ebola virus
Zika virus
Puerto Rican PRVABC-59
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Investigational
27838352
DrugRepV_3868BCX4430
NA
Ebola virus
Zika virus
Puerto Rican PRVABC-59
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Investigational
27838352
DrugRepV_3869BCX4430
NA
Ebola virus
Zika virus
Puerto Rican PRVABC-59
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Investigational
27838352
DrugRepV_3870BCX4430
NA
Ebola virus
Zika virus
Malaysian P 6-740
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Investigational
27838352
DrugRepV_3871BCX4430
NA
Ebola virus
Zika virus
Malaysian P 6-740
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Investigational
27838352
DrugRepV_3872BCX4430
NA
Ebola virus
Zika virus
Ugandan MR-766
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Investigational
27838352
DrugRepV_3873BCX4430
NA
Ebola virus
Zika virus
Ugandan MR-766
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Investigational
27838352
DrugRepV_3874BCX4430
NA
Ebola virus
Zika virus
Ugandan MR-766
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Investigational
27838352
DrugRepV_3883UV-1
NA
NA
Ebola virus
Zaire-Kikwit
NA
Plaque assay
Decrease (50 %)
NA
27908828
DrugRepV_3884UV-2
NA
NA
Ebola virus
Zaire-Kikwit
NA
Plaque assay
Decrease (50 %)
NA
27908828
DrugRepV_3885UV-3
NA
NA
Ebola virus
Zaire-Kikwit
NA
Plaque assay
Decrease (50 %)
NA
27908828
DrugRepV_3886UV-4
NA
NA
Ebola virus
Zaire-Kikwit
NA
Plaque assay
Decrease (50 %)
NA
27908828
DrugRepV_3887UV-5
NA
NA
Ebola virus
Zaire-Kikwit
NA
Plaque assay
Decrease (50 %)
NA
27908828
DrugRepV_3888UV-1
NA
NA
Marburg virus
Ci67
NA
Plaque assay
Decrease (50 %)
NA
27908828
DrugRepV_3889UV-2
NA
NA
Marburg virus
Ci67
NA
Plaque assay
Decrease (50 %)
NA
27908828
DrugRepV_3890UV-3
NA
NA
Marburg virus
Ci67
NA
Plaque assay
Decrease (50 %)
NA
27908828
DrugRepV_3891UV-4
NA
NA
Marburg virus
Ci67
NA
Plaque assay
Decrease (50 %)
NA
27908828
DrugRepV_3892UV-5
NA
NA
Marburg virus
Ci67
NA
Plaque assay
Decrease (50 %)
NA
27908828
DrugRepV_3893cp15
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3894cp15
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3895cp15
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3896cp15
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3897cp19
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3898cp19
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3899cp19
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3900cp19
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3901cp3
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3902cp5
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3903cp11
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3904cp13
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3905cp15
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3906cp16
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3907cp19
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3908cp3
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3909cp5
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3910cp11
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3911cp13
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3912cp15
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3913cp16
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3914cp19
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3915cp3
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3916cp5
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3917cp11
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3918cp13
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3919cp15
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3920cp16
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3921cp19
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3922CBS1129
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3923CBS1130
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3924CBS1131
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3925CBS1132
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3926CBS1133
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3927CBS1134
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3928CBS1135
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3929CBS1136
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3930CBS1137
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3931CBS1138
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3932CBS1139
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3933IHVR-19029
NA
NA
Zika virus
PRVABC-59
NA
qRT-PCR
Decrease (50 %)
NA
29253498
DrugRepV_3934IHVR-19029
NA
NA
Ebola virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
29253498
DrugRepV_3938GSK983
NA
NA
Ebola virus
NA
NA
Plaque assay
Decrease (50 %)
NA
29294299
DrugRepV_3939Angelicin
NA
NA
Ebola virus
NA
NA
Plaque assay
Decrease (50 %)
NA
29294299
DrugRepV_3940Benzoquinoline
NA
NA
Ebola virus
NA
NA
Plaque assay
Decrease (50 %)
NA
29294299
DrugRepV_3941SW539
NA
NA
Ebola virus
NA
NA
Plaque assay
Decrease (50 %)
NA
29294299
DrugRepV_3942SW320
NA
NA
Ebola virus
NA
NA
Plaque assay
Decrease (50 %)
NA
29294299
DrugRepV_3943SW351
NA
NA
Ebola virus
NA
NA
Plaque assay
Decrease (50 %)
NA
29294299
DrugRepV_3944SW491
NA
NA
Ebola virus
NA
NA
Plaque assay
Decrease (50 %)
NA
29294299
DrugRepV_3945SW490
NA
NA
Ebola virus
NA
NA
Plaque assay
Decrease (50 %)
NA
29294299
DrugRepV_3946SW388
NA
NA
Ebola virus
NA
NA
Plaque assay
Decrease (50 %)
NA
29294299
DrugRepV_3947SW386
NA
NA
Ebola virus
NA
NA
Plaque assay
Decrease (50 %)
NA
29294299
DrugRepV_3948SW349
NA
NA
Ebola virus
NA
NA
Plaque assay
Decrease (50 %)
NA
29294299
DrugRepV_3949SW991
NA
NA
Ebola virus
NA
NA
Plaque assay
Decrease (50 %)
NA
29294299
DrugRepV_3950SW456
NA
NA
Ebola virus
NA
NA
Plaque assay
Decrease (50 %)
NA
29294299
DrugRepV_395312N-p-dichlorobenzyl aloperine
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_395412N-o-methylbenzyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_395512N-2,4-dichlorobenzyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_395612N-3,5 -dichlorobenzyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_395712N-3,4-dichlorobenzyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_395812N-m-methoxybenzyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_395912N-benzyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_396012N-p-trifluoromethoxylbenzyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_396112N-p-fluorobenzyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_396212N-3,5-dichlorobenzoyl aloperine
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_396312N-p-chlorobenzoyl aloperine
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_396412N-3,4-dichlorobenzoyl aloperine
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_396512N-3,4-dichlorobenzenesulfonyl aloperine
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_396612N-3,5-dichlorobenzenesulfonyl aloperine
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_396712N-o-thiophenesulfonyl aloperine
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_396812N-m-cyanobenzenesulfonyl aloperine
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_396912N-p-chlorobenzenesulfonyl aloperine
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_397012N-p-chlorophenylethyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_397112N-3,4-dichlorophenylethyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_397212N-3,5-dichlorophenylethyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_397312N-3,4-dichlorohydrocinnamyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_397412N-3,5-dichlorohydrocinnamyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_397512N-p-chlorohydrocinnamyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_397612N-p-dichlorobenzyl aloperine
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_397712N-o-methylbenzyl aloperine dihydrochloride
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_397812N-2,4-dichlorobenzyl aloperine dihydrochloride
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_397912N-3,5 -dichlorobenzyl aloperine dihydrochloride
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_398012N-3,4-dichlorobenzyl aloperine dihydrochloride
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_398112N-m-methoxybenzyl aloperine dihydrochloride
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_398212N-benzyl aloperine dihydrochloride
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_398312N-p-trifluoromethoxylbenzyl aloperine dihydrochloride
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_398412N-p-fluorobenzyl aloperine dihydrochloride
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_398512N-3,5-dichlorobenzoyl aloperine
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_398612N-p-chlorobenzoyl aloperine
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_398712N-3,4-dichlorobenzoyl aloperine
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_398812N-3,4-dichlorobenzenesulfonyl aloperine
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_398912N-3,5-dichlorobenzenesulfonyl aloperine
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_399012N-o-thiophenesulfonyl aloperine
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_399112N-m-cyanobenzenesulfonyl aloperine
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_399212N-p-chlorobenzenesulfonyl aloperine
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_3996Tyrphostin AG1478
NA
NA
Lassa virus
NA
NA
Luciferase assay
Decrease (100 %)
NA
21947546
DrugRepV_3997Tyrphostin AG1478
NA
NA
Marburg virus
NA
NA
Luciferase assay
Decrease (100 %)
NA
21947546
DrugRepV_3998Tyrphostin AG1478
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (100 %)
NA
21947546
DrugRepV_3999Genistein-Tyrphostin AG1478
NA
NA
Lassa virus
NA
NA
Luciferase assay
Decrease (99 %)
NA
21947546
DrugRepV_4000Genistein-Tyrphostin AG1478
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (99 %)
NA
21947546
DrugRepV_4001FGI-103
NA
NA
Ebola virus
Zaire
NA
Plaque assay
Decrease (50 %)
NA
20211898
DrugRepV_4002FGI-103
NA
NA
Ebola virus
Sudan
NA
Plaque assay
Decrease (50 %)
NA
20211898
DrugRepV_4003FGI-103
NA
NA
Marburg virus
Ravn
NA
Plaque assay
Decrease (50 %)
NA
20211898
DrugRepV_4004FGI-103
NA
NA
Marburg virus
Ci67
NA
Plaque assay
Decrease (95 %)
NA
20211898
DrugRepV_4005FGI-103
NA
NA
Ebola virus
Zaire
NA
NA
Decrease
NA
20211898
DrugRepV_40062-APB
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4007A23187
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4008Di-Tert-Butylhydroquinone
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4009CA1001
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4011Ionomycin
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4012Ryanodine
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4013Thapsigargin
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4014Xestospongin C
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_40152-APB
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4016A23187
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4017Di-Tert-Butylhydroquinone
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4018CA1001
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4020Ionomycin
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4021Ryanodine
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4022Thapsigargin
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4023Xestospongin C
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4024Agatoxin
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4026Conotoxin
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
Investigational
20668647
DrugRepV_4028Lanthanum Chloride
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4032Tetrandrine
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
Experimental
20668647
DrugRepV_40345-N-ethyl isopropyl amiloride
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4036Benzamil
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4039Agatoxin
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4041Conotoxin
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
Investigational
20668647
DrugRepV_4043Lanthanum Chloride
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4047Tetrandrine
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
Experimental
20668647
DrugRepV_40495-N-ethyl isopropyl amiloride
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4051Benzamil
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_40547-octyl-indolactam
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4056Gliotoxin
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4057Oleic Acid
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
Approved, Investigational, Vet approved
20668647
DrugRepV_4059PKC Inhibitor
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4060PMA
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4061Rottlerin
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4062U73122
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_40637-octyl-indolactam
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4065Gliotoxin
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4066Oleic Acid
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
Approved, Investigational, Vet approved
20668647
DrugRepV_4068PKC Inhibitor
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4069PMA
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4070Rottlerin
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_4071U73122
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
NA
20668647
DrugRepV_407225-OH-cholecalciferol
NA
NA
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
Approved, Nutraceutical
20668647
DrugRepV_40734-OH-tamoxifen
NA
Breast cancer
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
Investigational
20668647
DrugRepV_4074Arg-vasopressin
NA
Enuresis, polyuria, diabetes insipidus, polydipsia and oesophageal varices with bleeding
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
Approved
20668647
DrugRepV_4075Bradykinin
NA
Hypertension and Diabetes Type 2
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
Investigational
20668647
DrugRepV_4077Cholecalciferol
NA
Vitamin D resistant rickets), hypoparathyroidism, and familial hypophosphatemia
Hendra virus
NA
NA
Immunolabeling assay
Decrease (50 %)
Approved
20668647
DrugRepV_408025-OH-cholecalciferol
NA
NA
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
Approved, Nutraceutical
20668647
DrugRepV_40814-OH-tamoxifen
NA
Breast cancer
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
Investigational
20668647
DrugRepV_4082Arg-vasopressin
NA
Enuresis, polyuria, diabetes insipidus, polydipsia and oesophageal varices with bleeding
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
Approved
20668647
DrugRepV_4083Bradykinin
NA
Hypertension and Diabetes Type 3
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
Investigational
20668647
DrugRepV_4085Cholecalciferol
NA
Vitamin D resistant rickets), hypoparathyroidism, and familial hypophosphatemia
Nipah virus
NA
NA
Immunolabeling assay
Decrease (50 %)
Approved
20668647
DrugRepV_41032-(4-tert-butylphenyl)-N-[(E)-(3,4-diethoxyphenyl)methylidene]cyclopropane-1-carbohydrazide
NA
NA
Chikungunya virus
NA
NA
CPE reduction assay
Decrease (50 %)
NA
23380636
DrugRepV_41042-(4-tert-butylphenyl)-N-[(E)-(3,5-dibromo-4-methoxyphenyl)methylidene]cyclopropane-1-carbohydrazide
NA
NA
Chikungunya virus
NA
NA
CPE reduction assay
Decrease (50 %)
NA
23380636
DrugRepV_41052-(4-tert-butylphenyl)-N-[(E)-[4-(diethylamino)-2-hydroxyphenyl]methylidene]cyclopropane-1-carbohydrazide
NA
NA
Chikungunya virus
NA
NA
CPE reduction assay
Decrease (50 %)
NA
23380636
DrugRepV_41062-(4-tert-butylphenyl)-N-[(E)-[4-(trifluoromethyl)phenyl]methylidene]cyclopropane-1-carbohydrazide
NA
NA
Chikungunya virus
NA
NA
CPE reduction assay
Decrease (50 %)
NA
23380636
DrugRepV_41072-(4-tert-butylphenyl)-N-[(E)-[4-(methylsulfanyl)phenyl]methylidene]cyclopropane-1-carbohydrazide
NA
NA
Chikungunya virus
NA
NA
CPE reduction assay
Decrease (50 %)
NA
23380636
DrugRepV_41082-(4-tert-butylphenyl)-N-[(E)-(4-methylphenyl)methylidene]cyclopropane-1-carbohydrazide
NA
NA
Chikungunya virus
NA
NA
CPE reduction assay
Decrease (50 %)
NA
23380636
DrugRepV_41092-(4-tert-butylphenyl)-N-[(1E)-2-[(1-methylnaphthalen-2-yl)oxy]ethylidene]cyclopropane-1-carbohydrazide
NA
NA
Chikungunya virus
NA
NA
CPE reduction assay
Decrease (50 %)
NA
23380636
DrugRepV_41102-(4-tert-butylphenyl)-N-[(E)-[4-(propan-2-yl)phenyl]methylidene]cyclopropane-1-carbohydrazide
NA
NA
Chikungunya virus
NA
NA
CPE reduction assay
Decrease (50 %)
NA
23380636
DrugRepV_41112-(4-tert-butylphenyl)-N-[(1E)-1-phenylpropylidene]cyclopropane-1-carbohydrazide
NA
NA
Chikungunya virus
NA
NA
CPE reduction assay
Decrease (50 %)
NA
23380636
DrugRepV_4112N-[(E)-(4-bromophenyl)methylidene]-2-phenylcyclopropane-1-carbohydrazide
NA
NA
Chikungunya virus
NA
NA
CPE reduction assay
Decrease (50 %)
NA
23380636
DrugRepV_4113N-[(E)-(4-hydroxyphenyl)methylidene]-2-phenylcyclopropane-1-carbohydrazide
NA
NA
Chikungunya virus
NA
NA
CPE reduction assay
Decrease (50 %)
NA
23380636
DrugRepV_4114N-[(E)-(4-cyclohexylphenyl)methylidene]-2-phenylcyclopropane-1-carbohydrazide
NA
NA
Chikungunya virus
NA
NA
CPE reduction assay
Decrease (50 %)
NA
23380636
DrugRepV_4115N-[(1E)-1-(4-methoxyphenyl)ethylidene]-2-phenylcyclopropane-1-carbohydrazide
NA
NA
Chikungunya virus
NA
NA
CPE reduction assay
Decrease (50 %)
NA
23380636
DrugRepV_4116(2E)-3-(4-tert-butylphenyl)-N-[(E)-(3,4-diethoxyphenyl)methylidene]prop-2-enehydrazide
NA
NA
Chikungunya virus
NA
NA
CPE reduction assay
Decrease (50 %)
NA
23380636
DrugRepV_4117Coumarin A
NA
NA
Chikungunya virus
Acol
NA
Plating method
Decrease (50 %)
NA
28100218
DrugRepV_4118Coumarin B
NA
NA
Chikungunya virus
Acol
NA
Plating method
Decrease (50 %)
NA
28100218
DrugRepV_4119Lupeol Acetate 26SK001
NA
NA
Chikungunya virus
Acol
NA
Plating method
Decrease (50 %)
NA
28100218
DrugRepV_4120Voacangine 26SK002
NA
NA
Chikungunya virus
Acol
NA
Plating method
Decrease (50 %)
NA
28100218
DrugRepV_4121Coumarin A
NA
NA
Chikungunya virus
Acol
NA
Plating method
Decrease (44 %)
NA
28100218
DrugRepV_4122Coumarin B
NA
NA
Chikungunya virus
Acol
NA
Plating method
Decrease (92.5 %)
NA
28100218
DrugRepV_4123Lupeol Acetate 26SK001
NA
NA
Chikungunya virus
Acol
NA
Plating method
Decrease (4.1 %)
NA
28100218
DrugRepV_4124Voacangine 26SK002
NA
NA
Chikungunya virus
Acol
NA
Plating method
Decrease (0.4 %)
NA
28100218
DrugRepV_41253-{3-[(1E)-1-(hydroxyimino)ethyl]phenyl}-5-methyl-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
899
NA
CPE inhibition assay
Decrease (50 %)
NA
28619679
DrugRepV_41263-{3-[(1E)-1-(methoxyimino)ethyl]phenyl}-5-methyl-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
899
NA
CPE inhibition assay
Decrease (50 %)
NA
28619679
DrugRepV_41275-ethyl-3-{3-[(1E)-1-(methoxyimino)ethyl]phenyl}-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
899
NA
CPE inhibition assay
Decrease (50 %)
NA
28619679
DrugRepV_41283-(3-acetylphenyl)-5-ethyl-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
899
NA
CPE inhibition assay
Decrease (50 %)
NA
28619679
DrugRepV_41295-(aminomethyl)-3-{3-[(1E)-1-(methoxyimino)ethyl]phenyl}-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
899
NA
CPE inhibition assay
Decrease (50 %)
NA
28619679
DrugRepV_41303-{3-[(1E)-1-(methoxyimino)ethyl]phenyl}-5-sulfanyl-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
899
NA
CPE inhibition assay
Decrease (50 %)
NA
28619679
DrugRepV_41313-{3-[(1E)-1-(methoxyimino)ethyl]phenyl}-5-(methylsulfanyl)-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
899
NA
CPE inhibition assay
Decrease (50 %)
NA
28619679
DrugRepV_41323-{3-[(1E)-1-(methoxyimino)ethyl]phenyl}-5-(methylamino)-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
899
NA
CPE inhibition assay
Decrease (50 %)
NA
28619679
DrugRepV_41335-ethyl-3-{3-[(1E)-1-{[2-(4-methylpiperazin-1-yl)ethoxy]imino}ethyl]phenyl}-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
899
NA
CPE inhibition assay
Decrease (50 %)
NA
28619679
DrugRepV_41345-ethyl-3-{3-[(1E)-1-{[2-(morpholin-4-yl)ethoxy]imino}ethyl]phenyl}-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
899
NA
CPE inhibition assay
Decrease (50 %)
NA
28619679
DrugRepV_41355-ethyl-3-{3-[(1E)-1-{[2-(thiomorpholin-4-yl)ethoxy]imino}ethyl]phenyl}-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
899
NA
CPE inhibition assay
Decrease (50 %)
NA
28619679
DrugRepV_41363-{3-[(1E)-1-{[2-(diethylamino)ethoxy]imino}ethyl]phenyl}-5-ethyl-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
899
NA
CPE inhibition assay
Decrease (50 %)
NA
28619679
DrugRepV_41373-{3-[(1E)-1-{[2-(cyclohexylamino)ethoxy]imino}ethyl]phenyl}-5-ethyl-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
899
NA
CPE inhibition assay
Decrease (50 %)
NA
28619679
DrugRepV_41385-ethyl-3-{3-[(1E)-1-{[2-(piperidin-1-yl)ethoxy]imino}ethyl]phenyl}-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
899
NA
CPE inhibition assay
Decrease (50 %)
NA
28619679
DrugRepV_41395-ethyl-3-{3-[(1E)-1-{[2-(pyrrolidin-1-yl)ethoxy]imino}ethyl]phenyl}-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
899
NA
CPE inhibition assay
Decrease (50 %)
NA
28619679
DrugRepV_41403-{3-[(1E)-1-({2-[4-(dimethylamino)piperidin-1-yl]ethoxy}imino)ethyl]phenyl}-5-ethyl-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
899
NA
CPE inhibition assay
Decrease (50 %)
NA
28619679
DrugRepV_41415-ethyl-3-{3-[(1E)-1-(methoxyimino)ethyl]phenyl}-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
Venturini
NA
qRT-PCR
Decrease (50 %)
NA
28619679
DrugRepV_41425-ethyl-3-{3-[(1E)-1-{[2-(morpholin-4-yl)ethoxy]imino}ethyl]phenyl}-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
Venturini
NA
qRT-PCR
Decrease (50 %)
NA
28619679
DrugRepV_41435-ethyl-3-{3-[(1E)-1-{[2-(piperidin-1-yl)ethoxy]imino}ethyl]phenyl}-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
Venturini
NA
qRT-PCR
Decrease (50 %)
NA
28619679
DrugRepV_41445-ethyl-3-{3-[(1E)-1-(methoxyimino)ethyl]phenyl}-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
Congo 95
NA
qRT-PCR
Decrease (50 %)
NA
28619679
DrugRepV_41455-ethyl-3-{3-[(1E)-1-{[2-(morpholin-4-yl)ethoxy]imino}ethyl]phenyl}-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
Congo 95
NA
qRT-PCR
Decrease (50 %)
NA
28619679
DrugRepV_41465-ethyl-3-{3-[(1E)-1-{[2-(piperidin-1-yl)ethoxy]imino}ethyl]phenyl}-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
Congo 95
NA
qRT-PCR
Decrease (50 %)
NA
28619679
DrugRepV_41475-ethyl-3-{3-[(1E)-1-(methoxyimino)ethyl]phenyl}-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
St. Martin 20235
NA
qRT-PCR
Decrease (50 %)
NA
28619679
DrugRepV_41485-ethyl-3-{3-[(1E)-1-{[2-(piperidin-1-yl)ethoxy]imino}ethyl]phenyl}-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
NA
NA
Chikungunya virus
St. Martin 20235
NA
qRT-PCR
Decrease (50 %)
NA
28619679
DrugRepV_41492-(4-tert-butylphenyl)-N-[(E)-(4-ethoxyphenyl)methylidene]cyclopropane-1-carbohydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_41502-(4-tert-butylphenyl)-N-[(E)-[4-(trifluoromethyl)phenyl]methylidene]cyclopropane-1-carbohydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4151N-[(E)-(4-hydroxyphenyl)methylidene]-2-phenylcyclopropane-1-carbohydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4152N-[(1E)-1-(4-cyclohexylphenyl)ethylidene]-2-phenylcyclopropane-1-carbohydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4153N-[(1E)-1-(4-methoxyphenyl)ethylidene]-2-phenylcyclopropane-1-carbohydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4154(2E)-3-(4-tert-butylphenyl)-N-[(E)-(3,4-diethoxyphenyl)methylidene]prop-2-enehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_41552-(4-tert-butylphenyl)-N-[(E)-(4-ethoxyphenyl)methylidene]cyclopropane-1-carbohydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_41562-(4-tert-butylphenyl)-N-[(E)-(4-hydroxyphenyl)methylidene]cyclopropane-1-carbohydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4157(2E)-3-(4-tert-butylphenyl)-N-[(E)-(4-ethoxyphenyl)methylidene]prop-2-enehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4158(2E)-3-(4-tert-butylphenyl)-N-[(E)-(4-methylphenyl)methylidene]prop-2-enehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4159(2E)-3-(4-methylphenyl)-N-[(E)-(4-methylphenyl)methylidene]prop-2-enehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4160(2E)-N-[(E)-(4-methylphenyl)methylidene]-3-phenylprop-2-enehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4161(2E)-3-(4-tert-butylphenyl)-N-[(E)-[4-(propan-2-yl)phenyl]methylidene]prop-2-enehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4162(2E)-3-(4-tert-butylphenyl)-N-[(E)-(4-tert-butylphenyl)methylidene]prop-2-enehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4163(2E)-3-(4-tert-butylphenyl)-N-[(1E)-1-(4-cyclohexylphenyl)ethylidene]prop-2-enehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4164(2E)-N-[(1E)-1-(4-cyclohexylphenyl)ethylidene]-3-phenylprop-2-enehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4165(2E)-3-(4-tert-butylphenyl)-N-[(E)-phenylmethylidene]prop-2-enehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4166(2E)-3-(4-tert-butylphenyl)-N-[(E)-(4-nitrophenyl)methylidene]prop-2-enehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4167(2E)-3-(4-tert-butylphenyl)-N-[(1E)-1-(4-chlorophenyl)ethylidene]prop-2-enehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4168(2E)-3-(4-tert-butylphenyl)-N-[(1E)-1-(pyrazin-2-yl)ethylidene]prop-2-enehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4169(2E)-3-(4-tert-butylphenyl)-N-[(1E)-1-(4-ethoxyphenyl)ethylidene]prop-2-enehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4170(2E)-N-[(1E)-1-{[1,1-biphenyl]-4-yl}ethylidene]-3-(4-tert-butylphenyl)prop-2-enehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4171(2E)-N-[(E)-(4-ethoxyphenyl)methylidene]-3-(4-methylphenyl)prop-2-enehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4172(2E)-3-(4-tert-butylphenyl)-N-{[4-(trifluoromethyl)phenyl]methyl}prop-2-enamide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4173(2E)-3-phenyl-N-{[4-(trifluoromethyl)phenyl]methyl}prop-2-enamide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4174(2E)-N-({[1,1-biphenyl]-4-yl}methyl)-3-(4-tert-butylphenyl)prop-2-enamide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4175(2E)-N-({[1,1-biphenyl]-4-yl}methyl)-3-phenylprop-2-enamide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_41763-(4-tert-butylphenyl)-N-[(E)-(4-ethoxyphenyl)methylidene]propanehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4177N-[(E)-(4-ethoxyphenyl)methylidene]-3-phenylpropanehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_41783-(4-tert-butylphenyl)-N-[(E)-(4-methylphenyl)methylidene]propanehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4179N-[(E)-(4-methylphenyl)methylidene]-3-phenylpropanehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_41803-(4-tert-butylphenyl)-N-[(E)-(4-hydroxyphenyl)methylidene]propanehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4181N-[(E)-(4-methylphenyl)methylidene]-3-phenylpropanehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_41823-(4-tert-butylphenyl)-N-[(1E)-1-(4-cyclohexylphenyl)ethylidene]propanehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_4183N-[(E)-(4-cyclohexylphenyl)methylidene]-3-phenylpropanehydrazide
NA
NA
Chikungunya virus
889
NA
CPE reduction assay
Decrease (50 %)
NA
29336951
DrugRepV_41841-(4-{2-[1-cyclohexyl-2-(furan-3-yl)-1H-1,3-benzodiazol-5-yl]-1,3-oxazol-5-yl}phenyl)pyrrolidin-2-one
NA
NA
Chikungunya virus
SL10571
NA
MTT assay
Decrease (50 %)
NA
28236746
DrugRepV_41861-(4-{2-[1-cyclohexyl-2-(furan-3-yl)-1H-1,3-benzodiazol-5-yl]-1,3-oxazol-5-yl}phenyl)pyrrolidin-2-one
NA
NA
Chikungunya virus
S27
NA
MTT assay
Decrease (50 %)
NA
28236746
DrugRepV_41881-(4-{2-[1-cyclohexyl-2-(furan-3-yl)-1H-1,3-benzodiazol-5-yl]-1,3-oxazol-5-yl}phenyl)pyrrolidin-2-one
NA
NA
Chikungunya virus
BaH306
NA
MTT assay
Decrease (50 %)
NA
28236746
DrugRepV_4190Phorbol
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_4191Phorbol-12-acetate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Experimental
25970561
DrugRepV_4192Phorbol-12-decanoate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_4193Phorbol-13-acetate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_4194Phorbol-13-butyrate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_4195Pphorbol-13-decanoate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_4196Phorbol-13-tetradecanoate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_4197Phorbol-12,13-diacetate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_4198Phorbol-12,13-dibutyrate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_4199Phorbol-12,13- dihexanoate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_4200Phorbol-12,13-didecanoate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_42014α-phorbol-12,13-didecanoate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_420212-O-tetradecanoylphorbol-13-acetate
NA
Cancer
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Phase II
25970561
DrugRepV_420312-O-tetradecanoyl-4?-phorbol-13-acetate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_420412-O- tiglylphorbol-13-decanoate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_420512-O-(N-methylanthranilate) phorbol-13-acetate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_4206Phorbol-13,20-diacetate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_420712,13-O,O-dinonanoylphorbol-20-homovanillate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_420812-O-phenylacetyl-13-O-acetylphorbol-20-homovanillate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_4209Phorbol-12,13,20-triacetate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_421020-oxo-20-deoxyphorbol-12,13-dibutyrate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_421112-O-tetradecanoyl-20-oxo-20-deoxyphorbol-13-acetate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_421212-deoxyphorbol-13-acetate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_421313-O-isobutyryl-12-deoxyphorbol-20-acetate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_421413-O-phenylacetyl-12-deoxyphorbol-20-acetate
NA
NA
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
25970561
DrugRepV_4218Resiniferatoxin
NA
Interstitial cystitis and urinary incontinence
Chikungunya virus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Investigational
25970561
DrugRepV_4220Arbidol
NA
NA
Chikungunya virus
LR2006 OPY1
NA
Immunoflourescence assay
Decrease (50 %)
Investigational
21440006
DrugRepV_4221HZ2a
NA
NA
Chikungunya virus
LR2006 OPY1
NA
Immunoflourescence assay
Decrease (50 %)
NA
21440006
DrugRepV_42226-bromo-4-(dimethylaminomethyl)-5-hydroxy-1-methyl-2-(phe- nylsulphonylmethyl)-1H-indole-3-carboxylate
NA
NA
Chikungunya virus
LR2006 OPY1
NA
Immunoflourescence assay
Decrease (50 %)
NA
21440006
DrugRepV_42236-bromo- 4-(dimethylaminomethyl)-5-hydroxy-1-methyl-2-(methylphenyl- sulphoxyde)-1H-indole-3-carboxylate
NA
NA
Chikungunya virus
LR2006 OPY1
NA
Immunoflourescence assay
Decrease (50 %)
NA
21440006
DrugRepV_4224(2E)-3-(4-tert-butylphenyl)-N-[(E)-(4-ethoxyphenyl)methylidene]prop-2-enehydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42253-[(E)-{[2-(4-methylphenyl)-1H-indol-3-yl]methylidene}amino]-1-(2-phenylethyl)thiourea
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4226(2E)-N-[(E)-(4-ethoxyphenyl)methylidene]-3-[4-(propan-2-yl)phenyl]prop-2-enehydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4227(2E)-N-[(E)-(4-ethoxyphenyl)methylidene]-3-[4-(trifluoromethyl)phenyl]prop-2-enehydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4228(2E)-N-[(E)-(4-ethoxyphenyl)methylidene]-3-(4-methoxyphenyl)prop-2-enehydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4229(2E)-3-{[1,1-biphenyl]-4-yl}-N-[(E)-(4-ethoxyphenyl)methylidene]prop-2-enehydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4230(2E)-N-[(E)-(4-methylphenyl)methylidene]-3-[4-(propan-2-yl)phenyl]prop-2-enehydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4231(2E)-N-[(E)-(4-methylphenyl)methylidene]-3-[4-(trifluoromethyl)phenyl]prop-2-enehydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4232(2E)-3-(4-methoxyphenyl)-N-[(E)-(4-methylphenyl)methylidene]prop-2-enehydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4233(2E)-3-{[1,1-biphenyl]-4-yl}-N-[(E)-(4-methylphenyl)methylidene]prop-2-enehydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4234(2E)-N-[(1E)-1-(4-cyclohexylphenyl)ethylidene]-3-[4-(propan-2-yl)phenyl]prop-2-enehydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4235(2E)-N-[(1E)-1-(4-cyclohexylphenyl)ethylidene]-3-[4-(trifluoromethyl)phenyl]prop-2-enehydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4236(2E)-N-[(1E)-1-(4-cyclohexylphenyl)ethylidene]-3-(4-methoxyphenyl)prop-2-enehydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4237(2E)-3-{[1,1-biphenyl]-4-yl}-N-[(1E)-1-(4-cyclohexylphenyl)ethylidene]prop-2-enehydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4238(2E)-N-[(E)-(4-hydroxyphenyl)methylidene]-3-[4-(propan-2-yl)phenyl]prop-2-enehydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4239N-[(E)-(4-ethoxyphenyl)methylidene]naphthalene-2-carbohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4240N-[(E)-(4-ethoxyphenyl)methylidene]quinoline-3-carbohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4241N-[(E)-(4-ethoxyphenyl)methylidene]quinoline-2-carbohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4242N-[(E)-(4-ethoxyphenyl)methylidene]-1H-indole-2-carbohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4243N-[(E)-(4-ethoxyphenyl)methylidene]-1H-1,3-benzodiazole-2-carbohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4244N-[(E)-(4-methylphenyl)methylidene]naphthalene-2-carbohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4245N-[(E)-(4-methylphenyl)methylidene]quinoline-3-carbohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4246N-[(E)-(4-methylphenyl)methylidene]quinoline-2-carbohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4247N-[(E)-(4-methylphenyl)methylidene]-1H-indole-2-carbohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4248N-[(E)-(4-methylphenyl)methylidene]-1H-1,3-benzodiazole-2-carbohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4249N-[(E)-(4-hydroxyphenyl)methylidene]naphthalene-2-carbohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4250N-[(E)-(4-hydroxyphenyl)methylidene]quinoline-3-carbohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4251N-[(E)-(4-hydroxyphenyl)methylidene]quinoline-2-carbohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4252N-[(E)-(4-hydroxyphenyl)methylidene]-1H-indole-2-carbohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4253N-[(E)-(4-hydroxyphenyl)methylidene]-1H-1,3-benzodiazole-2-carbohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4254N-[(1E)-1-(4-cyclohexylphenyl)ethylidene]naphthalene-2-carbohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4255N-[(1E)-1-(4-cyclohexylphenyl)ethylidene]quinoline-3-carbohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4256N-[(1E)-1-(4-cyclohexylphenyl)ethylidene]quinoline-2-carbohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4257N-[(1E)-1-(4-cyclohexylphenyl)ethylidene]-1H-indole-2-carbohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4258N-[(1E)-1-(4-cyclohexylphenyl)ethylidene]-1H-1,3-benzodiazole-2-carbohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42593-(4-tert-butylphenyl)-N-[(E)-(4-ethoxyphenyl)methylidene]-3-oxopropanehydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42603-(4-tert-butylphenyl)-N-[(E)-(4-methylphenyl)methylidene]-3-oxopropanehydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42613-(4-tert-butylphenyl)-N-[(E)-(4-hydroxyphenyl)methylidene]-3-oxopropanehydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42623-[(1E)-2-(4-tert-butylphenyl)ethenyl]-1-[(E)-[(4-ethoxyphenyl)methylidene]amino]urea
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42633-[(1E)-2-(4-tert-butylphenyl)ethenyl]-1-[(E)-[(4-methylphenyl)methylidene]amino]urea
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42643-[(1E)-2-(4-tert-butylphenyl)ethenyl]-1-[(E)-[(4-hydroxyphenyl)methylidene]amino]urea
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42653-[(1E)-2-(4-tert-butylphenyl)ethenyl]-1-[(E)-[1-(4-cyclohexylphenyl)ethylidene]amino]urea
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42661-[(E)-[(4-ethoxyphenyl)methylidene]amino]-3-(2-phenylethyl)thiourea
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42671-[(E)-[(4-methylphenyl)methylidene]amino]-3-(2-phenylethyl)thiourea
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42681-[(E)-[(4-hydroxyphenyl)methylidene]amino]-3-(2-phenylethyl)thiourea
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42691-[(E)-[1-(4-cyclohexylphenyl)ethylidene]amino]-3-(2-phenylethyl)thiourea
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42703-[(1E)-2-(4-tert-butylphenyl)ethenyl]-1-[(4-ethoxyphenyl)methyl]urea
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42713-[(1E)-2-(4-tert-butylphenyl)ethenyl]-1-[(4-methylphenyl)methyl]urea
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42721-benzyl-3-[(1E)-2-(4-tert-butylphenyl)ethenyl]urea
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42731-[(4-methoxyphenyl)methyl]-3-[(1E)-2-phenylethenyl]urea
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42741-[(4-methylphenyl)methyl]-3-[(1E)-2-phenylethenyl]urea
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42753-[(1E)-2-(4-tert-butylphenyl)ethenyl]-1-(4-methylphenyl)urea
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42763-[(1E)-2-(4-tert-butylphenyl)ethenyl]-1-(4-hydroxyphenyl)urea
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42771-(4-methylphenyl)-3-[(1E)-2-phenylethenyl]urea
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42781-(4-hydroxyphenyl)-3-[(1E)-2-phenylethenyl]urea
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4279N-[(2E)-3-(4-tert-butylphenyl)prop-2-enoyl]-4-ethoxybenzohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4280N-[(2E)-3-(4-tert-butylphenyl)prop-2-enoyl]-4-methylbenzohydrazide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42812-[(1E)-2-(4-tert-butylphenyl)ethenyl]-5-(4-ethoxyphenyl)-1,3,4-oxadiazole
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42822-[(1E)-2-(4-tert-butylphenyl)ethenyl]-5-(4-methylphenyl)-1,3,4-oxadiazole
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42832-[2-(4-tert-butylphenyl)ethyl]-5-(4-ethoxyphenyl)-1,3,4-oxadiazole
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42842-[2-(4-tert-butylphenyl)ethyl]-5-(4-methylphenyl)-1,3,4-oxadiazole
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42852-(4-ethoxyphenyl)-5-(2-phenylethyl)-1,3,4-oxadiazole
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42862-(4-methylphenyl)-5-(2-phenylethyl)-1,3,4-oxadiazole
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42874-{5-[2-(4-tert-butylphenyl)ethyl]-1,3,4-oxadiazol-2-yl}phenol
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42882-[(4-tert-butylphenyl)methyl]-5-(4-ethoxyphenyl)-1,3,4-oxadiazole
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42892-[(4-tert-butylphenyl)methyl]-5-(4-methylphenyl)-1,3,4-oxadiazole
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42904-(4-methylphenyl)-1-(2-phenylethyl)-1H-1,2,3-triazole
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4291(2E)-3-(4-tert-butylphenyl)-N-(5-methyl-1H-1,3-benzodiazol-2-yl)prop-2-enamide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4292(2E)-N-(1H-1,3-benzodiazol-2-yl)-3-(4-tert-butylphenyl)prop-2-enamide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_42933-(4-tert-butylphenyl)-N-(5-methyl-1H-1,3-benzodiazol-2-yl)propanamide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4294N-(1H-1,3-benzodiazol-2-yl)-3-(4-tert-butylphenyl)propanamide
NA
NA
Chikungunya virus
899
NA
CPE reduction assay
Decrease (50 %)
NA
29499487
DrugRepV_4299Fisetin
NA
Frail Elderly Syndrome
Chikungunya virus
NA
NA
NA
Decrease (50 %)
Experimental
27460167
DrugRepV_4300Quercetagetin
NA
NA
Chikungunya virus
NA
NA
NA
Decrease (50 %)
NA
27460167
DrugRepV_4302Carbocyclic adenosine
NA
NA
Ebola virus
Mayinga
NA
MTT assay
Decrease (50 %)
NA
9988190
DrugRepV_4303Carbocyclic 3-deazaadenosine
NA
NA
Ebola virus
Mayinga
NA
MTT assay
Decrease (50 %)
NA
9988190
DrugRepV_43049-[trans- 2,trans - 3 - dihydroxy - 4 - (methyl) - cyclopent - 4 - enyl] - 3 - deazaadenine
NA
NA
Ebola virus
Mayinga
NA
MTT assay
Decrease (50 %)
NA
9988190
DrugRepV_43059-[trans-2,trans-3-dihydroxy-4-hydroxymethyl-cyclopent-4-enyl]-adenine
NA
NA
Ebola virus
Mayinga
NA
MTT assay
Decrease (50 %)
NA
9988190
DrugRepV_43069-[trans-2,trans-3-dihydroxy-4-hydroxymethyl-cyclopent-4-enyl]-3-deazaadenine
NA
NA
Ebola virus
Mayinga
NA
MTT assay
Decrease (50 %)
NA
9988190
DrugRepV_43079-[trans-2,trans-3-dihydroxycyclopent-4-enyl]- adenine (DHCpAdo)
NA
NA
Ebola virus
Mayinga
NA
MTT assay
Decrease (50 %)
NA
9988190
DrugRepV_43089-[trans-2,trans-3-dihydroxycyclopent- 4-enyl]-3-deazaadenine (DHCp-c3Ado)
NA
NA
Ebola virus
Mayinga
NA
MTT assay
Decrease (50 %)
NA
9988190
DrugRepV_43094,5- didehydro-5-deoxy-5-fluoroadenosine (DDFA)
NA
NA
Ebola virus
Mayinga
NA
MTT assay
Decrease (50 %)
NA
9988190
DrugRepV_4311Guanosine Dialdehyde
NA
NA
Ebola virus
Mayinga
NA
MTT assay
Decrease (50 %)
NA
9988190
DrugRepV_4312Adenosine Dialdehyde
NA
NA
Ebola virus
Mayinga
NA
MTT assay
Decrease (50 %)
Approved, Investigational
9988190
DrugRepV_4314Carbocyclic 3-deazaadenosine
NA
NA
Ebola virus
Sudan (Boneface strain)
NA
Plaque reduction assay
Decrease (50 %)
NA
9988190
DrugRepV_43159-[trans-2,trans-3-dihydroxy-4-hydroxymethyl-cyclopent-4-enyl]-adenine
NA
NA
Ebola virus
Sudan (Boneface strain)
NA
Plaque reduction assay
Decrease (50 %)
NA
9988190
DrugRepV_43169-[trans-2,trans-3-dihydroxy-4-hydroxymethyl-cyclopent-4-enyl]-3-deazaadenine
NA
NA
Ebola virus
Sudan (Boneface strain)
NA
Plaque reduction assay
Decrease (50 %)
NA
9988190
DrugRepV_4317Carbocyclic 3-deazaadenosine
NA
NA
Ebola virus
EBO-Z
NA
Survival assay
Increase
NA
9988190
DrugRepV_4318FGI-106
NA
NA
Ebola virus
Zaire
NA
Plaque assay
Decrease (50 %)
NA
19523489
DrugRepV_4319FGI-106
NA
NA
Rift Valley fever virus
MP12
NA
Plaque assay
Decrease (50 %)
NA
19523489
DrugRepV_4320FGI-106
NA
NA
Ebola virus
Zaire
NA
Survival assay
Increase
NA
19523489
DrugRepV_4321N-(1,3-benzodioxol-5-ylmethyl)-2-(3-cyano-2-methyl-1H-indol-1-yl)acetamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (44.6 %)
NA
24501399
DrugRepV_4322N-benzyl-6-phenyl-2,3,4,9-tetrahydro-1H-carbazol-1-amine hydrochloride
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (32.6 %)
NA
24501399
DrugRepV_43239H-carbazol-3-amine
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (6.1 %)
NA
24501399
DrugRepV_43247-(1H-benzimidazol-2-ylthio)-8-methyl[1,3]dioxolo[4,5-g]quinolin-6(5H)-one
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (-3.8 %)
NA
24501399
DrugRepV_4325N-[2-(2-methoxyethyl)-1,2,3,4-tetrahydropyrazino[1,2-a]benzimidazol-8-yl]benzamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (-16 %)
NA
24501399
DrugRepV_4326tris[4-(dimethylamino)phenyl]methanol
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (31.8 %)
NA
24501399
DrugRepV_43276-chloro-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-2-(3-pyridinyl)-4-quinolinecarboxamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (31.8 %)
NA
24501399
DrugRepV_43281-(2-furoyl)-5-(2-furyl)-3-(3-methoxyphenyl)-4,5-dihydro-1H-pyrazole
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (-1.6 %)
NA
24501399
DrugRepV_43292-[(1H-benzimidazol-2-ylmethyl)thio]-1-[2-(4-methylphenoxy)ethyl]-1H-benzimidazole
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (-1.8 %)
NA
24501399
DrugRepV_4330N-(3-chloro-4-fluorophenyl)-N-[4-(4-morpholinylsulfonyl)phenyl]urea
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (66.3 %)
NA
24501399
DrugRepV_43314-{[(5-methyl-2-thienyl)methyl]amino}phenol
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (-12.6 %)
NA
24501399
DrugRepV_4332N-[5-(1H-benzimidazol-2-yl)-2-methylphenyl]-1,3-benzodioxole-5-carboxamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (-3.4 %)
NA
24501399
DrugRepV_4333N-[1-benzyl-2-oxo-2-(4-phenyl-1-piperazinyl)ethyl]benzamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (10.2 %)
NA
24501399
DrugRepV_43342-methoxy-N-[1-methyl-2-(1-pyrrolidinylmethyl)-1H-benzimidazol-5-yl]benzamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (8.6 %)
NA
24501399
DrugRepV_4335N-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-2-(2-naphthyloxy)acetamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (66.9 %)
NA
24501399
DrugRepV_4336N-(2,5-dimethoxyphenyl)-N-[4-(trifluoromethyl)phenyl]urea
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (9.6 %)
NA
24501399
DrugRepV_43374-{[(1H-benzimidazol-2-ylthio)acetyl]amino}phenyl thiocyanate
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (34 %)
NA
24501399
DrugRepV_4338N-(3,4-dichlorophenyl)-N-[3-(trifluoromethyl)phenyl]urea
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (11.6 %)
NA
24501399
DrugRepV_4339N-1,3-benzodioxol-5-yl-6-chloro-2-(3-pyridinyl)-4-quinolinecarboxamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (45.7 %)
NA
24501399
DrugRepV_4340N-(3-chlorophenyl)-N-(4-cyanophenyl)urea
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (10.1 %)
NA
24501399
DrugRepV_4341N-[4-(1H-benzimidazol-2-yl)phenyl]-2-chloro-5-(4H-1,2,4-triazol-4-yl)benzamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (-3.4 %)
NA
24501399
DrugRepV_4342N-[3-(aminocarbonyl)-5-benzyl-2-thienyl]-2-methyl-3-furamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (5.7 %)
NA
24501399
DrugRepV_43434,5-dimethyl-2-{[(5-propyl-3-thienyl)carbonyl]amino}-N-(3-pyridinylmethyl)-3-thiophenecarboxamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (-24.6 %)
NA
24501399
DrugRepV_43441-(isopropylamino)-3-(3-phenyl-4,5-dihydropyrazolo[4,3-a]carbazol-10(3H)-yl)-2-propanol
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (13.1 %)
NA
24501399
DrugRepV_43452-[(4-tert-butyl-1,3-thiazol-2-yl)amino]-8-quinolinol
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (6.4 %)
NA
24501399
DrugRepV_4346N-(aminocarbonyl)-2-{[(5-methyl-3-thienyl)carbonyl]amino}-3-thiophenecarboxamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (6.2 %)
NA
24501399
DrugRepV_43472-chloro-N-(4-phenyl-1,3-thiazol-2-yl)-5-(4H-1,2,4-triazol-4-yl)benzamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (10.7 %)
NA
24501399
DrugRepV_4348N-[3-(2-oxo-2H-chromen-3-yl)phenyl]-1,3-benzodioxole-5-carboxamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (2.1 %)
NA
24501399
DrugRepV_43494,5-dimethyl-2-[(phenoxyacetyl)amino]-N-(3-pyridinylmethyl)-3-thiophenecarboxamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (-0.6 %)
NA
24501399
DrugRepV_4350N-(4-{[(5-methyl-3-isoxazolyl)amino]sulfonyl}phenyl)-1-benzothiophene-3-carboxamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (-2.6 %)
NA
24501399
DrugRepV_43513-[(1H-benzimidazol-2-ylmethyl)thio]-9-benzyl-9H-[1,2,4]triazolo[4,3-a]benzimidazole
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (-6.1 %)
NA
24501399
DrugRepV_4352methyl N-[4,6-bis(isopropylamino)-1,3,5-triazin-2-yl]-N-cyanoglycinate
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (82.4 %)
NA
24501399
DrugRepV_4353N-(3,4-dichlorophenyl)-2-oxo-2,3-dihydro-1,3-benzoxazole-6-sulfonamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (33.4 %)
NA
24501399
DrugRepV_4354N-(3-pyridinylmethyl)dibenzo[b,d]furan-3-amine
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (25.4 %)
NA
24501399
DrugRepV_4355(1,3-benzodioxol-5-ylmethyl)[4-(1-pyrrolidinyl)phenyl]amine
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (10.5 %)
NA
24501399
DrugRepV_43564-methyl-5-phenyl-N-3-pyridinyl-2-thiophenecarboxamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (25.2 %)
NA
24501399
DrugRepV_4357N-(2,5-dimethoxyphenyl)-2-(2-oxo-1,3-benzoxazol-3(2H)-yl)acetamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (17.4 %)
NA
24501399
DrugRepV_43583-[(2,4-dichlorophenoxy)methyl]-N-(3-pyridinylmethyl)benzamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (26.8 %)
NA
24501399
DrugRepV_43595-phenyl-2-(2-phenylethyl)[1,2,4]triazolo[1,5-a]pyrimidin-7(4H)-one
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (-6.6 %)
NA
24501399
DrugRepV_43606-bromo-2-oxo-N-3-pyridinyl-2H-chromene-3-carboxamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (20.9 %)
NA
24501399
DrugRepV_43612-[(2-methyl-8-quinolinyl)amino]-4H-pyrido[3,2-e][1,3]thiazin-4-one
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (-12.1 %)
NA
24501399
DrugRepV_4362N-(3-chloro-4-fluorophenyl)-N-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (12.3 %)
NA
24501399
DrugRepV_43634-({[(3-chloro-4-fluorophenyl)amino]carbonyl}amino)-N-methylbenzenesulfonamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (1.8 %)
NA
24501399
DrugRepV_43642-(4-fluorophenyl)-N-(4-{[(4-methylphenyl)amino]sulfonyl}phenyl)acetamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (1.1 %)
NA
24501399
DrugRepV_43655-methyl-N-[4-(1-pyrrolidinylsulfonyl)phenyl]-3-thiophenecarboxamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (-0.3 %)
NA
24501399
DrugRepV_43662-amino-N-(3-chlorophenyl)-3-quinolinecarboxamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (-1.5 %)
NA
24501399
DrugRepV_43672-(1,3-benzodioxol-5-yl)-1-(1,3-benzodioxol-5-ylmethyl)-1H-benzimidazole
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (-15.9 %)
NA
24501399
DrugRepV_4368N-{3-[(benzylamino)carbonyl]phenyl}-5-methyl-3-thiophenecarboxamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (-11.5 %)
NA
24501399
DrugRepV_43698-chloro-N-[3-(3-methyl-1H-pyrazol-1-yl)propyl]-2-(2-pyridinyl)-4-quinolinecarboxamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (-11.7 %)
NA
24501399
DrugRepV_4370N-[4-(2,4-difluorophenyl)-1,3-thiazol-2-yl]-2-(2-thienyl)acetamide
NA
NA
Ebola virus
GP, amino acids 196 to 205
NA
CatL-Peptide cleavage
Decrease (8.05 %)
NA
24501399
DrugRepV_4371N-(1,3-benzodioxol-5-ylmethyl)-2-(3-cyano-2-methyl-1H-indol-1-yl)acetamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (24.79 %)
NA
24501399
DrugRepV_4372N-benzyl-6-phenyl-2,3,4,9-tetrahydro-1H-carbazol-1-amine hydrochloride
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (31.07 %)
NA
24501399
DrugRepV_43739H-carbazol-3-amine
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (8.2 %)
NA
24501399
DrugRepV_43747-(1H-benzimidazol-2-ylthio)-8-methyl[1,3]dioxolo[4,5-g]quinolin-6(5H)-one
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (37.87 %)
NA
24501399
DrugRepV_4375N-[2-(2-methoxyethyl)-1,2,3,4-tetrahydropyrazino[1,2-a]benzimidazol-8-yl]benzamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (-0.67 %)
NA
24501399
DrugRepV_4376tris[4-(dimethylamino)phenyl]methanol
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (108.4 %)
NA
24501399
DrugRepV_43776-chloro-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-2-(3-pyridinyl)-4-quinolinecarboxamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (39.17 %)
NA
24501399
DrugRepV_43781-(2-furoyl)-5-(2-furyl)-3-(3-methoxyphenyl)-4,5-dihydro-1H-pyrazole
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (5.24 %)
NA
24501399
DrugRepV_43792-[(1H-benzimidazol-2-ylmethyl)thio]-1-[2-(4-methylphenoxy)ethyl]-1H-benzimidazole
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (-2.7 %)
NA
24501399
DrugRepV_4380N-(3-chloro-4-fluorophenyl)-N-[4-(4-morpholinylsulfonyl)phenyl]urea
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (40.4 %)
NA
24501399
DrugRepV_43814-{[(5-methyl-2-thienyl)methyl]amino}phenol
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (-14.4 %)
NA
24501399
DrugRepV_4382N-[5-(1H-benzimidazol-2-yl)-2-methylphenyl]-1,3-benzodioxole-5-carboxamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (-7.77 %)
NA
24501399
DrugRepV_4383N-[1-benzyl-2-oxo-2-(4-phenyl-1-piperazinyl)ethyl]benzamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (0.34 %)
NA
24501399
DrugRepV_43842-methoxy-N-[1-methyl-2-(1-pyrrolidinylmethyl)-1H-benzimidazol-5-yl]benzamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (-9.26 %)
NA
24501399
DrugRepV_4385N-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-2-(2-naphthyloxy)acetamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (73.49 %)
NA
24501399
DrugRepV_4386N-(2,5-dimethoxyphenyl)-N-[4-(trifluoromethyl)phenyl]urea
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (-4.08 %)
NA
24501399
DrugRepV_43874-{[(1H-benzimidazol-2-ylthio)acetyl]amino}phenyl thiocyanate
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (7.92 %)
NA
24501399
DrugRepV_4388N-(3,4-dichlorophenyl)-N-[3-(trifluoromethyl)phenyl]urea
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (42.12 %)
NA
24501399
DrugRepV_4389N-1,3-benzodioxol-5-yl-6-chloro-2-(3-pyridinyl)-4-quinolinecarboxamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (32.88 %)
NA
24501399
DrugRepV_4390N-(3-chlorophenyl)-N-(4-cyanophenyl)urea
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (24.49 %)
NA
24501399
DrugRepV_4391N-[4-(1H-benzimidazol-2-yl)phenyl]-2-chloro-5-(4H-1,2,4-triazol-4-yl)benzamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (0.86 %)
NA
24501399
DrugRepV_4392N-[3-(aminocarbonyl)-5-benzyl-2-thienyl]-2-methyl-3-furamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (6.5 %)
NA
24501399
DrugRepV_43934,5-dimethyl-2-{[(5-propyl-3-thienyl)carbonyl]amino}-N-(3-pyridinylmethyl)-3-thiophenecarboxamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (-7.5 %)
NA
24501399
DrugRepV_43941-(isopropylamino)-3-(3-phenyl-4,5-dihydropyrazolo[4,3-a]carbazol-10(3H)-yl)-2-propanol
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (35.73 %)
NA
24501399
DrugRepV_43952-[(4-tert-butyl-1,3-thiazol-2-yl)amino]-8-quinolinol
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (-2.85 %)
NA
24501399
DrugRepV_4396N-(aminocarbonyl)-2-{[(5-methyl-3-thienyl)carbonyl]amino}-3-thiophenecarboxamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (37.33 %)
NA
24501399
DrugRepV_43972-chloro-N-(4-phenyl-1,3-thiazol-2-yl)-5-(4H-1,2,4-triazol-4-yl)benzamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (22.44 %)
NA
24501399
DrugRepV_4398N-[3-(2-oxo-2H-chromen-3-yl)phenyl]-1,3-benzodioxole-5-carboxamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (37.22 %)
NA
24501399
DrugRepV_43994,5-dimethyl-2-[(phenoxyacetyl)amino]-N-(3-pyridinylmethyl)-3-thiophenecarboxamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (33.41 %)
NA
24501399
DrugRepV_4400N-(4-{[(5-methyl-3-isoxazolyl)amino]sulfonyl}phenyl)-1-benzothiophene-3-carboxamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (7.38 %)
NA
24501399
DrugRepV_44013-[(1H-benzimidazol-2-ylmethyl)thio]-9-benzyl-9H-[1,2,4]triazolo[4,3-a]benzimidazole
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (-0.01 %)
NA
24501399
DrugRepV_4402methyl N-[4,6-bis(isopropylamino)-1,3,5-triazin-2-yl]-N-cyanoglycinate
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (90.92 %)
NA
24501399
DrugRepV_4403N-(3,4-dichlorophenyl)-2-oxo-2,3-dihydro-1,3-benzoxazole-6-sulfonamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (12.1 %)
NA
24501399
DrugRepV_4404N-(3-pyridinylmethyl)dibenzo[b,d]furan-3-amine
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (21.93 %)
NA
24501399
DrugRepV_4405(1,3-benzodioxol-5-ylmethyl)[4-(1-pyrrolidinyl)phenyl]amine
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (-8.72 %)
NA
24501399
DrugRepV_44064-methyl-5-phenyl-N-3-pyridinyl-2-thiophenecarboxamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (17.7 %)
NA
24501399
DrugRepV_4407N-(2,5-dimethoxyphenyl)-2-(2-oxo-1,3-benzoxazol-3(2H)-yl)acetamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (23.22 %)
NA
24501399
DrugRepV_44083-[(2,4-dichlorophenoxy)methyl]-N-(3-pyridinylmethyl)benzamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (23.55 %)
NA
24501399
DrugRepV_44095-phenyl-2-(2-phenylethyl)[1,2,4]triazolo[1,5-a]pyrimidin-7(4H)-one
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (3.55 %)
NA
24501399
DrugRepV_44106-bromo-2-oxo-N-3-pyridinyl-2H-chromene-3-carboxamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (32.65 %)
NA
24501399
DrugRepV_44112-[(2-methyl-8-quinolinyl)amino]-4H-pyrido[3,2-e][1,3]thiazin-4-one
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (3.23 %)
NA
24501399
DrugRepV_4412N-(3-chloro-4-fluorophenyl)-N-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (25.12 %)
NA
24501399
DrugRepV_44134-({[(3-chloro-4-fluorophenyl)amino]carbonyl}amino)-N-methylbenzenesulfonamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (-11.51 %)
NA
24501399
DrugRepV_44142-(4-fluorophenyl)-N-(4-{[(4-methylphenyl)amino]sulfonyl}phenyl)acetamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (5.7 %)
NA
24501399
DrugRepV_44155-methyl-N-[4-(1-pyrrolidinylsulfonyl)phenyl]-3-thiophenecarboxamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (-10.47 %)
NA
24501399
DrugRepV_44162-amino-N-(3-chlorophenyl)-3-quinolinecarboxamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (-2.95 %)
NA
24501399
DrugRepV_44172-(1,3-benzodioxol-5-yl)-1-(1,3-benzodioxol-5-ylmethyl)-1H-benzimidazole
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (-9.09 %)
NA
24501399
DrugRepV_4418N-{3-[(benzylamino)carbonyl]phenyl}-5-methyl-3-thiophenecarboxamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (-0.72 %)
NA
24501399
DrugRepV_44198-chloro-N-[3-(3-methyl-1H-pyrazol-1-yl)propyl]-2-(2-pyridinyl)-4-quinolinecarboxamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (-10.37 %)
NA
24501399
DrugRepV_4420N-[4-(2,4-difluorophenyl)-1,3-thiazol-2-yl]-2-(2-thienyl)acetamide
NA
NA
Hendra virus
F0, amino acids 105 to 114
NA
CatL-Peptide cleavage
Decrease (3.26 %)
NA
24501399
DrugRepV_4421N-(1,3-benzodioxol-5-ylmethyl)-2-(3-cyano-2-methyl-1H-indol-1-yl)acetamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (91.98 %)
NA
24501399
DrugRepV_4422N-benzyl-6-phenyl-2,3,4,9-tetrahydro-1H-carbazol-1-amine hydrochloride
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (98.65 %)
NA
24501399
DrugRepV_44239H-carbazol-3-amine
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (42.29 %)
NA
24501399
DrugRepV_44247-(1H-benzimidazol-2-ylthio)-8-methyl[1,3]dioxolo[4,5-g]quinolin-6(5H)-one
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (60.65 %)
NA
24501399
DrugRepV_4425N-[2-(2-methoxyethyl)-1,2,3,4-tetrahydropyrazino[1,2-a]benzimidazol-8-yl]benzamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (-0.15 %)
NA
24501399
DrugRepV_4426tris[4-(dimethylamino)phenyl]methanol
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (82.15 %)
NA
24501399
DrugRepV_44276-chloro-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-2-(3-pyridinyl)-4-quinolinecarboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (88.99 %)
NA
24501399
DrugRepV_44281-(2-furoyl)-5-(2-furyl)-3-(3-methoxyphenyl)-4,5-dihydro-1H-pyrazole
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (24.06 %)
NA
24501399
DrugRepV_44292-[(1H-benzimidazol-2-ylmethyl)thio]-1-[2-(4-methylphenoxy)ethyl]-1H-benzimidazole
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (57.39 %)
NA
24501399
DrugRepV_4430N-(3-chloro-4-fluorophenyl)-N-[4-(4-morpholinylsulfonyl)phenyl]urea
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (77.83 %)
NA
24501399
DrugRepV_44314-{[(5-methyl-2-thienyl)methyl]amino}phenol
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (1.34 %)
NA
24501399
DrugRepV_4432N-[5-(1H-benzimidazol-2-yl)-2-methylphenyl]-1,3-benzodioxole-5-carboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (76.53 %)
NA
24501399
DrugRepV_4433N-[1-benzyl-2-oxo-2-(4-phenyl-1-piperazinyl)ethyl]benzamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (14.51 %)
NA
24501399
DrugRepV_44342-methoxy-N-[1-methyl-2-(1-pyrrolidinylmethyl)-1H-benzimidazol-5-yl]benzamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (8.55 %)
NA
24501399
DrugRepV_4435N-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-2-(2-naphthyloxy)acetamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (79.93 %)
NA
24501399
DrugRepV_4436N-(2,5-dimethoxyphenyl)-N-[4-(trifluoromethyl)phenyl]urea
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (69.24 %)
NA
24501399
DrugRepV_44374-{[(1H-benzimidazol-2-ylthio)acetyl]amino}phenyl thiocyanate
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (65.51 %)
NA
24501399
DrugRepV_4438N-(3,4-dichlorophenyl)-N-[3-(trifluoromethyl)phenyl]urea
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (80.76 %)
NA
24501399
DrugRepV_4439N-1,3-benzodioxol-5-yl-6-chloro-2-(3-pyridinyl)-4-quinolinecarboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (65.73 %)
NA
24501399
DrugRepV_4440N-(3-chlorophenyl)-N-(4-cyanophenyl)urea
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (78.34 %)
NA
24501399
DrugRepV_4441N-[4-(1H-benzimidazol-2-yl)phenyl]-2-chloro-5-(4H-1,2,4-triazol-4-yl)benzamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (52.46 %)
NA
24501399
DrugRepV_4442N-[3-(aminocarbonyl)-5-benzyl-2-thienyl]-2-methyl-3-furamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (24.34 %)
NA
24501399
DrugRepV_44434,5-dimethyl-2-{[(5-propyl-3-thienyl)carbonyl]amino}-N-(3-pyridinylmethyl)-3-thiophenecarboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (39.61 %)
NA
24501399
DrugRepV_44441-(isopropylamino)-3-(3-phenyl-4,5-dihydropyrazolo[4,3-a]carbazol-10(3H)-yl)-2-propanol
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (44.31 %)
NA
24501399
DrugRepV_44452-[(4-tert-butyl-1,3-thiazol-2-yl)amino]-8-quinolinol
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (38.88 %)
NA
24501399
DrugRepV_4446N-(aminocarbonyl)-2-{[(5-methyl-3-thienyl)carbonyl]amino}-3-thiophenecarboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (38.54 %)
NA
24501399
DrugRepV_44472-chloro-N-(4-phenyl-1,3-thiazol-2-yl)-5-(4H-1,2,4-triazol-4-yl)benzamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (50.22 %)
NA
24501399
DrugRepV_4448N-[3-(2-oxo-2H-chromen-3-yl)phenyl]-1,3-benzodioxole-5-carboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (51.28 %)
NA
24501399
DrugRepV_44494,5-dimethyl-2-[(phenoxyacetyl)amino]-N-(3-pyridinylmethyl)-3-thiophenecarboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (39.55 %)
NA
24501399
DrugRepV_4450N-(4-{[(5-methyl-3-isoxazolyl)amino]sulfonyl}phenyl)-1-benzothiophene-3-carboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (33.84 %)
NA
24501399
DrugRepV_44513-[(1H-benzimidazol-2-ylmethyl)thio]-9-benzyl-9H-[1,2,4]triazolo[4,3-a]benzimidazole
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (23.55 %)
NA
24501399
DrugRepV_4452methyl N-[4,6-bis(isopropylamino)-1,3,5-triazin-2-yl]-N-cyanoglycinate
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (77.79 %)
NA
24501399
DrugRepV_4453N-(3,4-dichlorophenyl)-2-oxo-2,3-dihydro-1,3-benzoxazole-6-sulfonamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (56.45 %)
NA
24501399
DrugRepV_4454N-(3-pyridinylmethyl)dibenzo[b,d]furan-3-amine
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (47.55 %)
NA
24501399
DrugRepV_4455(1,3-benzodioxol-5-ylmethyl)[4-(1-pyrrolidinyl)phenyl]amine
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (-3.09 %)
NA
24501399
DrugRepV_44564-methyl-5-phenyl-N-3-pyridinyl-2-thiophenecarboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (72.37 %)
NA
24501399
DrugRepV_4457N-(2,5-dimethoxyphenyl)-2-(2-oxo-1,3-benzoxazol-3(2H)-yl)acetamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (47.94 %)
NA
24501399
DrugRepV_44583-[(2,4-dichlorophenoxy)methyl]-N-(3-pyridinylmethyl)benzamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (53.23 %)
NA
24501399
DrugRepV_44595-phenyl-2-(2-phenylethyl)[1,2,4]triazolo[1,5-a]pyrimidin-7(4H)-one
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (28.07 %)
NA
24501399
DrugRepV_44606-bromo-2-oxo-N-3-pyridinyl-2H-chromene-3-carboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (25.6 %)
NA
24501399
DrugRepV_44612-[(2-methyl-8-quinolinyl)amino]-4H-pyrido[3,2-e][1,3]thiazin-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (37.16 %)
NA
24501399
DrugRepV_4462N-(3-chloro-4-fluorophenyl)-N-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (61.47 %)
NA
24501399
DrugRepV_44634-({[(3-chloro-4-fluorophenyl)amino]carbonyl}amino)-N-methylbenzenesulfonamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (66.62 %)
NA
24501399
DrugRepV_44642-(4-fluorophenyl)-N-(4-{[(4-methylphenyl)amino]sulfonyl}phenyl)acetamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (32.44 %)
NA
24501399
DrugRepV_44655-methyl-N-[4-(1-pyrrolidinylsulfonyl)phenyl]-3-thiophenecarboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (30.53 %)
NA
24501399
DrugRepV_44662-amino-N-(3-chlorophenyl)-3-quinolinecarboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (47.39 %)
NA
24501399
DrugRepV_44672-(1,3-benzodioxol-5-yl)-1-(1,3-benzodioxol-5-ylmethyl)-1H-benzimidazole
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (49.81 %)
NA
24501399
DrugRepV_4468N-{3-[(benzylamino)carbonyl]phenyl}-5-methyl-3-thiophenecarboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (51.17 %)
NA
24501399
DrugRepV_44698-chloro-N-[3-(3-methyl-1H-pyrazol-1-yl)propyl]-2-(2-pyridinyl)-4-quinolinecarboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (41.66 %)
NA
24501399
DrugRepV_4470N-[4-(2,4-difluorophenyl)-1,3-thiazol-2-yl]-2-(2-thienyl)acetamide
NA
NA
Severe acute respiratory syndrome coronavirus
S, amino acids 674 to 683
NA
CatL-Peptide cleavage
Decrease (40.85 %)
NA
24501399
DrugRepV_4486Brincidofovir
NA
Viral infections
Ebola virus
EBOV-GFP
NA
Luciferase assay
Decrease (50 %)
Investigational
26526586
DrugRepV_4487CMX029
NA
NA
Ebola virus
EBOV-GFP
NA
Luciferase assay
Decrease (50 %)
NA
26526586
DrugRepV_4488CMX021
NA
NA
Ebola virus
EBOV-GFP
NA
Luciferase assay
Decrease (50 %)
NA
26526586
DrugRepV_4489CMX028
NA
NA
Ebola virus
EBOV-GFP
NA
Luciferase assay
Decrease (50 %)
NA
26526586
DrugRepV_4490CMX16669
NA
NA
Ebola virus
EBOV-GFP
NA
Luciferase assay
Decrease (50 %)
NA
26526586
DrugRepV_4491CMX16663
NA
NA
Ebola virus
EBOV-GFP
NA
Luciferase assay
Decrease (50 %)
NA
26526586
DrugRepV_4492CMX167
NA
NA
Ebola virus
EBOV-GFP
NA
Luciferase assay
Decrease (50 %)
NA
26526586
DrugRepV_4493CMX157
NA
NA
Ebola virus
EBOV-GFP
NA
Luciferase assay
Decrease (50 %)
NA
26526586
DrugRepV_4494CMX101
NA
NA
Ebola virus
EBOV-GFP
NA
Luciferase assay
Decrease (50 %)
NA
26526586
DrugRepV_4495CMX004
NA
NA
Ebola virus
EBOV-GFP
NA
Luciferase assay
Decrease (50 %)
NA
26526586
DrugRepV_4496CMX16689
NA
NA
Ebola virus
EBOV-GFP
NA
Luciferase assay
Decrease (50 %)
NA
26526586
DrugRepV_4500(1S,2R,5S)-5-{4-amino-1H-imidazo[4,5-c]pyridin-1-yl}-4-fluoro-3-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
Zaire
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4501(1S,2R,5R)-5-(6-amino-9H-purin-9-yl)-3-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
Zaire
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4502(1S,2R,5R)-5-{4-amino-1H-imidazo[4,5-c]pyridin-1-yl}-3-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
Zaire
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4503(1R,2S,5R)-3-(6-amino-9H-purin-9-yl)-5-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
Zaire
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4504(1R,2S,5R)-3-{4-amino-1H-imidazo[4,5-c]pyridin-1-yl}-5-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
Zaire
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4505(1S,2R,5S)-5-{4-amino-1H-imidazo[4,5-c]pyridin-1-yl}-4-fluoro-3-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4506(1S,2R,5R)-5-(6-amino-9H-purin-9-yl)-3-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4507(1S,2R,5R)-5-{4-amino-1H-imidazo[4,5-c]pyridin-1-yl}-3-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4508(1R,2S,5R)-3-(6-amino-9H-purin-9-yl)-5-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4509(1R,2S,5R)-3-{4-amino-1H-imidazo[4,5-c]pyridin-1-yl}-5-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4510(1S,2R,5S)-5-(6-amino-9H-purin-9-yl)-4-fluoro-3-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4511(1S,2R,5S)-5-{4-amino-1H-imidazo[4,5-c]pyridin-1-yl}-4-fluoro-3-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Influenza virus
NA
Pathway
NA
Decrease (50 %)
NA
30385162
DrugRepV_4519Alferon
NA
Condylomata acuminata
Severe acute respiratory syndrome coronavirus
NA
NA
Plaque reduction assay
Decrease (50 %)
Approved
15200845
DrugRepV_4525IFN-alphan3
NA
Condylomata acuminata
Severe acute respiratory syndrome coronavirus
NA
NA
CPE inhibition assay
Decrease (100 %)
Approved, Investigational
15200845
DrugRepV_45401-[4,5-dihydroxy-3-(hydroxymethyl)cyclopent-2-en-1-yl]-1H-1,2,4-triazole-3-carboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
16451078
DrugRepV_45411-[4,5-dihydroxy-3-(hydroxymethyl)cyclopent-2-en-1-yl]-1H-imidazole-4-carboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
16451078
DrugRepV_45421-[4,5-dihydroxy-3-(hydroxymethyl)cyclopent-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
16451078
DrugRepV_4543Alferon
NA
Condylomata acuminata
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Approved
16451078
DrugRepV_4547Aurintricarboxylic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
15961169
DrugRepV_4548DS5000
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
15961169
DrugRepV_4549Novaron
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
15961169
DrugRepV_4551S-Nitroso-N-acetylpenicillamine
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
15961169
DrugRepV_45527-(benzyloxy)-2-(3,4-dihydroxyphenyl)-3,5-dihydroxy-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45532-(3,4-dihydroxyphenyl)-7-[(2-fluorophenyl)methoxy]-3,5-dihydroxy-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45547-[(2-chlorophenyl)methoxy]-2-(3,4-dihydroxyphenyl)-3,5-dihydroxy-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45557-[(2-bromophenyl)methoxy]-2-(3,4-dihydroxyphenyl)-3,5-dihydroxy-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45562-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(2-iodophenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45572-({[2-(3,4-dihydroxyphenyl)-3,5-dihydroxy-4-oxo-4H-chromen-7-yl]oxy}methyl)benzonitrile
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45582-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(2-nitrophenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45592-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(2-methylphenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45602-(3,4-dihydroxyphenyl)-7-[(3-fluorophenyl)methoxy]-3,5-dihydroxy-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45617-[(3-chlorophenyl)methoxy]-2-(3,4-dihydroxyphenyl)-3,5-dihydroxy-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45627-[(3-bromophenyl)methoxy]-2-(3,4-dihydroxyphenyl)-3,5-dihydroxy-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45632-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(3-iodophenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45643-({[2-(3,4-dihydroxyphenyl)-3,5-dihydroxy-4-oxo-4H-chromen-7-yl]oxy}methyl)benzonitrile
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45652-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(3-nitrophenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45662-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(3-methylphenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45672-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(3-methoxyphenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45682-(3,4-dihydroxyphenyl)-7-[(4-fluorophenyl)methoxy]-3,5-dihydroxy-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45697-[(4-chlorophenyl)methoxy]-2-(3,4-dihydroxyphenyl)-3,5-dihydroxy-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45707-[(4-bromophenyl)methoxy]-2-(3,4-dihydroxyphenyl)-3,5-dihydroxy-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45712-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(4-iodophenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45724-({[2-(3,4-dihydroxyphenyl)-3,5-dihydroxy-4-oxo-4H-chromen-7-yl]oxy}methyl)benzonitrile
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45732-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(4-nitrophenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45742-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(4-methylphenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45752-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(4-methoxyphenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_4577Glycyrrhetinic Acid
NA
Apparent mineralocorticoid excess syndrome
Severe acute respiratory syndrome coronavirus
FFM1
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Investigational
15715493
DrugRepV_4578(2S,4aS,6aS,6bR,10S,12aS)-10-[(6-{[2-(benzylsulfanyl)-1-carboxyethyl]carbamoyl}-3-[(6-{[2-(benzylsulfanyl)-1-carboxyethyl]carbamoyl}-3,4,5-trihydroxyoxan-2-yl)oxy]-4,5-dihydroxyoxan-2-yl)oxy]-2,4a,6a,6b,9,9,12a-heptamethyl-13-oxo-1,2,3,4,4a,5,6,6a,6b
NA
NA
Severe acute respiratory syndrome coronavirus
FFM1
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
15715493
DrugRepV_4579(2S,4aS,6aS,6bR,10S,12aS)-10-[(6-{[2-(benzylsulfanyl)-1-carboxyethyl]carbamoyl}-3-[(6-{[2-(benzylsulfanyl)-1-carboxyethyl]carbamoyl}-3,4,5-trihydroxyoxan-2-yl)oxy]-4,5-dihydroxyoxan-2-yl)oxy]-2,4a,6a,6b,9,9,12a-heptamethyl-13-oxo-1,2,3,4,4a,5,6,6a,6b
NA
NA
Severe acute respiratory syndrome coronavirus
FFM1
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
15715493
DrugRepV_4580(2S,4aS,6aS,6bR,10S,12aS)-10-({4,5-dihydroxy-6-[({[(2S)-4-methyl-1-oxopentan-2-yl]carbamoyl}methyl)carbamoyl]-3-({3,4,5-trihydroxy-6-[({[(2S)-4-methyl-1-oxopentan-2-yl]carbamoyl}methyl)carbamoyl]oxan-2-yl}oxy)oxan-2-yl}oxy)-2,4a,6a,6b,9,9,12a-heptame
NA
NA
Severe acute respiratory syndrome coronavirus
FFM1
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
15715493
DrugRepV_45816-{[(3S,6aR,6bS,8aS,11S,14bS)-4,4,6a,6b,8a,11,14b-heptamethyl-11-{[(2S)-4-methyl-1-oxopentan-2-yl]carbamoyl}-14-oxo-1,2,3,4,4a,5,6,6a,6b,7,8,8a,9,10,11,12,12a,14,14a,14b-icosahydropicen-3-yl]oxy}-3,4-dihydroxy-N-[(2S)-4-methyl-1-oxopentan-2-yl]-5-[(3
NA
NA
Severe acute respiratory syndrome coronavirus
FFM1
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
15715493
DrugRepV_4582butyl (2S)-2-{[(2S,4aS,6aS,6bR,10S,12aS)-10-[(6-{[(2S)-1-butoxy-3-methyl-1-oxobutan-2-yl]carbamoyl}-3-[(6-{[(2S)-1-butoxy-3-methyl-1-oxobutan-2-yl]carbamoyl}-3,4,5-trihydroxyoxan-2-yl)oxy]-4,5-dihydroxyoxan-2-yl)oxy]-2,4a,6a,6b,9,9,12a-heptamethyl-13
NA
NA
Severe acute respiratory syndrome coronavirus
FFM1
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
15715493
DrugRepV_4583methyl (2S)-2-(2-{[(2S,4aS,6aS,6bR,10S,12aS)-10-({4,5-dihydroxy-6-[({[(2S)-1-methoxy-3-methyl-1-oxobutan-2-yl]carbamoyl}methyl)carbamoyl]-3-({3,4,5-trihydroxy-6-[({[(2S)-1-methoxy-3-methyl-1-oxobutan-2-yl]carbamoyl}methyl)carbamoyl]oxan-2-yl}oxy)oxan
NA
NA
Severe acute respiratory syndrome coronavirus
FFM1
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
15715493
DrugRepV_4584(4S)-4-{[(2S,4aS,6aS,6bR,10S,12aS)-10-[(6-{[(2S)-4-carboxy-1-oxobutan-2-yl]carbamoyl}-3-[(6-{[(2S)-4-carboxy-1-oxobutan-2-yl]carbamoyl}-3,4,5-trihydroxyoxan-2-yl)oxy]-4,5-dihydroxyoxan-2-yl)oxy]-2,4a,6a,6b,9,9,12a-heptamethyl-13-oxo-1,2,3,4,4a,5,6,6a
NA
NA
Severe acute respiratory syndrome coronavirus
FFM1
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
15715493
DrugRepV_4585butyl (2S)-2-{[(2S,4aS,6aS,6bR,10S,12aS)-10-[(6-{[(2S)-1-butoxy-1-oxopropan-2-yl]carbamoyl}-3-[(6-{[(2S)-1-butoxy-1-oxopropan-2-yl]carbamoyl}-3,4,5-trihydroxyoxan-2-yl)oxy]-4,5-dihydroxyoxan-2-yl)oxy]-2,4a,6a,6b,9,9,12a-heptamethyl-13-oxo-1,2,3,4,4a,
NA
NA
Severe acute respiratory syndrome coronavirus
FFM1
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
15715493
DrugRepV_4586(2S,4aS,6aS,6bR,10S,12aS)-10-{[4,5-dihydroxy-6-(2-hydroxyacetyl)-3-{[3,4,5-trihydroxy-6-(2-hydroxyacetyl)oxan-2-yl]oxy}oxan-2-yl]oxy}-2,4a,6a,6b,9,9,12a-heptamethyl-13-oxo-1,2,3,4,4a,5,6,6a,6b,7,8,8a,9,10,11,12,12a,12b,13,14b-icosahydropicene-2-carbo
NA
NA
Severe acute respiratory syndrome coronavirus
FFM1
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
15715493
DrugRepV_4587(2S,4aS,6aS,6bR,10S,12aS)-10-({4,5-dihydroxy-6-[(6-oxo-2-sulfanylidene-1,2,3,6-tetrahydropyrimidin-4-yl)carbamoyl]-3-({3,4,5-trihydroxy-6-[(6-oxo-2-sulfanylidene-1,2,3,6-tetrahydropyrimidin-4-yl)carbamoyl]oxan-2-yl}oxy)oxan-2-yl}oxy)-2,4a,6a,6b,9,9,1
NA
NA
Severe acute respiratory syndrome coronavirus
FFM1
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
15715493
DrugRepV_45885-{6-[(2-{[(3S,6aR,6bS,8aS,11S,14bS)-11-(2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl)-4,4,6a,6b,8a,11,14b-heptamethyl-14-oxo-1,2,3,4,4a,5,6,6a,6b,7,8,8a,9,10,11,12,12a,14,14a,14b-icosahydropicen-3-yl]oxy}-6-(2,4-dioxo-1,2,3,4-tetrahydropyrimidi
NA
NA
Severe acute respiratory syndrome coronavirus
FFM1
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
15715493
DrugRepV_4589methyl (2S,4aS,6aS,6bR,10S,12aS)-10-({6-[(hydrazinecarbonyl)carbonyl]-3-({6-[(hydrazinecarbonyl)carbonyl]-3,4,5-trihydroxyoxan-2-yl}oxy)-4,5-dihydroxyoxan-2-yl}oxy)-2,4a,6a,6b,9,9,12a-heptamethyl-13-oxo-1,2,3,4,4a,5,6,6a,6b,7,8,8a,9,10,11,12,12a,12b,
NA
NA
Severe acute respiratory syndrome coronavirus
FFM1
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
15715493
DrugRepV_4590methyl (2S,4aS,6aS,6bR,10S,12aS)-10-{[6-(2-azidoacetyl)-3-{[6-(2-azidoacetyl)-3,4,5-trihydroxyoxan-2-yl]oxy}-4,5-dihydroxyoxan-2-yl]oxy}-2,4a,6a,6b,9,9,12a-heptamethyl-13-oxo-1,2,3,4,4a,5,6,6a,6b,7,8,8a,9,10,11,12,12a,12b,13,14b-icosahydropicene-2-ca
NA
NA
Severe acute respiratory syndrome coronavirus
FFM1
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
15715493
DrugRepV_45912-{[(6aR,6bS,8aS,11S,14bS)-11-(acetyloxy)-4,4,6a,6b,8a,11,14b-heptamethyl-14-oxo-1,2,3,4,4a,5,6,6a,6b,7,8,8a,9,10,11,12,12a,14,14a,14b-icosahydropicen-3-yl]oxy}benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
FFM1
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
15715493
DrugRepV_45924-{[(6aR,6bS,8aS,11S,14bS)-11-(acetyloxy)-4,4,6a,6b,8a,11,14b-heptamethyl-14-oxo-1,2,3,4,4a,5,6,6a,6b,7,8,8a,9,10,11,12,12a,14,14a,14b-icosahydropicen-3-yl]oxy}-4-oxobutanoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
FFM1
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
15715493
DrugRepV_45933-(benzyloxy)-7-[(3-chlorophenyl)methoxy]-8-hydroxy-1,4-dihydronaphthalen-1-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Luciferase assay
Decrease (50 %)
NA
21925774
DrugRepV_45943-[(2-chlorophenyl)methoxy]-7-[(3-chlorophenyl)methoxy]-8-hydroxy-1,4-dihydronaphthalen-1-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Luciferase assay
Decrease (50 %)
NA
21925774
DrugRepV_45953,7-bis[(3-chlorophenyl)methoxy]-8-hydroxy-1,4-dihydronaphthalen-1-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Luciferase assay
Decrease (50 %)
NA
21925774
DrugRepV_45967-[(3-chlorophenyl)methoxy]-3-[(2,4-dichlorophenyl)methoxy]-8-hydroxy-1,4-dihydronaphthalen-1-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Luciferase assay
Decrease (50 %)
NA
21925774
DrugRepV_45977-[(3-chlorophenyl)methoxy]-8-hydroxy-3-[(2-iodophenyl)methoxy]-1,4-dihydronaphthalen-1-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Luciferase assay
Decrease (50 %)
NA
21925774
DrugRepV_45987-[(3-chlorophenyl)methoxy]-8-hydroxy-3-[(3-iodophenyl)methoxy]-1,4-dihydronaphthalen-1-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Luciferase assay
Decrease (50 %)
NA
21925774
DrugRepV_45992-[({6-[(3-chlorophenyl)methoxy]-5-hydroxy-4-oxo-1,4-dihydronaphthalen-2-yl}oxy)methyl]benzonitrile
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Luciferase assay
Decrease (50 %)
NA
21925774
DrugRepV_4600(2Z)-4-(3-{[(4-chlorophenyl)methyl]amino}phenyl)-2-hydroxy-4-oxobut-2-enoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Luciferase assay
Decrease (50 %)
NA
21925774
DrugRepV_46015,7-dihydroxy-3-[(3-nitrophenyl)methoxy]-2-phenyl-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Luciferase assay
Decrease (50 %)
NA
21925774
DrugRepV_46023-{[(3,5-dihydroxy-4-oxo-2-phenyl-4H-chromen-7-yl)oxy]methyl}benzonitrile
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Luciferase assay
Decrease (50 %)
NA
21925774
DrugRepV_46031H-1,2,3-benzotriazol-1-yl 1H-indole-5-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_46045-chloropyridin-3-yl 1H-indole-5-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_46055-chloropyridin-3-yl 1-acetyl-1H-indole-5-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_46065-chloropyridin-3-yl 1-(4-methylbenzenesulfonyl)-1H-indole-5-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_46075-chloropyridin-3-yl 1-(3-nitrobenzenesulfonyl)-1H-indole-5-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_46085-chloropyridin-3-yl1H-indole-6-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_46095-chloropyridin-3-yl 1H-indole-4-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_46105-chloropyridin-3-yl 1-acetyl-1H-indole-4-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_46115-chloropyridin-3-yl 1H-indole-7-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_46125-chloropyridin-3-yl (6R)-6-{[(tert-butoxy)carbonyl]amino}-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_46135-chloropyridin-3-yl 2-acetyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_4618Calpain VI inhibitor
NA
NA
Severe acute respiratory syndrome coronavirus
v2163
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
19853271
DrugRepV_4619Calpain VI inhibitor
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
19853271
DrugRepV_4620Calpain IV inhibitor
NA
NA
Severe acute respiratory syndrome coronavirus
v2163
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
19853271
DrugRepV_4621Calpain IV inhibitor
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
19853271
DrugRepV_4624Ampligen
NA
NA
Severe acute respiratory syndrome coronavirus
v2163
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
19853271
DrugRepV_4625Ampligen
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
19853271
DrugRepV_4626UDA
NA
NA
Severe acute respiratory syndrome coronavirus
v2163
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
19853271
DrugRepV_4627UDA
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
19853271
DrugRepV_4628EP128533
NA
NA
Severe acute respiratory syndrome coronavirus
v2163
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
19853271
DrugRepV_4629EP128533
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
19853271
DrugRepV_4631Ampligen
NA
NA
Severe acute respiratory syndrome coronavirus
v2163
NA
Survival assay
Increase
NA
19853271
DrugRepV_4632UDA
NA
NA
Severe acute respiratory syndrome coronavirus
v2163
NA
Survival assay
Increase
NA
19853271
DrugRepV_4633Cremaphor
NA
NA
Severe acute respiratory syndrome coronavirus
v2163
NA
Survival assay
No significant effect
NA
19853271
DrugRepV_4634TG-0205221
NA
SARS coronavirus
Severe acute respiratory syndrome coronavirus
Urbani
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
16884309
DrugRepV_4635ethyl (2E,4S)-4-[(2S)-3-(4-fluorophenyl)-2-[(2S)-3-methyl-2-[(5-methyl-1,2-oxazol-3-yl)formamido]butanamido]propanamido]-5-[(3S)-2-oxopyrrolidin-3-yl]pent-2-enoate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
16884309
DrugRepV_4636ethyl (2E,4S)-4-[(2S)-2-[(2S)-2-{[(benzyloxy)carbonyl]amino}-3-methylbutanamido]-3-phenylpropanamido]-5-[(3S)-2-oxopyrrolidin-3-yl]pent-2-enoate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
16884309
DrugRepV_4637ethyl (2E,4S)-4-[(2S)-2-[(2S)-2-{[(benzyloxy)carbonyl]amino}-3-methylbutanamido]-4-methylpentanamido]-5-[(3S)-2-oxopyrrolidin-3-yl]pent-2-enoate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
16884309
DrugRepV_4638ethyl (2E,4S)-4-[(2S)-2-[(2S)-2-{[(benzyloxy)carbonyl]amino}-3-(tert-butoxy)butanamido]-4-methylpentanamido]-5-[(3S)-2-oxopyrrolidin-3-yl]pent-2-enoate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
16884309
DrugRepV_4639TG-0205221
NA
SARS coronavirus
Severe acute respiratory syndrome coronavirus
Urbani
NA
Cytopathic effect (CPE) assay
Decrease (6.4 Log10)
NA
16884309
DrugRepV_4640TG-0205221
NA
SARS coronavirus
Severe acute respiratory syndrome coronavirus
Urbani
NA
Cytopathic effect (CPE) assay
Decrease
NA
16884309
DrugRepV_46415CI-IS-AC
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
20390088
DrugRepV_4642SPIII-5H
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
20390088
DrugRepV_4643SPIII-5Cl
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
20390088
DrugRepV_4644SPIII-5Br
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
20390088
DrugRepV_4645SPIII-5F
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
20390088
DrugRepV_4646SPIII-5Me
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
20390088
DrugRepV_4647SPIII-NA
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
20390088
DrugRepV_46546-Azauridine
NA
Cancer
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4657Kitasamycin
NA
Bacterial infections
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
Experimental
27909576
DrugRepV_4658SAM002589981
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4659SAM002564206
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4660SAM002564189
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4661SAM002554886
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4662SAM002548975
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4663SAM002548938
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4664SAM002264636
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4665SAM001247107
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4666SAM001247103
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4667SAM001247083
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4668SAM001247075
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4669SAM001247056
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4670SAM001247054
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4671SAM001247052
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4672SAM001247038
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4673SAM001246989
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4674SAM001246979
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4675SAM001246977
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4676SAM001246883
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4677SAM001246690
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4678SAM001246644
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4679SAM001246622
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4680SAM001246545
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease (50 %)
NA
27909576
DrugRepV_4681N-(4-hydroxyphenyl) retinamide
NA
NA
Zika virus
MR766
NA
Plaque assay
Decrease (90 %)
Investigational
29051080
DrugRepV_4682Arbidol
NA
Viral infection
Zika virus
MR766
NA
NA
Decrease (50 %)
Investigational
29895962
DrugRepV_46842-C-Methylcytidine
NA
Hepatitis C virus
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
Experimental
30061280
DrugRepV_46852-C-Methyladenosine
NA
NA
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
NA
30061280
DrugRepV_46862-C-Methylguanosine
NA
NA
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
NA
30061280
DrugRepV_46872-C-Methyluridine
NA
NA
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
NA
30061280
DrugRepV_46895-Fluoro-2-deoxyuridine
NA
Cancer
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
Approved
30061280
DrugRepV_46905-Fluorouridine
NA
Cancer
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
Experimental
30061280
DrugRepV_46915-Fluorocytidine
NA
Breast Cancer
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
Phase IV
30061280
DrugRepV_46932-O-Methylcytidine
NA
NA
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
NA
30061280
DrugRepV_46943-Deoxyadenosine
NA
Leukemia
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
Investigational
30061280
DrugRepV_46953-Deoxycytidine
NA
Cancer
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
Phase I
30061280
DrugRepV_46963-O-Methylguanosine
NA
NA
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
NA
30061280
DrugRepV_46973-O-Methyluridine
NA
NA
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
NA
30061280
DrugRepV_46989-(beta-D-Arabinofuranosyl)guanine
NA
NA
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
NA
30061280
DrugRepV_46992-C-Methylcytidine ProTide
NA
NA
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
NA
30061280
DrugRepV_47002-C-Methyluridine ProTide
NA
NA
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
NA
30061280
DrugRepV_47012-C-Methyladenosine ProTide
NA
NA
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
NA
30061280
DrugRepV_47023-Deoxyadenosine ProTide
NA
NA
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
NA
30061280
DrugRepV_47035-Fluorocytidine ProTide
NA
NA
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
NA
30061280
DrugRepV_47043-O-Methyluridine ProTide
NA
NA
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
NA
30061280
DrugRepV_47052-O-Methylcytidine ProTide
NA
NA
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
NA
30061280
DrugRepV_47063-Deoxycytidine ProTide
NA
NA
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
NA
30061280
DrugRepV_47073-Deoxy-3-fluoroguanosine ProTide
NA
NA
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
NA
30061280
DrugRepV_47082,4-dichloro-6-(3,4-dibromo-5-fluoro-1H-pyrrole-2-carbonyl)phenol
NA
NA
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
NA
30061280
DrugRepV_47102,4-dichloro-6-(3,4-dibromo-5-fluoro-1H-pyrrole-2-carbonyl)phenol
NA
NA
Zika virus
NA
NA
Immunoflourescence assay
Decrease
NA
30061280
DrugRepV_4711Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Zika virus
MR766
NA
Plaque assay
Decrease (50 %)
Investigational
27889529
DrugRepV_4713GSK369796
NA
NA
Zika virus
MR766
NA
Plaque assay
Decrease (50 %)
NA
27889529
DrugRepV_4714Nutlin-3
NA
NA
Middle East respiratory syndrome coronavirus
EMC/2012 strain
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
29795047
DrugRepV_4724Methotrimeprazine Maleate Salt
NA
NA
Middle East respiratory syndrome coronavirus
EMC/2012 strain
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved, Investigational
29795047
DrugRepV_4725N1-(4-pyridyl)-2-chloro-5-nitrobenzamide
NA
NA
Middle East respiratory syndrome coronavirus
EMC/2012 strain
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
29795047
DrugRepV_4729L-NAME
NA
Hypotension | Spinal Cord Injury
Middle East respiratory syndrome coronavirus
NA
NA
Plaque assay
Decrease (15 %)
Investigational
25487801
DrugRepV_4730AG490
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
Plaque assay
Decrease (17 %)
NA
25487801
DrugRepV_4731PKC-412
NA
Acute myeloid leukemia
Middle East respiratory syndrome coronavirus
NA
NA
Plaque assay
Decrease (33 %)
Approved, Investigational
25487801
DrugRepV_4732Ro 31-8220
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
Plaque assay
Decrease (73 %)
NA
25487801
DrugRepV_4733GF109203X
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
Plaque assay
Decrease (53 %)
NA
25487801
DrugRepV_4734SB203580
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
Plaque assay
Decrease (45 %)
NA
25487801
DrugRepV_4735U0126
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
Plaque assay
Decrease (50 %)
NA
25487801
DrugRepV_4736Wortmannin
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
Plaque assay
Decrease (40 %)
Experimental
25487801
DrugRepV_4738Bay 11-7082
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
Plaque assay
Decrease (28 %)
NA
25487801
DrugRepV_4739GW5074
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
Plaque assay
Decrease (50 %)
NA
25487801
DrugRepV_4740PP2
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
Plaque assay
Decrease (23 %)
NA
25487801
DrugRepV_4747tert-butyl 4-({[(1S)-3-methyl-1-{[(2S)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]carbamoyl}butyl]carbamoyl}oxy)piperidine-1-carboxylate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_4748sodium (2S)-2-[(2S)-2-{[({1-[(tert-butoxy)carbonyl]piperidin-4-yl}oxy)carbonyl]amino}-4-methylpentanamido]-1-hydroxy-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_47491-methanesulfonylpiperidin-4-yl N-[(1S)-3-methyl-1-{[(2S)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]carbamoyl}butyl]carbamate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_4750sodium (2S)-1-hydroxy-2-[(2S)-2-({[(1-methanesulfonylpiperidin-4-yl)oxy]carbonyl}amino)-4-methylpentanamido]-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_4751tert-butyl 4-benzyl-4-({[(1S)-3-methyl-1-{[(2S)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]carbamoyl}butyl]carbamoyl}oxy)piperidine-1-carboxylate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_4752sodium (2S)-2-[(2S)-2-{[({4-benzyl-1-[(tert-butoxy)carbonyl]piperidin-4-yl}oxy)carbonyl]amino}-4-methylpentanamido]-1-hydroxy-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_47534-benzyl-1-methanesulfonylpiperidin-4-yl N-[(1S)-3-methyl-1-{[(2S)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]carbamoyl}butyl]carbamate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_4754sodium (2S)-2-[(2S)-2-({[(4-benzyl-1-methanesulfonylpiperidin-4-yl)oxy]carbonyl}amino)-4-methylpentanamido]-1-hydroxy-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_4755tert-butyl 4-ethyl-4-({[(1S)-3-methyl-1-{[(2S)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]carbamoyl}butyl]carbamoyl}oxy)piperidine-1-carboxylate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_4756sodium (2S)-2-[(2S)-2-{[({1-[(tert-butoxy)carbonyl]-4-ethylpiperidin-4-yl}oxy)carbonyl]amino}-4-methylpentanamido]-1-hydroxy-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_4757ethyl 4-({[(1S)-3-methyl-1-{[(2S)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]carbamoyl}butyl]carbamoyl}oxy)piperidine-1-carboxylate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_4758sodium (2S)-2-[(2S)-2-[({[1-(ethoxycarbonyl)piperidin-4-yl]oxy}carbonyl)amino]-4-methylpentanamido]-1-hydroxy-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_4759tert-butyl 4-({[(1S)-3-methyl-1-{[(2S)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]carbamoyl}butyl]carbamoyl}oxy)piperidine-1-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_4760sodium (2S)-2-[(2S)-2-{[({1-[(tert-butoxy)carbonyl]piperidin-4-yl}oxy)carbonyl]amino}-4-methylpentanamido]-1-hydroxy-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_47611-methanesulfonylpiperidin-4-yl N-[(1S)-3-methyl-1-{[(2S)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]carbamoyl}butyl]carbamate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_4762sodium (2S)-1-hydroxy-2-[(2S)-2-({[(1-methanesulfonylpiperidin-4-yl)oxy]carbonyl}amino)-4-methylpentanamido]-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_4763tert-butyl 4-benzyl-4-({[(1S)-3-methyl-1-{[(2S)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]carbamoyl}butyl]carbamoyl}oxy)piperidine-1-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_4764sodium (2S)-2-[(2S)-2-{[({4-benzyl-1-[(tert-butoxy)carbonyl]piperidin-4-yl}oxy)carbonyl]amino}-4-methylpentanamido]-1-hydroxy-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_47654-benzyl-1-methanesulfonylpiperidin-4-yl N-[(1S)-3-methyl-1-{[(2S)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]carbamoyl}butyl]carbamate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_4766sodium (2S)-2-[(2S)-2-({[(4-benzyl-1-methanesulfonylpiperidin-4-yl)oxy]carbonyl}amino)-4-methylpentanamido]-1-hydroxy-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_4767tert-butyl 4-ethyl-4-({[(1S)-3-methyl-1-{[(2S)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]carbamoyl}butyl]carbamoyl}oxy)piperidine-1-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_4768sodium (2S)-2-[(2S)-2-{[({1-[(tert-butoxy)carbonyl]-4-ethylpiperidin-4-yl}oxy)carbonyl]amino}-4-methylpentanamido]-1-hydroxy-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_4769ethyl 4-({[(1S)-3-methyl-1-{[(2S)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]carbamoyl}butyl]carbamoyl}oxy)piperidine-1-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_4770sodium (2S)-2-[(2S)-2-[({[1-(ethoxycarbonyl)piperidin-4-yl]oxy}carbonyl)amino]-4-methylpentanamido]-1-hydroxy-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
FRET protease assay
Decrease (50 %)
NA
29544147
DrugRepV_4771sodium (2S)-2-[(2S)-2-{[({1-[(tert-butoxy)carbonyl]piperidin-4-yl}oxy)carbonyl]amino}-4-methylpentanamido]-1-hydroxy-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
Plaque assay
Decrease (50 %)
NA
29544147
DrugRepV_4772sodium (2S)-2-[(2S)-2-{[({4-benzyl-1-[(tert-butoxy)carbonyl]piperidin-4-yl}oxy)carbonyl]amino}-4-methylpentanamido]-1-hydroxy-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
Plaque assay
Decrease (50 %)
NA
29544147
DrugRepV_4775N-ethylmaleimide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Experimental
25542975
DrugRepV_4782IFN-universal
NA
NA
Middle East respiratory syndrome coronavirus
Hu/Jordan-N3/2012
NA
Virus yield reduction assay
Decrease (50 %)
NA
24323636
DrugRepV_47842-(5-{[(4Z)-1-(3-carboxyphenyl)-3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)-4-chlorobenzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47852-(5-{[(4Z)-1-(3-carboxyphenyl)-5-oxo-3-(trifluoromethyl)-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)-4-chlorobenzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47862-(5-{[(4Z)-1-(3-carboxyphenyl)-5-oxo-3-(trifluoromethyl)-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47872-(5-{[(4Z)-1-(3-carboxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)-4-chlorobenzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47884-chloro-2-(5-{[(4Z)-3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47894-chloro-2-(5-{[(4Z)-5-oxo-1,3-diphenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47904-chloro-2-(5-{[(4Z)-1-(4-fluorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47914-chloro-2-(5-{[(4Z)-5-oxo-3-phenyl-1-[4-(propan-2-yl)phenyl]-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47922-(5-{[(4Z)-1-(4-tert-butylphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)-4-chlorobenzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_4793(4Z)-1,3-diphenyl-4-[(5-phenylfuran-2-yl)methylidene]-4,5-dihydro-1H-pyrazol-5-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47943-[(4Z)-5-oxo-3-phenyl-4-[(5-phenylfuran-2-yl)methylidene]-4,5-dihydro-1H-pyrazol-1-yl]benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47953-[(4Z)-3-methyl-5-oxo-4-[(5-phenylfuran-2-yl)methylidene]-4,5-dihydro-1H-pyrazol-1-yl]benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47962-(5-{[(4Z)-5-oxo-1,3-diphenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47972-(5-{[(4Z)-1-(4-fluorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47982-(5-{[(4Z)-5-oxo-3-phenyl-1-[4-(propan-2-yl)phenyl]-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47992-(5-{[(4Z)-1-(4-tert-butylphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48002-(5-{[(4Z)-1-(4-cyanophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48012-(5-{[(4Z)-1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoicacid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48023-[(4Z)-4-[(furan-2-yl)methylidene]-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl]benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48032-(5-{[(4Z)-1-(3-carboxyphenyl)-3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)-4-chlorobenzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48042-(5-{[(4Z)-1-(3-carboxyphenyl)-5-oxo-3-(trifluoromethyl)-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)-4-chlorobenzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48052-(5-{[(4Z)-1-(3-carboxyphenyl)-5-oxo-3-(trifluoromethyl)-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48062-(5-{[(4Z)-1-(3-carboxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)-4-chlorobenzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48074-chloro-2-(5-{[(4Z)-3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48084-chloro-2-(5-{[(4Z)-5-oxo-1,3-diphenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48094-chloro-2-(5-{[(4Z)-1-(4-fluorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48104-chloro-2-(5-{[(4Z)-5-oxo-3-phenyl-1-[4-(propan-2-yl)phenyl]-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48112-(5-{[(4Z)-1-(4-tert-butylphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)-4-chlorobenzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_4812(4Z)-1,3-diphenyl-4-[(5-phenylfuran-2-yl)methylidene]-4,5-dihydro-1H-pyrazol-5-one
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48133-[(4Z)-5-oxo-3-phenyl-4-[(5-phenylfuran-2-yl)methylidene]-4,5-dihydro-1H-pyrazol-1-yl]benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48143-[(4Z)-3-methyl-5-oxo-4-[(5-phenylfuran-2-yl)methylidene]-4,5-dihydro-1H-pyrazol-1-yl]benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48152-(5-{[(4Z)-5-oxo-1,3-diphenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48162-(5-{[(4Z)-1-(4-fluorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48172-(5-{[(4Z)-5-oxo-3-phenyl-1-[4-(propan-2-yl)phenyl]-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48182-(5-{[(4Z)-1-(4-tert-butylphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48192-(5-{[(4Z)-1-(4-cyanophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48202-(5-{[(4Z)-1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoicacid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48213-[(4Z)-4-[(furan-2-yl)methylidene]-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl]benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_4828CTSL inhibitor
NA
NA
Ebola virus
NA
NA
Luciferase assay
Decrease (50 %)
NA
26953343
DrugRepV_48338-(trifluoromethyl)-9H-purin-6-amine
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
25746232
DrugRepV_48348-(trifluoromethyl)-9H-purin-6-amine
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
25746232
DrugRepV_48355-amino-2-methyl-N-[(1R)-1-(naphthalen-1-yl)ethyl]benzamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
25746232
DrugRepV_48362-methyl-5-[(methylamino)methyl]-N-[(1R)-1-(naphthalen-1-yl)ethyl]benzamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
25746232
DrugRepV_4837N-[(2H-1,3-benzodioxol-5-yl)methyl]-1-[(1R)-1-(naphthalen-1-yl)ethyl]piperidine-4-carboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
25746232
DrugRepV_4838N-[(2H-1,3-benzodioxol-5-yl)methyl]-1-[(1S)-1-(naphthalen-1-yl)ethyl]piperidine-4-carboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
25746232
DrugRepV_4839N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}thiophene-2-carboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4840N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}benzamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4841N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}cyclobutanecarboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4842N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}cyclohexanecarboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48432-(1H-1,2,3-benzotriazol-1-yl)-N-[4-(pyridin-4-yl)phenyl]-N-[(thiophen-3-yl)methyl]acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4844N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}-2-methylpropanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48452-(1H-1,2,3-benzotriazol-1-yl)-N-[4-(2-methoxypyridin-3-yl)phenyl]-N-[(thiophen-3-yl)methyl]acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4846N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}cyclopropanecarboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48472-(1H-1,2,3-benzotriazol-1-yl)-N-[4-(2-methoxypyrimidin-5-yl)phenyl]-N-[(thiophen-3-yl)methyl]acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4848N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}-2,2,2-trifluoroacetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48492-(1H-1,2,3-benzotriazol-1-yl)-N-[4-(pyridin-3-yl)phenyl]-N-[(thiophen-3-yl)methyl]acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48502-methylpropyl N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}carbamate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4851N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}propanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4852N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}-2-methoxyacetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4853N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}-3-methoxypropanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48542-(1H-1,2,3-benzotriazol-1-yl)-N-[4-(methylamino)phenyl]-N-[(thiophen-3-yl)methyl]acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48552-(1H-1,2,3-benzotriazol-1-yl)-N-[4-(benzylamino)phenyl]-N-[(thiophen-3-yl)methyl]acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4856N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}-2,2-dimethylpropanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48572-methyl-N-(4-{N-[(thiophen-3-yl)methyl]-2-(1H-1,2,3-triazol-1-yl)acetamido}phenyl)propanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4858methyl 2-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}-1H-pyrrole-1-carboxylate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (31 %)
NA
26190463
DrugRepV_48592-(1H-1,2,3-benzotriazol-1-yl)-N-{[1,1-biphenyl]-4-yl}-N-[(thiophen-3-yl)methyl]acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4860N-(4-tert-butylphenyl)-N-[(pyridin-3-yl)methyl]-1H-imidazole-4-carboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (49 %)
NA
26190463
DrugRepV_48612-methyl-N-{4-[2-(4-phenyl-1H-1,2,3-triazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}propanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (25 %)
NA
26190463
DrugRepV_4862N-(4-tert-butylphenyl)-N-[(pyridin-3-yl)methyl]furan-3-carboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (24 %)
NA
26190463
DrugRepV_48632-methyl-N-(4-{N-[(thiophen-3-yl)methyl]-2-[4-(trimethylsilyl)-1H-1,2,3-triazol-1-yl]acetamido}phenyl)propanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_4864N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1-methyl-1H-imidazol-4-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4865N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(benzylcarbamoyl)(3-fluorophenyl)methyl]acetamido]phenyl}-2-methylpropanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48662-[2-(1H-1,2,3-benzotriazol-1-yl)-N-(4-acetamidophenyl)acetamido]-N-tert-butyl-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4867N-tert-butyl-2-(N-{2-cyano-[1,1-biphenyl]-4-yl}-1-(furan-2-yl)formamido)-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4868N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(1H-indol-3-yl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4869N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}cyclopropanecarboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4870N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(benzylcarbamoyl)(3-fluorophenyl)methyl]acetamido]phenyl}cyclobutanecarboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4871N-tert-butyl-2-(N-{4-[(fluoromethoxy)methyl]phenyl}-2-(1H-indol-3-yl)acetamido)-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4872N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}benzamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4873N-tert-butyl-2-[2-(1H-indol-3-yl)-N-[4-(propan-2-yl)phenyl]acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4874N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(benzylcarbamoyl)(3-fluorophenyl)methyl]acetamido]phenyl}cyclopropanecarboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4875N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1,3-oxazol-5-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4876N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1H-imidazol-4-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4877N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4878N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1H-imidazol-4-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4879N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}-1,2-oxazole-5-carboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4880N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1H-imidazol-4-yl)formamido]-2-(pyrimidin-5-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4881N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}-2-methylpropanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4882N-{4-[2-(1H-1,3-benzodiazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}propanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48832-[2-(1H-1,2,3-benzotriazol-1-yl)-N-(4-acetamidophenyl)acetamido]-N-tert-butyl-2-(3-fluorophenyl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48842-[N-(4-aminophenyl)-2-(1H-1,2,3-benzotriazol-1-yl)acetamido]-N-tert-butyl-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4885(2S)-N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4886N-{4-[2-(1H-1,3-benzodiazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}-2-methylpropanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4887N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1,3-oxazol-5-yl)formamido]-2-(pyrimidin-5-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4888N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}thiophene-2-carboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (26 %)
NA
26190463
DrugRepV_4889N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}cyclobutanecarboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (20 %)
NA
26190463
DrugRepV_4890N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}cyclohexanecarboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4891N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}propanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (34 %)
NA
26190463
DrugRepV_4892N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}-2,2-dimethylpropanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4893N-tert-butyl-2-[1-(4-cyanophenyl)-N-(4-fluorophenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (53 %)
NA
26190463
DrugRepV_4894N-tert-butyl-2-[N-cyclopropyl-2-(1H-indol-3-yl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (49 %)
NA
26190463
DrugRepV_4895N-tert-butyl-2-[N-cyclopropyl-2-(pyridin-3-yl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (48 %)
NA
26190463
DrugRepV_4896N-tert-butyl-2-[N-(4-fluorophenyl)-2-(pyridin-3-yl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (47 %)
NA
26190463
DrugRepV_4897N-tert-butyl-2-[N-cyclopropyl-1-(furan-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (43 %)
NA
26190463
DrugRepV_4898N-tert-butyl-2-{N-cyclopropyl-1-[5-(trifluoromethyl)pyridin-2-yl]formamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (42 %)
NA
26190463
DrugRepV_4899N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(pyrazin-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (41 %)
NA
26190463
DrugRepV_4900N-tert-butyl-2-{N-[4-(propan-2-yl)phenyl]-2-(pyridin-3-yl)acetamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (41 %)
NA
26190463
DrugRepV_4901N-tert-butyl-2-[N-(4-fluorophenyl)-2-(1H-indol-3-yl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (41 %)
NA
26190463
DrugRepV_4902N-tert-butyl-2-[N-(4-fluorophenyl)-1-(furan-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (41 %)
NA
26190463
DrugRepV_4903(2S)-2-{N-[4-(butan-2-yl)phenyl]-1-(furan-2-yl)formamido}-N-tert-butyl-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (39 %)
NA
26190463
DrugRepV_4904N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(pyridazin-4-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (35 %)
NA
26190463
DrugRepV_4905N-tert-butyl-2-[1-(3-methylfuran-2-yl)-N-[4-(propan-2-yl)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (36 %)
NA
26190463
DrugRepV_4906N-tert-butyl-2-[1-(furan-2-yl)-N-[4-(propan-2-yl)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (34 %)
NA
26190463
DrugRepV_49072-[2-(1H-1,2,3-benzotriazol-1-yl)-N-(4-acetamidophenyl)acetamido]-2-(3-fluorophenyl)-N-phenylacetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (32 %)
NA
26190463
DrugRepV_4908N-tert-butyl-2-{N-[4-(difluoromethoxy)phenyl]-1-(furan-2-yl)formamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (31 %)
NA
26190463
DrugRepV_4909N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(1H-indol-3-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (31 %)
NA
26190463
DrugRepV_4910N-tert-butyl-2-[1-(furan-2-yl)-N-[4-(1H-pyrrol-3-yl)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (31 %)
NA
26190463
DrugRepV_4911N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1,3-oxazol-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (30 %)
NA
26190463
DrugRepV_4912N-tert-butyl-2-[N-(4-fluorophenyl)-1-[5-(trifluoromethyl)pyridin-2-yl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (29 %)
NA
26190463
DrugRepV_4913N-tert-butyl-2-{N-[4-(fluoromethoxy)phenyl]-2-(pyridin-3-yl)acetamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (29 %)
NA
26190463
DrugRepV_4914[(tert-butylcarbamoyl)(pyridin-3-yl)methyl](4-tert-butylphenyl)carbamic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (29 %)
NA
26190463
DrugRepV_49152-[2-(1H-1,3-benzodiazol-1-yl)-N-(4-methanesulfonamidophenyl)acetamido]-N-tert-butyl-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (28 %)
NA
26190463
DrugRepV_4916N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1H-pyrazol-5-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (28 %)
NA
26190463
DrugRepV_4917N-tert-butyl-2-[1-(4-cyanophenyl)-N-[4-(propan-2-yl)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (28 %)
NA
26190463
DrugRepV_4918N-tert-butyl-2-{N-[4-(3,5-dimethyl-1,2-oxazol-4-yl)phenyl]-1-(furan-2-yl)formamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (28 %)
NA
26190463
DrugRepV_4919N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (28 %)
NA
26190463
DrugRepV_49202-[2-(1H-1,2,3-benzotriazol-1-yl)-N-(4-methanesulfonamidophenyl)acetamido]-N-tert-butyl-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (27 %)
NA
26190463
DrugRepV_4921N-tert-butyl-2-[N-(4-acetamidophenyl)-2-(1H-1,2,3-triazol-1-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (27 %)
NA
26190463
DrugRepV_4922N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(4-chlorophenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (27 %)
NA
26190463
DrugRepV_4923N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(5-methylfuran-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (26 %)
NA
26190463
DrugRepV_4924N-tert-butyl-2-[2-(naphthalen-1-yl)-N-[4-(propan-2-yl)phenyl]acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (26 %)
NA
26190463
DrugRepV_4925N-tert-butyl-2-(4-tert-butylphenyl)-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (26 %)
NA
26190463
DrugRepV_4926N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(naphthalen-1-yl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (26 %)
NA
26190463
DrugRepV_4927N-tert-butyl-2-{N-[4-(fluoromethoxy)phenyl]-2-(1H-indol-3-yl)acetamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (25 %)
NA
26190463
DrugRepV_4928N-tert-butyl-2-{N-[4-(propan-2-yl)phenyl]-1-(5,6,7,8-tetrahydronaphthalen-1-yl)formamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (25 %)
NA
26190463
DrugRepV_4929N-tert-butyl-2-[2-(1H-indol-3-yl)-N-[4-(propan-2-yl)phenyl]acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (25 %)
NA
26190463
DrugRepV_4930N-tert-butyl-2-[1-(furan-2-yl)-N-[4-(2-methylpropoxy)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (25 %)
NA
26190463
DrugRepV_49312-{N-[4-(benzyloxy)phenyl]-1-(furan-2-yl)formamido}-N-tert-butyl-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (25 %)
NA
26190463
DrugRepV_4932N-tert-butyl-2-{N-[4-(propan-2-yl)phenyl]-2-(pyridin-3-yl)acetamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (24 %)
NA
26190463
DrugRepV_4933N-tert-butyl-2-[N-(4-fluorophenyl)-2-(pyridin-3-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (24 %)
NA
26190463
DrugRepV_4934N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(1H-imidazol-4-yl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (24 %)
NA
26190463
DrugRepV_4935N-tert-butyl-2-{N-[4-(difluoromethoxy)phenyl]-1-(1H-indazol-3-yl)formamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (24 %)
NA
26190463
DrugRepV_4936N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(pyridin-3-yl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (23 %)
NA
26190463
DrugRepV_4937N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1H-indazol-3-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (23 %)
NA
26190463
DrugRepV_4938N-tert-butyl-2-(N-{2,6-difluoro-[1,1-biphenyl]-4-yl}-1-(furan-2-yl)formamido)-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (23 %)
NA
26190463
DrugRepV_4939N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-methoxyacetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (23 %)
NA
26190463
DrugRepV_4940N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(pyridin-3-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (23 %)
NA
26190463
DrugRepV_4941N-tert-butyl-2-[1-(4-cyanophenyl)-N-cyclopropylformamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (23 %)
NA
26190463
DrugRepV_4942N-tert-butyl-2-[N-(4-fluorophenyl)-1-(5,6,7,8-tetrahydronaphthalen-1-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (22 %)
NA
26190463
DrugRepV_4943N-tert-butyl-2-[N-cyclopropyl-2-(naphthalen-1-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (22 %)
NA
26190463
DrugRepV_4944N-tert-butyl-2-[N-(4-fluorophenyl)-2-(naphthalen-1-yl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (22 %)
NA
26190463
DrugRepV_4945N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1H-imidazol-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (22 %)
NA
26190463
DrugRepV_49462-(N-{[1,1-biphenyl]-4-yl}-1-(furan-2-yl)formamido)-N-tert-butyl-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (22 %)
NA
26190463
DrugRepV_4947N-tert-butyl-2-[N-(4-fluorophenyl)-2-(1H-indol-3-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (22 %)
NA
26190463
DrugRepV_4948N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(5,6,7,8-tetrahydronaphthalen-1-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4949N-tert-butyl-2-[N-cyclopropyl-1-(1H-indazol-3-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4950N-tert-butyl-2-{N-[4-(fluoromethoxy)phenyl]-2-(naphthalen-1-yl)acetamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4951N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(4-fluorophenyl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4952N-tert-butyl-2-[1-(1H-indazol-3-yl)-N-[4-(propan-2-yl)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4953N-tert-butyl-2-[1-(4-cyanophenyl)-N-[4-(propan-2-yl)phenyl]formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4954N-tert-butyl-2-[N-cyclopropyl-1-(1H-indazol-3-yl)formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4955N-tert-butyl-2-[1-(furan-2-yl)-N-{4-[(1E)-2-phenylethenyl]phenyl}formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4956N-tert-butyl-2-{N-[4-(fluoromethoxy)phenyl]-1-(5,6,7,8-tetrahydronaphthalen-2-yl)formamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4957(2R)-2-{N-[4-(butan-2-yl)phenyl]-1-(furan-2-yl)formamido}-N-tert-butyl-2-(pyridin-4-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (20 %)
NA
26190463
DrugRepV_4958N-tert-butyl-2-[N-(4-acetamidophenyl)-2-[4-(trimethylsilyl)-1H-1,2,3-triazol-1-yl]acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (20 %)
NA
26190463
DrugRepV_49592-{N-[4-(butan-2-yloxy)phenyl]-1-(furan-2-yl)formamido}-N-tert-butyl-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (20 %)
NA
26190463
DrugRepV_4960N-tert-butyl-2-[1-(4-cyanophenyl)-N-cyclopropylformamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (20 %)
NA
26190463
DrugRepV_4961N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-phenylacetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (20 %)
NA
26190463
DrugRepV_4962N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (20 %)
NA
26190463
DrugRepV_4963N-tert-butyl-2-{N-[4-(propan-2-yl)phenyl]-1-(5,6,7,8-tetrahydronaphthalen-1-yl)formamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (20 %)
NA
26190463
DrugRepV_4964N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (19 %)
NA
26190463
DrugRepV_49652-[1-(1-benzofuran-3-yl)-N-(4-tert-butylphenyl)formamido]-N-tert-butyl-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (19 %)
NA
26190463
DrugRepV_4966N-tert-butyl-2-[N-(4-acetamidophenyl)-2-(4-phenyl-1H-1,2,3-triazol-1-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (19 %)
NA
26190463
DrugRepV_4967N-tert-butyl-2-[N-(4-fluorophenyl)-1-[5-(trifluoromethyl)pyridin-2-yl]formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (19 %)
NA
26190463
DrugRepV_4968N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (19 %)
NA
26190463
DrugRepV_4969N-tert-butyl-2-[1-(furan-2-yl)-N-(4-phenoxyphenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (19 %)
NA
26190463
DrugRepV_49702-methylpropyl N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}carbamate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (19 %)
NA
26190463
DrugRepV_4971N-(4-{N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]-2-(2-methyl-1H-imidazol-1-yl)acetamido}phenyl)propanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (19 %)
NA
26190463
DrugRepV_4972N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(oxolan-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4973N-tert-butyl-2-[N-cyclopropyl-1-(5,6,7,8-tetrahydronaphthalen-1-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_49742-[N-(4-aminophenyl)-2-(1H-1,3-benzodiazol-1-yl)acetamido]-N-tert-butyl-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4975N-tert-butyl-2-(N-{2,3-difluoro-[1,1-biphenyl]-4-yl}-1-(furan-2-yl)formamido)-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4976N-tert-butyl-2-{N-[4-(fluoromethoxy)phenyl]-1-[5-(trifluoromethyl)pyridin-2-yl]formamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4977N-tert-butyl-2-[1-(furan-2-yl)-N-[4-(propan-2-yl)phenyl]formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4978N-tert-butyl-2-[N-cyclopropyl-1-(furan-2-yl)formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4979N-tert-butyl-2-[1-(furan-2-yl)-N-[4-(3-methoxyphenoxy)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4980N-(4-{N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]-2-(2-methyl-1H-imidazol-1-yl)acetamido}phenyl)-2-methylpropanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4981N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1H-pyrrol-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4982N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(4-cyanophenyl)formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4983N-tert-butyl-2-{N-[4-(propan-2-yl)phenyl]-1-[6-(trifluoromethyl)pyridin-3-yl]formamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4984N-tert-butyl-2-{N-[4-(fluoromethoxy)phenyl]-2-(pyridin-3-yl)acetamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_49852-[N-(adamantan-1-yl)-1-(furan-2-yl)formamido]-N-tert-butyl-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4986N-tert-butyl-2-[N-(4-fluorophenyl)-1-(5,6,7,8-tetrahydronaphthalen-1-yl)formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_4987N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1H-pyrazol-3-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_4988N-tert-butyl-2-[N-(4-acetamidophenyl)-2-(2-methyl-1H-imidazol-1-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_4989tert-butyl 2-(4-{N-[(tert-butylcarbamoyl)(pyridin-3-yl)methyl]furan-2-amido}phenyl)-1H-pyrrole-1-carboxylate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_4990N-tert-butyl-2-{N-[4-(difluoromethoxy)phenyl]-1-(1H-indazol-3-yl)formamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_4991N-tert-butyl-2-[N-cyclopropyl-2-(1H-indol-3-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_49922-[N-(4-aminophenyl)-2-(2-methyl-1H-imidazol-1-yl)acetamido]-N-tert-butyl-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_4993N-tert-butyl-2-{N-[4-(fluoromethoxy)phenyl]-2-(naphthalen-1-yl)acetamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_4994N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-[6-(trifluoromethyl)pyridin-3-yl]formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_4995N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(3-methoxyphenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_4996N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(2-methoxyphenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_4997N-tert-butyl-2-(N-{3-cyano-[1,1-biphenyl]-4-yl}-1-(furan-2-yl)formamido)-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_4998N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(pyrimidin-5-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_4999N-tert-butyl-2-[N-(4-fluorophenyl)-1-(furan-2-yl)formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_50002-[N-(adamantan-1-yl)-2-(1H-1,2,3-benzotriazol-1-yl)acetamido]-N-benzyl-2-(3-fluorophenyl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_5001N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(thiophen-3-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_5002N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-[5-(trifluoromethyl)furan-2-yl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_5003N-tert-butyl-2-[N-cyclopropyl-2-(pyridin-3-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_5004N-tert-butyl-2-[1-(4-cyanophenyl)-N-[4-(fluoromethoxy)phenyl]formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_5005N-tert-butyl-2-(N-{2,4-difluoro-[1,1-biphenyl]-4-yl}-1-(furan-2-yl)formamido)-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_5006N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1H-indazol-3-yl)formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_5007N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1H-pyrrol-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_5008N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(4-methoxyphenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_50092-[N-(4-benzenesulfonamidophenyl)-1-(furan-2-yl)formamido]-N-tert-butyl-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_5010N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(1H-1,2,3-triazol-4-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_50112-(N-{bicyclo[2.2.1]heptan-2-yl}-1-(furan-2-yl)formamido)-N-tert-butyl-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_5012N-tert-butyl-2-{N-[4-(2-fluoropyridin-4-yl)phenyl]-1-(furan-2-yl)formamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_50132-[2-(1H-1,2,3-benzotriazol-1-yl)-N-{bicyclo[2.2.1]heptan-2-yl}acetamido]-N-tert-butyl-2-(3-fluorophenyl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_5014N-tert-butyl-2-[1-(furan-2-yl)-N-[4-(pyridin-3-yl)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_50152-[2-(1H-1,3-benzodiazol-1-yl)-N-(4-tert-butylphenyl)acetamido]-N-tert-butyl-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_5016N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(naphthalen-1-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_5017N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-[6-(trifluoromethyl)pyridin-3-yl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_5018N-tert-butyl-2-{N-[4-(fluoromethoxy)phenyl]-1-(5,6,7,8-tetrahydronaphthalen-1-yl)formamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_5019N-tert-butyl-2-{N-[4-(propan-2-yl)phenyl]-1-[6-(trifluoromethyl)pyridin-3-yl]formamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_5020N-tert-butyl-2-{N-[4-(fluoromethoxy)phenyl]-1-[6-(trifluoromethyl)pyridin-3-yl]formamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_5021N-tert-butyl-2-[1-(4-cyanophenyl)-N-[4-(fluoromethoxy)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_5022N-tert-butyl-2-[N-(4-fluorophenyl)-2-(naphthalen-1-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_5023N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(5,6,7,8-tetrahydronaphthalen-1-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (14 %)
NA
26190463
DrugRepV_5024N-tert-butyl-2-[N-(4-fluorophenyl)-1-(1H-indazol-3-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (14 %)
NA
26190463
DrugRepV_5025N-tert-butyl-2-(N-{4-cyano-[1,1-biphenyl]-4-yl}-1-(furan-2-yl)formamido)-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (14 %)
NA
26190463
DrugRepV_5026N-(4-{N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]-2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetamido}phenyl)-2-methylpropanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (14 %)
NA
26190463
DrugRepV_50272-[N-(adamantan-1-yl)-2-(1H-1,2,3-benzotriazol-1-yl)acetamido]-N-tert-butyl-2-(3-fluorophenyl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (14 %)
NA
26190463
DrugRepV_50282-[2-(1H-1,3-benzodiazol-1-yl)-N-(4-acetamidophenyl)acetamido]-N-tert-butyl-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (14 %)
NA
26190463
DrugRepV_50292-{N-[4-(benzyloxy)phenyl]-1-(furan-2-yl)formamido}-N-tert-butyl-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (14 %)
NA
26190463
DrugRepV_5030N-tert-butyl-2-[N-cyclopropyl-1-(5,6,7,8-tetrahydronaphthalen-1-yl)formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (14 %)
NA
26190463
DrugRepV_5031N-tert-butyl-2-[1-(furan-2-yl)-N-[4-(pyrimidin-5-yl)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (14 %)
NA
26190463
DrugRepV_50322-[N-(4-aminophenyl)-2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetamido]-N-tert-butyl-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (14 %)
NA
26190463
DrugRepV_5033N-tert-butyl-2-{N-[4-(difluoromethoxy)phenyl]-1-(furan-2-yl)formamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (13 %)
NA
26190463
DrugRepV_5034N-tert-butyl-2-[N-(4-methanesulfonamidophenyl)-2-(2-methyl-1H-imidazol-1-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (13 %)
NA
26190463
DrugRepV_5035N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(pyrimidin-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (13 %)
NA
26190463
DrugRepV_5036N-tert-butyl-2-[2-(naphthalen-1-yl)-N-[4-(propan-2-yl)phenyl]acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (13 %)
NA
26190463
DrugRepV_5037N-tert-butyl-2-[1-(furan-2-yl)-N-[4-(propan-2-yloxy)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (13 %)
NA
26190463
DrugRepV_5038N-tert-butyl-2-[1-(4-cyanophenyl)-N-(4-fluorophenyl)formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (13 %)
NA
26190463
DrugRepV_5039N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(pyridin-3-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (13 %)
NA
26190463
DrugRepV_5040N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(pyridin-4-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (13 %)
NA
26190463
DrugRepV_5041N-[(tert-butylcarbamoyl)(pyridin-3-yl)methyl]-N-(4-tert-butylphenyl)-3,3,3-trifluoropropanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (13 %)
NA
26190463
DrugRepV_5042N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(5-chlorofuran-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (12 %)
NA
26190463
DrugRepV_5043N-tert-butyl-2-{N-cyclopropyl-1-[6-(trifluoromethyl)pyridin-3-yl]formamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (12 %)
NA
26190463
DrugRepV_5044N-tert-butyl-2-[N-(4-ethoxyphenyl)-1-(furan-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (12 %)
NA
26190463
DrugRepV_5045N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(1H-pyrazol-4-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (12 %)
NA
26190463
DrugRepV_50462-[2-(1H-1,2,3-benzotriazol-1-yl)-N-{bicyclo[2.2.1]heptan-2-yl}acetamido]-N-benzyl-2-(3-fluorophenyl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (12 %)
NA
26190463
DrugRepV_5047N-tert-butyl-2-(N-{3,4-difluoro-[1,1-biphenyl]-4-yl}-1-(furan-2-yl)formamido)-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (12 %)
NA
26190463
DrugRepV_5048N-tert-butyl-2-[1-(furan-2-yl)-N-(4-methanesulfonamidophenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (12 %)
NA
26190463
DrugRepV_5049N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(pyridin-3-yl)formamido]-2-(pyridin-2-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (12 %)
NA
26190463
DrugRepV_5050N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(4-hydroxyphenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (11 %)
NA
26190463
DrugRepV_5051N-tert-butyl-2-[N-(4-fluorophenyl)-1-(1H-indazol-3-yl)formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (11 %)
NA
26190463
DrugRepV_5052N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(2-methyl-1H-imidazol-1-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (11 %)
NA
26190463
DrugRepV_5053N-tert-butyl-2-[N-cyclopropyl-2-(naphthalen-1-yl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (11 %)
NA
26190463
DrugRepV_5054N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (11 %)
NA
26190463
DrugRepV_5055N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(4-cyanophenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (11 %)
NA
26190463
DrugRepV_5056N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(2-hydroxyphenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (11 %)
NA
26190463
DrugRepV_5057N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(1H-pyrazol-5-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (11 %)
NA
26190463
DrugRepV_5058N-tert-butyl-2-[1-(1H-indazol-3-yl)-N-[4-(propan-2-yl)phenyl]formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (11 %)
NA
26190463
DrugRepV_5059N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(3-hydroxyphenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (10 %)
NA
26190463
DrugRepV_5060N-tert-butyl-2-[1-(furan-2-yl)-N-(4-propoxyphenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (10 %)
NA
26190463
DrugRepV_5061N-tert-butyl-2-[1-(furan-2-yl)-N-(4-methoxyphenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (10 %)
NA
26190463
DrugRepV_5062N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(1H-imidazol-4-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (9 %)
NA
26190463
DrugRepV_50632-[2-(1H-1,2,3-benzotriazol-1-yl)-N-(4-tert-butylphenyl)acetamido]-N-tert-butyl-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (9 %)
NA
26190463
DrugRepV_50642-[N-(4-benzylphenyl)-1-(furan-2-yl)formamido]-N-tert-butyl-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (8 %)
NA
26190463
DrugRepV_5065N-(4-{N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]-2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetamido}phenyl)propanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (8 %)
NA
26190463
DrugRepV_5066N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(6-methylpyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (8 %)
NA
26190463
DrugRepV_5067N-tert-butyl-2-[N-cyclohexyl-1-(furan-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (6 %)
NA
26190463
DrugRepV_5068Alisporivir
NA
Hepatitis C virus
Middle East respiratory syndrome coronavirus
EMC/2012
NA
Virus yield reduction assay
Decrease (50 %)
Investigational
27840112
DrugRepV_5069Alisporivir
NA
Hepatitis C virus
Middle East respiratory syndrome coronavirus
N3/Jordan
NA
CPE inhibition assay
Decrease (50 %)
Investigational
27840112
DrugRepV_5070Alisporivir
NA
Hepatitis C virus
Severe acute respiratory syndrome coronavirus
MA-15
NA
CPE inhibition assay
Decrease (50 %)
Investigational
27840112
DrugRepV_5089S-Nitroso-N-acetylpenicillamine
NA
NA
Crimean-Congo hemorrhagic fever virus
IbAr 10200
NA
Immunoflourescence assay
Decrease (>90 %)
NA
16632039
DrugRepV_5090S-Nitroso-N-acetylpenicillamine
NA
NA
Crimean-Congo hemorrhagic fever virus
IbAr 10200
NA
Western blot
Decrease
NA
16632039
DrugRepV_5091S-Nitroso-N-acetylpenicillamine
NA
NA
Crimean-Congo hemorrhagic fever virus
IbAr 10200
NA
Real-time PCR
Decrease
NA
16632039
DrugRepV_51002-Deoxy-2-fluorocytidine
NA
NA
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
Decrease (50 %)
NA
29024765
DrugRepV_51022-Chloroadenosine
NA
NA
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
Increase (-26 %)
NA
29024765
DrugRepV_51032-Deoxy-2-fluorocytidine
NA
NA
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
Decrease (98 %)
NA
29024765
DrugRepV_51042-C-Methylcytidine
NA
HCV
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (4 %)
Experimental
29024765
DrugRepV_51052-C-Methyluridine
NA
NA
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
Increase (-9 %)
NA
29024765
DrugRepV_51062-O-Methylcytidine
NA
NA
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (7 %)
NA
29024765
DrugRepV_51072-O-Methyluridine
NA
NA
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (7 %)
NA
29024765
DrugRepV_51083-Deazauridine
NA
NA
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (19 %)
NA
29024765
DrugRepV_51105-Azidouridine
NA
NA
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (28 %)
NA
29024765
DrugRepV_51115-Bromouridine
NA
NA
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (1 %)
NA
29024765
DrugRepV_51125-Chlorouridine
NA
NA
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (0 %)
NA
29024765
DrugRepV_51135-Fluorouridine
NA
Cancer
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (7 %)
Experimental
29024765
DrugRepV_51145-Methylcytidine
NA
NA
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (6 %)
NA
29024765
DrugRepV_51156-Aza-2-thiouridine
NA
NA
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (17 %)
NA
29024765
DrugRepV_51166-Azauridine
NA
Cancer
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (36 %)
NA
29024765
DrugRepV_51177-DMA
NA
NA
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (26 %)
NA
29024765
DrugRepV_51188-Azaadenosine
NA
NA
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
Decrease (92 %)
NA
29024765
DrugRepV_51198-Azidoadenosine
NA
NA
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
Decrease (87 %)
NA
29024765
DrugRepV_5122BCX4430
NA
Ebola virus
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (18 %)
Investigational
29024765
DrugRepV_5129PSI-6130
NA
NA
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
Increase (-6 %)
NA
29024765
DrugRepV_5130PSI-6206
NA
NA
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
Increase (-1 %)
NA
29024765
DrugRepV_5131PSI-7976
NA
NA
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (9 %)
NA
29024765
DrugRepV_5133R-1479
NA
NA
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (15 %)
NA
29024765
DrugRepV_5135RO-9187
NA
NA
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (12 %)
NA
29024765
DrugRepV_5141PF-4708671
NA
NA
Rift Valley fever virus
MP12ΔNSs-Luc
NA
Luciferase assay
Decrease (50 %)
NA
29652799
DrugRepV_5142Pteridinone
NA
NA
Rift Valley fever virus
MP12ΔNSs-Luc
NA
Luciferase assay
Increase (50 %)
NA
29652799
DrugRepV_5143PF-4708671-BI-D1870
NA
NA
Rift Valley fever virus
MP12ΔNSs-Luc
NA
Luciferase assay
Decrease (50 %)
NA
29652799
DrugRepV_5144SB203580
NA
NA
Rift Valley fever virus
MP12ΔNSs-Luc
NA
Luciferase assay
Decrease (50 %)
NA
29652799
DrugRepV_5145PD0325901
NA
Melanoma | Solid Tumour | Solid Tumors | Advanced Cancer | Breast Neoplasms
Rift Valley fever virus
MP12ΔNSs-Luc
NA
Luciferase assay
Decrease (50 %)
Investigational
29652799
DrugRepV_5147Rapamycin-SB203580
NA
NA
Rift Valley fever virus
MP12ΔNSs-Luc
NA
Luciferase assay
Decrease (50 %)
NA
29652799
DrugRepV_5148Rapamycin-PD0325901
NA
NA
Rift Valley fever virus
MP12ΔNSs-Luc
NA
Luciferase assay
Decrease (50 %)
NA
29652799
DrugRepV_5149PF-4708671
NA
NA
Rift Valley fever virus
MP12
NA
Western blot
Decrease
NA
29652799
DrugRepV_5150PF-4708671
NA
NA
Rift Valley fever virus
MP12
NA
Plaque assay
No significant effect (0.5 log pfu/ml)
NA
29652799
DrugRepV_5151PF-4708671-BI-D1870
NA
NA
Rift Valley fever virus
MP12
NA
Western blot
Decrease
NA
29652799
DrugRepV_5152PF-4708671-BI-D1870
NA
NA
Rift Valley fever virus
MP12
NA
Plaque assay
Decrease (2 log pfu/ml)
NA
29652799
DrugRepV_5153SB203580
NA
NA
Rift Valley fever virus
MP12
NA
Western blot
No significant effect
NA
29652799
DrugRepV_5154SB203580
NA
NA
Rift Valley fever virus
MP12
NA
Plaque assay
No significant effect (<0.5log pfu/ml)
NA
29652799
DrugRepV_5155PD0325901
NA
Melanoma | Solid Tumour | Solid Tumors | Advanced Cancer | Breast Neoplasms
Rift Valley fever virus
MP12
NA
Western blot
Decrease
Investigational
29652799
DrugRepV_5156PD0325901
NA
Melanoma | Solid Tumour | Solid Tumors | Advanced Cancer | Breast Neoplasms
Rift Valley fever virus
MP12
NA
Plaque assay
No significant effect (0.5log pfu/ml)
Investigational
29652799
DrugRepV_5158Rapamycin-SB203580
NA
NA
Rift Valley fever virus
MP12
NA
Plaque assay
Decrease (>3log pfu/ml)
NA
29652799
DrugRepV_5159Rapamycin-PD0325901
NA
NA
Rift Valley fever virus
MP12
NA
Plaque assay
Decrease (3log pfu/ml)
NA
29652799
DrugRepV_5160Benzavir-2
NA
NA
Rift Valley fever virus
rRVFV?NSs::Katushka
NA
Fluorescence-based assay
Decrease (50 %)
NA
29386590
DrugRepV_5161Benzavir-1
NA
NA
Rift Valley fever virus
rRVFV?NSs::Katushka
NA
Fluorescence-based assay
Decrease (50 %)
NA
29386590
DrugRepV_51622-[[4-chloro-2-[(2-fluorobenzoyl)amino]benzoyl]amino]benzoic acid
NA
NA
Rift Valley fever virus
rRVFV?NSs::Katushka
NA
Fluorescence-based assay
Decrease (50 %)
NA
29386590
DrugRepV_51632-[[2-(2,2-dimethylpropanoylamino)benzoyl]amino]benzoic acid
NA
NA
Rift Valley fever virus
rRVFV?NSs::Katushka
NA
Fluorescence-based assay
No significant effect (50 %)
NA
29386590
DrugRepV_51642-[[2-(cyclohexanecarbonylamino)benzoyl]amino]benzoic acid
NA
NA
Rift Valley fever virus
rRVFV?NSs::Katushka
NA
Fluorescence-based assay
No significant effect (50 %)
NA
29386590
DrugRepV_51713-(2,3-Diphenyl-1H-indol-1-yl)-N-(3-hydroxybenzylidene) propanohydrazide
NA
NA
Rift Valley fever virus
rRVFVΔNSs::Katushka
NA
Fluorescence-based assay
Decrease (50 %)
NA
26762502
DrugRepV_51721-(3,5-Di-tert-butyl-4-hydroxyphenyl)-2-(2-imino-3-(4-methylbenzyl)-2,3- dihydro-1H-benzimidazol-1-yl)ethanone hydrobromide
NA
NA
Rift Valley fever virus
rRVFVΔNSs::Katushka
NA
Fluorescence-based assay
Decrease (50 %)
NA
26762502
DrugRepV_51734-Hydroxy-3-methoxybenzaldehyde (4-(3,4-dimethoxyphenyl)-6-phenyl-2- pyrimidinyl)hydrazone
NA
NA
Rift Valley fever virus
rRVFVΔNSs::Katushka
NA
Fluorescence-based assay
Decrease (50 %)
NA
26762502
DrugRepV_51741-(3,4-Dichlorophenyl)-3-(4-(3,4-dimethoxyphenyl)-1-methylpyrrolidin-3- yl)urea
NA
NA
Rift Valley fever virus
rRVFVΔNSs::Katushka
NA
Fluorescence-based assay
Decrease (50 %)
NA
26762502
DrugRepV_51752-Chloro-N-(2-(5-(trifluoromethyl)-1,3,4-thiadiazol-2-ylcarbamoyl)phenyl) benzamide
NA
NA
Rift Valley fever virus
rRVFVΔNSs::Katushka
NA
Fluorescence-based assay
Decrease (50 %)
NA
26762502
DrugRepV_51762-(4-Bromo-5-chlorothiophene-2-sulfonamido)-N-(4-fluorophenyl) benzamide
NA
NA
Rift Valley fever virus
rRVFVΔNSs::Katushka
NA
Fluorescence-based assay
Decrease (50 %)
NA
26762502
DrugRepV_5180C795-0925
NA
NA
Rift Valley fever virus
ZH501
NA
Immunoflourescence assay
Decrease (50 %)
NA
25144302
DrugRepV_5181D011-2120
NA
NA
Rift Valley fever virus
ZH501
NA
Immunoflourescence assay
Decrease (50 %)
NA
25144302
DrugRepV_5182F694-1532
NA
NA
Rift Valley fever virus
ZH501
NA
Immunoflourescence assay
Decrease (50 %)
NA
25144302
DrugRepV_5183G202-0362
NA
NA
Rift Valley fever virus
ZH501
NA
Immunoflourescence assay
Decrease (50 %)
NA
25144302
DrugRepV_5186C795-0925
NA
NA
Rift Valley fever virus
ZH501
NA
Immunoflourescence assay
Decrease (50 %)
NA
25144302
DrugRepV_5187D011-2120
NA
NA
Rift Valley fever virus
ZH501
NA
Immunoflourescence assay
Decrease (50 %)
NA
25144302
DrugRepV_5188F694-1532
NA
NA
Rift Valley fever virus
ZH501
NA
Immunoflourescence assay
Decrease (50 %)
NA
25144302
DrugRepV_5189G202-0362
NA
NA
Rift Valley fever virus
ZH501
NA
Immunoflourescence assay
Decrease (50 %)
NA
25144302
DrugRepV_5192C795-0925
NA
NA
Ebola virus
Zaire
NA
Immunoflourescence assay
Decrease (50 %)
NA
25144302
DrugRepV_5193D011-2120
NA
NA
Ebola virus
Zaire
NA
Immunoflourescence assay
Decrease (50 %)
NA
25144302
DrugRepV_5194F694-1532
NA
NA
Ebola virus
Zaire
NA
Immunoflourescence assay
Decrease (50 %)
NA
25144302
DrugRepV_5195G202-0362
NA
NA
Ebola virus
Zaire
NA
Immunoflourescence assay
Decrease (50 %)
NA
25144302
DrugRepV_5197C795-0925
NA
NA
Marburg virus
Ci67
NA
Immunoflourescence assay
Decrease (50 %)
NA
25144302
DrugRepV_5198D011-2120
NA
NA
Marburg virus
Ci67
NA
Immunoflourescence assay
Decrease (50 %)
NA
25144302
DrugRepV_5199F694-1532
NA
NA
Marburg virus
Ci67
NA
Immunoflourescence assay
Decrease (50 %)
NA
25144302
DrugRepV_5200G202-0362
NA
NA
Marburg virus
Ci67
NA
Immunoflourescence assay
Decrease (50 %)
NA
25144302
DrugRepV_5202C795-0925
NA
NA
Lassa virus
Josiah
NA
Immunoflourescence assay
Decrease (50 %)
NA
25144302
DrugRepV_5203D011-2120
NA
NA
Lassa virus
Josiah
NA
Immunoflourescence assay
Decrease (50 %)
NA
25144302
DrugRepV_5204F694-1532
NA
NA
Lassa virus
Josiah
NA
Immunoflourescence assay
Decrease (50 %)
NA
25144302
DrugRepV_5208Curcumin
NA
Depressive disorder
Rift Valley fever virus
MP12
NA
Plaque assay
Decrease (3 log pfu/ml)
Approved
22847000
DrugRepV_5209SC-514
NA
NA
Rift Valley fever virus
MP12
NA
Plaque assay
Decrease (<1 log pfu/ml)
NA
22847000
DrugRepV_5210Curcumin
NA
Depressive disorder
Rift Valley fever virus
ZH501
NA
Plaque assay
Decrease (4 log pfu/ml)
Approved
22847000
DrugRepV_5211Curcumin
NA
Depressive disorder
Rift Valley fever virus
MP12
NA
Plaque assay
Decrease (5 log pfu/ml)
Approved
22847000
DrugRepV_5213Quinacrine Dihydrochloride
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Rift Valley fever virus
NA
NA
RVFV nucleocapsid (N) protein RNA-binding activity
Decrease (50 %)
Investigational
22644268
DrugRepV_5214N-methyl-2,3-diphenyl-1,2,4-thiadiazol-5-imine;hydrobromide
NA
NA
Rift Valley fever virus
NA
NA
RVFV nucleocapsid (N) protein RNA-binding activity
Decrease (50 %)
NA
22644268
DrugRepV_52154-(3,6-dioxocyclohexa-1,4-dien-1-yl)benzoic acid
NA
NA
Rift Valley fever virus
NA
NA
RVFV nucleocapsid (N) protein RNA-binding activity
Decrease (50 %)
NA
22644268
DrugRepV_5216BTB 11461
NA
NA
Rift Valley fever virus
NA
NA
RVFV nucleocapsid (N) protein RNA-binding activity
Decrease (50 %)
NA
22644268
DrugRepV_5226Ribamidine
NA
NA
Crimean-Congo hemorrhagic fever virus
IbAr 10200
NA
Neutral red uptake assay
Decrease (50 %)
Investigational
15026198
DrugRepV_52276-Azauridine
NA
Cancer
Crimean-Congo hemorrhagic fever virus
IbAr 10200
NA
Neutral red uptake assay
Decrease (50 %)
NA
15026198
DrugRepV_5228Selenazofurin
NA
NA
Crimean-Congo hemorrhagic fever virus
IbAr 10200
NA
Neutral red uptake assay
Decrease (50 %)
NA
15026198
DrugRepV_5231Ribamidine
NA
NA
Crimean-Congo hemorrhagic fever virus
Spu 128/81
NA
Neutral red uptake assay
Decrease (50 %)
Investigational
15026198
DrugRepV_52326-Azauridine
NA
Cancer
Crimean-Congo hemorrhagic fever virus
Spu 128/81
NA
Neutral red uptake assay
Decrease (50 %)
NA
15026198
DrugRepV_5233Selenazofurin
NA
NA
Crimean-Congo hemorrhagic fever virus
Spu 128/81
NA
Neutral red uptake assay
Decrease (50 %)
NA
15026198
DrugRepV_5236Ribamidine
NA
NA
Crimean-Congo hemorrhagic fever virus
Hy-13
NA
Neutral red uptake assay
Decrease (50 %)
Investigational
15026198
DrugRepV_52376-Azauridine
NA
Cancer
Crimean-Congo hemorrhagic fever virus
Hy-13
NA
Neutral red uptake assay
Decrease (50 %)
NA
15026198
DrugRepV_5238Selenazofurin
NA
NA
Crimean-Congo hemorrhagic fever virus
Hy-13
NA
Neutral red uptake assay
Decrease (50 %)
NA
15026198
DrugRepV_5241Ribamidine
NA
NA
Crimean-Congo hemorrhagic fever virus
UG3010
NA
Neutral red uptake assay
Decrease (50 %)
Investigational
15026198
DrugRepV_52426-Azauridine
NA
Cancer
Crimean-Congo hemorrhagic fever virus
UG3010
NA
Neutral red uptake assay
Decrease (50 %)
NA
15026198
DrugRepV_5243Selenazofurin
NA
NA
Crimean-Congo hemorrhagic fever virus
UG3010
NA
Neutral red uptake assay
Decrease (50 %)
NA
15026198
DrugRepV_5245Cytarabine
NA
Leukemia
Variola virus
Harvey
NA
Focus forming assay
Decrease (82.3 %)
Approved
198636
DrugRepV_5246Cytarabine
NA
Leukemia
Variola virus
Harvey
NA
Focus forming assay
Decrease (30.2 %)
Approved
198636
DrugRepV_52476-Azauridine
NA
Cancer
Variola virus
Harvey
NA
Focus forming assay
Decrease (1.2 %)
NA
198636
DrugRepV_5248Cytarabine
NA
Leukemia
Variola virus
Yamamoto P
NA
Focus forming assay
Decrease (66.1 %)
Approved
198636
DrugRepV_52496-Azauridine
NA
Cancer
Variola virus
Yamamoto P
NA
Focus forming assay
Decrease (2.9 %)
NA
198636
DrugRepV_5250Cytarabine
NA
Leukemia
Variola virus
Butler
NA
Focus forming assay
Decrease (44.4 %)
Approved
198636
DrugRepV_52516-Azauridine
NA
Cancer
Variola virus
Butler
NA
Focus forming assay
No significant effect (No inhibition %)
NA
198636
DrugRepV_5253beta-D-cyclopentenyl cytosine
NA
NA
Variola virus
Bangladesh 1975
NA
NA
Decrease (50 %)
NA
14604375
DrugRepV_5254beta-D-cyclopentenyl cytosine
NA
NA
Variola virus
7124
NA
NA
Decrease (50 %)
NA
14604375
DrugRepV_5255beta-D-cyclopentenyl-5-iodocytidine
NA
NA
Variola virus
Bangladesh 1975
NA
NA
Decrease (50 %)
NA
14604375
DrugRepV_5256beta-D-cyclopentenyl-5-iodocytidine
NA
NA
Variola virus
7124
NA
NA
Decrease (50 %)
NA
14604375
DrugRepV_5257beta-D-Cyclopentenyl-5-chlorocytidine
NA
NA
Variola virus
Bangladesh 1975
NA
NA
Decrease (50 %)
NA
14604375
DrugRepV_5258beta-D-Cyclopentenyl-5-chlorocytidine
NA
NA
Variola virus
7124
NA
NA
Decrease (50 %)
NA
14604375
DrugRepV_5259beta-D-cyclopentenyl-5-bromocytidine
NA
NA
Variola virus
Bangladesh 1975
NA
NA
Decrease (50 %)
NA
14604375
DrugRepV_5260beta-D-cyclopentenyl-5-bromocytidine
NA
NA
Variola virus
7124
NA
NA
Decrease (50 %)
NA
14604375
DrugRepV_5261Delphinidin Chloride
NA
NA
Zika virus
MR766
NA
Plaque assay
Decrease (102 Log)
NA
28744282
DrugRepV_5263Delphinidin Chloride
NA
NA
Zika virus
PA259459
NA
Plaque assay
Decrease
NA
28744282
DrugRepV_5265Tetra-O-methyl nordihydroguaiaretic acid (M4N)
NA
Brain and Central Nervous System Tumors
Zika virus
PA259459
NA
Plaque assay
Decrease (50 %)
Investigational
28507114
DrugRepV_5266Tetra-O-methyl nordihydroguaiaretic acid (M4N)
NA
Brain and Central Nervous System Tumors
Zika virus
PA259459
NA
Plaque assay
Decrease (50 %)
Investigational
28507114
DrugRepV_526725-Hydroxycholesterol
NA
NA
Lassa virus
Josiah
NA
TCID50 assay
Decrease (>1.1 Log)
Experimental
27999160
DrugRepV_526825-Hydroxycholesterol
NA
NA
Lassa virus
Josiah
NA
TCID50 assay
Decrease (1.4 Log)
Experimental
27999160
DrugRepV_52731-{[2-(benzyloxy)ethoxy]methyl}-1H-imidazole-4,5-dicarbonitrile
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_5274diethyl {[2-(4,5-dicyano-1H-imidazol-1-yl)ethoxy]methyl}phosphonate
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_5275diethyl {2-[(4,5-dicyano-1H-imidazol-1-yl)methoxy]ethyl}phosphonate
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_52761-[(2-bromoethoxy)methyl]-1H-imidazole-4,5-dicarbonitrile
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_52772-[(4,5-dicyano-1H-imidazol-1-yl)methoxy]ethyl acetate
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_52781-[(2-hydroxyethoxy)methyl]-1H-imidazole-4,5-dicarbonitrile
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_52791-[(2R,5S)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-1H-imidazole-4,5-dicarbonitrile
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_5280{2-[4,5-bis(methoxycarbonyl)-1H-imidazol-1-yl]ethoxy}phosphonic acid
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_52814,5-dimethyl 1-[(2R,5S)-4-hydroxy-5-(hydroxymethyl)oxolan-2-yl]-1H-imidazole-4,5-dicarboxylate
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_52824,5-dimethyl 1-(2-hydroxyethyl)-1H-imidazole-4,5-dicarboxylate
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_52834,5-dimethyl 1-[2-(acetyloxy)ethyl]-1H-imidazole-4,5-dicarboxylate
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_52844,5-dimethyl 1-[(2R,5S)-3,4-bis(acetyloxy)-5-[(acetyloxy)methyl]oxolan-2-yl]-1H-imidazole-4,5-dicarboxylate
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_52854,5-dimethyl 1-[(2R,5S)-3,4-bis(benzoyloxy)-5-[(benzoyloxy)methyl]oxolan-2-yl]-1H-imidazole-4,5-dicarboxylate
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_52864,5-dimethyl 1-[(2R,5S)-4-(4-methylbenzoyloxy)-5-[(4-methylbenzoyloxy)methyl]oxolan-2-yl]-1H-imidazole-4,5-dicarboxylate
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_52871-(2-hydroxyethyl)-1H-imidazole-4,5-dicarboxylic acid
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_52881-{[2-(benzyloxy)ethoxy]methyl}-1H-imidazole-4,5-dicarboxylic acid
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_52891-[(2R,5S)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-1H-imidazole-4,5-dicarbohydrazide
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_52901-[(2R,5S)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-1H-imidazole-4,5-dicarboxamide
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_52911-{[2-(benzyloxy)ethoxy]methyl}-1H-imidazole-4,5-dicarbonitrile
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (90 %)
NA
15451189
DrugRepV_5292diethyl {[2-(4,5-dicyano-1H-imidazol-1-yl)ethoxy]methyl}phosphonate
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (90 %)
NA
15451189
DrugRepV_5293diethyl {2-[(4,5-dicyano-1H-imidazol-1-yl)methoxy]ethyl}phosphonate
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (90 %)
NA
15451189
DrugRepV_52941-[(2-bromoethoxy)methyl]-1H-imidazole-4,5-dicarbonitrile
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (90 %)
NA
15451189
DrugRepV_52952-[(4,5-dicyano-1H-imidazol-1-yl)methoxy]ethyl acetate
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (90 %)
NA
15451189
DrugRepV_52961-[(2-hydroxyethoxy)methyl]-1H-imidazole-4,5-dicarbonitrile
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (90 %)
NA
15451189
DrugRepV_52971-[(2R,5S)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-1H-imidazole-4,5-dicarbonitrile
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (90 %)
NA
15451189
DrugRepV_5298{2-[4,5-bis(methoxycarbonyl)-1H-imidazol-1-yl]ethoxy}phosphonic acid
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (90 %)
NA
15451189
DrugRepV_52994,5-dimethyl 1-[(2R,5S)-4-hydroxy-5-(hydroxymethyl)oxolan-2-yl]-1H-imidazole-4,5-dicarboxylate
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (90 %)
NA
15451189
DrugRepV_53004,5-dimethyl 1-(2-hydroxyethyl)-1H-imidazole-4,5-dicarboxylate
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (90 %)
NA
15451189
DrugRepV_53014,5-dimethyl 1-[2-(acetyloxy)ethyl]-1H-imidazole-4,5-dicarboxylate
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (90 %)
NA
15451189
DrugRepV_53024,5-dimethyl 1-[(2R,5S)-3,4-bis(acetyloxy)-5-[(acetyloxy)methyl]oxolan-2-yl]-1H-imidazole-4,5-dicarboxylate
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (90 %)
NA
15451189
DrugRepV_53034,5-dimethyl 1-[(2R,5S)-3,4-bis(benzoyloxy)-5-[(benzoyloxy)methyl]oxolan-2-yl]-1H-imidazole-4,5-dicarboxylate
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (90 %)
NA
15451189
DrugRepV_53044,5-dimethyl 1-[(2R,5S)-4-(4-methylbenzoyloxy)-5-[(4-methylbenzoyloxy)methyl]oxolan-2-yl]-1H-imidazole-4,5-dicarboxylate
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (90 %)
NA
15451189
DrugRepV_53051-(2-hydroxyethyl)-1H-imidazole-4,5-dicarboxylic acid
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (90 %)
NA
15451189
DrugRepV_53061-{[2-(benzyloxy)ethoxy]methyl}-1H-imidazole-4,5-dicarboxylic acid
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (90 %)
NA
15451189
DrugRepV_53071-[(2R,5S)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-1H-imidazole-4,5-dicarbohydrazide
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (90 %)
NA
15451189
DrugRepV_53081-[(2R,5S)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-1H-imidazole-4,5-dicarboxamide
NA
NA
Lassa virus
AV
NA
Real-time PCR
Decrease (90 %)
NA
15451189
DrugRepV_53091-{[2-(benzyloxy)ethoxy]methyl}-1H-imidazole-4,5-dicarbonitrile
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_5310diethyl {[2-(4,5-dicyano-1H-imidazol-1-yl)ethoxy]methyl}phosphonate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_5311diethyl {2-[(4,5-dicyano-1H-imidazol-1-yl)methoxy]ethyl}phosphonate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53121-[(2-bromoethoxy)methyl]-1H-imidazole-4,5-dicarbonitrile
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53132-[(4,5-dicyano-1H-imidazol-1-yl)methoxy]ethyl acetate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53141-[(2-hydroxyethoxy)methyl]-1H-imidazole-4,5-dicarbonitrile
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53151-[(2R,5S)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-1H-imidazole-4,5-dicarbonitrile
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_5316{2-[4,5-bis(methoxycarbonyl)-1H-imidazol-1-yl]ethoxy}phosphonic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53174,5-dimethyl 1-[(2R,5S)-4-hydroxy-5-(hydroxymethyl)oxolan-2-yl]-1H-imidazole-4,5-dicarboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53184,5-dimethyl 1-(2-hydroxyethyl)-1H-imidazole-4,5-dicarboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53194,5-dimethyl 1-[2-(acetyloxy)ethyl]-1H-imidazole-4,5-dicarboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53204,5-dimethyl 1-[(2R,5S)-3,4-bis(acetyloxy)-5-[(acetyloxy)methyl]oxolan-2-yl]-1H-imidazole-4,5-dicarboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53214,5-dimethyl 1-[(2R,5S)-3,4-bis(benzoyloxy)-5-[(benzoyloxy)methyl]oxolan-2-yl]-1H-imidazole-4,5-dicarboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53224,5-dimethyl 1-[(2R,5S)-4-(4-methylbenzoyloxy)-5-[(4-methylbenzoyloxy)methyl]oxolan-2-yl]-1H-imidazole-4,5-dicarboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53231-(2-hydroxyethyl)-1H-imidazole-4,5-dicarboxylic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53241-{[2-(benzyloxy)ethoxy]methyl}-1H-imidazole-4,5-dicarboxylic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53251-[(2R,5S)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-1H-imidazole-4,5-dicarbohydrazide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53261-[(2R,5S)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-1H-imidazole-4,5-dicarboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53271-{[2-(benzyloxy)ethoxy]methyl}-1H-imidazole-4,5-dicarbonitrile
NA
NA
Ebola virus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_5328diethyl {[2-(4,5-dicyano-1H-imidazol-1-yl)ethoxy]methyl}phosphonate
NA
NA
Ebola virus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_5329diethyl {2-[(4,5-dicyano-1H-imidazol-1-yl)methoxy]ethyl}phosphonate
NA
NA
Ebola virus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53301-[(2-bromoethoxy)methyl]-1H-imidazole-4,5-dicarbonitrile
NA
NA
Ebola virus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53312-[(4,5-dicyano-1H-imidazol-1-yl)methoxy]ethyl acetate
NA
NA
Ebola virus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53321-[(2-hydroxyethoxy)methyl]-1H-imidazole-4,5-dicarbonitrile
NA
NA
Ebola virus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53331-[(2R,5S)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-1H-imidazole-4,5-dicarbonitrile
NA
NA
Ebola virus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_5334{2-[4,5-bis(methoxycarbonyl)-1H-imidazol-1-yl]ethoxy}phosphonic acid
NA
NA
Ebola virus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53354,5-dimethyl 1-[(2R,5S)-4-hydroxy-5-(hydroxymethyl)oxolan-2-yl]-1H-imidazole-4,5-dicarboxylate
NA
NA
Ebola virus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53364,5-dimethyl 1-(2-hydroxyethyl)-1H-imidazole-4,5-dicarboxylate
NA
NA
Ebola virus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53374,5-dimethyl 1-[2-(acetyloxy)ethyl]-1H-imidazole-4,5-dicarboxylate
NA
NA
Ebola virus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53384,5-dimethyl 1-[(2R,5S)-3,4-bis(acetyloxy)-5-[(acetyloxy)methyl]oxolan-2-yl]-1H-imidazole-4,5-dicarboxylate
NA
NA
Ebola virus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53394,5-dimethyl 1-[(2R,5S)-3,4-bis(benzoyloxy)-5-[(benzoyloxy)methyl]oxolan-2-yl]-1H-imidazole-4,5-dicarboxylate
NA
NA
Ebola virus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53404,5-dimethyl 1-[(2R,5S)-4-(4-methylbenzoyloxy)-5-[(4-methylbenzoyloxy)methyl]oxolan-2-yl]-1H-imidazole-4,5-dicarboxylate
NA
NA
Ebola virus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53411-(2-hydroxyethyl)-1H-imidazole-4,5-dicarboxylic acid
NA
NA
Ebola virus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53421-{[2-(benzyloxy)ethoxy]methyl}-1H-imidazole-4,5-dicarboxylic acid
NA
NA
Ebola virus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53431-[(2R,5S)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-1H-imidazole-4,5-dicarbohydrazide
NA
NA
Ebola virus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53441-[(2R,5S)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-1H-imidazole-4,5-dicarboxamide
NA
NA
Ebola virus
NA
NA
Real-time PCR
Decrease (50 %)
NA
15451189
DrugRepV_53455-ethynyl-1-beta-D-ribofuranosylimidazole-4-carboxamide
NA
NA
Lassa virus
AV
NA
RT-PCR
Decrease (50 %)
NA
21616094
DrugRepV_53465-ethynyl-1-beta-D-ribofuranosylimidazole-4-carboxamide
NA
NA
Lassa virus
AV
NA
RT-PCR
Decrease (50 %)
NA
21616094
DrugRepV_53475-ethynyl-1-beta-D-ribofuranosylimidazole-4-carboxamide
NA
NA
Lassa virus
AV
NA
RT-PCR
Decrease (50 %)
NA
21616094
DrugRepV_53485-ethynyl-1-beta-D-ribofuranosylimidazole-4-carboxamide
NA
NA
Lassa virus
AV
NA
RT-PCR
Decrease (50 %)
NA
21616094
DrugRepV_53495-ethynyl-1-beta-D-ribofuranosylimidazole-4-carboxamide
NA
NA
Ebola virus
NA
NA
RT-PCR
Decrease (50 %)
NA
21616094
DrugRepV_53505-ethynyl-1-beta-D-ribofuranosylimidazole-4-carboxamide
NA
NA
Ebola virus
NA
NA
RT-PCR
Decrease (50 %)
NA
21616094
DrugRepV_53515-ethynyl-1-beta-D-ribofuranosylimidazole-4-carboxamide
NA
NA
Ebola virus
NA
NA
RT-PCR
Decrease (50 %)
NA
21616094
DrugRepV_53525-ethynyl-1-beta-D-ribofuranosylimidazole-4-carboxamide
NA
NA
Ebola virus
NA
NA
RT-PCR
Decrease (50 %)
NA
21616094
DrugRepV_53535-ethynyl-1-beta-D-ribofuranosylimidazole-4-carboxamide
NA
NA
Lassa virus
AV
NA
RT-PCR
Decrease (90 %)
NA
21616094
DrugRepV_53545-ethynyl-1-beta-D-ribofuranosylimidazole-4-carboxamide
NA
NA
Lassa virus
AV
NA
RT-PCR
Decrease (90 %)
NA
21616094
DrugRepV_53555-ethynyl-1-beta-D-ribofuranosylimidazole-4-carboxamide
NA
NA
Lassa virus
AV
NA
RT-PCR
Decrease (90 %)
NA
21616094
DrugRepV_53565-ethynyl-1-beta-D-ribofuranosylimidazole-4-carboxamide
NA
NA
Lassa virus
AV
NA
RT-PCR
Decrease (90 %)
NA
21616094
DrugRepV_53575-ethynyl-1-beta-D-ribofuranosylimidazole-4-carboxamide
NA
NA
Ebola virus
NA
NA
RT-PCR
Decrease (90 %)
NA
21616094
DrugRepV_53585-ethynyl-1-beta-D-ribofuranosylimidazole-4-carboxamide
NA
NA
Ebola virus
NA
NA
RT-PCR
Decrease (90 %)
NA
21616094
DrugRepV_53595-ethynyl-1-beta-D-ribofuranosylimidazole-4-carboxamide
NA
NA
Ebola virus
NA
NA
RT-PCR
Decrease (90 %)
NA
21616094
DrugRepV_53605-ethynyl-1-beta-D-ribofuranosylimidazole-4-carboxamide
NA
NA
Ebola virus
NA
NA
RT-PCR
Decrease (90 %)
NA
21616094
DrugRepV_53772-deoxy-2-fluorocytidine
NA
NA
Lassa virus
Josiah
NA
Minigenome assays
Decrease (50 %)
NA
27771389
DrugRepV_53785-fluorouridine
NA
Cancer
Lassa virus
Josiah
NA
Minigenome assays
Decrease (50 %)
Experimental
27771389
DrugRepV_53798-Azaadenosine
NA
NA
Lassa virus
Josiah
NA
Minigenome assays
Decrease (50 %)
NA
27771389
DrugRepV_53808-Azidoadenosine
NA
NA
Lassa virus
Josiah
NA
Minigenome assays
Decrease (50 %)
NA
27771389
DrugRepV_5381Toyocamycin
NA
NA
Lassa virus
Josiah
NA
Minigenome assays
Decrease (50 %)
Experimental
27771389
DrugRepV_53826-Azauridine
NA
Cancer
Lassa virus
Josiah
NA
Minigenome assays
Decrease (50 %)
NA
27771389
DrugRepV_53838-Azaadenosine
NA
NA
Ebola virus
Ebola virus/H.sapiens-rec/LBR/2014/ Makona-L2014
NA
Minigenome assays
Decrease (50 %)
NA
27771389
DrugRepV_5384Toyocamycin
NA
NA
Ebola virus
Ebola virus/H.sapiens-rec/LBR/2014/ Makona-L2015
NA
Minigenome assays
Decrease (50 %)
Experimental
27771389
DrugRepV_53856-Azauridine
NA
Cancer
Ebola virus
Ebola virus/H.sapiens-rec/LBR/2014/ Makona-L2016
NA
Minigenome assays
Decrease (50 %)
NA
27771389
DrugRepV_5386Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Ebola virus
NA
NA
qRT-PCR
Decrease
Investigational
31307979
DrugRepV_5387Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Chikungunya virus
NA
NA
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_5388Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Ebola virus
NA
NA
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_5389Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Influenza virus
NA
Pathway
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_5390Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_5391Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Rift Valley fever virus
NA
NA
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_5392Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Zika virus
NA
NA
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_5393Zoniporide
NA
NA
Lassa virus
Josiah
NA
Luciferase assay
Decrease (50 %)
NA
30700611
DrugRepV_5394Zoniporide
NA
NA
Ebola virus
Mayinga
NA
Luciferase assay
Decrease (50 %)
NA
30700611
DrugRepV_5399Apilimod
NA
Crohn's disease | Psoriasis | Psoriatic disorders
Lassa virus
Josiah
NA
Luciferase assay
Decrease (50 %)
Investigational
30700611
DrugRepV_5400Apilimod
NA
Crohn's disease | Psoriasis | Psoriatic disorders
Ebola virus
Mayinga
NA
Luciferase assay
Decrease (50 %)
Investigational
30700611
DrugRepV_5401Arbidol
NA
Viral infection
Lassa virus
Josiah
NA
Luciferase assay
Decrease (50 %)
Investigational
30700611
DrugRepV_5402Arbidol
NA
Viral infection
Ebola virus
Mayinga
NA
Luciferase assay
Decrease (50 %)
Investigational
30700611
DrugRepV_5410Desethylamodiaquine
NA
NA
Zika virus
PLCal_ZV
NA
MTT assay
Decrease (50 %)
NA
30801742
DrugRepV_5411Desethylchloroquine
NA
NA
Zika virus
PLCal_ZV
NA
MTT assay
Decrease (50 %)
NA
30801742
DrugRepV_5413Desethylamodiaquine
NA
NA
Zika virus
MR 766
NA
MTT assay
Decrease (50 %)
NA
30801742
DrugRepV_5414Desethylchloroquine
NA
NA
Zika virus
MR 766
NA
MTT assay
Decrease (50 %)
NA
30801742
DrugRepV_5416Desethylamodiaquine
NA
NA
Zika virus
PRVABC59
NA
MTT assay
Decrease (50 %)
NA
30801742
DrugRepV_5417Desethylchloroquine
NA
NA
Zika virus
PRVABC59
NA
MTT assay
Decrease (50 %)
NA
30801742
DrugRepV_5420Losmapimod
NA
Chronic Obstructive Pulmonary Disease
Lassa virus
Josiah
NA
TCID50 assay
Decrease (50 %)
Investigational
30953674
DrugRepV_5421Losmapimod
NA
Chronic Obstructive Pulmonary Disease
Lassa virus
Josiah
NA
RT-qPCR
Decrease (50 %)
Investigational
30953674
DrugRepV_5422Losmapimod
NA
Chronic Obstructive Pulmonary Disease
Lassa virus
LP
NA
NA
Decrease (50 %)
Investigational
30953674
DrugRepV_5423Losmapimod
NA
Chronic Obstructive Pulmonary Disease
Lassa virus
803213
NA
NA
Decrease (50 %)
Investigational
30953674
DrugRepV_5424Losmapimod
NA
Chronic Obstructive Pulmonary Disease
Lassa virus
GA391
NA
NA
Decrease (50 %)
Investigational
30953674
DrugRepV_5425Losmapimod
NA
Chronic Obstructive Pulmonary Disease
Lassa virus
Josiah
NA
NA
Decrease (50 %)
Investigational
30953674
DrugRepV_5426ST-193
NA
NA
Lassa virus
LP
NA
NA
Decrease (50 %)
NA
30953674
DrugRepV_5427ST-193
NA
NA
Lassa virus
803213
NA
NA
Decrease (50 %)
NA
30953674
DrugRepV_5428ST-193
NA
NA
Lassa virus
GA391
NA
NA
Decrease (50 %)
NA
30953674
DrugRepV_5429ST-193
NA
NA
Lassa virus
Josiah
NA
NA
Decrease (50 %)
NA
30953674
DrugRepV_5431Gallium nitrate
NA
NA
Influenza virus
A/Puerto Rico/8/34 (PR8)
Pathway
Plaque reduction assay
Decrease (50 %)
Approved, Investigational
31244822
DrugRepV_5435Gallium nitrate
NA
NA
Influenza virus
pdm09A/Mexico/InDRE4487/2009
Pathway
Plaque reduction assay
Decrease (50 %)
Approved, Investigational
31244822
DrugRepV_5439Gallium nitrate
NA
NA
Influenza virus
A/Victoria/36/2011
Pathway
Plaque reduction assay
Decrease (50 %)
Approved, Investigational
31244822
DrugRepV_5443Gallium nitrate
NA
NA
Influenza virus
A/Puerto Rico/8/34 (PR8)
Pathway
Virus inhibition assay
Decrease (5.3 log)
Approved, Investigational
31244822
DrugRepV_5447Gallium nitrate
NA
NA
Influenza virus
pdm09A/Mexico/InDRE4487/2009
Pathway
Virus inhibition assay
Decrease (5.2 log)
Approved, Investigational
31244822
DrugRepV_5451Gallium nitrate
NA
NA
Influenza virus
A/Victoria/36/2011
Pathway
Virus inhibition assay
Decrease (5.5 log)
Approved, Investigational
31244822
DrugRepV_5477Nafamostat
NA
Blood vessel coagulation | Hemorrhagic lesions
SARS Coronavirus-2
nCoV- 2019BetaCoV/Wuhan/WIV04/2019
NA
qRT-PCR
Decrease (50 %)
Investigational
32020029
DrugRepV_5479Beta-D-N4-hydroxycytidine
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
Plaque assay
Decrease (50 %)
NA
31578288
DrugRepV_5482RK-33
NA
NA
Zika virus
Asian/Cook Islands/2014
NA
Plaque assay
Decrease (50 %)
NA
31936642
DrugRepV_5483RK-33
NA
NA
Zika virus
Asian/Cook Islands/2014
NA
qRT-PCR
Decrease (50 %)
NA
31936642
DrugRepV_5487Novobiocin
NA
Staphylococci infections
Zika virus
NA
NA
Flow cytometry
Decrease (50 %)
Approved, Investigational, Vet approved
31786251
DrugRepV_5495Winthrop
NA
NA
Ebola virus
NA
NA
Cell based assay
Decrease (50 %)
NA
31882748
DrugRepV_5496Winthrop
NA
NA
Ebola virus
NA
NA
Cell based assay
Decrease (50 %)
NA
31882748
DrugRepV_5497Winthrop
NA
NA
Ebola virus
NA
NA
Cell based assay
Decrease (50 %)
NA
31882748
DrugRepV_5498N-Desethylamodiaquine hydrochloride
NA
NA
Ebola virus
NA
NA
Cell based assay
Decrease (50 %)
NA
31882748
DrugRepV_5499N-Desethylamodiaquine hydrochloride
NA
NA
Ebola virus
NA
NA
Cell based assay
Decrease (50 %)
NA
31882748
DrugRepV_5500N-Desethylamodiaquine hydrochloride
NA
NA
Ebola virus
NA
NA
Cell based assay
Decrease (50 %)
NA
31882748
DrugRepV_5501Dihydroartimesinin
NA
Malaria
Ebola virus
NA
NA
Cell based assay
Decrease (50 %)
Experimental, Investigational
31882748
DrugRepV_5502Dihydroartimesinin
NA
Malaria
Ebola virus
NA
NA
Cell based assay
Decrease (50 %)
Experimental, Investigational
31882748
DrugRepV_5506Anthralin
NA
Psoriasis
Influenza virus
H1N1
Pathway
TCID50 assay
Decrease (99 %)
Approved
32132985
DrugRepV_5507Anthralin
NA
Psoriasis
Influenza virus
H1N1
Pathway
TCID50 assay
Decrease (99 %)
Approved
32132985
DrugRepV_5508Amuvatinib
NA
Cancer
Lassa virus
NA
NA
Gaussia luciferase (Gluc) Glow assay
Decrease (50 %)
Investigational
31786250
DrugRepV_5510Azoxystrobin
NA
Fungal infections
Lassa virus
NA
NA
Gaussia luciferase (Gluc) Glow assay
Decrease (50 %)
Experimental
31786250
DrugRepV_5511Buparvaquone
NA
NA
Lassa virus
NA
NA
Gaussia luciferase (Gluc) Glow assay
Decrease (50 %)
NA
31786250
DrugRepV_5512Dequalinium chloride hydrate
NA
NA
Lassa virus
NA
NA
Gaussia luciferase (Gluc) Glow assay
Decrease (50 %)
NA
31786250
DrugRepV_5513Manassantin A
NA
NA
Lassa virus
NA
NA
Gaussia luciferase (Gluc) Glow assay
Decrease (50 %)
NA
31786250
DrugRepV_5514Monensin sodium salt
NA
NA
Lassa virus
NA
NA
Gaussia luciferase (Gluc) Glow assay
Decrease (50 %)
Experimental, Vet approved
31786250
DrugRepV_5515Mubritinib
NA
Lung Neoplasm, Renal Neoplasm, Breast Neoplasm, Ovarian Neoplasm, and Pancreatic Neoplasm
Lassa virus
NA
NA
Gaussia luciferase (Gluc) Glow assay
Decrease (50 %)
Investigational
31786250
DrugRepV_5519Rotenone
NA
NA
Lassa virus
NA
NA
Gaussia luciferase (Gluc) Glow assay
Decrease (50 %)
Vet approved
31786250
DrugRepV_5520Spautin-1
NA
NA
Lassa virus
NA
NA
Gaussia luciferase (Gluc) Glow assay
Decrease (50 %)
NA
31786250
DrugRepV_5521Valinomycin
NA
NA
Lassa virus
NA
NA
Gaussia luciferase (Gluc) Glow assay
Decrease (50 %)
Experimental
31786250
DrugRepV_5523Tryptanthrin
NA
NA
Lassa virus
NA
NA
Gaussia luciferase (Gluc) Glow assay
Decrease (50 %)
NA
31786250
DrugRepV_5531JQ1
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5532RVX-208
NA
Diabetes, Atherosclerosis, and Coronary Artery Disease
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5533Silmitasertib
NA
Medulloblastoma
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Investigational
32353859
DrugRepV_5534TMCB
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5535Apicidin
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5538E-52862
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5539PD-144418
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5540RS-PPCC
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5541PB28
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5547H-89
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5548Merimepodib
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Investigational
32353859
DrugRepV_5552XL413
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5553CCT 365623
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5556ZINC1775962367
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5557ZINC4326719
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5558ZINC4511851
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5559ZINC95559591
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5560AC-55541
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5561AZ8838
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5563GB110
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5564S-verapamil
NA
Hypertension (high blood pressure) | Angina (chest pain) | Arrhythmia (heart rhythm disorders).
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved
32353859
DrugRepV_5565AZ3451
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5566ABBV-744
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5567dBET6
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5568MZ1
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5569CPI-0610
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5570Sapanisertib
NA
Tumor
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Investigational
32353859
DrugRepV_5572Zotatifin
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5573Verdinexor
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Investigational
32353859
DrugRepV_5576WDB002
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5577Sanglifehrin A
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Experimental
32353859
DrugRepV_5579Pevonedistat
NA
Lymphoma
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Investigational
32353859
DrugRepV_5580Ternatin 4
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_55814E2RCat
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5582Tomivosertib
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Investigational
32353859
DrugRepV_5583(2R,5S,11S,14S,17R,18R,21E)-2-(2-aminoethyl)-18-methoxy-11,17-dimethyl-14-(propan-2-yl)-3-oxa-9,12,15,28-tetraazatricyclo[21.3.1.1?,?]octacosa-1(26),21,23(27),24-tetraene-4,10,13,16-tetrone
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5584N-(5-{3-[(4-Hydroxyphenyl)sulfamoyl]-4-methoxyphenyl}-4-methyl-1,3-thiazol-2-yl)-2,2-dimethylpropanamide
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5585PS3061
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5586IHVR-19029
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5590Nafamostat
NA
Blood vessel coagulation | Hemorrhagic lesions
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Investigational
32353859
DrugRepV_5604Sunitinib-Erlotinib
NA
NA
Dengue virus
N124D/K128E
Pathway
NA
Increase
NA
28240606
DrugRepV_5605Sunitinib-Erlotinib
NA
NA
Dengue virus
N124D/K128E
Pathway
Real-time PCR
Decrease (11 Fold)
NA
28240606
DrugRepV_5615AMG-458
NA
Cancer
Dengue virus
New Guinea C
Pathway
Immunoflourescence assay
Decrease (60 %)
NA
28099856
DrugRepV_5616AMG-458
NA
Cancer
Dengue virus
New Guinea C
Pathway
Immunoflourescence assay
No significant effect (40 %)
NA
28099856
DrugRepV_5617AMG-458
NA
Cancer
Dengue virus
New Guinea C
Pathway
Immunoflourescence assay
No significant effect (5 %)
NA
28099856
DrugRepV_5708R1479
NA
NA
Dengue virus
MY-10340
Pathway
Plaque assay
Decrease (50 %)
NA
24257621
DrugRepV_5709Sunitinib-Erlotinib
NA
NA
Dengue virus
NA
Pathway
Survival assay
Increase
NA
29753658
DrugRepV_5710Sunitinib-Erlotinib
NA
NA
Dengue virus
NA
Pathway
Plaque assay
Decrease (>5 Log (pfu/g))
NA
29753658
DrugRepV_5714Carrageenan
NA
NA
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
NA
20973722
DrugRepV_5715Tannic Acid
NA
Cold sores | Diaper rash | Fever blisters | Poison ivy
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
Approved
20973722
DrugRepV_5716Tannic Acid
NA
Cold sores | Diaper rash | Fever blisters | Poison ivy
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
Approved
20973722
DrugRepV_5717Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
Investigational
20973722
DrugRepV_5718Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
Investigational
20973722
DrugRepV_5721BIBU 1361
NA
NA
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
NA
20973722
DrugRepV_5722BIBU 1361
NA
NA
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
NA
20973722
DrugRepV_57243-[(4-chloro-phenyl)-phenyl-methoxy]-tropane
NA
NA
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
NA
20973722
DrugRepV_57253-[(4-chloro-phenyl)-phenyl-methoxy]-tropane
NA
NA
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
NA
20973722
DrugRepV_5727H-89
NA
NA
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
NA
20973722
DrugRepV_5728H-89
NA
NA
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
NA
20973722
DrugRepV_5729MPP
NA
NA
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
NA
20973722
DrugRepV_5730MPP
NA
NA
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
NA
20973722
DrugRepV_5734W-9
NA
NA
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
NA
20973722
DrugRepV_5735W-9
NA
NA
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
NA
20973722
DrugRepV_5736AZ 10417808
NA
NA
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
NA
20973722
DrugRepV_5737AZ 10417808
NA
NA
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
NA
20973722
DrugRepV_5738Niguldipine
NA
NA
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
Experimental
20973722
DrugRepV_5739Niguldipine
NA
NA
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
Experimental
20973722
DrugRepV_57403a-bis-(4-fluorophenyl) Methoxytropane
NA
NA
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
NA
20973722
DrugRepV_5741LE 135
NA
NA
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
NA
20973722
DrugRepV_5742LE 135
NA
NA
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
NA
20973722
DrugRepV_5761Myriocin
NA
Bacterial infections
Dengue virus
NGC
Pathway
Plaque assay
No significant effect
NA
25313218
DrugRepV_5762Fenretinide-Myriocin
NA
NA
Dengue virus
NGC
Pathway
Plaque assay
Decrease (4 Logs)
NA
25313218
DrugRepV_5763Butylated Hydroxyanisole
NA
Antioxidant
Dengue virus
NGC
Pathway
Plaque assay
No significant effect
NA
25313218
DrugRepV_5764Fenretinide-Butylated Hydroxyanisole
NA
NA
Dengue virus
NGC
Pathway
Plaque assay
Decrease (1.5 Logs)
NA
25313218
DrugRepV_5766Fenretinide-Vitamin C
NA
NA
Dengue virus
NGC
Pathway
Plaque assay
Decrease (3 Logs)
NA
25313218
DrugRepV_5775Allantoin
NA
NA
Dengue virus
Singapore isolates
Pathway
Plaque assay
Decrease (78 %)
Approved
25251726
DrugRepV_5777Brucine
NA
NA
Dengue virus
Singapore isolates
Pathway
Plaque assay
Decrease (75 %)
NA
25251726
DrugRepV_5778Dicloxacillium Sodium
NA
Bacterial infections
Dengue virus
Singapore isolates
Pathway
Plaque assay
Decrease (72 %)
Approved
25251726
DrugRepV_5780Acrisorcin
NA
NA
Dengue virus
Singapore isolates
Pathway
Plaque assay
Decrease (72 %)
NA
25251726
DrugRepV_5782Oxantel Pamoate
NA
NA
Dengue virus
Singapore isolates
Pathway
Plaque assay
Decrease (68 %)
NA
25251726
DrugRepV_5787Lasalocid Sodium
NA
NA
Dengue virus
Singapore isolates
Pathway
Plaque assay
Decrease (62 %)
NA
25251726
DrugRepV_5803Lapachaone Alpha
NA
NA
Dengue virus
NA
Pathway
Immunoflourescence assay
Decrease (98.84 %)
NA
22155902
DrugRepV_5809Shikonin
NA
NA
Dengue virus
NA
Pathway
Immunoflourescence assay
Decrease (78.94 %)
NA
22155902
DrugRepV_5811Chelerythrine Chloride
NA
NA
Dengue virus
NA
Pathway
Immunoflourescence assay
Decrease (73.36 %)
NA
22155902
DrugRepV_5812Skimmianine
NA
NA
Dengue virus
NA
Pathway
Immunoflourescence assay
Decrease (61.96 %)
NA
22155902
DrugRepV_5816Tunicamycin B
NA
Bacterial infections
Dengue virus
NA
Pathway
Immunoflourescence assay
Decrease (55.01 %)
Experimental
22155902
DrugRepV_5817Acivicin
NA
Cancer
Dengue virus
NA
Pathway
Immunoflourescence assay
Decrease (54.32 %)
Phase I
22155902
DrugRepV_5821Gitoxigenin
NA
NA
Dengue virus
NA
Pathway
Immunoflourescence assay
Decrease (49.01 %)
NA
22155902
DrugRepV_5822Kainic Acid
NA
Neuroexcitatory
Dengue virus
NA
Pathway
Immunoflourescence assay
Decrease (48.87 %)
NA
22155902
DrugRepV_5825Diacetoxyscirpenol
NA
NA
Dengue virus
NA
Pathway
Immunoflourescence assay
Decrease (45.55 %)
NA
22155902
DrugRepV_5826Austricin
NA
NA
Dengue virus
NA
Pathway
Immunoflourescence assay
Decrease (45.01 %)
NA
22155902
DrugRepV_5827Valinomycin
NA
NA
Dengue virus
NA
Pathway
Immunoflourescence assay
Decrease (43.34 %)
Experimental
22155902
DrugRepV_5828Thapsigargin
NA
NA
Dengue virus
NA
Pathway
Immunoflourescence assay
Decrease (42.9 %)
NA
22155902
DrugRepV_5829Strophanthidin Acetate
NA
NA
Dengue virus
NA
Pathway
Immunoflourescence assay
Decrease (41.96 %)
NA
22155902
DrugRepV_5831Echinomycin
NA
Bacterial infections
Dengue virus
NA
Pathway
Immunoflourescence assay
Decrease (41.52 %)
NA
22155902
DrugRepV_5832Chromomycin A3
NA
NA
Dengue virus
NA
Pathway
Immunoflourescence assay
Decrease (40.87 %)
NA
22155902
DrugRepV_5835Strophanthidin Acetate
NA
NA
Dengue virus
NA
Pathway
Immunoflourescence assay
Decrease (50 %)
NA
22155902
DrugRepV_5839Strophanthidin Acetate
NA
NA
Dengue virus
NA
Pathway
Immunoflourescence assay
Decrease (98 %)
NA
22155902
DrugRepV_5843Strophanthidin Acetate
NA
NA
Dengue virus
NA
Pathway
Plaque assay
Decrease (5 Logs reduction)
NA
22155902
DrugRepV_5890Quinacrine Mustard
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Dengue virus
NA
Pathway
Plaque assay
Decrease (> 99 %)
Experimental
24680954
DrugRepV_5908Quinacrine Mustard
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Dengue virus
NA
Pathway
Plaque assay
Decrease (50 %)
Experimental
24680954
DrugRepV_5969ZX-2401
NA
Rhinovirus 1A | Rhinovirus 30 | Rhinovirus 13 | Rhinovirus 8 | Rhinovirus 2
Dengue virus
New Guinea
Pathway
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
16199098
DrugRepV_5975Deoxynojirimycin
NA
NA
Dengue virus
FGA/89
Pathway
Focus immunoassay
Decrease (80 %)
NA
10590151
DrugRepV_6001U18666A
NA
NA
Dengue virus
New Guinea
Pathway
Plaque assay
Decrease (3 Log (pfu/ml))
NA
22146564
DrugRepV_6002U18666A
NA
NA
Dengue virus
Replicon systen
Pathway
Luciferase reporter assay
Decrease (50 %)
NA
22146564
DrugRepV_6003U18666A
NA
NA
Dengue virus
Replicon systen
Pathway
Luciferase reporter assay
Decrease (50 %)
NA
22146564
DrugRepV_6006Chebulagic Acid
NA
Immunosuppressive and hepatoprotective
Dengue virus
16681
Pathway
Plaque assay
Decrease (50 %)
NA
23924316
DrugRepV_6008Chebulagic Acid
NA
Immunosuppressive and hepatoprotective
Dengue virus
16681
Pathway
Plaque assay
Decrease (100 %)
NA
23924316
DrugRepV_6013N-nonyl-deoxynojirimycin
NA
NA
Dengue virus
PL046
Pathway
FITC- assay
Decrease (98 %)
NA
11907199
DrugRepV_6014N-nonyl-deoxynojirimycin
NA
NA
Dengue virus
PL046
Pathway
Plaque assay
Decrease (4 Log)
NA
11907199
DrugRepV_6015N-nonyl-deoxynojirimycin
NA
NA
Dengue virus
PL046
Pathway
Western blot
Decrease (Decrease Band Intensity)
NA
11907199
DrugRepV_6016N-nonyl-deoxynojirimycin
NA
NA
Dengue virus
PL046
Pathway
Western blot
Decrease (Decrease Band Intensity)
NA
11907199
DrugRepV_6017N-nonyl-deoxynojirimycin
NA
NA
Dengue virus
PL046
Pathway
Real-time PCR
Decrease (Decrease Ct Value)
NA
11907199
DrugRepV_6018N-nonyl-deoxynojirimycin
NA
NA
Dengue virus
PL046
Pathway
Real-time PCR
Decrease (Decrease Ct Value)
NA
11907199
DrugRepV_60384-(5-(4-Fluorophenyl)-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60394-(5-(2-chlorophenyl)-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60404-(5-(3-chlorophenyl)-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60414-(3-Phenyl-5-(o-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60424-(3-Phenyl-5-(p-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60434-(3-(4-phenoxyphenyl)-5-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60444-(5-(2-fluorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60454-(5-(3-fluorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60464-(5-(4-fluorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60474-(5-(2-chlorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60484-(5-(3-chlorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60494-(5-(4-chlorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60504-(3-(4-phenoxyphenyl)-5-(o-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60514-(3-(4-phenoxyphenyl)-5-(m-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60524-(3-(4-phenoxyphenyl)-5-(p-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60534-(3-(4-(benzyloxy)phenyl)-5-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60544-(3-(4-(benzyloxy)phenyl)-5-(2-fluorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60554-(3-(4-(benzyloxy)phenyl)-5-(3-fluorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60564-(3-(4-(benzyloxy)phenyl)-5-(4-fluorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60574-(3-(4-(benzyloxy)phenyl)-5-(2-chlorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60584-(3-(4-(benzyloxy)phenyl)-5-(3-chlorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60594-(3-(4-(benzyloxy)phenyl)-5-(4-chlorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60604-(3-(4-(benzyloxy)phenyl)-5-(o-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60614-(3-(4-(benzyloxy)phenyl)-5-(m-tolyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_60624-(3-(4-(benzyloxy)phenyl)-5-(p-tolyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Dengue virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_6064N2-(4-fluorophenyl)-N3-(4-methyl-2-(3-methyl-1H-pyrazol- 5-yl)phenyl) pyrazine-2,3 dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6065N2-(4-methyl-2-(3-methyl-1H-pyrazol-5-yl)phenyl)-N3-(p- tolyl)pyrazine-2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6066N2-(4-fluorophenyl)-N3-(4-methyl-2-(thiophen-2-yl)phenyl) pyrazine-2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6067N2-(4-methyl-2-(thiophen-2-yl)phenyl)-N3-(p-tolyl) pyrazine-2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6068N2-(4-fluorophenyl)-N3-(4-methyl-2-(5-methylthiophen-2-yl)phenyl)pyrazine-2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6069N2-(4-methyl-2-(5-methylthiophen-2-yl)phenyl)-N3-(p- tolyl)pyrazine-2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6070N2-(4-fluorophenyl)-N3-(4-methyl-2-(thiophen-3-yl) phenyl)pyrazine-2,3- dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6071N2-(4-methyl-2-(thiophen-3-yl)phenyl)-N3-(p-tolyl) pyrazine-2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6072N2-(4-fluorophenyl)-N3-(2-(thiophen-3-yl)benzyl)pyrazine- 2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6073N2-(2-(thiophen-3-yl)benzyl)-N3-(p-tolyl)pyrazine-2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6074N2-(4-fluorophenyl)-N3-(4-(thiophen-3-yl)benzyl)pyrazine-2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6075N2-(4-(thiophen-3-yl)benzyl)-N3-(p-tolyl)pyrazine-2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6076N2-(4-fluorophenyl)-N3-(2-(3-methyl-1H-pyrazol-5-yl) phenyl)pyrazine-2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6077N2-(2-(3-methyl-1H-pyrazol-5-yl)phenyl)-N3-(p-tolyl) pyrazine-2,3-di-carboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6078N1-(4-fluorophenyl)-N2-(4-methyl-2-(3-methyl-1H-pyrazol-5-yl)phenyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6079N1-(4-fluorophenyl)-N2-(4-methyl-2-(thiophen-2-yl) phenyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6080N1-(4-methyl-2-(3-methyl-1H-pyrazol-5-yl)phenyl)-N2-(p- tolyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6081N1-(4-methyl-2-(thiophen-2-yl)phenyl)-N2-(p-tolyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6082N1-(4-methyl-2-(5-methylthiophen-2-yl)phenyl)-N2-(p- tolyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6083N1-(4-fluorophenyl)-N2-(4-methyl-2-(5-methylthiophen-2- yl)phenyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6084N1-(4-methyl-2-(thiophen-3-yl)phenyl)-N2-(p-tolyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6085N1-(4-fluorophenyl)-N2-(4-methyl-2-(thiophen-3-yl) phenyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6086N1-(4-fluorophenyl)-N2-(2-(thiophen-3-yl)benzyl) phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6087N1-(2-(thiophen-3-yl)benzyl)-N2-(p-tolyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6088N1-(4-fluorophenyl)-N2-(4-(thiophen-3-yl)benzyl) phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6089N1-(4-(thiophen-3-yl)benzyl)-N2-(p-tolyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6090N1-(4-fluorophenyl)-N2-(2-(3-methyl-1H-pyrazol-5-yl) phenyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6091N1-(2-(3-methyl-1H-pyrazol-5-yl)phenyl)-N2-(p-tolyl) phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_60922-(4-fluorobenzamido)-N-(4-methyl-2-(thiophen-3-yl) phenyl)benzamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_60932-(4-fluorobenzamido)-N-(4-methyl-2-(5-methylthiophen- 2-yl)phenyl)benzamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_60942-(4-fluorobenzamido)-N-(4-methyl-2-(pyridin-4-yl)phenyl) benzamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_60952-(4-fluorobenzamido)-N-(4-methyl-2-(pyridin-3-yl)phenyl) benzamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6097SA-3
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
qRT-PCR
Decrease (50 %)
NA
20837762
DrugRepV_6098SA-11
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
qRT-PCR
Decrease (50 %)
NA
20837762
DrugRepV_6099SA-17
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
qRT-PCR
Decrease (50 %)
NA
20837762
DrugRepV_6100SA-17
NA
NA
Dengue virus
New Guinea C
Pathway
qRT-PCR
Decrease (50 %)
NA
20837762
DrugRepV_6101CM-10-18
NA
NA
Dengue virus
New Guinea C
Pathway
MTT assay
Decrease (50 %)
NA
23578725
DrugRepV_6102IHVR11029
NA
NA
Dengue virus
New Guinea C
Pathway
MTT assay
Decrease (50 %)
NA
23578725
DrugRepV_6103IHVR17028
NA
NA
Dengue virus
New Guinea C
Pathway
MTT assay
Decrease (50 %)
NA
23578725
DrugRepV_6104IHVR19029
NA
NA
Dengue virus
New Guinea C
Pathway
MTT assay
Decrease (50 %)
NA
23578725
DrugRepV_6105BCX4430
NA
Ebola virus
Dengue virus
New Guinea C
Pathway
RT-PCR
Decrease (50 %)
Investigational
24590073
DrugRepV_6106IHVR-19029
NA
NA
Dengue virus
NA
Pathway
qRT-PCR
Decrease (50 %)
NA
29253498
DrugRepV_6107Coumarin A
NA
NA
Dengue virus
NG
Pathway
RT-PCR
Decrease (50 %)
NA
28100218
DrugRepV_6108Coumarin B
NA
NA
Dengue virus
NG
Pathway
RT-PCR
Decrease (50 %)
NA
28100218
DrugRepV_6109Lupeol Acetate 26SK001
NA
NA
Dengue virus
NG
Pathway
RT-PCR
Decrease (50 %)
NA
28100218
DrugRepV_6110Voacangine 26SK002
NA
NA
Dengue virus
NG
Pathway
RT-PCR
Decrease (50 %)
NA
28100218
DrugRepV_6111Coumarin A
NA
NA
Dengue virus
NG
Pathway
RT-PCR
Decrease (37.1 %)
NA
28100218
DrugRepV_6112Coumarin B
NA
NA
Dengue virus
NG
Pathway
RT-PCR
Decrease (99.25 %)
NA
28100218
DrugRepV_6113Lupeol Acetate 26SK001
NA
NA
Dengue virus
NG
Pathway
RT-PCR
Decrease (23 %)
NA
28100218
DrugRepV_6114Voacangine 26SK002
NA
NA
Dengue virus
NG
Pathway
RT-PCR
Decrease (23 %)
NA
28100218
DrugRepV_6117FGI-106
NA
NA
Dengue virus
NA
Pathway
Flow cytometry
Decrease (50 %)
NA
19523489
DrugRepV_6118FGI-106
NA
NA
Dengue virus
NA
Pathway
Flow cytometry
Decrease (50 %)
NA
19523489
DrugRepV_6119FGI-106
NA
NA
Dengue virus
NA
Pathway
Flow cytometry
Decrease (50 %)
NA
19523489
DrugRepV_6120FGI-106
NA
NA
Dengue virus
NA
Pathway
Flow cytometry
Decrease (50 %)
NA
19523489
DrugRepV_6121Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Dengue virus
NA
Pathway
Plaque assay
Decrease (50 %)
Investigational
27889529
DrugRepV_6123GSK369796
NA
NA
Dengue virus
NA
Pathway
Plaque assay
Decrease (50 %)
NA
27889529
DrugRepV_6124Tomatidine
NA
NA
Dengue virus
16681
Pathway
MTT assay
Decrease (50 %)
NA
30468746
DrugRepV_6125Tomatidine
NA
NA
Dengue virus
16007
Pathway
MTT assay
Decrease (50 %)
NA
30468746
DrugRepV_6126Tomatidine
NA
NA
Dengue virus
H87
Pathway
MTT assay
Decrease (50 %)
NA
30468746
DrugRepV_6127Tomatidine
NA
NA
Dengue virus
1036
Pathway
MTT assay
Decrease (50 %)
NA
30468746
DrugRepV_6130VGTI-A3
NA
NA
Dengue virus
New Guinea C
Pathway
Focus forming assay
Decrease (90 %)
NA
29709563
DrugRepV_6131VGTI-A3-03
NA
NA
Dengue virus
New Guinea C
Pathway
Focus forming assay
Decrease (90 %)
NA
29709563
DrugRepV_6132Ribavirin Nucleobase
NA
NA
Dengue virus
New Guinea C
Pathway
DENV replicon assay
Decrease (50 %)
NA
29672522
DrugRepV_6133Mizoribine Nucleobase
NA
NA
Dengue virus
New Guinea C
Pathway
DENV replicon assay
Decrease (50 %)
NA
29672522
DrugRepV_6134T-1105
NA
Zika virus
Dengue virus
New Guinea C
Pathway
DENV replicon assay
Decrease (50 %)
NA
29672522
DrugRepV_6135Diaminopurine
NA
NA
Dengue virus
New Guinea C
Pathway
DENV replicon assay
Decrease (50 %)
NA
29672522
DrugRepV_6140T-1106
NA
Yellow Fever virus
Dengue virus
New Guinea C
Pathway
DENV replicon assay
Decrease (50 %)
NA
29672522
DrugRepV_6141Diaminopurine Riboside
NA
NA
Dengue virus
New Guinea C
Pathway
DENV replicon assay
Decrease (50 %)
NA
29672522
DrugRepV_6142T-1105
NA
Zika virus
Dengue virus
New Guinea C
Pathway
Titer reduction assay
Decrease (50 %)
NA
29672522
DrugRepV_6143T-1106
NA
Yellow Fever virus
Dengue virus
New Guinea C
Pathway
Titer reduction assay
Decrease (50 %)
NA
29672522
DrugRepV_61445,7-dichloro-2-(propan-2-yl)quinolin-8-ol
NA
NA
Dengue virus
NA
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
29547522
DrugRepV_61455,7-dichloro-2-(2-methylpropyl)quinolin-8-ol
NA
NA
Dengue virus
NA
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
29547522
DrugRepV_6150AR-12
NA
Solid Tumors and Lymphoma
Dengue virus
NA
Pathway
qRT-PCR
Decrease
Phase I
28666323
DrugRepV_6151AR-12
NA
Solid Tumors and Lymphoma
Dengue virus
NA
Pathway
qRT-PCR
Decrease
Phase I
28666323
DrugRepV_6152AR-12
NA
Solid Tumors and Lymphoma
Dengue virus
NA
Pathway
qRT-PCR
Decrease
Phase I
28666323
DrugRepV_6153AR-12
NA
Solid Tumors and Lymphoma
Dengue virus
NA
Pathway
qRT-PCR
Decrease
Phase I
28666323
DrugRepV_6154Schisandrin A
NA
NA
Dengue virus
NA
Pathway
qRT-PCR
Decrease (50 %)
NA
28338050
DrugRepV_6155Schisandrin B
NA
NA
Dengue virus
NA
Pathway
qRT-PCR
Decrease (50 %)
NA
28338050
DrugRepV_6156Schisandrin C
NA
NA
Dengue virus
NA
Pathway
qRT-PCR
Decrease (50 %)
NA
28338050
DrugRepV_6157Schisandrin A
NA
NA
Dengue virus
NA
Pathway
Survival assay
Decrease
NA
28338050
DrugRepV_61605hydroxyl-6,7,3,4,5-pentamethoxyflavone
NA
NA
Dengue virus
16681
Pathway
MTT assay
Decrease (50 %)
NA
22068705
DrugRepV_61615,3-dihydroxy-6,7,4,5-tetramethoxyflavone
NA
NA
Dengue virus
16681
Pathway
MTT assay
Decrease (50 %)
NA
22068705
DrugRepV_6162BZ-TRP-TSC
NA
NA
Dengue virus
NA
Pathway
MTT assay
Decrease (85 %)
NA
27490721
DrugRepV_6163BZ-TRP-TSC
NA
NA
Dengue virus
NA
Pathway
MTT assay
Decrease (76 %)
NA
27490721
DrugRepV_6164BZ-TRP-TSC
NA
NA
Dengue virus
NA
Pathway
MTT assay
Decrease (65 %)
NA
27490721
DrugRepV_6165BZ-TRP-TSC
NA
NA
Dengue virus
NA
Pathway
MTT assay
Decrease (76 %)
NA
27490721
DrugRepV_6166Thiosemicarbazide
NA
NA
Dengue virus
NA
Pathway
Immunoflourescence assay
Decrease
NA
27490721
DrugRepV_61694-{1-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]-3-(4-methoxyphenyl)-4,5-dihydro-1H-pyrazol-5-yl}-2-methoxyphenol
NA
NA
Dengue virus
NA
Pathway
CPE reduction assay
Decrease (50 %)
NA
25791449
DrugRepV_61704-[1-(4-{[1,1-biphenyl]-4-yl}-1,3-thiazol-2-yl)-5-phenyl-4,5-dihydro-1H-pyrazol-3-yl]phenol
NA
NA
Dengue virus
NA
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
25791449
DrugRepV_61714-[1-(4-{[1,1-biphenyl]-4-yl}-1,3-thiazol-2-yl)-3-(4-methoxyphenyl)-4,5-dihydro-1H-pyrazol-5-yl]-2-methoxyphenol
NA
NA
Dengue virus
NA
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
25791449
DrugRepV_61724-[1-(4-{[1,1-biphenyl]-4-yl}-1,3-thiazol-2-yl)-3-(4-methoxyphenyl)-4,5-dihydro-1H-pyrazol-5-yl]phenol
NA
NA
Dengue virus
NA
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
25791449
DrugRepV_61734-[(1E)-1-{2-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]hydrazin-1-ylidene}ethyl]phenol
NA
NA
Dengue virus
NA
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
25791449
DrugRepV_61744-{[1,1-biphenyl]-4-yl}-2-[(2E)-2-[1-(4-methoxyphenyl)ethylidene]hydrazin-1-yl]-1,3-thiazole
NA
NA
Dengue virus
NA
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
25791449
DrugRepV_61754-{[1,1-biphenyl]-4-yl}-2-[(2E)-2-[1-(4-nitrophenyl)ethylidene]hydrazin-1-yl]-1,3-thiazole
NA
NA
Dengue virus
NA
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
25791449
DrugRepV_61764-{[1,1-biphenyl]-4-yl}-2-[(2E)-2-(phenylmethylidene)hydrazin-1-yl]-1,3-thiazole
NA
NA
Dengue virus
NA
Pathway
CPE reduction assay
Decrease (50 %)
NA
25791449
DrugRepV_61774-[(E)-[2-(4-{[1,1-biphenyl]-4-yl}-1,3-thiazol-2-yl)hydrazin-1-ylidene]methyl]phenol
NA
NA
Dengue virus
NA
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
25791449
DrugRepV_6179(1S,2R,3S,4S)-3,4-dihydroxy-2-(hydroxymethyl)-1-[(2S,3S,4R,5R,6S)-2,4,5,6,7-pentahydroxy-3-(sulfonatooxy)heptyl]thiolan-1-ium
NA
NA
Dengue virus
ThNH-7/93
Pathway
Fluorescent focus-forming assay
Decrease (50 %)
NA
22784856
DrugRepV_6180(1R,2R,3S,4S)-1-[(2S,3S,4R,5R,6S)-2,3,4,5,6,7-hexahydroxyheptyl]-3,4-dihydroxy-2-(hydroxymethyl)thiolan-1-ium chloride
NA
NA
Dengue virus
ThNH-7/93
Pathway
Fluorescent focus-forming assay
Decrease (50 %)
NA
22784856
DrugRepV_61812 -C-methyladenosine
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
Cell proliferation assay
Decrease (50 %)
NA
17662475
DrugRepV_6184UV-4B
NA
NA
Dengue virus
NA
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
26946111
DrugRepV_6185UV-4B
NA
NA
Dengue virus
16681
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
26946111
DrugRepV_6186UV-4B
NA
NA
Dengue virus
NA
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
26946111
DrugRepV_6187UV-4B
NA
NA
Dengue virus
NA
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
26946111
DrugRepV_6193STK332077
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
26807547
DrugRepV_6194STK529754
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
26807547
DrugRepV_6195STK530661
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
26807547
DrugRepV_6196(2S)-6-amino-2-[(2S)-6-amino-2-[(2S)-2-[(2S,3R)-2-[(2S)-2-acetamido-5-[(prop-1-en-2-yl)amino]pentanamido]-3-hydroxybutanamido]-3-hydroxypropanamido]hexanamido]-N-[(1S)-4-carbamimidamido-1-carbamoylbutyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Cell based assay
Decrease (5.31 ± 0.06 Log PFU/ml)
NA
25823617
DrugRepV_6197(E)-N-[(E)-({4-[(E)-{[(diaminomethylidene)amino]imino}methyl]phenyl}methylidene)amino]ethanimidamide
NA
NA
Dengue virus
NA
Pathway
Cell based assay
Decrease (5.37 ± 0.15 Log PFU/ml)
NA
25823617
DrugRepV_6198(2S)-6-amino-N-[(1S)-4-carbamimidamido-1-[(5-carbamimidamido-1-oxopentan-2-yl)carbamoyl]butyl]-2-[(2S)-2-(phenylformamido)propanamido]hexanamide
NA
NA
Dengue virus
NA
Pathway
Cell based assay
Decrease (5.38 ± 0.10 Log PFU/ml)
NA
25823617
DrugRepV_61997-[(phenylamino)(pyridin-2-yl)methyl]quinolin-8-ol
NA
NA
Dengue virus
NA
Pathway
Cell based assay
Decrease (5.34 ± 0.15 Log PFU/ml)
NA
25823617
DrugRepV_62001,8-dihydroxy-4,5-dinitro-9,10-dihydroanthracene-9,10-dione
NA
NA
Dengue virus
NA
Pathway
Cell based assay
Decrease (50 %)
NA
25823617
DrugRepV_62014-carbamimidamidophenyl 4-carbamimidamidobenzoate
NA
NA
Dengue virus
NA
Pathway
Cell based assay
Decrease (5.30 ± 0.10 Log PFU/ml)
NA
25823617
DrugRepV_62024-nitrophenyl 4-carbamimidamidobenzoate
NA
NA
Dengue virus
NA
Pathway
Cell based assay
Decrease (5.41 ± 0.17 Log PFU/ml)
NA
25823617
DrugRepV_6203(2E)-2-cyano-3-(4-hydroxyphenyl)prop-2-enamide
NA
NA
Dengue virus
NA
Pathway
Cell based assay
Decrease (5.46 ± 0.15 Log PFU/ml)
NA
25823617
DrugRepV_62044-[2-(2,4-dinitrophenyl)diazen-1-yl]naphthalen-1-ol
NA
NA
Dengue virus
NA
Pathway
Cell based assay
Decrease (5.49 ± 0.26 Log PFU/ml)
NA
25823617
DrugRepV_62051-ethyl-2-[(1E)-3-[(2Z)-1-ethyl-1H,2H-naphtho[1,2-d][1,3]oxazol-2-ylidene]prop-1-en-1-yl]naphtho[1,2-d][1,3]oxazol-1-ium
NA
NA
Dengue virus
NA
Pathway
Cell based assay
Decrease (50 %)
NA
25823617
DrugRepV_6206(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-(phenylformamido)pentanamido]-N-[(1R)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Cell based assay
Decrease (5.35 ± 0.21 Log PFU/ml)
NA
25823617
DrugRepV_6207(4R,7S,10S,13S,16S,22R)-22-amino-10,16-bis(4-aminobutyl)-13-(3-carbamimidamidopropyl)-7-(hydroxymethyl)-6,9,12,15,18,21-hexaoxo-1,2-dithia-5,8,11,14,17,20-hexaazacyclotricosane-4-carboxylic acid
NA
NA
Dengue virus
NA
Pathway
Cell based assay
Decrease (5.46 ± 0.35 Log PFU/ml)
NA
25823617
DrugRepV_62081-[N-(2-ethylhexyl)carbamimidamido]-N-(6-{N-[N-(2-ethylhexyl)carbamimidoyl]carbamimidamido}hexyl)methanimidamide
NA
NA
Dengue virus
NA
Pathway
Cell based assay
Decrease (5.62 ± 0.20 Log PFU/ml)
NA
25823617
DrugRepV_6209(1R,2R,4S,5S,8R,10E,12S,13S,14E,16E,20R,21R,24S)-6-[(2S)-butan-2-yl]-21,24-dihydroxy-12-{[(2R,4S,6S)-5-{[(2S,4S,5S,6S)-5-hydroxy-4-methoxy-6-methyloxan-2-yl]oxy}-4-methoxy-6-methyloxan-2-yl]oxy}-5,11,13,22-tetramethyl-3,7,19-trioxaspiro[oxane-2,6-tet
NA
NA
Dengue virus
NA
Pathway
Cell based assay
Decrease
NA
25823617
DrugRepV_6210(1R,2R,4S,5S,6S,8R,10E,13S,14E,16E,20R,21E,24S)-6-cyclohexyl-24-hydroxy-12-{[(2R,4S,5S,6S)-5-hydroxy-4-methoxy-6-methyloxan-2-yl]oxy}-21-(hydroxyimino)-5,11,13,22-tetramethyl-3,7,19-trioxaspiro[oxane-2,6-tetracyclo[15.6.1.14,8.0
NA
NA
Dengue virus
NA
Pathway
Cell based assay
Decrease
NA
25823617
DrugRepV_62212-chloro-10-(prop-2-en-1-yl)-9,10-dihydroacridin-9-one
NA
NA
Dengue virus
Hawaii
Pathway
Virus yield inhibition assay
Decrease (50 %)
NA
25908170
DrugRepV_62222-chloro-10-(prop-2-en-1-yl)-9,10-dihydroacridin-9-one
NA
NA
Dengue virus
New Guinea C
Pathway
Virus yield inhibition assay
Decrease (50 %)
NA
25908170
DrugRepV_62232-chloro-10-(prop-2-en-1-yl)-9,10-dihydroacridin-9-one
NA
NA
Dengue virus
H87
Pathway
Virus yield inhibition assay
Decrease (50 %)
NA
25908170
DrugRepV_62242-chloro-10-(prop-2-en-1-yl)-9,10-dihydroacridin-9-one
NA
NA
Dengue virus
8124
Pathway
Virus yield inhibition assay
Decrease (50 %)
NA
25908170
DrugRepV_62276-MPTF
NA
NA
Dengue virus
16681
Pathway
Plaque assay
Decrease (2.05 * 106 pfu/ml)
NA
7201778
DrugRepV_6228Sinefungin
NA
NA
Dengue virus
NA
Pathway
2-O-MTase assays
Decrease (50 %)
Experimental
23769894
DrugRepV_6229AdoHcy
NA
NA
Dengue virus
NA
Pathway
2-O-MTase assays
Decrease (50 %)
Experimental
23769894
DrugRepV_6230Aurintricarboxylic acid
NA
NA
Dengue virus
NA
Pathway
2-O-MTase assays
Decrease (50 %)
NA
23769894
DrugRepV_62315,50 -Methylene-disalicylic acid
NA
NA
Dengue virus
NA
Pathway
2-O-MTase assays
Decrease (50 %)
NA
23769894
DrugRepV_6232YK 51
NA
NA
Dengue virus
New Guinea C
Pathway
CPE inhibition assay
Decrease (92 %)
NA
20567498
DrugRepV_6233YK 73
NA
NA
Dengue virus
New Guinea C
Pathway
CPE inhibition assay
Decrease (90 %)
NA
20567498
DrugRepV_6234YK 73x
NA
NA
Dengue virus
New Guinea C
Pathway
CPE inhibition assay
Decrease (91 %)
NA
20567498
DrugRepV_6235YK 101
NA
NA
Dengue virus
New Guinea C
Pathway
CPE inhibition assay
Decrease (94 %)
NA
20567498
DrugRepV_6236YK 38
NA
NA
Dengue virus
New Guinea C
Pathway
CPE inhibition assay
Decrease (83 %)
NA
20567498
DrugRepV_6237YK 38
NA
NA
Dengue virus
New Guinea C
Pathway
Virus plaque assay
Decrease (3.2 * 103 pfu/ml)
NA
20567498
DrugRepV_6238YK 51
NA
NA
Dengue virus
New Guinea C
Pathway
Virus plaque assay
Decrease (3.4 * 103 pfu/ml)
NA
20567498
DrugRepV_6239YK 73
NA
NA
Dengue virus
New Guinea C
Pathway
Virus plaque assay
Decrease (3.5 * 103 pfu/ml)
NA
20567498
DrugRepV_6240YK 73x
NA
NA
Dengue virus
New Guinea C
Pathway
Virus plaque assay
Decrease (2.8 * 103 pfu/ml)
NA
20567498
DrugRepV_6241YK 101
NA
NA
Dengue virus
New Guinea C
Pathway
Virus plaque assay
Decrease (2.6 * 103 pfu/ml)
NA
20567498
DrugRepV_62429-benzyl-6-[(1-methyl-4-nitro-4,5-dihydro-1H-imidazol-5-yl)methyl]-9H-purin-2-amine
NA
NA
Dengue virus
NA
Pathway
Luciferase assay
Decrease (50 %)
NA
19053243
DrugRepV_62432-{[(3-nitrophenyl)methyl]sulfanyl}-9H-purin-6-ol
NA
NA
Dengue virus
NA
Pathway
Luciferase assay
Decrease (50 %)
NA
19053243
DrugRepV_62442-({[2-(4-chlorophenyl)-1,3-thiazol-4-yl]methyl}sulfanyl)aniline
NA
NA
Dengue virus
NA
Pathway
Luciferase assay
Decrease (50 %)
NA
19053243
DrugRepV_62451-(4-Bromophenyl)-2-(ethylamino)-2-methylpropyl hydrodisulfide
NA
NA
Dengue virus
NA
Pathway
Luciferase assay
Decrease (50 %)
NA
19053243
DrugRepV_6246N-[4-(4-aminobenzenesulfonyl)phenyl]pyridine-3-carboxamide
NA
NA
Dengue virus
NA
Pathway
Luciferase assay
Decrease (50 %)
NA
19053243
DrugRepV_62472-(2-{2-[(2E,5E)-3-ethyl-4-oxo-5-[(phenylamino)methylidene]-1,3-thiazolidin-2-ylidene]hydrazin-1-yl}-1,3-thiazol-5-yl)-N-(2-methylphenyl)acetamide
NA
NA
Dengue virus
NA
Pathway
Luciferase assay
Decrease (50 %)
NA
19053243
DrugRepV_6248(2E)-3-(3,4-dichlorophenyl)-1-[2-(3,5-diphenyl-1H-pyrazol-1-yl)-4-methyl-1,3-thiazol-5-yl]prop-2-en-1-one
NA
NA
Dengue virus
NA
Pathway
Luciferase assay
Decrease (50 %)
NA
19053243
DrugRepV_62492-{[5-(4-{[(4-chlorophenyl)methylidene]amino}phenyl)-1,3,4-oxadiazol-2-yl]sulfanyl}-N-(2-nitrophenyl)acetamide
NA
NA
Dengue virus
NA
Pathway
Luciferase assay
Decrease (50 %)
NA
19053243
DrugRepV_62501,3-bis({4-[(1E)-1-(carbamimidamidoimino)ethyl]phenyl})urea
NA
NA
Dengue virus
NA
Pathway
Luciferase assay
Decrease (50 %)
NA
19053243
DrugRepV_62513-{[(4-chlorophenyl)methyl]sulfanyl}-5-[(4,5-dichloro-1H-imidazol-1-yl)methyl]-4-methyl-4H-1,2,4-triazole
NA
NA
Dengue virus
NGC
Pathway
Plaque assay
Decrease (50 %)
NA
19781577
DrugRepV_62522-({[5-(5-methyl-3-phenyl-1,2-oxazol-4-yl)-1,2,4-oxadiazol-3-yl]methyl}sulfanyl)pyridin-1-ium-1-olate
NA
NA
Dengue virus
NGC
Pathway
Plaque assay
Decrease (50 %)
NA
19781577
DrugRepV_62531-(4-chlorophenyl)-2-({5-[(4,5-dichloro-1H-imidazol-1-yl)methyl]-1,3,4-oxadiazol-2-yl}sulfanyl)ethan-1-one
NA
NA
Dengue virus
NGC
Pathway
Plaque assay
Decrease (50 %)
NA
19781577
DrugRepV_62541-(2-chlorophenyl)-3-{2-[(4,5-dichloro-1H-imidazol-1-yl)methyl]-1,3-thiazol-4-yl}urea
NA
NA
Dengue virus
NGC
Pathway
Plaque assay
Decrease (50 %)
NA
19781577
DrugRepV_62552-chloro-6-(4-chlorophenoxy)-4-{4-methyl-5-[(1E)-1-(2-phenylhydrazin-1-ylidene)ethyl]-1,3-thiazol-2-yl}pyridine
NA
NA
Dengue virus
NGC
Pathway
Plaque assay
Decrease (50 %)
NA
19781577
DrugRepV_6260HHA
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
Flow cytometry
Decrease (50 %)
NA
19264337
DrugRepV_6261GNA
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
Flow cytometry
Decrease (50 %)
NA
19264337
DrugRepV_6262UDA
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
Flow cytometry
Decrease (50 %)
NA
19264337
DrugRepV_6264Mannan
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
Flow cytometry
Decrease (50 %)
NA
19264337
DrugRepV_6265HHA
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
RT-PCR
Decrease (50 %)
NA
19264337
DrugRepV_6266GNA
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
RT-PCR
Decrease (50 %)
NA
19264337
DrugRepV_6267UDA
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
RT-PCR
Decrease (50 %)
NA
19264337
DrugRepV_6269Mannan
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
RT-PCR
Decrease (50 %)
NA
19264337
DrugRepV_6270HHA
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
Flow cytometry
Decrease (50 %)
NA
19264337
DrugRepV_6271GNA
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
Flow cytometry
Decrease (50 %)
NA
19264337
DrugRepV_6272UDA
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
Flow cytometry
Decrease (50 %)
NA
19264337
DrugRepV_6274Mannan
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
Flow cytometry
Decrease (50 %)
NA
19264337
DrugRepV_6275HHA
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
RT-PCR
Decrease (50 %)
NA
19264337
DrugRepV_6276GNA
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
RT-PCR
Decrease (50 %)
NA
19264337
DrugRepV_6277UDA
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
RT-PCR
Decrease (50 %)
NA
19264337
DrugRepV_6279Mannan
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
RT-PCR
Decrease (50 %)
NA
19264337
DrugRepV_6280G3d
NA
NA
Dengue virus
NGC
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6281C2S-3
NA
NA
Dengue virus
NGC
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6283DS8000
NA
NA
Dengue virus
NGC
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6284G3d
NA
NA
Dengue virus
NGC
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6285C2S-3
NA
NA
Dengue virus
NGC
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6287DS8000
NA
NA
Dengue virus
NGC
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6288G3d
NA
NA
Dengue virus
NGC
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6289C2S-3
NA
NA
Dengue virus
NGC
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6291DS8000
NA
NA
Dengue virus
NGC
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6292G3d
NA
NA
Dengue virus
NGC
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6293C2S-3
NA
NA
Dengue virus
NGC
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6295DS8000
NA
NA
Dengue virus
NGC
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6296G3d
NA
NA
Dengue virus
H87
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6297C2S-3
NA
NA
Dengue virus
H87
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6299DS8000
NA
NA
Dengue virus
H87
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6300G3d
NA
NA
Dengue virus
H87
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6301C2S-3
NA
NA
Dengue virus
H87
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6303DS8000
NA
NA
Dengue virus
H87
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6304G3d
NA
NA
Dengue virus
H87
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6305C2S-3
NA
NA
Dengue virus
H87
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6307DS8000
NA
NA
Dengue virus
H87
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6308G3d
NA
NA
Dengue virus
H87
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6309C2S-3
NA
NA
Dengue virus
H87
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6311DS8000
NA
NA
Dengue virus
H87
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
15911027
DrugRepV_6313PI-88
NA
Hepatocellular carcinoma | Liver cancer | Melanoma | Multiple myeloma
Dengue virus
NGC
Pathway
Flow cytometry
Decrease (53 %)
Investigational
16309754
DrugRepV_6315PPS
NA
NA
Dengue virus
NGC
Pathway
Flow cytometry
Decrease (76 %)
NA
16309754
DrugRepV_6316Lapachaone Alpha
NA
NA
Dengue virus
New Guinea C
Pathway
Immunoflourescence assay
Decrease (98.84 %)
NA
22155902
DrugRepV_6322Shikonin
NA
NA
Dengue virus
New Guinea C
Pathway
Immunoflourescence assay
Decrease (78.94 %)
NA
22155902
DrugRepV_6324Chelerythrine Chloride
NA
NA
Dengue virus
New Guinea C
Pathway
Immunoflourescence assay
Decrease (73.36 %)
NA
22155902
DrugRepV_6325Skimmianine
NA
NA
Dengue virus
New Guinea C
Pathway
Immunoflourescence assay
Decrease (61.96 %)
NA
22155902
DrugRepV_6329Tunicamycin B
NA
Bacterial infections
Dengue virus
New Guinea C
Pathway
Immunoflourescence assay
Decrease (55.01 %)
Experimental
22155902
DrugRepV_6330Acivicin
NA
Cancer
Dengue virus
New Guinea C
Pathway
Immunoflourescence assay
Decrease (54.32 %)
Phase I
22155902
DrugRepV_6334Gitoxigenin
NA
NA
Dengue virus
New Guinea C
Pathway
Immunoflourescence assay
Decrease (49.01 %)
NA
22155902
DrugRepV_6335Kainic acid
NA
Neuroexcitatory
Dengue virus
New Guinea C
Pathway
Immunoflourescence assay
Decrease (48.87 %)
NA
22155902
DrugRepV_6338Diacetoxyscirpenol
NA
NA
Dengue virus
New Guinea C
Pathway
Immunoflourescence assay
Decrease (45.55 %)
NA
22155902
DrugRepV_6339Austricin
NA
NA
Dengue virus
New Guinea C
Pathway
Immunoflourescence assay
Decrease (45.01 %)
NA
22155902
DrugRepV_6340Valinomycin
NA
NA
Dengue virus
New Guinea C
Pathway
Immunoflourescence assay
Decrease (43.34 %)
Experimental
22155902
DrugRepV_6341Thapsigargin
NA
NA
Dengue virus
New Guinea C
Pathway
Immunoflourescence assay
Decrease (42.9 %)
NA
22155902
DrugRepV_6344Echinomycin
NA
Bacterial infections
Dengue virus
New Guinea C
Pathway
Immunoflourescence assay
Decrease (41.52 %)
NA
22155902
DrugRepV_6345Chromomycin A3
NA
NA
Dengue virus
New Guinea C
Pathway
Immunoflourescence assay
Decrease (40.87 %)
NA
22155902
DrugRepV_6346AM404
NA
Pain and Fever
Dengue virus
New Guinea C (NGC)
Pathway
NA
Decrease (50 %)
Phase IV
26856827
DrugRepV_6349(2S)-6-amino-2-[(2S)-2-[(4-{[(5Z)-3-butyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]-5-carbamimidamidopentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6350(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-cyclopentyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6351(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-cyclohexyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6352methyl 2-[(5Z)-5-[(4-{[(1S)-1-{[(1S)-5-amino-1-{[(1S)-1-carbamoylpentyl]carbamoyl}pentyl]carbamoyl}-4-carbamimidamidobutyl]carbamoyl}phenyl)methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoate
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6353(2S)-6-amino-2-[(2S)-2-[(4-{[(5Z)-3-benzyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]-5-carbamimidamidopentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6354(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-[(4-methylphenyl)methyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6355(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-[(4-methoxyphenyl)methyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6356(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-[(4-fluorophenyl)methyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6357(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-[(4-chlorophenyl)methyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6358(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-4-oxo-3-(2-phenylethyl)-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6359(2S)-6-amino-2-[(2S)-2-[(4-{[(5Z)-3-butyl-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]-5-carbamimidamidopentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6360(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-cyclopentyl-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6361(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-cyclohexyl-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_63622-[(5Z)-5-[(4-{[(1S)-1-{[(1S)-5-amino-1-{[(1S)-1-carbamoylpentyl]carbamoyl}pentyl]carbamoyl}-4-carbamimidamidobutyl]carbamoyl}phenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl acetate
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6363(2S)-6-amino-2-[(2S)-2-[(4-{[(5Z)-3-benzyl-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]-5-carbamimidamidopentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6364(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-[(4-methylphenyl)methyl]-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6365(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-[(4-methoxyphenyl)methyl]-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6366(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-[(4-fluorophenyl)methyl]-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6367(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-[(4-chlorophenyl)methyl]-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6368(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-2,4-dioxo-3-(2-phenylethyl)-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6369(2S)-N-[(5S,8S)-1-amino-11-carbamimidamido-6,7-dioxo-8-(phenylformamido)undecan-5-yl]-2-hydrazinylhexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6370(2S)-N-[(5S,8S)-1-amino-11-carbamimidamido-6,7-dioxo-8-[(thiophen-2-yl)formamido]undecan-5-yl]-2-hydrazinylhexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6371(2S)-N-[(5S,8S)-1-amino-11-carbamimidamido-8-({4-[(1E)-2-cyano-2-(cyclopropylcarbamoyl)eth-1-en-1-yl]phenyl}formamido)-6,7-dioxoundecan-5-yl]-2-hydrazinylhexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6372(2S)-N-[(5S,8S)-1-amino-11-carbamimidamido-8-({4-[(1E)-2-carbamoyleth-1-en-1-yl]phenyl}formamido)-6,7-dioxoundecan-5-yl]-2-hydrazinylhexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6373(2S)-N-[(5S,8S)-1-amino-11-carbamimidamido-6,7-dioxo-8-[(2E)-3-phenylprop-2-enamido]undecan-5-yl]-2-hydrazinylhexanamide
NA
NA
Dengue virus
NA
Pathway
Protease Assay
Decrease (50 %)
NA
24083834
DrugRepV_6374(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6375(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-methyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6376(2S)-6-amino-2-[(2S)-2-[(4-{[(5Z)-3-butyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]-5-carbamimidamidopentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6377(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-cyclopentyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6378(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-cyclohexyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6379methyl 2-[(5Z)-5-[(4-{[(1S)-1-{[(1S)-5-amino-1-{[(1S)-1-carbamoylpentyl]carbamoyl}pentyl]carbamoyl}-4-carbamimidamidobutyl]carbamoyl}phenyl)methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoate
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6380(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-4-oxo-3-(prop-2-en-1-yl)-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6381(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-(2-hydroxyethyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6382(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-(4-methoxyphenyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6383(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-(4-chlorophenyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6384(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-[(4-methoxyphenyl)methyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6385(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-[(4-chlorophenyl)methyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6386(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-4-oxo-3-(2-phenylethyl)-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6387(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6388(2S)-6-amino-2-[(2S)-2-[(4-{[(5Z)-3-butyl-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]-5-carbamimidamidopentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6389(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-cyclopentyl-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6390(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-(2-hydroxyethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6391(2S)-6-amino-2-[(2S)-2-[(4-{[(5Z)-3-benzyl-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]-5-carbamimidamidopentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6392(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-3-[(4-chlorophenyl)methyl]-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6393(2S)-6-amino-2-[(2S)-5-carbamimidamido-2-[(4-{[(5Z)-2,4-dioxo-3-(2-phenylethyl)-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]pentanamido]-N-[(1S)-1-carbamoylpentyl]hexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6394(2S)-N-[(4S,7S)-1-amino-7-{[1-(4-{[(5Z)-3-benzyl-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}phenyl)ethenyl]amino}-10-carbamimidamido-5,6-dioxodecan-4-yl]-2-hydrazinylhexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6395(2S)-N-[(5S,8S)-1-amino-11-carbamimidamido-6,7-dioxo-8-[(3-{[(5Z)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]undecan-5-yl]-2-hydrazinylhexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6396(2S)-N-[(5S,8S)-1-amino-11-carbamimidamido-8-[(3-{[(5Z)-3-cyclopentyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}phenyl)formamido]-6,7-dioxoundecan-5-yl]-2-hydrazinylhexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6397(2S)-N-[(5S,8S)-1-amino-11-carbamimidamido-8-[(2S)-2-[(5Z)-5-[(3,4-dimethoxyphenyl)methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-3-phenylpropanamido]-6,7-dioxoundecan-5-yl]-2-hydrazinylhexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6398(2S)-N-[(5S,8S)-1-amino-11-carbamimidamido-8-(2-{3-[(4-methoxyphenyl)methyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-yl}acetamido)-6,7-dioxoundecan-5-yl]-2-hydrazinylhexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6399(2S)-N-[(5S,8S)-1-amino-11-carbamimidamido-8-{2-[(5Z)-3-[(4-methoxyphenyl)methyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]acetamido}-6,7-dioxoundecan-5-yl]-2-hydrazinylhexanamide
NA
NA
Dengue virus
NA
Pathway
Renilla luciferase assay
Decrease (50 %)
NA
24083834
DrugRepV_6400HHA
NA
NA
Dengue virus
D1/H/IMTSSA/98/606
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6401HHA
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6402HHA
NA
NA
Dengue virus
H87
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6403HHA
NA
NA
Dengue virus
Dak HD 34 460
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6404HHA
NA
NA
Dengue virus
D1/H/IMTSSA/98/606
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6405HHA
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6406HHA
NA
NA
Dengue virus
H87
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6407HHA
NA
NA
Dengue virus
Dak HD 34 460
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6408GNA
NA
NA
Dengue virus
D1/H/IMTSSA/98/606
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6409GNA
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6410GNA
NA
NA
Dengue virus
H87
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6411GNA
NA
NA
Dengue virus
Dak HD 34 460
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6412GNA
NA
NA
Dengue virus
D1/H/IMTSSA/98/606
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6413GNA
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6414GNA
NA
NA
Dengue virus
H87
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6415GNA
NA
NA
Dengue virus
Dak HD 34 460
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6416UDA
NA
NA
Dengue virus
D1/H/IMTSSA/98/606
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6417UDA
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6418UDA
NA
NA
Dengue virus
H87
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6419UDA
NA
NA
Dengue virus
Dak HD 34 460
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6420UDA
NA
NA
Dengue virus
D1/H/IMTSSA/98/606
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6421UDA
NA
NA
Dengue virus
New Guinea C (NGC)
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6422UDA
NA
NA
Dengue virus
H87
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6423UDA
NA
NA
Dengue virus
Dak HD 34 460
Pathway
RT-PCR
Decrease (50 %)
NA
21738755
DrugRepV_6424Carbenoxolone disodium
NA
Digestive tract ulcers
Dengue virus
Hawaii
Pathway
TCID50 assay
Decrease (500 Fold)
Experimental
27155198
DrugRepV_6425Carbenoxolone disodium
NA
Digestive tract ulcers
Dengue virus
New Guinea C
Pathway
TCID50 assay
Decrease (2000 Fold)
Experimental
27155198
DrugRepV_6426Cdt yellow
NA
NA
Dengue virus
NGC
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_6427Cdt white
NA
NA
Dengue virus
NGC
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_6428Crotoxin
NA
NA
Dengue virus
NGC
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_6429Crotapotin
NA
NA
Dengue virus
NGC
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_6430Crotamin
NA
NA
Dengue virus
NGC
Pathway
NA
Decrease (11 %)
NA
21723310
DrugRepV_6431Convulxin
NA
NA
Dengue virus
NGC
Pathway
NA
Decrease (5 %)
NA
21723310
DrugRepV_6432PLA2-IC
NA
NA
Dengue virus
NGC
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_6433PLA2-IC
NA
NA
Dengue virus
NGC
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_6434Cdt yellow
NA
NA
Dengue virus
NGC
Pathway
Virucidal assay
Decrease (50 %)
NA
21723310
DrugRepV_6435Cdt white
NA
NA
Dengue virus
NGC
Pathway
Virucidal assay
Decrease (50 %)
NA
21723310
DrugRepV_6436Crotoxin
NA
NA
Dengue virus
NGC
Pathway
Virucidal assay
Decrease (50 %)
NA
21723310
DrugRepV_6437Crotapotin
NA
NA
Dengue virus
NGC
Pathway
Virucidal assay
Decrease (50 %)
NA
21723310
DrugRepV_6438Crotamin
NA
NA
Dengue virus
NGC
Pathway
Virucidal assay
Decrease (33 %)
NA
21723310
DrugRepV_6439Convulxin
NA
NA
Dengue virus
NGC
Pathway
Virucidal assay
Decrease (32 %)
NA
21723310
DrugRepV_6440PLA2-IC
NA
NA
Dengue virus
NGC
Pathway
Virucidal assay
Decrease (50 %)
NA
21723310
DrugRepV_6441PLA2-IC
NA
NA
Dengue virus
NGC
Pathway
Virucidal assay
Decrease (50 %)
NA
21723310
DrugRepV_6442Cdt yellow
NA
NA
Dengue virus
NGC
Pathway
Adsorption assay
Decrease (50 %)
NA
21723310
DrugRepV_6443Cdt white
NA
NA
Dengue virus
NGC
Pathway
Adsorption assay
Decrease (50 %)
NA
21723310
DrugRepV_6444Crotoxin
NA
NA
Dengue virus
NGC
Pathway
Adsorption assay
Decrease (50 %)
NA
21723310
DrugRepV_6445Crotapotin
NA
NA
Dengue virus
NGC
Pathway
Adsorption assay
Decrease (50 %)
NA
21723310
DrugRepV_6446Crotamin
NA
NA
Dengue virus
NGC
Pathway
Adsorption assay
Decrease (100 %)
NA
21723310
DrugRepV_6447Convulxin
NA
NA
Dengue virus
NGC
Pathway
Adsorption assay
Decrease (100 %)
NA
21723310
DrugRepV_6448PLA2-IC
NA
NA
Dengue virus
NGC
Pathway
Adsorption assay
Decrease (50 %)
NA
21723310
DrugRepV_6449PLA2-IC
NA
NA
Dengue virus
NGC
Pathway
Adsorption assay
Decrease (50 %)
NA
21723310
DrugRepV_6450Cdt yellow
NA
NA
Dengue virus
NGC
Pathway
Internalization assay
Decrease (50 %)
NA
21723310
DrugRepV_6451Cdt white
NA
NA
Dengue virus
NGC
Pathway
Internalization assay
Decrease (50 %)
NA
21723310
DrugRepV_6452Crotoxin
NA
NA
Dengue virus
NGC
Pathway
Internalization assay
Decrease (50 %)
NA
21723310
DrugRepV_6453Crotapotin
NA
NA
Dengue virus
NGC
Pathway
Internalization assay
Decrease (41 %)
NA
21723310
DrugRepV_6454Crotamin
NA
NA
Dengue virus
NGC
Pathway
Internalization assay
Decrease (46 %)
NA
21723310
DrugRepV_6455Convulxin
NA
NA
Dengue virus
NGC
Pathway
Internalization assay
Decrease (2.3 %)
NA
21723310
DrugRepV_6456PLA2-IC
NA
NA
Dengue virus
NGC
Pathway
Internalization assay
Decrease (50 %)
NA
21723310
DrugRepV_6457PLA2-IC
NA
NA
Dengue virus
NGC
Pathway
Internalization assay
Decrease (50 %)
NA
21723310
DrugRepV_6458(3E)-N-tert-butyl-2-oxo-4-phenylbut-3-enamide
NA
NA
Dengue virus
NA
Pathway
Protease assay
Decrease (26.3 %)
NA
21641807
DrugRepV_6459(3E)-N-tert-butyl-3-methyl-2-oxo-4-phenylbut-3-enamide
NA
NA
Dengue virus
NA
Pathway
Protease assay
Decrease (25.6 %)
NA
21641807
DrugRepV_6460(3E)-N-tert-butyl-2-oxo-4-(thiophen-2-yl)but-3-enamide
NA
NA
Dengue virus
NA
Pathway
Protease assay
Decrease (27.6 %)
NA
21641807
DrugRepV_6461(3E)-N-tert-butyl-4-(4-methoxyphenyl)-2-oxobut-3-enamide
NA
NA
Dengue virus
NA
Pathway
Protease assay
Decrease (16.7 %)
NA
21641807
DrugRepV_6462(3E)-N-tert-butyl-4-(3,4-dimethoxyphenyl)-2-oxobut-3-enamide
NA
NA
Dengue virus
NA
Pathway
Protease assay
Decrease (36.1 %)
NA
21641807
DrugRepV_6463(3E)-N-tert-butyl-4-(4-hydroxyphenyl)-2-oxobut-3-enamide
NA
NA
Dengue virus
NA
Pathway
Protease assay
Decrease (37.6 %)
NA
21641807
DrugRepV_6464(3E)-4-(4-aminophenyl)-N-tert-butyl-2-oxobut-3-enamide
NA
NA
Dengue virus
NA
Pathway
Protease assay
Decrease (40.6 %)
NA
21641807
DrugRepV_6465(3E)-N-tert-butyl-4-(4-chlorophenyl)-2-oxobut-3-enamide
NA
NA
Dengue virus
NA
Pathway
Protease assay
Decrease (15.9 %)
NA
21641807
DrugRepV_6466(3E)-N-tert-butyl-4-(1H-indol-3-yl)-2-oxobut-3-enamide
NA
NA
Dengue virus
NA
Pathway
Protease assay
Decrease (39.1 %)
NA
21641807
DrugRepV_6467(3E)-N-tert-butyl-4-[4-(dimethylamino)phenyl]-2-oxobut-3-enamide
NA
NA
Dengue virus
NA
Pathway
Protease assay
Decrease (13.8 %)
NA
21641807
DrugRepV_6468(3E)-N-cyclopropyl-2-oxo-4-phenylbut-3-enamide
NA
NA
Dengue virus
NA
Pathway
Protease assay
Decrease (31.2 %)
NA
21641807
DrugRepV_64692-[(3E)-2-oxo-4-phenylbut-3-enamido]ethyl acetate
NA
NA
Dengue virus
NA
Pathway
Protease assay
Decrease (35.8 %)
NA
21641807
DrugRepV_6470(3E)-2-oxo-4-phenyl-N-(1-phenylethyl)but-3-enamide
NA
NA
Dengue virus
NA
Pathway
Protease assay
Decrease (0 %)
NA
21641807
DrugRepV_6471methyl 3-hydroxy-2-[(3E)-2-oxo-4-phenylbut-3-enamido]propanoate
NA
NA
Dengue virus
NA
Pathway
Protease assay
Decrease (35.1 %)
NA
21641807
DrugRepV_6472Delphinidin Chloride
NA
NA
Dengue virus
NA
Pathway
Plaque assay
Decrease
NA
28744282
DrugRepV_6474N-nonyl-deoxynojirimycin
NA
NA
Dengue virus
New Guinea C
Pathway
Yield reduction assay
Decrease (50 %)
NA
17354651
DrugRepV_6475N-pentyl-(1-hydroxycyclohexyl)-DNJ
NA
NA
Dengue virus
New Guinea C
Pathway
Yield reduction assay
Decrease (50 %)
NA
17354651
DrugRepV_6476N-Propylcyclohexyl-DNJ
NA
NA
Dengue virus
New Guinea C
Pathway
Yield reduction assay
Decrease (50 %)
NA
17354651
DrugRepV_6477N-Butylcyclohexyl-DNJ
NA
NA
Dengue virus
New Guinea C
Pathway
Yield reduction assay
Decrease (50 %)
NA
17354651
DrugRepV_6479N-acetyl cysteine
NA
Acetaminophen poisoning
Dengue virus
NA
Pathway
Cell viability assay
Decrease (50 %)
Approved
30928439
DrugRepV_6480Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Dengue virus
NA
Pathway
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_6487KX2-391
NA
Colon cancer | Pancreatic cancer | Prostate cancer | Breast cancer
Human immunodeficiency virus
HXB2 luciferase reporter virus
Pathway
Luciferase reporter assay
Decrease (80 %)
Investigational
26807966
DrugRepV_6488KX2-391
NA
Colon cancer | Pancreatic cancer | Prostate cancer | Breast cancer
Human immunodeficiency virus
JR-FL luciferase reporter virus
Pathway
Luciferase reporter assay
Decrease (90 %)
Investigational
26807966
DrugRepV_6496Decitabine
NA
Myelodysplastic syndromes +Different types of Cancer
Human immunodeficiency virus
NA
Pathway
Plaque assay
Decrease (73 %)
NA
20610712
DrugRepV_6498Decitabine
NA
NA
Human immunodeficiency virus
NA
Pathway
Plaque assay
Decrease (75 %)
NA
20610712
DrugRepV_6500Decitabine
NA
Myelodysplastic syndromes +Different types of Cancer
Human immunodeficiency virus
NA
Pathway
Real-time PCR
Decrease
NA
20610712
DrugRepV_68674-(3,5-Diphenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68684-(5-(2-Fluorophenyl)-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68694-(5-(3-fluorophenyl)-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68704-(5-(4-Fluorophenyl)-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68714-(5-(2-chlorophenyl)-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68724-(5-(3-chlorophenyl)-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68734-(5-(4-chlorophenyl)-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68744-(3-Phenyl-5-(o-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68754-(3-Phenyl-5-(m-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68764-(3-Phenyl-5-(p-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68774-(3-(4-phenoxyphenyl)-5-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68784-(5-(2-fluorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68794-(5-(3-fluorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68804-(5-(4-fluorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68814-(5-(2-chlorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68824-(5-(3-chlorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68834-(5-(4-chlorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68844-(3-(4-phenoxyphenyl)-5-(o-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68854-(3-(4-phenoxyphenyl)-5-(m-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68864-(3-(4-phenoxyphenyl)-5-(p-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68874-(3-(4-(benzyloxy)phenyl)-5-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68884-(3-(4-(benzyloxy)phenyl)-5-(2-fluorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68894-(3-(4-(benzyloxy)phenyl)-5-(3-fluorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68904-(3-(4-(benzyloxy)phenyl)-5-(4-fluorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68914-(3-(4-(benzyloxy)phenyl)-5-(2-chlorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68924-(3-(4-(benzyloxy)phenyl)-5-(3-chlorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68934-(3-(4-(benzyloxy)phenyl)-5-(4-chlorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68944-(3-(4-(benzyloxy)phenyl)-5-(o-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68954-(3-(4-(benzyloxy)phenyl)-5-(m-tolyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_68964-(3-(4-(benzyloxy)phenyl)-5-(p-tolyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Human immunodeficiency virus
NA
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_6897Phorbol
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6898Phorbol-12-acetate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6899Phorbol-12-decanoate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6900Phorbol-13-acetate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6901Phorbol-13-butyrate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6902Phorbol-13-decanoate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6903Phorbol-13-tetradecanoate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6904Phorbol-12,13-diacetate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6905Phorbol-12,13-dibutyrate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6906Phorbol-12,13- dihexanoate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6907Phorbol-12,13-didecanoate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_69084α-phorbol-12,13-didecanoate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_690912-O-tetradecanoylphorbol-13-acetate
NA
Cancer
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
Phase II
25970561
DrugRepV_691012-O-tetradecanoyl-4γ-phorbol-13-acetate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_691112-O- tiglylphorbol-13-decanoate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_691212-O-(N-methylanthranilate) phorbol-13-acetate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6913Phorbol-13,20-diacetate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_691412,13-O,O-dinonanoylphorbol-20-homovanillate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_691512-O-phenylacetyl-13-O-acetylphorbol-20-homovanillate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6916Phorbol-12,13,20-triacetate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_691720-oxo-20-deoxyphorbol-12,13-dibutyrate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_691812-O-tetradecanoyl-20-oxo-20-deoxyphorbol-13-acetate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_691912-deoxyphorbol-13-acetate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_692013-O-isobutyryl-12-deoxyphorbol-20-acetate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_692113-O-phenylacetyl-12-deoxyphorbol-20-acetate
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6925Resiniferatoxin
NA
Interstitial cystitis and urinary incontinence
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
Investigational
25970561
DrugRepV_6927Phorbol
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6928Phorbol-12-acetate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6929Phorbol-12-decanoate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6930Phorbol-13-acetate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6931Phorbol-13-butyrate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6932Pphorbol-13-decanoate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6933Phorbol-13-tetradecanoate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6934Phorbol-12,13-diacetate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6935Phorbol-12,13-dibutyrate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6936Phorbol-12,13- dihexanoate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6937Phorbol-12,13-didecanoate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_69384α-phorbol-12,13-didecanoate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_693912-O-tetradecanoylphorbol-13-acetate
NA
Cancer
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
Phase II
25970561
DrugRepV_694012-O-tetradecanoyl-4?-phorbol-13-acetate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_694112-O- tiglylphorbol-13-decanoate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_694212-O-(N-methylanthranilate) phorbol-13-acetate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6943Phorbol-13,20-diacetate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_694412,13-O,O-dinonanoylphorbol-20-homovanillate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_694512-O-phenylacetyl-13-O-acetylphorbol-20-homovanillate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6946Phorbol-12,13,20-triacetate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_694720-oxo-20-deoxyphorbol-12,13-dibutyrate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_694812-O-tetradecanoyl-20-oxo-20-deoxyphorbol-13-acetate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_694912-deoxyphorbol-13-acetate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_695013-O-isobutyryl-12-deoxyphorbol-20-acetate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_695113-O-phenylacetyl-12-deoxyphorbol-20-acetate
NA
NA
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
NA
25970561
DrugRepV_6955Resiniferatoxin
NA
Interstitial cystitis and urinary incontinence
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
Investigational
25970561
DrugRepV_6957FGI-106
NA
NA
Human immunodeficiency virus
NA
Pathway
Luciferase assay
Decrease (50 %)
NA
19523489
DrugRepV_6964(1S,2R,3S)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]uracil
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6965(1S,2R,3S)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]thymine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6966(1S,2R,3S)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]-5-fluorouracil
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6967(1S,2R,3S)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]cytosine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6968(1S,2R,3S)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]-5-fluorocytosine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6969L-Neplanocin A
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6970(1S,2R,3S)-9-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl] hypoxanthine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6971(1S,2R,3S)-9-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]guanine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6972Cyclopentenyl nucleosides
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6973(1R,2S,3R)-9-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl] hypoxanthine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6974(1R,2S,3R)-9-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]guanine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6975(1S,2R,3S)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]uracil
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6976(1R,2S,3R)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]thymine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6977(1R,2S,3R)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]-5-fluorouracil
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6978(1R,2S,3R)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]cytosine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6979(1R,2S,3R)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]-5-fluorocytosine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6980Octadecyloxyethyl benzyl 9-[(2-phosphonomethoxy)ethyl]guanine
NA
NA
Human immunodeficiency virus
NA
Pathway
RT-PCR
Decrease (50 %)
NA
27933957
DrugRepV_69813-azido-2,3-dideoxyuridine
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_69821-(4-azido-5-hydroxyoxolan-2-yl)-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_69831-(4-azido-5-hydroxyoxolan-2-yl)-5-(trifluoromethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_69842- deoxy-5-fluorouridine
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_69852- deoxy-5-bromouridine
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_69862-deoxy-5-iodouridine
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_69873-Azido-2,3-dideoxy-5-aminouridine Hydrochloride
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_69883-Azido-2,3-dideoxy-5-(methylamino)uridine hydrochloride
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_69893-Azido-2,3-dideoxy-5-(dimethylamino)uridine hydrochloride
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_69903-Azido-2,3-dideoxy-5-hydroxyuridine
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_69913-Azido-2,3-dideoxy-5-methoxyuridine
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_69923-Azido-2,3-dideoxy-5-ethoxyuridine
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_69933-Azido-2,3-dideoxy-5-(2-propynyloxy)uridine
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_69943-Azido-2,3-dideoxy-5-(propenyloxy)uridine
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_69953-Azido-2,3-dideoxy-5-[(cyanomethyl)oxy]uridine
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_69963-Azido-2,3-dideoxy-5-thiocyanatouridine
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_69973-Azido-2,3-dideoxy-5-(methylthio)uridine
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_69982-deoxycytidine
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_69992-deoxy-5-fluorocytidine
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_70002,-deoxy-5-methylcytidine
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_70013-(3-Oxo-l-propenyI)-3-azido-3-deoxyThymidine
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_70023-Azido-3-deoxy-6-azaThymidine
NA
NA
Human immunodeficiency virus
LAV
Pathway
RT assay
Decrease (50 %)
NA
3339606
DrugRepV_70472-Aminobiphenyl borate
NA
NA
Japanese encephalitis virus
AT31
Pathway
Immunoflourescence assay
Decrease (18 %)
NA
28814523
DrugRepV_70491,2-bis-(o-aminophenoxy)-ethane-N,N,N,N-tetraacetic Acid
NA
NA
Japanese encephalitis virus
AT31
Pathway
Immunoflourescence assay
Decrease (60 %)
NA
28814523
DrugRepV_70512-Aminobiphenyl borate
NA
NA
Japanese encephalitis virus
AT31
Pathway
Immunoflourescence assay
Decrease (20 %)
NA
28814523
DrugRepV_70531,2-bis-(o-aminophenoxy)-ethane-N,N,N,N-tetraacetic Acid
NA
NA
Japanese encephalitis virus
AT31
Pathway
Immunoflourescence assay
Decrease (45 %)
NA
28814523
DrugRepV_7068Quinacrine Mustard
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
West Nile virus
NA
Pathway
Plaque assay
Decrease (> 99 %)
Experimental
24680954
DrugRepV_7086Quinacrine Mustard
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
West Nile virus
NA
Pathway
Plaque assay
Decrease (50 %)
Experimental
24680954
DrugRepV_7097Abamectin
NA
Helmintic infection
Yellow fever virus
17D
Pathway
Plaque assay
Decrease (5.3 Log)
Terminated
26752081
DrugRepV_7098Berberine
NA
Parasitic and fungal infection
Yellow fever virus
17D
Pathway
Plaque assay
No significant effect (No significant effect Log)
Approved
26752081
DrugRepV_7103Chebulagic Acid
NA
Immunosuppressive and hepatoprotective
Measles virus
IC323
Pathway
EGFP assay
Decrease (50 %)
NA
23924316
DrugRepV_7105Chebulagic Acid
NA
Immunosuppressive and hepatoprotective
Measles virus
IC323
Pathway
EGFP assay
Decrease (80 %)
NA
23924316
DrugRepV_7107Arbidol
NA
Viral infection
Polio virus
NA
Pathway
Plaque assay
Decrease (50 %)
Phase IV
22028179
DrugRepV_7108N-nonyl-deoxynojirimycin
NA
NA
Japanese encephalitis virus
RP-9
Pathway
Immunoflourescence assay
Decrease (90 %)
NA
11907199
DrugRepV_7109N-nonyl-deoxynojirimycin
NA
NA
Japanese encephalitis virus
RP-9
Pathway
Plaque assay
Decrease (3 Logs)
NA
11907199
DrugRepV_7110N-nonyl-deoxynojirimycin
NA
NA
Japanese encephalitis virus
RP-9
Pathway
LDH assay
No significant effect
NA
11907199
DrugRepV_7111N-nonyl-deoxynojirimycin
NA
NA
Japanese encephalitis virus
RP-9
Pathway
Western blot
No significant effect (No significant effect Band Intensity)
NA
11907199
DrugRepV_7112N-nonyl-deoxynojirimycin
NA
NA
Japanese encephalitis virus
RP-9
Pathway
Western blot
No significant effect (No significant effect Band Intensity)
NA
11907199
DrugRepV_7113N-nonyl-deoxynojirimycin
NA
NA
Japanese encephalitis virus
RP-9
Pathway
Survival assay
Increase
NA
11907199
DrugRepV_71154-(3,5-Diphenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71164-(5-(2-Fluorophenyl)-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71174-(5-(3-fluorophenyl)-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71184-(5-(4-Fluorophenyl)-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71194-(5-(2-chlorophenyl)-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71204-(5-(3-chlorophenyl)-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71214-(5-(4-chlorophenyl)-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71224-(3-Phenyl-5-(o-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71234-(3-Phenyl-5-(m-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71244-(3-Phenyl-5-(p-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71254-(3-(4-phenoxyphenyl)-5-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71264-(5-(2-fluorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71274-(5-(3-fluorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71284-(5-(4-fluorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71294-(5-(2-chlorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71304-(5-(3-chlorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71314-(5-(4-chlorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71324-(3-(4-phenoxyphenyl)-5-(o-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71334-(3-(4-phenoxyphenyl)-5-(m-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71344-(3-(4-phenoxyphenyl)-5-(p-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71354-(3-(4-(benzyloxy)phenyl)-5-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71364-(3-(4-(benzyloxy)phenyl)-5-(2-fluorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71374-(3-(4-(benzyloxy)phenyl)-5-(3-fluorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71384-(3-(4-(benzyloxy)phenyl)-5-(4-fluorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71394-(3-(4-(benzyloxy)phenyl)-5-(2-chlorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71404-(3-(4-(benzyloxy)phenyl)-5-(3-chlorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71414-(3-(4-(benzyloxy)phenyl)-5-(4-chlorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71424-(3-(4-(benzyloxy)phenyl)-5-(o-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71434-(3-(4-(benzyloxy)phenyl)-5-(m-tolyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71444-(3-(4-(benzyloxy)phenyl)-5-(p-tolyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
Yellow fever virus
17D
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71454-(5-(4-Fluorophenyl)-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71464-(5-(2-chlorophenyl)-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71474-(5-(3-chlorophenyl)-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71484-(3-Phenyl-5-(o-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71494-(3-Phenyl-5-(p-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71504-(3-(4-phenoxyphenyl)-5-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71514-(5-(2-fluorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71524-(5-(3-fluorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71534-(5-(4-fluorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71544-(5-(2-chlorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71554-(5-(3-chlorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71564-(5-(4-chlorophenyl)-3-(4-phenoxyphenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71574-(3-(4-phenoxyphenyl)-5-(o-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71584-(3-(4-phenoxyphenyl)-5-(m-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71594-(3-(4-phenoxyphenyl)-5-(p-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71604-(3-(4-(benzyloxy)phenyl)-5-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71614-(3-(4-(benzyloxy)phenyl)-5-(2-fluorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71624-(3-(4-(benzyloxy)phenyl)-5-(3-fluorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71634-(3-(4-(benzyloxy)phenyl)-5-(4-fluorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71644-(3-(4-(benzyloxy)phenyl)-5-(2-chlorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71654-(3-(4-(benzyloxy)phenyl)-5-(3-chlorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71664-(3-(4-(benzyloxy)phenyl)-5-(4-chlorophenyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71674-(3-(4-(benzyloxy)phenyl)-5-(o-tolyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71684-(3-(4-(benzyloxy)phenyl)-5-(m-tolyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_71694-(3-(4-(benzyloxy)phenyl)-5-(p-tolyl)-4,5-dihydro-1H-pyrazol-1- yl)benzenesulfonamide
NA
NA
West Nile virus
Clinical isolate
Pathway
MTT assay
Decrease (50 %)
NA
29028528
DrugRepV_7173N2-(4-fluorophenyl)-N3-(4-methyl-2-(thiophen-2-yl)phenyl) pyrazine-2,3-dicarboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7174N2-(4-fluorophenyl)-N3-(4-methyl-2-(thiophen-3-yl) phenyl)pyrazine-2,3- dicarboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7175N2-(4-methyl-2-(thiophen-3-yl)phenyl)-N3-(p-tolyl) pyrazine-2,3-dicarboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7176N2-(4-fluorophenyl)-N3-(2-(thiophen-3-yl)benzyl)pyrazine- 2,3-dicarboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7177N2-(2-(thiophen-3-yl)benzyl)-N3-(p-tolyl)pyrazine-2,3-dicarboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7178N2-(4-fluorophenyl)-N3-(4-(thiophen-3-yl)benzyl)pyrazine-2,3-dicarboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7179N2-(4-(thiophen-3-yl)benzyl)-N3-(p-tolyl)pyrazine-2,3-dicarboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7180N2-(4-fluorophenyl)-N3-(2-(3-methyl-1H-pyrazol-5-yl) phenyl)pyrazine-2,3-dicarboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7181N2-(2-(3-methyl-1H-pyrazol-5-yl)phenyl)-N3-(p-tolyl) pyrazine-2,3-di-carboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7182N1-(4-fluorophenyl)-N2-(4-methyl-2-(3-methyl-1H-pyrazol-5-yl)phenyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7183N1-(4-fluorophenyl)-N2-(4-methyl-2-(thiophen-2-yl) phenyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7184N1-(4-methyl-2-(3-methyl-1H-pyrazol-5-yl)phenyl)-N2-(p- tolyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7185N1-(4-methyl-2-(thiophen-2-yl)phenyl)-N2-(p-tolyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7186N1-(4-methyl-2-(5-methylthiophen-2-yl)phenyl)-N2-(p- tolyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7187N1-(4-fluorophenyl)-N2-(4-methyl-2-(5-methylthiophen-2- yl)phenyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7188N1-(4-methyl-2-(thiophen-3-yl)phenyl)-N2-(p-tolyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7189N1-(4-fluorophenyl)-N2-(4-methyl-2-(thiophen-3-yl) phenyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7190N1-(4-fluorophenyl)-N2-(2-(thiophen-3-yl)benzyl) phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7191N1-(2-(thiophen-3-yl)benzyl)-N2-(p-tolyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7192N1-(4-fluorophenyl)-N2-(4-(thiophen-3-yl)benzyl) phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7193N1-(4-(thiophen-3-yl)benzyl)-N2-(p-tolyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7194N1-(4-fluorophenyl)-N2-(2-(3-methyl-1H-pyrazol-5-yl) phenyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7195N1-(2-(3-methyl-1H-pyrazol-5-yl)phenyl)-N2-(p-tolyl) phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_71962-(4-fluorobenzamido)-N-(4-methyl-2-(thiophen-3-yl) phenyl)benzamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_71972-(4-fluorobenzamido)-N-(4-methyl-2-(5-methylthiophen- 2-yl)phenyl)benzamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_71982-(4-fluorobenzamido)-N-(4-methyl-2-(pyridin-4-yl)phenyl) benzamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_71992-(4-fluorobenzamido)-N-(4-methyl-2-(pyridin-3-yl)phenyl) benzamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7200CCG-4088
NA
NA
Yellow fever virus
YFV 17D
Pathway
HTS assay
Decrease (50 %)
NA
19651907
DrugRepV_7201CCG-3394
NA
NA
Yellow fever virus
YFV 17D
Pathway
HTS assay
Decrease (50 %)
NA
19651907
DrugRepV_7202CCG-3925
NA
NA
Yellow fever virus
YFV 17D
Pathway
HTS assay
Decrease (50 %)
NA
19651907
DrugRepV_7203CCG-7648
NA
NA
Yellow fever virus
YFV 17D
Pathway
HTS assay
Decrease (50 %)
NA
19651907
DrugRepV_7204CCG-6269
NA
NA
Yellow fever virus
YFV 17D
Pathway
HTS assay
Decrease (50 %)
NA
19651907
DrugRepV_7205CCG-3374
NA
NA
Yellow fever virus
YFV 17D
Pathway
HTS assay
Decrease (50 %)
NA
19651907
DrugRepV_7206CCG-4088
NA
NA
Yellow fever virus
YFV 17D
Pathway
qRT-PCR
Decrease (20 Fold)
NA
19651907
DrugRepV_7207CCG-3394
NA
NA
Yellow fever virus
YFV 17D
Pathway
qRT-PCR
Decrease (15 Fold)
NA
19651907
DrugRepV_7208CCG-4088
NA
NA
Yellow fever virus
YFV 17D
Pathway
Immunoflourescence assay
Decrease
NA
19651907
DrugRepV_7209CCG-3394
NA
NA
Yellow fever virus
YFV 17D
Pathway
Immunoflourescence assay
Decrease
NA
19651907
DrugRepV_7210CCG-6269
NA
NA
Yellow fever virus
YFV 17D
Pathway
Luciferase assay
Decrease (87 %)
NA
19651907
DrugRepV_7211CCG-3394
NA
NA
Yellow fever virus
YFV 17D
Pathway
Luciferase assay
Decrease (92 %)
NA
19651907
DrugRepV_7212CCG-4088
NA
NA
Yellow fever virus
YFV 17D
Pathway
Luciferase assay
Decrease (90 %)
NA
19651907
DrugRepV_7213CCG-3394
NA
NA
Yellow fever virus
YFV 17D
Pathway
Luciferase assay
Decrease (38 %)
NA
19651907
DrugRepV_7214CCG-4088
NA
NA
Yellow fever virus
YFV 17D
Pathway
Luciferase assay
Decrease (48 %)
NA
19651907
DrugRepV_7215CCG-4088
NA
NA
Yellow fever virus
YFV 17D
Pathway
Luciferase assay
Decrease (42 %)
NA
19651907
DrugRepV_7217SA-3
NA
NA
Yellow fever virus
17D
Pathway
qRT-PCR
Decrease (50 %)
NA
20837762
DrugRepV_7218SA-11
NA
NA
Yellow fever virus
17D
Pathway
qRT-PCR
Decrease (50 %)
NA
20837762
DrugRepV_7219SA-17
NA
NA
Yellow fever virus
17D
Pathway
qRT-PCR
Decrease (50 %)
NA
20837762
DrugRepV_7220SA-17
NA
NA
Yellow fever virus
17D
Pathway
qRT-PCR
Decrease (50 %)
NA
20837762
DrugRepV_72212-(3-chlorophenoxy) acetaldehydethiosemicarbazone
NA
NA
Yellow fever virus
NA
Pathway
Plaque reduction assay
Decrease (60 %)
NA
28068627
DrugRepV_72222-(3,4-dichlorophen oxy) acetaldehydethiosemicarbazone
NA
NA
Yellow fever virus
NA
Pathway
Plaque reduction assay
Decrease (78 %)
NA
28068627
DrugRepV_72232-(2,3-dichlorophenoxy) acetaldehyde thiosemicarbazone
NA
NA
Yellow fever virus
NA
Pathway
Plaque reduction assay
Decrease (70 %)
NA
28068627
DrugRepV_72242-(4-(4-fluorophenyl)thiazol-2-yl)hydrazono)ethyl)isoindoline-1,3-dione
NA
NA
Yellow fever virus
NA
Pathway
Plaque reduction assay
Decrease (40 %)
NA
28068627
DrugRepV_72252-(4-(4-chlorophenyl) thiazol-2-yl)hydrazono)ethyl)isoindoline-1,3-dione
NA
NA
Yellow fever virus
NA
Pathway
Plaque reduction assay
Decrease (55 %)
NA
28068627
DrugRepV_72262-(3-chlorophenoxy) acetaldehydethiosemicarbazone
NA
NA
Yellow fever virus
NA
Pathway
Flow cytometry
Decrease (17 %)
NA
28068627
DrugRepV_72272-(3,4-dichlorophen oxy) acetaldehydethiosemicarbazone
NA
NA
Yellow fever virus
NA
Pathway
Flow cytometry
Decrease (22 %)
NA
28068627
DrugRepV_72282-(2,3-dichlorophenoxy) acetaldehyde thiosemicarbazone
NA
NA
Yellow fever virus
NA
Pathway
Flow cytometry
Decrease (14 %)
NA
28068627
DrugRepV_72292-(4-(4-fluorophenyl)thiazol-2-yl)hydrazono)ethyl)isoindoline-1,3-dione
NA
NA
Yellow fever virus
NA
Pathway
Flow cytometry
Decrease (10 %)
NA
28068627
DrugRepV_72302-(4-(4-chlorophenyl) thiazol-2-yl)hydrazono)ethyl)isoindoline-1,3-dione
NA
NA
Yellow fever virus
NA
Pathway
Flow cytometry
Decrease (3 %)
NA
28068627
DrugRepV_72312-(3-chlorophenoxy) acetaldehydethiosemicarbazone
NA
NA
Yellow fever virus
NA
Pathway
Flow cytometry
Increase
NA
28068627
DrugRepV_72322-(3,4-dichlorophen oxy) acetaldehydethiosemicarbazone
NA
NA
Yellow fever virus
NA
Pathway
Flow cytometry
Increase
NA
28068627
DrugRepV_72332-(2,3-dichlorophenoxy) acetaldehyde thiosemicarbazone
NA
NA
Yellow fever virus
NA
Pathway
Flow cytometry
Increase
NA
28068627
DrugRepV_72342-(4-(4-fluorophenyl)thiazol-2-yl)hydrazono)ethyl)isoindoline-1,3-dione
NA
NA
Yellow fever virus
NA
Pathway
Flow cytometry
Increase
NA
28068627
DrugRepV_72352-(4-(4-chlorophenyl) thiazol-2-yl)hydrazono)ethyl)isoindoline-1,3-dione
NA
NA
Yellow fever virus
NA
Pathway
Flow cytometry
Increase
NA
28068627
DrugRepV_72362-(3-chlorophenoxy) acetaldehydethiosemicarbazone
NA
NA
Yellow fever virus
NA
Pathway
Immunoflourescence assay
Decrease
NA
28068627
DrugRepV_72372-(3,4-dichlorophen oxy) acetaldehydethiosemicarbazone
NA
NA
Yellow fever virus
NA
Pathway
Immunoflourescence assay
Decrease
NA
28068627
DrugRepV_7238BCX4430
NA
Ebola virus
Measles virus
Chicago
Pathway
RT-PCR
Decrease (50 %)
Investigational
24590073
DrugRepV_7239BCX4430
NA
Ebola virus
Yellow fever virus
17D
Pathway
RT-PCR
Decrease (50 %)
Investigational
24590073
DrugRepV_7240BCX4430
NA
Ebola virus
Japanese encephalitis virus
SA14
Pathway
RT-PCR
Decrease (50 %)
Investigational
24590073
DrugRepV_7242IHVR-19029
NA
NA
Yellow fever virus
17D
Pathway
qRT-PCR
Decrease (50 %)
NA
29253498
DrugRepV_7243BCX4430
NA
Ebola virus
Yellow fever virus
17D
Pathway
NA
Decrease (50 %)
Investigational
27095300
DrugRepV_72441-[4,5-dihydroxy-3-(hydroxymethyl)cyclopent-2-en-1-yl]-1H-1,2,4-triazole-3-carboxamide
NA
NA
West Nile virus
NA
Pathway
NA
Decrease (50 %)
NA
16451078
DrugRepV_72451-[4,5-dihydroxy-3-(hydroxymethyl)cyclopent-2-en-1-yl]-1H-1,2,4-triazole-3-carboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
16451078
DrugRepV_72461-[4,5-dihydroxy-3-(hydroxymethyl)cyclopent-2-en-1-yl]-1H-imidazole-4-carboxamide
NA
NA
West Nile virus
NA
Pathway
NA
Decrease (50 %)
NA
16451078
DrugRepV_72471-[4,5-dihydroxy-3-(hydroxymethyl)cyclopent-2-en-1-yl]-1H-imidazole-4-carboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
16451078
DrugRepV_72481-[4,5-dihydroxy-3-(hydroxymethyl)cyclopent-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
NA
NA
West Nile virus
NA
Pathway
NA
Decrease (50 %)
NA
16451078
DrugRepV_72491-[4,5-dihydroxy-3-(hydroxymethyl)cyclopent-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
16451078
DrugRepV_72513-{[(4-chlorophenyl)methyl]sulfanyl}-5-[(4,5-dichloro-1H-imidazol-1-yl)methyl]-4-methyl-4H-1,2,4-triazole
NA
NA
West Nile virus
Kunjin
Pathway
Plaque assay
Decrease (50 %)
NA
19781577
DrugRepV_72522-({[5-(5-methyl-3-phenyl-1,2-oxazol-4-yl)-1,2,4-oxadiazol-3-yl]methyl}sulfanyl)pyridin-1-ium-1-olate
NA
NA
West Nile virus
Kunjin
Pathway
Plaque assay
Decrease (50 %)
NA
19781577
DrugRepV_72531-(4-chlorophenyl)-2-({5-[(4,5-dichloro-1H-imidazol-1-yl)methyl]-1,3,4-oxadiazol-2-yl}sulfanyl)ethan-1-one
NA
NA
West Nile virus
Kunjin
Pathway
Plaque assay
Decrease (50 %)
NA
19781577
DrugRepV_72541-(2-chlorophenyl)-3-{2-[(4,5-dichloro-1H-imidazol-1-yl)methyl]-1,3-thiazol-4-yl}urea
NA
NA
West Nile virus
Kunjin
Pathway
Plaque assay
Decrease (50 %)
NA
19781577
DrugRepV_72552-chloro-6-(4-chlorophenoxy)-4-{4-methyl-5-[(1E)-1-(2-phenylhydrazin-1-ylidene)ethyl]-1,3-thiazol-2-yl}pyridine
NA
NA
West Nile virus
Kunjin
Pathway
Plaque assay
Decrease (50 %)
NA
19781577
DrugRepV_72563-{[(4-chlorophenyl)methyl]sulfanyl}-5-[(4,5-dichloro-1H-imidazol-1-yl)methyl]-4-methyl-4H-1,2,4-triazole
NA
NA
Yellow fever virus
17D
Pathway
Plaque assay
Decrease (50 %)
NA
19781577
DrugRepV_72572-({[5-(5-methyl-3-phenyl-1,2-oxazol-4-yl)-1,2,4-oxadiazol-3-yl]methyl}sulfanyl)pyridin-1-ium-1-olate
NA
NA
Yellow fever virus
17D
Pathway
Plaque assay
Decrease (50 %)
NA
19781577
DrugRepV_72581-(4-chlorophenyl)-2-({5-[(4,5-dichloro-1H-imidazol-1-yl)methyl]-1,3,4-oxadiazol-2-yl}sulfanyl)ethan-1-one
NA
NA
Yellow fever virus
17D
Pathway
Plaque assay
Decrease (50 %)
NA
19781577
DrugRepV_72591-(2-chlorophenyl)-3-{2-[(4,5-dichloro-1H-imidazol-1-yl)methyl]-1,3-thiazol-4-yl}urea
NA
NA
Yellow fever virus
17D
Pathway
Plaque assay
Decrease (50 %)
NA
19781577
DrugRepV_72602-chloro-6-(4-chlorophenoxy)-4-{4-methyl-5-[(1E)-1-(2-phenylhydrazin-1-ylidene)ethyl]-1,3-thiazol-2-yl}pyridine
NA
NA
Yellow fever virus
17D
Pathway
Plaque assay
Decrease (50 %)
NA
19781577
DrugRepV_7263PI-88
NA
Hepatocellular carcinoma | Liver cancer | Melanoma | Multiple myeloma
Japanese encephalitis virus
Nakayama
Pathway
Flow cytometry
Decrease (66 %)
Investigational
16309754
DrugRepV_7265PPS
NA
NA
Japanese encephalitis virus
Nakayama
Pathway
Flow cytometry
Decrease (70 %)
NA
16309754
DrugRepV_7266PI-88
NA
Hepatocellular carcinoma | Liver cancer | Melanoma | Multiple myeloma
West Nile virus
NY-99
Pathway
Flow cytometry
Decrease (66 %)
Investigational
16309754
DrugRepV_7267Cdt yellow
NA
NA
Yellow fever virus
17D
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_7268Cdt white
NA
NA
Yellow fever virus
17D
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_7269Crotoxin
NA
NA
Yellow fever virus
17D
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_7270Crotapotin
NA
NA
Yellow fever virus
17D
Pathway
NA
Decrease (43 %)
NA
21723310
DrugRepV_7271Crotamin
NA
NA
Yellow fever virus
17D
Pathway
NA
Decrease (20 %)
NA
21723310
DrugRepV_7272Convulxin
NA
NA
Yellow fever virus
17D
Pathway
NA
Decrease (22 %)
NA
21723310
DrugRepV_7273PLA2-IC
NA
NA
Yellow fever virus
17D
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_7274PLA2-IC
NA
NA
Yellow fever virus
17D
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_7275Cdt yellow
NA
NA
Yellow fever virus
17D
Pathway
Virucidal assay
Decrease (50 %)
NA
21723310
DrugRepV_7276Cdt white
NA
NA
Yellow fever virus
17D
Pathway
Virucidal assay
Decrease (50 %)
NA
21723310
DrugRepV_7277Crotoxin
NA
NA
Yellow fever virus
17D
Pathway
Virucidal assay
Decrease (50 %)
NA
21723310
DrugRepV_7278Crotapotin
NA
NA
Yellow fever virus
17D
Pathway
Virucidal assay
Decrease (50 %)
NA
21723310
DrugRepV_7279Crotamin
NA
NA
Yellow fever virus
17D
Pathway
Virucidal assay
Decrease (14.34 %)
NA
21723310
DrugRepV_7280Convulxin
NA
NA
Yellow fever virus
17D
Pathway
Virucidal assay
Decrease (25.5 %)
NA
21723310
DrugRepV_7281PLA2-IC
NA
NA
Yellow fever virus
17D
Pathway
Virucidal assay
Decrease (50 %)
NA
21723310
DrugRepV_7282PLA2-IC
NA
NA
Yellow fever virus
17D
Pathway
Virucidal assay
Decrease (50 %)
NA
21723310
DrugRepV_7283Cdt yellow
NA
NA
Yellow fever virus
17D
Pathway
Adsorption assay
Decrease (50 %)
NA
21723310
DrugRepV_7284Cdt white
NA
NA
Yellow fever virus
17D
Pathway
Adsorption assay
Decrease (50 %)
NA
21723310
DrugRepV_7285Crotoxin
NA
NA
Yellow fever virus
17D
Pathway
Adsorption assay
Decrease (50 %)
NA
21723310
DrugRepV_7286Crotapotin
NA
NA
Yellow fever virus
17D
Pathway
Adsorption assay
Decrease (50 %)
NA
21723310
DrugRepV_7287Crotamin
NA
NA
Yellow fever virus
17D
Pathway
Adsorption assay
Decrease (50 %)
NA
21723310
DrugRepV_7288Convulxin
NA
NA
Yellow fever virus
17D
Pathway
Adsorption assay
Decrease (50 %)
NA
21723310
DrugRepV_7289PLA2-IC
NA
NA
Yellow fever virus
17D
Pathway
Adsorption assay
Decrease (50 %)
NA
21723310
DrugRepV_7290PLA2-IC
NA
NA
Yellow fever virus
17D
Pathway
Adsorption assay
Decrease (50 %)
NA
21723310
DrugRepV_7291Cdt yellow
NA
NA
Yellow fever virus
17D
Pathway
Internalization assay
Decrease (50 %)
NA
21723310
DrugRepV_7292Cdt white
NA
NA
Yellow fever virus
17D
Pathway
Internalization assay
Decrease (50 %)
NA
21723310
DrugRepV_7293Crotoxin
NA
NA
Yellow fever virus
17D
Pathway
Internalization assay
Decrease (50 %)
NA
21723310
DrugRepV_7294Crotapotin
NA
NA
Yellow fever virus
17D
Pathway
Internalization assay
Decrease (50 %)
NA
21723310
DrugRepV_7295Crotamin
NA
NA
Yellow fever virus
17D
Pathway
Internalization assay
Decrease (32 %)
NA
21723310
DrugRepV_7296Convulxin
NA
NA
Yellow fever virus
17D
Pathway
Internalization assay
Decrease (-70 %)
NA
21723310
DrugRepV_7297PLA2-IC
NA
NA
Yellow fever virus
17D
Pathway
Internalization assay
Decrease (50 %)
NA
21723310
DrugRepV_7298PLA2-IC
NA
NA
Yellow fever virus
17D
Pathway
Internalization assay
Decrease (46 %)
NA
21723310
DrugRepV_7299(3E)-N-tert-butyl-2-oxo-4-phenylbut-3-enamide
NA
NA
West Nile virus
NA
Pathway
Protease assay
Decrease (20 %)
NA
21641807
DrugRepV_7300(3E)-N-tert-butyl-3-methyl-2-oxo-4-phenylbut-3-enamide
NA
NA
West Nile virus
NA
Pathway
Protease assay
Decrease (0 %)
NA
21641807
DrugRepV_7301(3E)-N-tert-butyl-2-oxo-4-(thiophen-2-yl)but-3-enamide
NA
NA
West Nile virus
NA
Pathway
Protease assay
Decrease (20.3 %)
NA
21641807
DrugRepV_7302(3E)-N-tert-butyl-4-(4-methoxyphenyl)-2-oxobut-3-enamide
NA
NA
West Nile virus
NA
Pathway
Protease assay
Decrease (27.3 %)
NA
21641807
DrugRepV_7303(3E)-N-tert-butyl-4-(3,4-dimethoxyphenyl)-2-oxobut-3-enamide
NA
NA
West Nile virus
NA
Pathway
Protease assay
Decrease (31 %)
NA
21641807
DrugRepV_7304(3E)-N-tert-butyl-4-(4-hydroxyphenyl)-2-oxobut-3-enamide
NA
NA
West Nile virus
NA
Pathway
Protease assay
Decrease (31.4 %)
NA
21641807
DrugRepV_7305(3E)-4-(4-aminophenyl)-N-tert-butyl-2-oxobut-3-enamide
NA
NA
West Nile virus
NA
Pathway
Protease assay
Decrease (39.5 %)
NA
21641807
DrugRepV_7306(3E)-N-tert-butyl-4-(4-chlorophenyl)-2-oxobut-3-enamide
NA
NA
West Nile virus
NA
Pathway
Protease assay
Decrease (6.3 %)
NA
21641807
DrugRepV_7307(3E)-N-tert-butyl-4-(1H-indol-3-yl)-2-oxobut-3-enamide
NA
NA
West Nile virus
NA
Pathway
Protease assay
Decrease (40.6 %)
NA
21641807
DrugRepV_7308(3E)-N-tert-butyl-4-[4-(dimethylamino)phenyl]-2-oxobut-3-enamide
NA
NA
West Nile virus
NA
Pathway
Protease assay
Decrease (33.9 %)
NA
21641807
DrugRepV_7309(3E)-N-cyclopropyl-2-oxo-4-phenylbut-3-enamide
NA
NA
West Nile virus
NA
Pathway
Protease assay
Decrease (20 %)
NA
21641807
DrugRepV_73102-[(3E)-2-oxo-4-phenylbut-3-enamido]ethyl acetate
NA
NA
West Nile virus
NA
Pathway
Protease assay
Decrease (29.8 %)
NA
21641807
DrugRepV_7311(3E)-2-oxo-4-phenyl-N-(1-phenylethyl)but-3-enamide
NA
NA
West Nile virus
NA
Pathway
Protease assay
Decrease (12.2 %)
NA
21641807
DrugRepV_7312methyl 3-hydroxy-2-[(3E)-2-oxo-4-phenylbut-3-enamido]propanoate
NA
NA
West Nile virus
NA
Pathway
Protease assay
Decrease (27.5 %)
NA
21641807
DrugRepV_7313CW-33A
NA
NA
Japanese encephalitis virus
T1P1
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
30413749
DrugRepV_7314CW-33
NA
NA
Japanese encephalitis virus
T1P1
Pathway
Virus yield reduction assay
Decrease (50 %)
NA
30413749
DrugRepV_7315CW-33A
NA
NA
Japanese encephalitis virus
T1P1
Pathway
Plaque assay
Decrease (50 %)
NA
30413749
DrugRepV_7316CW-33
NA
NA
Japanese encephalitis virus
T1P1
Pathway
Plaque assay
Decrease (50 %)
NA
30413749
DrugRepV_7319MJ-47
NA
NA
Japanese encephalitis virus
JEVSRIP
Pathway
Flow cytometry
Decrease (50 %)
NA
28394283
DrugRepV_7320N-(6-methanesulfonyl-1,3-benzothiazol-2-yl)-4-[(4-nitro-1H-pyrazol-1-yl)methyl]benzamide
NA
NA
Japanese encephalitis virus
NS3 helicase
Pathway
Flow cytometry
Decrease (79 %)
NA
27679979
DrugRepV_7321N-[6-({[(thiophen-2-yl)formamido]methanethioyl}amino)-1,3-benzothiazol-2-yl]butanamide
NA
NA
Japanese encephalitis virus
NS3 helicase
Pathway
Flow cytometry
Decrease (73 %)
NA
27679979
DrugRepV_7322N-(6-methanesulfonyl-1,3-benzothiazol-2-yl)-4-[(4-nitro-1H-pyrazol-1-yl)methyl]benzamide
NA
NA
Japanese encephalitis virus
P3
Pathway
Western blot
Decrease (70.1 %)
NA
27679979
DrugRepV_7323N-[6-({[(thiophen-2-yl)formamido]methanethioyl}amino)-1,3-benzothiazol-2-yl]butanamide
NA
NA
Japanese encephalitis virus
P3
Pathway
Western blot
Decrease (94.8 %)
NA
27679979
DrugRepV_7324N-(6-methanesulfonyl-1,3-benzothiazol-2-yl)-4-[(4-nitro-1H-pyrazol-1-yl)methyl]benzamide
NA
NA
Japanese encephalitis virus
P3
Pathway
Immunoflourescence assay
Decrease (86.71 %)
NA
27679979
DrugRepV_7325N-[6-({[(thiophen-2-yl)formamido]methanethioyl}amino)-1,3-benzothiazol-2-yl]butanamide
NA
NA
Japanese encephalitis virus
P3
Pathway
Immunoflourescence assay
Decrease (89.3 %)
NA
27679979
DrugRepV_7326N-(6-methanesulfonyl-1,3-benzothiazol-2-yl)-4-[(4-nitro-1H-pyrazol-1-yl)methyl]benzamide
NA
NA
Japanese encephalitis virus
P3
Pathway
Plaque assay
Decrease (2 log pfu/ml)
NA
27679979
DrugRepV_7327N-[6-({[(thiophen-2-yl)formamido]methanethioyl}amino)-1,3-benzothiazol-2-yl]butanamide
NA
NA
Japanese encephalitis virus
P3
Pathway
Plaque assay
Decrease (2 log pfu/ml)
NA
27679979
DrugRepV_7328N-(6-methanesulfonyl-1,3-benzothiazol-2-yl)-4-[(4-nitro-1H-pyrazol-1-yl)methyl]benzamide
NA
NA
Japanese encephalitis virus
P3
Pathway
Cell viability assay
Decrease (50 %)
NA
27679979
DrugRepV_7329N-[6-({[(thiophen-2-yl)formamido]methanethioyl}amino)-1,3-benzothiazol-2-yl]butanamide
NA
NA
Japanese encephalitis virus
P3
Pathway
Cell viability assay
Decrease (50 %)
NA
27679979
DrugRepV_7330CW-33
NA
NA
Japanese encephalitis virus
T1P1
Pathway
Cytopathic effect (CPE) assay
Decrease
NA
27563890
DrugRepV_7331CW-33
NA
NA
Japanese encephalitis virus
T1P1
Pathway
Cytopathic effect (CPE) assay
Decrease
NA
27563890
DrugRepV_7332CW-33
NA
NA
Japanese encephalitis virus
T1P1
Pathway
Plaque assay
Decrease (5 times pfu/ml)
NA
27563890
DrugRepV_7333CW-33
NA
NA
Japanese encephalitis virus
T1P1
Pathway
Plaque assay
Decrease (3 times pfu/ml)
NA
27563890
DrugRepV_7334CW-33
NA
NA
Japanese encephalitis virus
T1P1
Pathway
Plaque assay
Decrease (50 %)
NA
27563890
DrugRepV_7335FGIN-1-27
NA
NA
Japanese encephalitis virus
P3
Pathway
Plaque assay
Decrease (2 log %)
NA
24348901
DrugRepV_7338FGIN-1-27
NA
NA
Japanese encephalitis virus
P3
Pathway
Immunoflourescence assay
Decrease (80 %)
NA
24348901
DrugRepV_7341FGIN-1-27
NA
NA
Japanese encephalitis virus
P3
Pathway
Luminescence assay
Decrease (50 %)
NA
24348901
DrugRepV_7348Indigo
NA
NA
Japanese encephalitis virus
T1P1
Pathway
Plaque assay
Decrease (50 %)
NA
22911608
DrugRepV_7349Indirubin
NA
NA
Japanese encephalitis virus
T1P1
Pathway
Plaque assay
Decrease (50 %)
Investigational
22911608
DrugRepV_7350Indirubin
NA
NA
Japanese encephalitis virus
Beijing-1
Pathway
Survival assay
Increase
Investigational
22911608
DrugRepV_7351NG-monomethyl-L-arginine
NA
Obesity | Type 2 Diabetes | Ocular Physiology | Regional Blood Flow
Japanese encephalitis virus
78668A
Pathway
Survival assay
Decrease
Approved, Investigational
10762444
DrugRepV_7352N-nitro-L-arginine methyl ester
NA
NA
Japanese encephalitis virus
RP-9
Pathway
Survival assay
Decrease
NA
9188590
DrugRepV_7353S-nitroso-N-acetylpenicillamine
NA
NA
Japanese encephalitis virus
NT109
Pathway
Plaque assay
Decrease (3 log pfu/ml)
NA
9188590
DrugRepV_7354Glycine-Zn
NA
NA
Japanese encephalitis virus
Nakayama
Pathway
Paralysis
Increase (16.37 %)
NA
14011545
DrugRepV_7355DL-Phenylalanine-Zn
NA
NA
Japanese encephalitis virus
Nakayama
Pathway
Paralysis
No significant effect (3.63 %)
NA
14011545
DrugRepV_7356L-Leucine-Zn
NA
NA
Japanese encephalitis virus
Nakayama
Pathway
Paralysis
No significant effect (3.63 %)
NA
14011545
DrugRepV_7357DL-Aspartic acid -Zn
NA
NA
Japanese encephalitis virus
Nakayama
Pathway
Paralysis
Decrease (23.63 %)
NA
14011545
DrugRepV_7358DL-Asparagine-Zn
NA
NA
Japanese encephalitis virus
Nakayama
Pathway
Paralysis
Decrease (36.36 %)
NA
14011545
DrugRepV_7359DL-Alanine-Zn
NA
NA
Japanese encephalitis virus
Nakayama
Pathway
Paralysis
Increase (9 %)
NA
14011545
DrugRepV_7360L-Cysteine-Zn
NA
NA
Japanese encephalitis virus
Nakayama
Pathway
Paralysis
Decrease (18.18 %)
NA
14011545
DrugRepV_7361DL-Lysine-Zn
NA
NA
Japanese encephalitis virus
Nakayama
Pathway
Paralysis
Increase (9 %)
NA
14011545
DrugRepV_7362L-Tyrosine-Zn
NA
NA
Japanese encephalitis virus
Nakayama
Pathway
Paralysis
No significant effect (10 %)
NA
14011545
DrugRepV_7363DL-Methionine-Zn
NA
NA
Japanese encephalitis virus
Nakayama
Pathway
Paralysis
Increase (20 %)
NA
14011545
DrugRepV_73642-Picolinic acid-Zn
NA
NA
Japanese encephalitis virus
Nakayama
Pathway
Paralysis
Increase (0.45 %)
NA
14011545
DrugRepV_7365Guanidine-Zn
NA
NA
Japanese encephalitis virus
Nakayama
Pathway
Paralysis
Increase (9.5 %)
NA
14011545
DrugRepV_7366Diethyl Dithiocarbamic Acid-Zn
NA
NA
Japanese encephalitis virus
Nakayama
Pathway
Paralysis
Increase (27.72 %)
NA
14011545
DrugRepV_7367Diphenylthiocarbazone-Zn
NA
NA
Japanese encephalitis virus
Nakayama
Pathway
Paralysis
Increase (12.14 %)
NA
14011545
DrugRepV_73688-Hydroxyquinoline-Zn
NA
NA
Japanese encephalitis virus
Nakayama
Pathway
Paralysis
No significant effect (8.6 %)
NA
14011545
DrugRepV_73693,4-Dimercaptotoluene-Zn
NA
NA
Japanese encephalitis virus
Nakayama
Pathway
Paralysis
Increase (10 %)
NA
14011545
DrugRepV_73701,10-Phenanthroline-Zn
NA
NA
Japanese encephalitis virus
Nakayama
Pathway
Paralysis
No significant effect (5 %)
NA
14011545
DrugRepV_73711,10-Phenanthroline-3,4-dimercaptotoluene-Zn
NA
NA
Japanese encephalitis virus
Nakayama
Pathway
Paralysis
Decrease (35 %)
NA
14011545
DrugRepV_7372Luteolin
NA
NA
Japanese encephalitis virus
SX09S01
Pathway
Plaque assay
Decrease (50 %)
NA
27126774
DrugRepV_7373Luteolin
NA
NA
Japanese encephalitis virus
SX09S01
Pathway
Plaque assay
Decrease (2 log Log PFU/ml)
NA
27126774
DrugRepV_7374Luteolin
NA
NA
Japanese encephalitis virus
SX09S01
Pathway
Western blot
Decrease
NA
27126774
DrugRepV_7375Chrysophanol
NA
NA
Japanese encephalitis virus
T1P1
Pathway
Plaque assay
Decrease (50 %)
NA
24395532
DrugRepV_7376Aloe-emodin
NA
NA
Japanese encephalitis virus
T1P1
Pathway
Plaque assay
Decrease (50 %)
NA
24395532
DrugRepV_7377Aloe-emodin
NA
NA
Japanese encephalitis virus
T1P1
Pathway
Plaque assay
Decrease (50 %)
NA
18701259
DrugRepV_7378Aloe-emodin
NA
NA
Japanese encephalitis virus
T1P1
Pathway
Plaque assay
Decrease (50 %)
NA
18701259
DrugRepV_7379Shikonin
NA
NA
Japanese encephalitis virus
T1P1
Pathway
Plaque assay
Decrease (50 %)
NA
18701259
DrugRepV_7380Shikonin
NA
NA
Japanese encephalitis virus
T1P1
Pathway
Plaque assay
Decrease (50 %)
NA
18701259
DrugRepV_7381Arecoline
NA
NA
Japanese encephalitis virus
T1P1
Pathway
Plaque assay
Decrease (50 %)
Experimental
18701259
DrugRepV_7382Arecoline
NA
NA
Japanese encephalitis virus
T1P1
Pathway
Plaque assay
Decrease (50 %)
Experimental
18701259
DrugRepV_7383Hesperetin
NA
NA
Japanese encephalitis virus
T1P1
Pathway
Plaque assay
Decrease (50 %)
Experimental
18701259
DrugRepV_7384Dehydroepiandrosterone
NA
Schizophrenia
Japanese encephalitis virus
NT113
Pathway
Plaque assay
Decrease
Approved
16099910
DrugRepV_7385Dehydroepiandrosterone
NA
Schizophrenia
Japanese encephalitis virus
NT113
Pathway
Slot Blot analysis
Decrease
Approved
16099910
DrugRepV_7386Dehydroepiandrosterone
NA
Schizophrenia
Japanese encephalitis virus
NT113
Pathway
Western blot
Decrease
Approved
16099910
DrugRepV_7387SCH16-Ribavirin
NA
NA
Japanese encephalitis virus
P20778
Pathway
Cytopathic effect (CPE) assay
Decrease
NA
22738253
DrugRepV_7388SCH16-Mycophenolic acid
NA
NA
Japanese encephalitis virus
P20778
Pathway
Cytopathic effect (CPE) assay
Decrease
NA
22738253
DrugRepV_7389Delphinidin Chloride
NA
NA
West Nile virus
NY-99
Pathway
Plaque assay
Decrease (O.6 Log)
NA
28744282
DrugRepV_7390Cyanidin Chloride
NA
NA
West Nile virus
NY-99
Pathway
Plaque assay
No significant effect (No significant effect Log)
NA
28744282
DrugRepV_7392Epicatechin
NA
Pre-diabetes
West Nile virus
NY-99
Pathway
Plaque assay
No significant effect (No significant effect Log)
Investigational
28744282
DrugRepV_7393Epigallocatechin
NA
NA
West Nile virus
NY-99
Pathway
Plaque assay
Decrease (0.5 Log)
Experimental
28744282
DrugRepV_7395Delphinidin Chloride
NA
NA
West Nile virus
NY-99
Pathway
RT-PCR
Decrease (0.7 Copies/cell)
NA
28744282
DrugRepV_7397Nordihydroguaiaretic Acid
NA
Actinic keratoses
West Nile virus
NY-99
Pathway
Plaque assay
Decrease (50 %)
Approved, Investigational
28507114
DrugRepV_7398Nordihydroguaiaretic Acid
NA
Actinic keratoses
West Nile virus
NY-99
Pathway
Plaque assay
Decrease (50 %)
Approved, Investigational
28507114
DrugRepV_7400PF-429242
NA
NA
West Nile virus
NY-99
Pathway
Plaque assay
Decrease (0.4 Log)
NA
28507114
DrugRepV_7401Fatostatin
NA
NA
West Nile virus
NY-99
Pathway
Plaque assay
Decrease (0.7 Log)
NA
28507114
DrugRepV_7402Zileuton
NA
Asthma
West Nile virus
NY-99
Pathway
Plaque assay
No significant change (No significant change Log)
Approved / Withdrawn
28507114
DrugRepV_7403BCX4430
NA
Ebola virus
West Nile virus
Eg101
Pathway
Plaque assay
Decrease (50 %)
Investigational
28336346
DrugRepV_7404BCX4430 Hydrochloride
NA
Ebola virus
West Nile virus
Eg101
Pathway
Plaque assay
Decrease (50 %)
Investigational
28336346
DrugRepV_7405(1S,2R,3S)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]uracil
NA
NA
West Nile virus
New York isolate
Pathway
CPE inhibition assay
Decrease (50 %)
NA
11689085
DrugRepV_7406(1S,2R,3S)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]thymine
NA
NA
West Nile virus
New York isolate
Pathway
CPE inhibition assay
Decrease (50 %)
NA
11689085
DrugRepV_7407(1S,2R,3S)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]-5-fluorouracil
NA
NA
West Nile virus
New York isolate
Pathway
CPE inhibition assay
Decrease (50 %)
NA
11689085
DrugRepV_7408(1S,2R,3S)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]cytosine
NA
NA
West Nile virus
New York isolate
Pathway
CPE inhibition assay
Decrease (50 %)
NA
11689085
DrugRepV_7409(1S,2R,3S)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]-5-fluorocytosine
NA
NA
West Nile virus
New York isolate
Pathway
CPE inhibition assay
Decrease (50 %)
NA
11689085
DrugRepV_7410L-Neplanocin A
NA
NA
West Nile virus
New York isolate
Pathway
CPE inhibition assay
Decrease (50 %)
NA
11689085
DrugRepV_7411(1S,2R,3S)-9-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl] hypoxanthine
NA
NA
West Nile virus
New York isolate
Pathway
CPE inhibition assay
Decrease (50 %)
NA
11689085
DrugRepV_7412(1S,2R,3S)-9-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]guanine
NA
NA
West Nile virus
New York isolate
Pathway
CPE inhibition assay
Decrease (50 %)
NA
11689085
DrugRepV_7413Cyclopentenyl nucleosides
NA
NA
West Nile virus
New York isolate
Pathway
CPE inhibition assay
Decrease (50 %)
NA
11689085
DrugRepV_7414(1R,2S,3R)-9-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl] hypoxanthine
NA
NA
West Nile virus
New York isolate
Pathway
CPE inhibition assay
Decrease (50 %)
NA
11689085
DrugRepV_7415(1R,2S,3R)-9-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]guanine
NA
NA
West Nile virus
New York isolate
Pathway
CPE inhibition assay
Decrease (50 %)
NA
11689085
DrugRepV_7416(1S,2R,3S)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]uracil
NA
NA
West Nile virus
New York isolate
Pathway
CPE inhibition assay
Decrease (50 %)
NA
11689085
DrugRepV_7417(1R,2S,3R)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]thymine
NA
NA
West Nile virus
New York isolate
Pathway
CPE inhibition assay
Decrease (50 %)
NA
11689085
DrugRepV_7418(1R,2S,3R)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]-5-fluorouracil
NA
NA
West Nile virus
New York isolate
Pathway
CPE inhibition assay
Decrease (50 %)
NA
11689085
DrugRepV_7419(1R,2S,3R)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]cytosine
NA
NA
West Nile virus
New York isolate
Pathway
CPE inhibition assay
Decrease (50 %)
NA
11689085
DrugRepV_7420(1R,2S,3R)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]-5-fluorocytosine
NA
NA
West Nile virus
New York isolate
Pathway
CPE inhibition assay
Decrease (50 %)
NA
11689085
DrugRepV_7421N-nonyl-deoxynojirimycin
NA
NA
West Nile virus
NA
Pathway
Yield reduction assay
Decrease (50 %)
NA
17354651
DrugRepV_7422N-pentyl-(1-hydroxycyclohexyl)-DNJ
NA
NA
West Nile virus
NA
Pathway
Yield reduction assay
Decrease (50 %)
NA
17354651
DrugRepV_7423N-Propylcyclohexyl-DNJ
NA
NA
West Nile virus
NA
Pathway
Yield reduction assay
Decrease (50 %)
NA
17354651
DrugRepV_7424N-Butylcyclohexyl-DNJ
NA
NA
West Nile virus
NA
Pathway
Yield reduction assay
Decrease (50 %)
NA
17354651
DrugRepV_74266-Azauridine
NA
Cancer
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_74276-Azauridine
NA
Cancer
West Nile virus
Uganda strain B 956
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_74286-Azauridine triacetate
NA
NA
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_74296-Azauridine triacetate
NA
NA
West Nile virus
Uganda strain B 956
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_7430Pyrazofurin
NA
NA
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_7431Pyrazofurin
NA
NA
West Nile virus
Uganda strain B 956
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_74322-Thio-6-azauridine
NA
NA
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_74332-Thio-6-azauridine
NA
NA
West Nile virus
Uganda strain B 956
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_74346-Azauridine
NA
Cancer
West Nile virus
New York
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_74356-Azauridine
NA
Cancer
West Nile virus
Uganda strain B 956
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_74366-Azauridine triacetate
NA
NA
West Nile virus
New York
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_74376-Azauridine triacetate
NA
NA
West Nile virus
Uganda strain B 956
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_7438Pyrazofurin
NA
NA
West Nile virus
New York
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_7439Pyrazofurin
NA
NA
West Nile virus
Uganda strain B 956
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_74402-Thio-6-azauridine
NA
NA
West Nile virus
New York
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_74412-Thio-6-azauridine
NA
NA
West Nile virus
Uganda strain B 956
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_74423-Deazaguanosine
NA
NA
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_7445Ribamidine
NA
NA
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_7446Ribamidine
NA
NA
West Nile virus
Uganda strain B 956
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_7449Selenazofurin
NA
NA
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_7450Selenazofurin
NA
NA
West Nile virus
Uganda strain B 956
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_7452beta-Methylene TAD
NA
NA
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_7453beta-Methylene TAD
NA
NA
West Nile virus
Uganda strain B 956
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_74543-Deazaguanosine
NA
NA
West Nile virus
New York
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_7457Ribamidine
NA
NA
West Nile virus
New York
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_7458Ribamidine
NA
NA
West Nile virus
Uganda strain B 956
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_7461Selenazofurin
NA
NA
West Nile virus
New York
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_7462Selenazofurin
NA
NA
West Nile virus
Uganda strain B 956
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_7464beta-Methylene TAD
NA
NA
West Nile virus
New York
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_7465beta-Methylene TAD
NA
NA
West Nile virus
Uganda strain B 956
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_74663-Deazauridine
NA
NA
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_74673-Deazauridine
NA
NA
West Nile virus
Uganda strain B 956
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_7468Cyclopentenylcytosine
NA
NA
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_7469Cyclopentenylcytosine
NA
NA
West Nile virus
Uganda strain B 956
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_74703-Deazauridine
NA
NA
West Nile virus
New York
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_74713-Deazauridine
NA
NA
West Nile virus
Uganda strain B 956
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_7472Cyclopentenylcytosine
NA
NA
West Nile virus
New York
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_7473Cyclopentenylcytosine
NA
NA
West Nile virus
Uganda strain B 956
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_74805-fluorouridine
NA
Cancer
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
Experimental
12076755
DrugRepV_74815-fluorouridine
NA
Cancer
West Nile virus
New York
Pathway
NR assay
Decrease (50 %)
Experimental
12076755
DrugRepV_7482(S )-DHPA
NA
NA
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_7483(S )-DHPA
NA
NA
West Nile virus
Uganda strain B 956
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_74843-Deazaneplanocin A
NA
NA
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_7485(S )-DHPA
NA
NA
West Nile virus
New York
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_7486(S )-DHPA
NA
NA
West Nile virus
Uganda strain B 956
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_74873-Deazaneplanocin A
NA
NA
West Nile virus
New York
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_74886-Bromotoyocamycin
NA
NA
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_7489Formycin B
NA
NA
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
Experimental
12076755
DrugRepV_74906-Bromotoyocamycin
NA
NA
West Nile virus
New York
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_7491Formycin B
NA
NA
West Nile virus
New York
Pathway
NR assay
Decrease (50 %)
Experimental
12076755
DrugRepV_74922-Thiouracil
NA
NA
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_7494Cyclopentyluracil
NA
NA
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_7495Dihydro-5-azacytidine
NA
NA
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_7496Uridine 2,3-dialdehyde
NA
NA
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_74972-Thiouracil
NA
NA
West Nile virus
New York
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_7499Cyclopentyluracil
NA
NA
West Nile virus
New York
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_7500Dihydro-5-azacytidine
NA
NA
West Nile virus
New York
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_7501Uridine 2,3-dialdehyde
NA
NA
West Nile virus
New York
Pathway
NR assay
Decrease (50 %)
NA
12076755
DrugRepV_75026-Azauridine
NA
Cancer
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_75036-Azauridine triacetate
NA
NA
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_7504Pyrazofurin
NA
NA
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_7505Selenazofurin
NA
NA
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_7508Cyclopentenylcytosine
NA
NA
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
NA
12076755
DrugRepV_75096-Azauridine
NA
Cancer
West Nile virus
New York
Pathway
Virus yield reduction assay
Decrease (90 %)
NA
12076755
DrugRepV_7510Pyrazofurin
NA
NA
West Nile virus
New York
Pathway
Virus yield reduction assay
Decrease (90 %)
NA
12076755
DrugRepV_7513Cyclopentenylcytosine
NA
NA
West Nile virus
New York
Pathway
Virus yield reduction assay
Decrease (90 %)
NA
12076755
DrugRepV_7514Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Polio virus
NA
Pathway
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_7515Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
West Nile virus
NA
Pathway
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_7516Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_7517Aloe-emodin
NA
NA
Enterovirus
EV71
Pathway
Plaque assay
Decrease (50 %)
NA
18701259
DrugRepV_7518Aloe-emodin
NA
NA
Enterovirus
EV71
Pathway
Plaque assay
Decrease (50 %)
NA
18701259
DrugRepV_7520beta-D-cyclopentenyl cytosine
NA
NA
Vaccinia virus
Copenhagen
Pathway
NA
Decrease (50 %)
NA
14604375
DrugRepV_7521beta-D-cyclopentenyl-5-iodocytidine
NA
NA
Vaccinia virus
Copenhagen
Pathway
NA
Decrease (50 %)
NA
14604375
DrugRepV_7522beta-D-Cyclopentenyl-5-chlorocytidine
NA
NA
Vaccinia virus
Copenhagen
Pathway
NA
Decrease (50 %)
NA
14604375
DrugRepV_7523beta-D-cyclopentenyl-5-bromocytidine
NA
NA
Vaccinia virus
Copenhagen
Pathway
NA
Decrease (50 %)
NA
14604375
DrugRepV_7524Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Vaccinia virus
NA
Pathway
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_7575Merimepodib
NA
NA
SARS Coronavirus-2
SARS-CoV-2 USA-WA1/2020
NA
RT-PCR
Decrease (50 %)
Investigational
32438446
DrugRepV_7576Merimepodib
NA
NA
SARS Coronavirus-2
SARS-CoV-2 USA-WA1/2020
NA
RT-PCR
Decrease (90 %)
Investigational
32438446
DrugRepV_7664Cetilistat
NA
Obesity
SARS Coronavirus-2
NA
Plaque reduction assay
Decrease (50 %)
Investigational
32473310
DrugRepV_7668Cetilistat
NA
Obesity
SARS Coronavirus-2
NA
Viral load reduction assay
Decrease (90 %)
Investigational
32473310
DrugRepV_7673ROC-325
NA
NA
SARS Coronavirus-2
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
32511355
DrugRepV_7690S1RA
NA
NA
SARS Coronavirus-2
NA
NA
Decrease (50 %)
NA
32577649
DrugRepV_7693Z-FA-FMK
NA
NA
SARS Coronavirus-2
NA
NA
Decrease (50 %)
NA
32577649
DrugRepV_7694Lactoferrin
NA
NA
SARS Coronavirus-2
NA
NA
Decrease (50 %)
NA
32577649
DrugRepV_7695Nafamostat
NA
Blood vessel coagulation | Hemorrhagic lesions
SARS Coronavirus-2
NA
NA
Decrease (50 %)
Investigational
32532094
DrugRepV_7696Immunoglobulin F(ab’)2
NA
NA
SARS Coronavirus-2
NA
NA
Decrease (50 %)
NA
32659292
DrugRepV_7697Unfractionated Heparin
NA
Prophylaxis and Venous thrombosis
SARS Coronavirus-2
NA
NA
Decrease (50 %)
Approved, Investigational
32577638
DrugRepV_7698UFH-de6S
NA
NA
SARS Coronavirus-2
NA
NA
Decrease (50 %)
NA
32577638
DrugRepV_7700Enoxaparin-de6S
NA
NA
SARS Coronavirus-2
NA
NA
Decrease (50 %)
NA
32577638
DrugRepV_7701Pegasys
NA
Hepatitis C Virus
SARS Coronavirus-2
NA
Plaque reduction assay
Decrease (50 %)
Approved, Investigational
32532085
DrugRepV_7705Immukin
NA
Chronic granulomatous disease and Osteopetrosis
SARS Coronavirus-2
NA
Plaque reduction assay
Decrease (50 %)
Approved, Investigational
32532085
DrugRepV_770625-Hydroxycholesterol
NA
NA
SARS Coronavirus-2
NA
NA
Plaque reduction assay
Decrease (50 %)
Experimental
32532085
DrugRepV_7707AM580
NA
NA
SARS Coronavirus-2
NA
Plaque reduction assay
Decrease (50 %)
NA
32532085
DrugRepV_7710AMG-2674
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7713DS-6930
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7714Elopiprazole
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7715Hanfangchin A
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7716KW 8232
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7717N-tert-Butylisoquine
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7718R 82913
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
Experimental
32707573
DrugRepV_7719SB-616234A
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7720SDZ-62-434
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7721SL-11128
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7722YH-1238
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7724AMG-2674
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7727Elopiprazole
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7728Hanfangchin A
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7729MLN-3897
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7730KW 8232
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7731N-tert-Butylisoquine
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7732SB-616234A
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7733SDZ-62-434
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7734SL-11128
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_77368-(2-Chlorostyryl)caffeine
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7737AMG-2674
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7739Elopiprazole
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7740Hanfangchin A
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7741KW 8232
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7742MLN-3897
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7743N-tert-Butylisoquine
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7744SB-616234A
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7745SDZ-62-434
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7746YH-1238
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7748Apilimod
NA
Crohn's disease | Psoriasis | Psoriatic disorders
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
Investigational
32707573
DrugRepV_7749VBY-825
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7750ONO 5334
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7751Z LVG CHN2
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7752MDL 28170
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7753SL-11128
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7755DS-6930
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7756R 82913
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
Experimental
32707573
DrugRepV_7757Hanfangchin A
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7758SB-616234A
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7759MLN-3897
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7760VBY-825
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7761Apilimod
NA
Crohn's disease | Psoriasis | Psoriatic disorders
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
Investigational
32707573
DrugRepV_7762VBY-825
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7763ONO 5334
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7764Z LVG CHN2
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7765MDL 28170
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7766Apilimod
NA
Crohn's disease | Psoriasis | Psoriatic disorders
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
Investigational
32707573
DrugRepV_7767VBY-825
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7768ONO 5334
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7769Z LVG CHN2
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7770MDL 28170
NA
NA
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
NA
32707573
DrugRepV_7773Galidesivir
NA
Ebolavirus
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Investigational
32687696
DrugRepV_7775Camostat mesylate
NA
Pancreatitis
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Experimental
32687696
DrugRepV_7776Nafamostat Mesylate
NA
Blood vessel coagulation | Hemorrhagic lesions
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Investigational
32687696
DrugRepV_7778Apilimod
NA
Crohn's disease | Psoriasis | Psoriatic disorders
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Investigational
32687696
DrugRepV_7788SSAA09E3
NA
NA
Severe acute respiratory syndrome coronavirus
Toronto-2
NA
Dose-dependence fluorescence inhibition assay
Decrease (50 %)
NA
23678171
DrugRepV_7789SSAA09E1
NA
NA
Severe acute respiratory syndrome coronavirus
Toronto-2
NA
Dose-dependence fluorescence inhibition assay
Decrease (50 %)
NA
23678171
DrugRepV_7790SSAA09E2
NA
NA
Severe acute respiratory syndrome coronavirus
Toronto-2
NA
Dose-dependence fluorescence inhibition assay
Decrease (50 %)
NA
23678171
DrugRepV_7791Ferruginol
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Cell based assay
Decrease (50 %)
NA
17663539
DrugRepV_7792Dehydroabieta-7-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_7793Cryptojaponol
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_77948beta-hydroxyabieta-9(11),13- dien-12-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_77957beta-hydroxydeoxycryptojaponol
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_77966,7-dehydroroyleanone
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_77973beta,12-diacetoxyabieta-6,8,11,13- tetraene
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_7798Pinusolidic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_7799Forskolin
NA
Smooth muscle relaxant
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Experimental, Investigational
17663539
DrugRepV_7800Cedrane-3beta,12-diol
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_7801alpha-cadinol
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_7802Betulinic acid
NA
Dysplastic Nevus Syndrome
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Investigational
17663539
DrugRepV_7803Betulonic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_7804Hinokinin
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_7805Savinin
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_7806Honokiol
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_7807Magnolol
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_7808Curcumin
NA
Depressive disorder
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Approved
17663539
DrugRepV_7810Valinomycin
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Experimental
17663539
DrugRepV_78132-aminobenzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric assay
Decrease (50 %)
Experimental
16638531
DrugRepV_78142-(5-bromopyridin-3-yl)-1-[5-(4-chlorophenyl)furan-2-yl]-2-fluoroethanone
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
18295820
DrugRepV_7815ML188
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Luminescent Cell Viability Assay
Decrease (50 %)
NA
23231439
DrugRepV_7816ML300
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_78172-(benzotriazol-1-yl)-N-(4-phenylphenyl)-N-(thiophen-3-ylmethyl)acetamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_78185-Chloro-pyridin-3-yl Furan-2-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric assay
Decrease (50 %)
NA
17381079
DrugRepV_78195-Chloropyridin-3-yl Benzofuran-2-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric assay
Decrease (50 %)
NA
17381079
DrugRepV_78205-Bromo-pyridin-3-yl Furan-2-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric assay
Decrease (50 %)
NA
17381079
DrugRepV_78215-Chloro-pyridin-3-yl-1H-indole-2-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric assay
Decrease (50 %)
NA
17381079
DrugRepV_78225-Chloropyridin-3-yl-benzo-(b)-thiophene-2-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric assay
Decrease (50 %)
NA
17381079
DrugRepV_78235-Chloropyridin-3-yl-thiazole-4-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric assay
Decrease (50 %)
NA
17381079
DrugRepV_78245-Chloropyridin-3-yl-3-methoxybenzoate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric assay
Decrease (50 %)
NA
17381079
DrugRepV_78255-Chloropyridin-3-yl-5-(4-chlorophenyl)furan-2-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric assay
Decrease (50 %)
NA
17381079
DrugRepV_7826N-[4-[[2-(benzotriazol-1-yl)acetyl]-(thiophen-3-ylmethyl)amino]phenyl]propanamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_7827N-[4-[[2-(benzotriazol-1-yl)acetyl]-(thiophen-3-ylmethyl)amino]phenyl]-2-methylpropanamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_7828N-{4-[(1H-Benzotriazol-1-ylacetyl)(3-thienylmethyl)amino]phenyl}-2,2-dimethylpropanamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_7829N-[4-[[2-(benzotriazol-1-yl)acetyl]-(thiophen-3-ylmethyl)amino]phenyl]-3-methoxypropanamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_7830N-[4-[[2-(benzotriazol-1-yl)acetyl]-(thiophen-3-ylmethyl)amino]phenyl]cyclobutanecarboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_7831N-[4-[[2-(benzotriazol-1-yl)acetyl]-(thiophen-3-ylmethyl)amino]phenyl]cyclohexanecarboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_7832N-[4-[[2-(benzotriazol-1-yl)acetyl]-(thiophen-3-ylmethyl)amino]phenyl]benzamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_78332-methylpropyl N-[4-[[2-(benzotriazol-1-yl)acetyl]-(thiophen-3-ylmethyl)amino]phenyl]carbamate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_78342-(benzotriazol-1-yl)-N-[4-(methylamino)phenyl]-N-(thiophen-3-ylmethyl)acetamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_78352-(benzotriazol-1-yl)-N-[4-(benzylamino)phenyl]-N-(thiophen-3-ylmethyl)acetamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_78362-(benzotriazol-1-yl)-N-(4-pyridin-3-ylphenyl)-N-(thiophen-3-ylmethyl)acetamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_78372-(benzotriazol-1-yl)-N-[4-(2-methoxypyridin-3-yl)phenyl]-N-(thiophen-3-ylmethyl)acetamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_78382-(benzotriazol-1-yl)-N-(4-pyridin-4-ylphenyl)-N-(thiophen-3-ylmethyl)acetamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_78392-(benzotriazol-1-yl)-N-[4-(2-methoxypyrimidin-5-yl)phenyl]-N-(thiophen-3-ylmethyl)acetamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_7840benzyl N-[(2S)-1-[[(2S)-3-methyl-1-[[(2S)-4-methyl-1-oxo-1-[(4,4,4-trifluoro-3-oxo-1-phenylbutan-2-yl)amino]pentan-2-yl]amino]-1-oxobutan-2-yl]amino]-1-oxopropan-2-yl]carbamate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease (50 %)
NA
23747811
DrugRepV_7841(4S)-4-[[(2S)-2-[[(2S,3S)-2-[[(2S)-2-acetamido-3-methylbutanoyl]amino]-3-phenylmethoxybutanoyl]amino]-4-methylpentanoyl]amino]-N,N-dimethyl-6-(5-nitro-1,4-dioxo-3H-phthalazin-2-yl)-5-oxohexanamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease (50 %)
NA
23747811
DrugRepV_7842methyl (E,4S)-4-[[(2S)-4-methyl-2-[[(2S)-3-methyl-2-(phenylmethoxycarbonylamino)butanoyl]amino]pentanoyl]amino]-5-[(3S)-2-oxopyrrolidin-3-yl]pent-2-enoate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease (50 %)
NA
23747811
DrugRepV_7843ethyl 3-[(3-amino-3-oxopropyl)-[[(2R,5S)-2-benzyl-7-methyl-4-oxo-5-(phenylmethoxycarbonylamino)octanoyl]amino]carbamoyl]oxirane-2-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7844(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-hydroxypropanoyl]amino]propanoyl]amino]-N-[(2S)-3-cyclohexyl-1-[[(2S)-1-(1H-imidazol-5-yl)-3-oxopropan-2-yl]amino]-1-oxopropan-2-yl]-3-methylbutanamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease (50 %)
NA
23747811
DrugRepV_7845N-[(Benzyloxy)carbonyl]valyl-N-[1-oxo-3-(2-oxo-3-pyrrolidinyl)-1-(1,3-thiazol-2-yl)-2-propanyl]leucinamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7846N-[(Benzyloxy)carbonyl]-L-valyl-N-{(2S)-1-(1,3-benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxo-3-pyrrolidinyl]-2-propanyl}-D-leucinamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease (50 %)
NA
23747811
DrugRepV_7847N-{[3-(Dimethylamino)phenoxy]acetyl}-L-valyl-N-{(2S)-1-(1,3-benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxo-3-pyrrolidinyl]-2-propanyl}-L-leucinamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_78482-[2,3-Dichloro-4-(2-methylenebutanoyl)phenoxy]-N-(2-methyl-2-propanyl)acetamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7849Cinanserin
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease (50 %)
NA
23747811
DrugRepV_78505-Chloro-3-pyridinyl 1H-indole-2-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease (50 %)
NA
23747811
DrugRepV_78511-(2-Naphthylmethyl)-2,3-dioxo-5-indolinecarboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease (50 %)
NA
23747811
DrugRepV_78521-[(1H-Indol-5-ylcarbonyl)oxy]-1H-benzotriazole
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_78534-(4-Chlorophenyl)-2-[(4-nitrobenzyl)sulfanyl]-6-oxo-1,6-dihydro-5-pyrimidinecarbonitrile
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease (50 %)
NA
23747811
DrugRepV_78544-{(Z)-[1-(4-Fluorophenyl)-5-oxo-3-phenyl-1,5-dihydro-4H-pyrazol-4-ylidene]methyl}benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease (50 %)
NA
23747811
DrugRepV_78553-Benzyl-1-[(6,7-dimethyl-2-oxo-1,2-dihydro-3-quinolinyl)methyl]-1-[2-(2-methylphenyl)ethyl]urea
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease (50 %)
NA
23747811
DrugRepV_7856N-{(2S)-1-(1,3-Benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxo-3-pyrrolidinyl]-2-propanyl}-N2-(3-methylbutanoyl)-L-leucinamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7857tert-butyl N-[(2S)-1-[[(2S)-1-(1,3-benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7858benzyl N-[(2S)-1-[[(2S)-1-(1,3-benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease (50 %)
NA
23747811
DrugRepV_7859benzyl N-[(2S)-1-[[(2S)-1-(1,3-benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]amino]-1-oxohexan-2-yl]carbamate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7860benzyl N-[(2S)-1-[[(2S)-1-(1,3-benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]carbamate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7861Benzyl [(2S,3R)-1-({(2S)-1-(1,3-benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxo-3-pyrrolidinyl]-2-propanyl}amino)-3-methyl-1-oxo-2-pentanyl]carbamate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7862benzyl N-[(2S)-1-[[(2S)-1-(1,3-benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]amino]-4-methylsulfanyl-1-oxobutan-2-yl]carbamate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7863benzyl N-[(2S)-1-[[(2S)-1-(1,3-benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]carbamate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7864(2S)-N-[(2S)-1-(1,3-benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]-4-methyl-2-[(2-phenylacetyl)amino]pentanamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7865(2S)-N-[(2S)-1-(1,3-benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]-2-[[2-(4-methoxyphenyl)acetyl]amino]-4-methylpentanamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease (50 %)
NA
23747811
DrugRepV_7866(2S)-N-[(2S)-1-(1,3-benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]-2-[3-(4-methoxyphenyl)propanoylamino]-4-methylpentanamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7867N-{(2S)-1-(1,3-Benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxo-3-pyrrolidinyl]-2-propanyl}-N2-[3-(3-pyridinyl)propanoyl]-L-leucinamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7868N-{(2S)-1-(1,3-Benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxo-3-pyrrolidinyl]-2-propanyl}-N~2~-[(2E)-3-phenyl-2-propenoyl]-L-leucinamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7869N-{(2S)-1-(1,3-Benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxo-3-pyrrolidinyl]-2-propanyl}-N~2~-[(2E)-3-(4-methoxyphenyl)-2-propenoyl]-L-leucinamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7870N-{(2S)-1-(1,3-Benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxo-3-pyrrolidinyl]-2-propanyl}-N~2~-[(2E)-3-(3,4-dimethoxyphenyl)-2-propenoyl]-L-leucinamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7871(2S)-N-[(2S)-1-(1,3-benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]-4-methyl-2-[(2-phenoxyacetyl)amino]pentanamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease (50 %)
NA
23747811
DrugRepV_7872N-{(2S)-1-(1,3-Benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxo-3-pyrrolidinyl]-2-propanyl}-N~2~-[(4-methoxyphenoxy)acetyl]-L-leucinamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7873(2S)-N-[(2S)-1-(1,3-benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]-2-[[2-(4-hydroxyphenoxy)acetyl]amino]-4-methylpentanamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7874N-{(2S)-1-(1,3-Benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxo-3-pyrrolidinyl]-2-propanyl}-N~2~-{[3-(dimethylamino)phenoxy]acetyl}-L-leucinamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7875(2S)-N-[(2S)-1-(1,3-benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]-2-[[2-(4-methoxyanilino)acetyl]amino]-4-methylpentanamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7876(2S)-N-[(2S)-1-(1,3-benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]-2-[[2-(3-methoxyanilino)acetyl]amino]-4-methylpentanamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease (50 %)
NA
23747811
DrugRepV_7877(2S)-N-[(2S)-1-(1,3-benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]-2-[[2-(2-methoxyanilino)acetyl]amino]-4-methylpentanamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease (50 %)
NA
23747811
DrugRepV_7878benzyl N-[(2S)-4-methyl-1-oxo-1-[[(2S)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]-1-(5-phenyl-1,3-thiazol-2-yl)propan-2-yl]amino]pentan-2-yl]carbamate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7879N~2~-[(Benzyloxy)carbonyl]-N-{(2S)-1-[5-(4-methylphenyl)-1,3-thiazol-2-yl]-1-oxo-3-[(3S)-2-oxo-3-pyrrolidinyl]-2-propanyl}-L-leucinamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7880benzyl N-[(2S)-1-[[(2S)-1-[5-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_7881benzyl N-[(2S)-1-[[(2S)-1-[5-(2-methoxyphenyl)-1,3-thiazol-2-yl]-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
Fluorometric protease inhibitory assay
Decrease
NA
23747811
DrugRepV_78825-chloropyridin-3-yl 5-(4-chlorophenyl)oxolane-2-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_78835-chloropyridin-3-yl 5-(4-nitrophenyl)oxolane-2-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_78845-chloropyridin-3-yl 5-(4-chloro-2-nitrophenyl)oxolane-2-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_78855-chloropyridin-3-yl 5-(2-nitrophenyl)oxolane-2-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_78865-chloropyridin-3-yl 5-(3-nitrophenyl)oxolane-2-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_7887(5-chloropyridin-3-yl) pyridine-4-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_7888(5-chloropyridin-3-yl) pyridine-3-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_7889(5-chloropyridin-3-yl) 4-chlorobenzoate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_7890(5-chloropyridin-3-yl) 2-nitrobenzoate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_7891(5-chloropyridin-3-yl) 3-nitrobenzoate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_78925-Chloro-3-pyridinyl 1-naphthoate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_7893(5-chloropyridin-3-yl) 2-oxochromene-3-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_7895Rotenone
NA
NA
Lassa virus
NA
NA
GLuc assay
Decrease (50 %)
Vet approved
31786250
DrugRepV_7899Lycorine
NA
NA
Japanese encephalitis virus
NA
Pathway
NA
Decrease (50 %)
NA
31871089
DrugRepV_7900Cephalotaxlen
NA
NA
Japanese encephalitis virus
NA
Pathway
NA
Decrease (50 %)
NA
31871089
DrugRepV_7901Schisandrin B
NA
NA
Japanese encephalitis virus
NA
Pathway
NA
Decrease (50 %)
NA
31871089
DrugRepV_7902Procyanidin
NA
NA
Japanese encephalitis virus
NA
Pathway
NA
Decrease (50 %)
NA
31871089
DrugRepV_7903Emodin
NA
Polycystic Kidney
Japanese encephalitis virus
NA
Pathway
NA
Decrease (50 %)
Investigational
31871089
DrugRepV_7904Schisandrin B
NA
NA
Japanese encephalitis virus
NA
Pathway
NA
Decrease (50 %)
NA
31871089
DrugRepV_7905RK-33
NA
NA
Dengue virus
New Guinea C
Pathway
Plaque assay
Decrease (50 %)
NA
31936642
DrugRepV_7906RK-33
NA
NA
Zika virus
Asian/Cook Islands/2014
NA
Plaque assay
Decrease (50 %)
NA
31936642
DrugRepV_7907RK-33
NA
NA
West Nile virus
Kunjin
Pathway
Plaque assay
Decrease (50 %)
NA
31936642
DrugRepV_7908Antimycin A
NA
NA
Influenza virus
A/Puerto Rico/8/34
Pathway
MTT assay
Decrease (50 %)
NA
31941776
DrugRepV_7909Brequinar
NA
NA
Influenza virus
A/Puerto Rico/8/34
Pathway
MTT assay
Decrease (50 %)
Experimental
31941776
DrugRepV_79106-Azauridine
NA
Cancer
Influenza virus
A/Puerto Rico/8/34
Pathway
MTT assay
Decrease (50 %)
NA
31941776
DrugRepV_7911Azaribine
NA
Psoriasis
Influenza virus
A/Puerto Rico/8/34
Pathway
MTT assay
Decrease (50 %)
NA
31941776
DrugRepV_7912Pyrazofurin
NA
NA
Influenza virus
A/Puerto Rico/8/34
Pathway
MTT assay
Decrease (50 %)
NA
31941776
DrugRepV_7913AVN-944
NA
Cancer
Influenza virus
A/Puerto Rico/8/34
Pathway
MTT assay
Decrease (50 %)
Investigational
31941776
DrugRepV_7914Mycophenolate mofetil
NA
Organ rejection (immunosuppressants)
Influenza virus
A/Puerto Rico/8/34
Pathway
MTT assay
Decrease (50 %)
Approved, Investigational
31941776
DrugRepV_7918Antimycin A
NA
NA
Influenza virus
B/Brisbane/60/08
Pathway
MTT assay
Decrease (50 %)
NA
31941776
DrugRepV_7919Brequinar
NA
NA
Influenza virus
B/Brisbane/60/08
Pathway
MTT assay
Decrease (50 %)
Experimental
31941776
DrugRepV_79206-Azauridine
NA
Cancer
Influenza virus
B/Brisbane/60/08
Pathway
MTT assay
Decrease (50 %)
NA
31941776
DrugRepV_7921Azaribine
NA
Psoriasis
Influenza virus
B/Brisbane/60/08
Pathway
MTT assay
Decrease (50 %)
NA
31941776
DrugRepV_7922Pyrazofurin
NA
NA
Influenza virus
B/Brisbane/60/08
Pathway
MTT assay
Decrease (50 %)
NA
31941776
DrugRepV_7923AVN-944
NA
Cancer
Influenza virus
B/Brisbane/60/08
Pathway
MTT assay
Decrease (50 %)
Investigational
31941776
DrugRepV_7924Mycophenolate mofetil
NA
Organ rejection (immunosuppressants)
Influenza virus
B/Brisbane/60/08
Pathway
MTT assay
Decrease (50 %)
Approved, Investigational
31941776
DrugRepV_7926Antimycin A
NA
NA
Influenza virus
A/Puerto Rico/8/34
Pathway
MTT assay
Decrease (50 %)
NA
31941776
DrugRepV_7927Brequinar
NA
NA
Influenza virus
A/Puerto Rico/8/34
Pathway
MTT assay
Decrease (50 %)
Experimental
31941776
DrugRepV_79286-Azauridine
NA
Cancer
Influenza virus
A/Puerto Rico/8/34
Pathway
MTT assay
Decrease (50 %)
NA
31941776
DrugRepV_7929Azaribine
NA
Psoriasis
Influenza virus
A/Puerto Rico/8/34
Pathway
MTT assay
Decrease (50 %)
NA
31941776
DrugRepV_7930Pyrazofurin
NA
NA
Influenza virus
A/Puerto Rico/8/34
Pathway
MTT assay
Decrease (50 %)
NA
31941776
DrugRepV_7931AVN-944
NA
Cancer
Influenza virus
A/Puerto Rico/8/34
Pathway
MTT assay
Decrease (50 %)
Investigational
31941776
DrugRepV_7932Mycophenolate mofetil
NA
Organ rejection (immunosuppressants)
Influenza virus
A/Puerto Rico/8/34
Pathway
MTT assay
Decrease (50 %)
Approved, Investigational
31941776
DrugRepV_7934Antimycin A
NA
NA
Influenza virus
A/New Caledonia/20/1999
Pathway
MTT assay
Decrease (50 %)
NA
31941776
DrugRepV_7935Brequinar
NA
NA
Influenza virus
A/New Caledonia/20/1999
Pathway
MTT assay
Decrease (50 %)
Experimental
31941776
DrugRepV_79366-Azauridine
NA
Cancer
Influenza virus
A/New Caledonia/20/1999
Pathway
MTT assay
Decrease (50 %)
NA
31941776
DrugRepV_7937Azaribine
NA
Psoriasis
Influenza virus
A/New Caledonia/20/1999
Pathway
MTT assay
Decrease (50 %)
NA
31941776
DrugRepV_7938Pyrazofurin
NA
NA
Influenza virus
A/New Caledonia/20/1999
Pathway
MTT assay
Decrease (50 %)
NA
31941776
DrugRepV_7939AVN-944
NA
Cancer
Influenza virus
A/New Caledonia/20/1999
Pathway
MTT assay
Decrease (50 %)
Investigational
31941776
DrugRepV_7940Mycophenolate mofetil
NA
Organ rejection (immunosuppressants)
Influenza virus
A/New Caledonia/20/1999
Pathway
MTT assay
Decrease (50 %)
Approved, Investigational
31941776
DrugRepV_7942DHBNH
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79433-[(E)-{[(3,4-dihydroxyphenyl)formamido]imino}methyl]-[1,1'-biphenyl]-4-carboxylic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7944(3E)-3-{2-[4-(3,4-dihydroxyphenyl)-1,3-thiazol-2-yl]hydrazin-1-ylidene}-2,3-dihydro-1H-indol-2-one
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79454-[2-[(2-hydroxy-1H-indol-3-yl)diazenyl]-1,3-thiazol-4-yl]benzonitrile
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7946NSC727447
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7947NSC732665
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79482-(3,4-Dihydroxyphenyl)-1,5,6,7,8,9-hexahydro-4H-cyclohepta[4,5]thieno[2,3-d]pyrimidin-4-one
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79492-(3,4-dihydroxybenzamido)-N-(pyridin-2-yl)-4H,5H,6H,7H,8H-cyclohepta[b]thiophene-3-carboxamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79505-(3,4-dihydroxyphenyl)-4-oxa-8-thia-6-azatricyclo[7.4.0.0²,?]trideca-1(9),2(7),5,10,12-pentaen-3-one
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7951(E)-3-(3,4-dihydroxyphenyl)-N-[(Z)-octadec-9-enyl]prop-2-enamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79524-Butoxy-N-(5-methyl-7-phenyl-4,7-dihydro[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79534-Butyl-N-(5-methyl-7-phenyl-4,7-dihydro[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79544-butyl-N-{5-methyl-7-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79552-fluoro-N-{5-methyl-7-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7956N-{5-methyl-7-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-4-nitrobenzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79574-amino-N-{5-methyl-7-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79583,4-dimethoxy-N-{5-methyl-7-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79593,4-dihydroxy-N-{5-methyl-7-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79602-fluoro-N-{7-methyl-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7961N-{7-methyl-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-4-nitrobenzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79624-amino-N-{7-methyl-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79633,4-dimethoxy-N-{7-methyl-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79643,4-dihydroxy-N-{7-methyl-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79654-butyl-N-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7966N-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-2-fluorobenzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7967N-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-4-nitrobenzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79684-amino-N-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7969N-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-3,4-dimethoxybenzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7970N-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-3,4-dihydroxybenzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7971N-{5,7-diphenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-3,4-dihydroxybenzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7972N-[7-(3,4-dihydroxyphenyl)-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7973N-benzoyl-N-[7-(3,4-dimethoxyphenyl)-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7974N-(3,4-dihydroxyphenyl)-5-methyl-7-phenyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7975N-(3,4-dihydroxyphenyl)-7-methyl-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79882-(6-{[1-carboxy-2-(2-phenyl-1H-indol-3-yl)ethyl]carbamoyl}-4-(2-{[1-carboxy-2-(2-phenyl-1H-indol-3-yl)ethyl]carbamoyl}ethyl)-4-nitrohexanamido)-3-(2-phenyl-1H-indol-3-yl)propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79892-[6-({1-carboxy-2-[2-(2-fluorophenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(2-fluorophenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]-3-[2-(2-fluorophenyl)-1H-indol-3-yl]propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79902-[6-({1-carboxy-2-[2-(4-nitrophenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(4-nitrophenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]-3-[2-(4-nitrophenyl)-1H-indol-3-yl]propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79913-[2-(4-bromophenyl)-1H-indol-3-yl]-2-[6-({2-[2-(4-bromophenyl)-1H-indol-3-yl]-1-carboxyethyl}carbamoyl)-4-[2-({2-[2-(4-bromophenyl)-1H-indol-3-yl]-1-carboxyethyl}carbamoyl)ethyl]-4-nitrohexanamido]propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79922-{6-[(1-carboxy-2-{2-[4-(trifluoromethyl)phenyl]-1H-indol-3-yl}ethyl)carbamoyl]-4-{2-[(1-carboxy-2-{2-[4-(trifluoromethyl)phenyl]-1H-indol-3-yl}ethyl)carbamoyl]ethyl}-4-nitrohexanamido}-3-{2-[4-(trifluoromethyl)phenyl]-1H-indol-3-yl}propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79932-[6-({1-carboxy-2-[2-(4-methoxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(4-methoxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]-3-[2-(4-methoxyphenyl)-1H-indol-3-yl]propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79943-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79954-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79965-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzene-1,3-dicarboxylic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79973-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79984-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79995-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzene-1
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80003-(1-benzyl-1H-indol-3-yl)-2-(6-{[2-(1-benzyl-1H-indol-3-yl)-1-carboxyethyl]carbamoyl}-4-(2-{[2-(1-benzyl-1H-indol-3-yl)-1-carboxyethyl]carbamoyl}ethyl)-4-nitrohexanamido)propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80012-{6-[(1-carboxy-2-{1-[(4-fluorophenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]-4-{2-[(1-carboxy-2-{1-[(4-fluorophenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]ethyl}-4-nitrohexanamido}-3-{1-[(4-fluorophenyl)methyl]-1H-indol-3-yl}propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80024-{[3-(2-carboxy-2-{6-[(1-carboxy-2-{1-[(4-carboxyphenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]-4-{2-[(1-carboxy-2-{1-[(4-carboxyphenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]ethyl}-4-nitrohexanamido}ethyl)-1H-indol-1-yl]methyl}benzoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80034-[(3-{2-carboxy-2-[3-(3-{2-[(1-carboxy-2-{1-[(4-carboxyphenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]ethoxy}-2,2-bis({2-[(1-carboxy-2-{1-[(4-carboxyphenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]ethoxy}methyl)propoxy)propanamido]ethyl}-1H-indol-1-yl)me
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80042-(6-{[1-carboxy-2-(2-phenyl-1H-indol-3-yl)ethyl]carbamoyl}-4-(2-{[1-carboxy-2-(2-phenyl-1H-indol-3-yl)ethyl]carbamoyl}ethyl)-4-nitrohexanamido)-3-(2-phenyl-1H-indol-3-yl)propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80052-[6-({1-carboxy-2-[2-(2-fluorophenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(2-fluorophenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]-3-[2-(2-fluorophenyl)-1H-indol-3-yl]propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80062-[6-({1-carboxy-2-[2-(4-nitrophenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(4-nitrophenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]-3-[2-(4-nitrophenyl)-1H-indol-3-yl]propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80073-[2-(4-bromophenyl)-1H-indol-3-yl]-2-[6-({2-[2-(4-bromophenyl)-1H-indol-3-yl]-1-carboxyethyl}carbamoyl)-4-[2-({2-[2-(4-bromophenyl)-1H-indol-3-yl]-1-carboxyethyl}carbamoyl)ethyl]-4-nitrohexanamido]propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80082-{6-[(1-carboxy-2-{2-[4-(trifluoromethyl)phenyl]-1H-indol-3-yl}ethyl)carbamoyl]-4-{2-[(1-carboxy-2-{2-[4-(trifluoromethyl)phenyl]-1H-indol-3-yl}ethyl)carbamoyl]ethyl}-4-nitrohexanamido}-3-{2-[4-(trifluoromethyl)phenyl]-1H-indol-3-yl}propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80092-[6-({1-carboxy-2-[2-(4-methoxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(4-methoxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]-3-[2-(4-methoxyphenyl)-1H-indol-3-yl]propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80103-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80114-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80125-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzene-1,3-dicarboxylic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80133-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80144-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80155-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzene-1
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80163-(1-benzyl-1H-indol-3-yl)-2-(6-{[2-(1-benzyl-1H-indol-3-yl)-1-carboxyethyl]carbamoyl}-4-(2-{[2-(1-benzyl-1H-indol-3-yl)-1-carboxyethyl]carbamoyl}ethyl)-4-nitrohexanamido)propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80172-{6-[(1-carboxy-2-{1-[(4-fluorophenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]-4-{2-[(1-carboxy-2-{1-[(4-fluorophenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]ethyl}-4-nitrohexanamido}-3-{1-[(4-fluorophenyl)methyl]-1H-indol-3-yl}propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80184-{[3-(2-carboxy-2-{6-[(1-carboxy-2-{1-[(4-carboxyphenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]-4-{2-[(1-carboxy-2-{1-[(4-carboxyphenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]ethyl}-4-nitrohexanamido}ethyl)-1H-indol-1-yl]methyl}benzoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80194-[(3-{2-carboxy-2-[3-(3-{2-[(1-carboxy-2-{1-[(4-carboxyphenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]ethoxy}-2,2-bis({2-[(1-carboxy-2-{1-[(4-carboxyphenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]ethoxy}methyl)propoxy)propanamido]ethyl}-1H-indol-1-yl)me
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80202-(6-{[1-carboxy-2-(2-phenyl-1H-indol-3-yl)ethyl]carbamoyl}-4-(2-{[1-carboxy-2-(2-phenyl-1H-indol-3-yl)ethyl]carbamoyl}ethyl)-4-nitrohexanamido)-3-(2-phenyl-1H-indol-3-yl)propanoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80212-[6-({1-carboxy-2-[2-(2-fluorophenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(2-fluorophenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]-3-[2-(2-fluorophenyl)-1H-indol-3-yl]propanoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80222-[6-({1-carboxy-2-[2-(4-nitrophenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(4-nitrophenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]-3-[2-(4-nitrophenyl)-1H-indol-3-yl]propanoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80233-[2-(4-bromophenyl)-1H-indol-3-yl]-2-[6-({2-[2-(4-bromophenyl)-1H-indol-3-yl]-1-carboxyethyl}carbamoyl)-4-[2-({2-[2-(4-bromophenyl)-1H-indol-3-yl]-1-carboxyethyl}carbamoyl)ethyl]-4-nitrohexanamido]propanoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80242-{6-[(1-carboxy-2-{2-[4-(trifluoromethyl)phenyl]-1H-indol-3-yl}ethyl)carbamoyl]-4-{2-[(1-carboxy-2-{2-[4-(trifluoromethyl)phenyl]-1H-indol-3-yl}ethyl)carbamoyl]ethyl}-4-nitrohexanamido}-3-{2-[4-(trifluoromethyl)phenyl]-1H-indol-3-yl}propanoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80252-[6-({1-carboxy-2-[2-(4-methoxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(4-methoxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]-3-[2-(4-methoxyphenyl)-1H-indol-3-yl]propanoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80263-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80274-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80285-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzene-1,3-dicarboxylic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80293-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80304-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80315-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzene-1
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80324-[(3-{2-carboxy-2-[3-(3-{2-[(1-carboxy-2-{1-[(4-carboxyphenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]ethoxy}-2,2-bis({2-[(1-carboxy-2-{1-[(4-carboxyphenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]ethoxy}methyl)propoxy)propanamido]ethyl}-1H-indol-1-yl)me
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80332-[6-({1-carboxy-2-[2-(4-nitrophenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(4-nitrophenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]-3-[2-(4-nitrophenyl)-1H-indol-3-yl]propanoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (90 %)
NA
31809045
DrugRepV_80343-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (90 %)
NA
31809045
DrugRepV_80355-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzene-1,3-dicarboxylic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (90 %)
NA
31809045
DrugRepV_80363-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (90 %)
NA
31809045
DrugRepV_80374-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (90 %)
NA
31809045
DrugRepV_80385-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzene-1
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (90 %)
NA
31809045
DrugRepV_8039MADAL-385
NA
NA
Enterovirus
11316
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80405-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzene-1,3-dicarboxylic acid
NA
NA
Enterovirus
11316
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80413-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Enterovirus
11316
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80425-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzene-1
NA
NA
Enterovirus
11316
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_8043MADAL-385
NA
NA
Enterovirus
TW/70902/08
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80445-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzene-1,3-dicarboxylic acid
NA
NA
Enterovirus
TW/70902/08
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80453-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Enterovirus
TW/70902/08
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80465-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzene-1
NA
NA
Enterovirus
TW/70902/08
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_8047MADAL-385
NA
NA
Enterovirus
H08300 461; 812
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80485-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzene-1,3-dicarboxylic acid
NA
NA
Enterovirus
H08300 461; 812
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80493-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Enterovirus
H08300 461; 812
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80505-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzene-1
NA
NA
Enterovirus
H08300 461; 812
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_8051MADAL-385
NA
NA
Enterovirus
TW/1956/05
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80525-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzene-1,3-dicarboxylic acid
NA
NA
Enterovirus
TW/1956/05
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80533-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Enterovirus
TW/1956/05
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80545-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzene-1
NA
NA
Enterovirus
TW/1956/05
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80554-{[6-chloro-4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80564-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80574-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80584-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80594-{[6-chloro-4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80604-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80614-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80624-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80634-{[6-chloro-4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80644-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80654-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80664-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80674-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80684-{[4-({2-chloro-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-fluorophenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80694-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80704-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80714-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80724-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-dimethylphenyl}amino)-6-methoxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80734-{[4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)-6-methoxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80744-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-methoxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80754-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-hydroxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80764-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-nitroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80774-{[7-chloro-4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80784-{[7-chloro-4-({2-chloro-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-fluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80794-{[7-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80804-{[7-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80814-{[7-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80824-{[4-({2-amino-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-methylphenyl}amino)-7-chloroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80834-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-dimethylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80844-{[4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80854-{[4-({2-chloro-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-fluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80864-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80874-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80884-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80894-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80904-{[4-({2-chloro-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-fluorophenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80914-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80924-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80934-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80944-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-dimethylphenyl}amino)-6-methoxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80954-{[4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)-6-methoxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80964-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-methoxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80974-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-hydroxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80984-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-nitroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80994-{[7-chloro-4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81004-{[7-chloro-4-({2-chloro-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-fluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81014-{[7-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81024-{[7-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81034-{[7-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81044-{[4-({2-amino-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-methylphenyl}amino)-7-chloroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81054-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-dimethylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81064-{[4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81074-{[4-({2-chloro-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-fluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81084-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81094-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81104-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81114-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81124-{[4-({2-chloro-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-fluorophenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81134-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81144-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81154-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81164-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-dimethylphenyl}amino)-6-methoxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81174-{[4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)-6-methoxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81184-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-methoxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81194-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-hydroxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81204-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-nitroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81214-{[7-chloro-4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81224-{[7-chloro-4-({2-chloro-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-fluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81234-{[7-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81244-{[7-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81254-{[7-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81264-{[4-({2-amino-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-methylphenyl}amino)-7-chloroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81274-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-dimethylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81284-{[4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81294-{[4-({2-chloro-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-fluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81304-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81314-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81324-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_8133StemRegenin 1
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (68.1 %)
NA
32708182
DrugRepV_8135ICG-001
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (80.9 %)
NA
32708182
DrugRepV_8137NSC 319726
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (99.8 %)
NA
32708182
DrugRepV_8139RITA
NA
Cancer
Vaccinia virus
NA
Pathway
NA
Decrease (50.2 %)
NA
32708182
DrugRepV_8143Monensin sodium salt
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (96.7 %)
Experimental, Vet approved
32708182
DrugRepV_81453-Deazaneplanocin A
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (76.8 %)
NA
32708182
DrugRepV_8148Azaguanine-8
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (12.7 %)
Experimental
32708182
DrugRepV_8149Cytarabine
NA
Leukemia
Vaccinia virus
NA
Pathway
NA
Decrease (99.8 %)
Approved
32708182
DrugRepV_8151Cyclocytidine Hydrochloride
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (99.8 %)
NA
32708182
DrugRepV_8156Triapine
NA
Leukemia, Lung Cancer, Kidney Cancer, Prostate Cancer, and Pancreatic Cancer
Vaccinia virus
NA
Pathway
NA
Decrease (99.9 %)
Investigational
32708182
DrugRepV_8158Apigenin
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (54.8 %)
Experimental
32708182
DrugRepV_8159Avasimibe
NA
Peripheral vascular disease
Vaccinia virus
NA
Pathway
NA
Decrease (50.9 %)
Investigational
32708182
DrugRepV_8160Cyclosporin A
NA
Bone marrow transplant rejection
Vaccinia virus
NA
Pathway
NA
Decrease (67.2 %)
Approved, Investigational, Vet approved
32708182
DrugRepV_8161ML130
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (35.9 %)
NA
32708182
DrugRepV_8162PAC-1
NA
Lymphoma, Melanoma, Solid Tumors, Breast Cancer, and Thoracic Cancers
Vaccinia virus
NA
Pathway
NA
Decrease (95.5 %)
Investigational
32708182
DrugRepV_8163ABT-263
NA
Solid Tumors, Non-Hodgkin's Lymphoma, EGFR Activating Mutation, Chronic Lymphoid Leukemia, and Hematological Malignancies
Vaccinia virus
NA
Pathway
NA
Decrease (33.1 %)
Investigational
32708182
DrugRepV_8164ABT-737
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (26.6 %)
NA
32708182
DrugRepV_8165PF-2545920
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (33.7 %)
NA
32708182
DrugRepV_8168TPCA-1
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (78.5 %)
NA
32708182
DrugRepV_8170PTC-209
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (90.7 %)
NA
32708182
DrugRepV_8171Selisistat
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (30.5 %)
NA
32708182
DrugRepV_8172Salinomycin
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (92.5 %)
Vet approved
32708182
DrugRepV_8173Dapivirine
NA
Acquired immunodeficiency syndrome
Vaccinia virus
NA
Pathway
NA
Decrease (41.7 %)
Investigational
32708182
DrugRepV_8174CCG 50014
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (35.8 %)
NA
32708182
DrugRepV_8175Mocetinostat
NA
Lymphoma, Urothelial Carcinoma, Relapsed and Refractory, Myelodysplastic Syndrome, and Metastatic Leiomyosarcoma
Vaccinia virus
NA
Pathway
NA
Decrease (46.9 %)
Investigational
32708182
DrugRepV_8177UK 383367
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (17 %)
NA
32708182
DrugRepV_8178Lonafarnib
NA
Solid tumors, leukemia (unspecified), and lung cancer
Vaccinia virus
NA
Pathway
NA
Decrease (36.2 %)
Investigational
32708182
DrugRepV_8179BX-912
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (42.3 %)
NA
32708182
DrugRepV_8180URB597
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (21.7 %)
NA
32708182
DrugRepV_8181Anagrelide HCl
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (58.4 %)
NA
32708182
DrugRepV_8185Ganetespib
NA
BREAST CANCER, Small Cell Lung Cancer, Acute Myeloid Leukaemia, and Myelodysplastic Syndrome
Vaccinia virus
NA
Pathway
NA
Decrease (99.7 %)
Investigational
32708182
DrugRepV_8186PF-04929113
NA
Cancer/tumors
Vaccinia virus
NA
Pathway
NA
Decrease (99.4 %)
Investigational
32708182
DrugRepV_8187NMS-E973
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (99.1 %)
NA
32708182
DrugRepV_8188XL888
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (99.6 %)
NA
32708182
DrugRepV_8189Tanespimycin
NA
Leukemia (myeloid) and solid tumors.
Vaccinia virus
NA
Pathway
NA
Decrease (99.4 %)
Investigational
32708182
DrugRepV_8190VER-49009
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (98.9 %)
NA
32708182
DrugRepV_8191SNX2112
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (99.4 %)
NA
32708182
DrugRepV_8192BIIB021
NA
Tumors and Lymphoma
Vaccinia virus
NA
Pathway
NA
Decrease (99.8 %)
Investigational
32708182
DrugRepV_8194NVP-BEP800
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (98.8 %)
NA
32708182
DrugRepV_8195AUY922
NA
Lymphoma, Breast Cancer, Metastatic Disease, Advanced Solid Tumors, and Hematologic Neoplasms
Vaccinia virus
NA
Pathway
NA
Decrease (99.8 %)
Investigational
32708182
DrugRepV_8196KW-2478
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (92.7 %)
NA
32708182
DrugRepV_8198ABT-751
NA
Lung Cancer
Vaccinia virus
NA
Pathway
NA
Decrease (81.5 %)
Investigational
32708182
DrugRepV_8199Epothilone A
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (27.3 %)
NA
32708182
DrugRepV_8200Amygdalin
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (58.3 %)
NA
32708182
DrugRepV_8201Kaempferol
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (64.7 %)
NA
32708182
DrugRepV_8202ENMD-2076
NA
Breast cancer, leukemia (unspecified), lung cancer, and solid tumors
Vaccinia virus
NA
Pathway
NA
Decrease (72.3 %)
Investigational
32708182
DrugRepV_8203AMG-900
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (50.4 %)
NA
32708182
DrugRepV_8204MLN8054
NA
Colon Neoplasm, Breast Neoplasm, Bladder Neoplasm, Pancreatic Neoplasm, and Advanced Malignancies
Vaccinia virus
NA
Pathway
NA
Decrease (36.2 %)
Investigational
32708182
DrugRepV_8205Ibrutinib
NA
Mantle cell lymphoma
Vaccinia virus
NA
Pathway
NA
Decrease (74.9 %)
Approved
32708182
DrugRepV_8206CNX-774
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (70 %)
NA
32708182
DrugRepV_8207AR-A014418
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (47.9 %)
Experimental
32708182
DrugRepV_8208CGP 57380
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (58.1 %)
NA
32708182
DrugRepV_8210HMN-214
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (58.9 %)
NA
32708182
DrugRepV_8211TG003
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (46.7 %)
NA
32708182
DrugRepV_8212Skepinone-L
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (47.1 %)
NA
32708182
DrugRepV_8213TAK-632
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (65.2 %)
NA
32708182
DrugRepV_8214YM201636
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (56.3 %)
NA
32708182
DrugRepV_8215MK-2461
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (57 %)
NA
32708182
DrugRepV_8217SP600125
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (50.5 %)
NA
32708182
DrugRepV_8218SKI II
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (65.1 %)
NA
32708182
DrugRepV_8219PKI-402
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (44.9 %)
NA
32708182
DrugRepV_8220BEZ235
NA
Cancer, Solid Tumor, Renal Cancer, Breast Cancer, and Cowden Syndrome
Vaccinia virus
NA
Pathway
NA
Decrease (37.4 %)
Investigational
32708182
DrugRepV_8221WYE-125132
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (67.6 %)
NA
32708182
DrugRepV_8222OSI-027
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (68.3 %)
Investigational
32708182
DrugRepV_8223Torin 1
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (57.3 %)
NA
32708182
DrugRepV_8224Ku-0063794
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (55.3 %)
NA
32708182
DrugRepV_8225AZD2014
NA
Advanced Gastric Adenocarcinoma
Vaccinia virus
NA
Pathway
NA
Decrease (70.3 %)
Investigational
32708182
DrugRepV_8228KX2-391
NA
Colon cancer | Pancreatic cancer | Prostate cancer | Breast cancer
Vaccinia virus
NA
Pathway
NA
Decrease (65.1 %)
Investigational
32708182
DrugRepV_8230PP1
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (35.8 %)
NA
32708182
DrugRepV_8231AZ 960
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (82.1 %)
NA
32708182
DrugRepV_8232LY2784544
NA
Myelofibrosis, Polycythemia Vera, Primary Myelofibrosis, Thrombocythemia, Essential, and Myeloproliferative Disorders
Vaccinia virus
NA
Pathway
NA
Decrease (65.7 %)
Investigational
32708182
DrugRepV_8233WHI-P154
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (66.3 %)
NA
32708182
DrugRepV_8234Cyt387
NA
Polycythemia Vera, Primary Myelofibrosis, Post-Polycythemia Vera, Essential Thrombocythemia, and Primary Myelofibrosis (PMF)
Vaccinia virus
NA
Pathway
NA
Decrease (45.2 %)
Investigational
32708182
DrugRepV_8235KPT-276
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (27.6 %)
NA
32708182
DrugRepV_8236KPT-185
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (26.2 %)
NA
32708182
DrugRepV_8237Phloretin
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (-27 %)
Experimental
32708182
DrugRepV_8242SC144
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (98.4 %)
NA
32708182
DrugRepV_8243Daidzein
NA
Dietary supplement
Vaccinia virus
NA
Pathway
NA
Decrease (32.2 %)
Experimental
32708182
DrugRepV_8244Delanzomib
NA
Solid Tumors, Multiple Myeloma, and Lymphoma, Non-Hodgkin.
Vaccinia virus
NA
Pathway
NA
Decrease (99.7 %)
Investigational
32708182
DrugRepV_8245MLN9708
NA
Multiple myeloma
Vaccinia virus
NA
Pathway
NA
Decrease (99.6 %)
Approved, Investigational
32708182
DrugRepV_8246Oprozomib
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (99.5 %)
Investigational
32708182
DrugRepV_8247MG-132
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (98.9 %)
NA
32708182
DrugRepV_8248MLN2238
NA
Multiple myeloma
Vaccinia virus
NA
Pathway
NA
Decrease (99.7 %)
Approved, Investigational
32708182
DrugRepV_8249ONX-0914
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (99.5 %)
NA
32708182
DrugRepV_8250Amonafide
NA
Breast cancer, ovarian cancer, and prostate cancer
Vaccinia virus
NA
Pathway
NA
Decrease (99.3 %)
Investigational
32708182
DrugRepV_8253Golvatinib
NA
Platinum-Resistant Squamous Cell Carcinoma of the Head and Neck
Vaccinia virus
NA
Pathway
NA
Decrease (79.8 %)
Investigational
32708182
DrugRepV_8255AG 1296
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (53.2 %)
NA
32708182
DrugRepV_8256NVP-TAE226
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (91.5 %)
NA
32708182
DrugRepV_8257Cabozantinib malate
NA
Metastatic medullary thyroid cancer
Vaccinia virus
NA
Pathway
NA
Decrease (79.3 %)
NA
32708182
DrugRepV_8258XL-184
NA
Thyroid cancer
Vaccinia virus
NA
Pathway
NA
Decrease (64.2 %)
Approved, Investigational
32708182
DrugRepV_8259Linifanib
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (60.5 %)
NA
32708182
DrugRepV_8260TKI-258
NA
Multiple myeloma and solid tumors
Vaccinia virus
NA
Pathway
NA
Decrease (67.6 %)
Investigational
32708182
DrugRepV_8261AZD4547
NA
Cancer
Vaccinia virus
NA
Pathway
NA
Decrease (81.5 %)
Investigational
32708182
DrugRepV_8262AG-1024
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (71.8 %)
NA
32708182
DrugRepV_8263BMS-754807
NA
Solid Tumors
Vaccinia virus
NA
Pathway
NA
Decrease (61.8 %)
Investigational
32708182
DrugRepV_8265Butein
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (62.6 %)
NA
32708182
DrugRepV_8266CO-1686 (AVL-301)
NA
Nonsmall Cell Lung Cancer, Non-small Cell Lung Cancer, and Locally Advanced or Metastatic Non-small Cell Lung Cancer
Vaccinia virus
NA
Pathway
NA
Decrease (74.3 %)
NA
32708182
DrugRepV_8267PD168393
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (67.2 %)
Experimental
32708182
DrugRepV_8268PD153035 HCl
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (74.7 %)
NA
32708182
DrugRepV_8270Desmethyl Erlotinib
NA
Cancer
Vaccinia virus
NA
Pathway
NA
Decrease (75.5 %)
Approved, Investigational
32708182
DrugRepV_8271OSI-420
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (46.7 %)
NA
32708182
DrugRepV_8274WZ8040
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (96.4 %)
NA
32708182
DrugRepV_82821-(2-fluorophenyl)-3-(4-(4-isopentyl-1H-1,2,3-triazol-1-yl)phenyl)urea
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_82831-(3-fluorophenyl)-3-(4-(4-isopentyl-1H-1,2,3-triazol-1-yl)phenyl)urea
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_82841-(4-(4-(ethoxymethyl)-1H-1,2,3-triazol-1-yl)phenyl)-3-(3-fluorophenyl)urea
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_82851-(3-fluorophenyl)-3-(4-(4-(3-oxobutyl)-1H-1,2,3-triazol-1-yl)phenyl)urea
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_82861-(4-(4-butyl-1H-1,2,3-triazol-1-yl)phenyl)-3-(3-fluorophenyl)urea
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_8287N-(2-(3-(4-(4-butyl-1H-1,2,3-triazol-1-yl)phenyl)ureido)phenyl)methanesulfonamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_82881-(4-(4-isopentyl-1H-1,2,3-triazol-1-yl)phenyl)-3-o-tolylurea
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_82891-(4-(4-hexyl-1H-1,2,3-triazol-1-yl)phenyl)-3-(2-(trifluoromethyl)phenyl)urea)
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_82903-(4-(ethoxymethyl)-1H-1,2,3-triazol-1-yl)-N-(2-morpholinophenyl)benzenesulfonamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_8291ethyl 3-((3-(4-(ethoxymethyl)-1H-1,2,3-triazol-1-yl)phenyl)sulfonamido)benzoate
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_82923-((3-(4-(ethoxymethyl)-1H-1,2,3-triazol-1-yl)phenyl)sulfonamido)benzoic acid
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_82933-(4-butyl-1H-1,2,3-triazol-1-yl)-N-(2-(methylsulfonamido)phenyl)benzenesulfonamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_8315Tenatoprazole
NA
NA
Human immunodeficiency virus
NA
Pathway
Western blot
Decrease (50 %)
NA
32132561
DrugRepV_8317Roscovitine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31866007
DrugRepV_8318Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
Investigational
31866007
DrugRepV_8319Kenpaullone
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31866007
DrugRepV_8320SB743921
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31866007
DrugRepV_83213-Deazauridine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31866007
DrugRepV_83222’-C-Methylcytidine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31866007
DrugRepV_8323Alisporivir
NA
Hepatitis C virus
SARS Coronavirus-2
Experimental
NA
Viral RNA reduction assay
Decrease (50 %)
Investigational
32376613
DrugRepV_8324Alisporivir
NA
Hepatitis C virus
SARS Coronavirus-2
Experimental
NA
Viral RNA reduction assay
Decrease (90 %)
Investigational
32376613
DrugRepV_83274-ethynyl-2-fluoro-2-deoxyadenosine
NA
NA
SARS Coronavirus-2
Experimental
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
32429580
DrugRepV_8328Alovudine
NA
HIV
SARS Coronavirus-2
Experimental
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Investigational
32429580
DrugRepV_83295-O-(12-thioethydodecanoyl)FLT
NA
NA
SARS Coronavirus-2
Experimental
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
32429580
DrugRepV_83315-O-(tetradecanoyl)3TC
NA
NA
SARS Coronavirus-2
Experimental
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
32429580
DrugRepV_83335-O-(tetradecanoyl)FTC
NA
NA
SARS Coronavirus-2
Experimental
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
NA
32429580
DrugRepV_8335Nafamostat
NA
Blood vessel coagulation | Hemorrhagic lesions
SARS Coronavirus-2
NA
NA
Decrease (50 %)
Investigational
32596694
DrugRepV_8337Gabexate
NA
Cancer, ischemia-reperfusion injury, and pancreatitis
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Investigational
32596694
DrugRepV_8339((4-((3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8340((4-((2,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8341((4-((3,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_83424-((4-((2,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8343((4-((3-fluoro-2-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8344((4-((3-fluoro-3-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8345((4-((3-fluoro-4-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8346((4-((3-fluoro-2-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8347((4-((3-fluoro-3-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8348((4-((3-fluoro-4-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino) benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8349((4-((2-chloro-3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino) benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8350((4-((4-chloro-3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8351((4-((3-fluoro-2-(trifluoromethyl)-[1,1-biphenyl]-4-yl)(hydroxylimino)methyl)pyrimidin-2-yl) amino)benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8352((4-((3-fluoro-4-(trifluoromethyl)-[1,1-biphenyl]-4-yl)(hydroxylimino)methyl)pyrimidin-2-yl) amino)benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8353((4-((3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8354((4-((2,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8355((4-((3,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_83564-((4-((2,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8357((4-((3-fluoro-2-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8358((4-((3-fluoro-3-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8359((4-((3-fluoro-4-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8360((4-((3-fluoro-2-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8361((4-((3-fluoro-3-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8362((4-((3-fluoro-4-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino) benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8363((4-((2-chloro-3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino) benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8364((4-((4-chloro-3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8365((4-((3-fluoro-2-(trifluoromethyl)-[1,1-biphenyl]-4-yl)(hydroxylimino)methyl)pyrimidin-2-yl) amino)benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8366((4-((3-fluoro-4-(trifluoromethyl)-[1,1-biphenyl]-4-yl)(hydroxylimino)methyl)pyrimidin-2-yl) amino)benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8367((4-((3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
L100I
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8368((4-((2,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
L100I
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8369((4-((3,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
L100I
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_83704-((4-((2,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
L100I
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8371((4-((3-fluoro-2-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
L100I
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8372((4-((3-fluoro-3-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
L100I
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8373((4-((3-fluoro-4-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
L100I
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8374((4-((3-fluoro-2-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
L100I
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8375((4-((3-fluoro-3-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
L100I
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8376((4-((3-fluoro-4-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino) benzonitrile
NA
NA
Human immunodeficiency virus
L100I
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8377((4-((2-chloro-3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino) benzonitrile
NA
NA
Human immunodeficiency virus
L100I
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8378((4-((4-chloro-3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
L100I
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8379((4-((3-fluoro-2-(trifluoromethyl)-[1,1-biphenyl]-4-yl)(hydroxylimino)methyl)pyrimidin-2-yl) amino)benzonitrile
NA
NA
Human immunodeficiency virus
L100I
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8380((4-((3-fluoro-4-(trifluoromethyl)-[1,1-biphenyl]-4-yl)(hydroxylimino)methyl)pyrimidin-2-yl) amino)benzonitrile
NA
NA
Human immunodeficiency virus
L100I
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8381((4-((3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8382((4-((2,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8383((4-((3,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_83844-((4-((2,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8385((4-((3-fluoro-2-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8386((4-((3-fluoro-3-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8387((4-((3-fluoro-4-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8388((4-((3-fluoro-2-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8389((4-((3-fluoro-3-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8390((4-((3-fluoro-4-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino) benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8391((4-((2-chloro-3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino) benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8392((4-((4-chloro-3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8393((4-((3-fluoro-2-(trifluoromethyl)-[1,1-biphenyl]-4-yl)(hydroxylimino)methyl)pyrimidin-2-yl) amino)benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8394((4-((3-fluoro-4-(trifluoromethyl)-[1,1-biphenyl]-4-yl)(hydroxylimino)methyl)pyrimidin-2-yl) amino)benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8395((4-((3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y181C
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8396((4-((2,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y181C
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8397((4-((3,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y181C
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_83984-((4-((2,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y181C
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8399((4-((3-fluoro-2-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y181C
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8400((4-((3-fluoro-3-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y181C
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8401((4-((3-fluoro-4-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y181C
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8402((4-((3-fluoro-2-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y181C
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8403((4-((3-fluoro-3-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y181C
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8404((4-((3-fluoro-4-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino) benzonitrile
NA
NA
Human immunodeficiency virus
Y181C
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8405((4-((2-chloro-3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino) benzonitrile
NA
NA
Human immunodeficiency virus
Y181C
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8406((4-((4-chloro-3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y181C
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8407((4-((3-fluoro-2-(trifluoromethyl)-[1,1-biphenyl]-4-yl)(hydroxylimino)methyl)pyrimidin-2-yl) amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y181C
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8408((4-((3-fluoro-4-(trifluoromethyl)-[1,1-biphenyl]-4-yl)(hydroxylimino)methyl)pyrimidin-2-yl) amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y181C
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8409((4-((3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y188L
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8410((4-((2,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y188L
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8411((4-((3,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y188L
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_84124-((4-((2,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y188L
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8413((4-((3-fluoro-2-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y188L
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8414((4-((3-fluoro-3-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y188L
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8415((4-((3-fluoro-4-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y188L
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8416((4-((3-fluoro-2-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y188L
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8417((4-((3-fluoro-3-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y188L
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8418((4-((3-fluoro-4-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino) benzonitrile
NA
NA
Human immunodeficiency virus
Y188L
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8419((4-((2-chloro-3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino) benzonitrile
NA
NA
Human immunodeficiency virus
Y188L
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8420((4-((4-chloro-3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y188L
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8421((4-((3-fluoro-2-(trifluoromethyl)-[1,1-biphenyl]-4-yl)(hydroxylimino)methyl)pyrimidin-2-yl) amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y188L
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8422((4-((3-fluoro-4-(trifluoromethyl)-[1,1-biphenyl]-4-yl)(hydroxylimino)methyl)pyrimidin-2-yl) amino)benzonitrile
NA
NA
Human immunodeficiency virus
Y188L
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8423((4-((3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
F227L + V106A
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8424((4-((2,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
F227L + V106A
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8425((4-((3,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
F227L + V106A
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_84264-((4-((2,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
F227L + V106A
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8427((4-((3-fluoro-2-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
F227L + V106A
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8428((4-((3-fluoro-3-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
F227L + V106A
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8429((4-((3-fluoro-4-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
F227L + V106A
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8430((4-((3-fluoro-2-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
F227L + V106A
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8431((4-((3-fluoro-3-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
F227L + V106A
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8432((4-((3-fluoro-4-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino) benzonitrile
NA
NA
Human immunodeficiency virus
F227L + V106A
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8433((4-((2-chloro-3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino) benzonitrile
NA
NA
Human immunodeficiency virus
F227L + V106A
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8434((4-((4-chloro-3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
F227L + V106A
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8435((4-((3-fluoro-2-(trifluoromethyl)-[1,1-biphenyl]-4-yl)(hydroxylimino)methyl)pyrimidin-2-yl) amino)benzonitrile
NA
NA
Human immunodeficiency virus
F227L + V106A
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8436((4-((3-fluoro-4-(trifluoromethyl)-[1,1-biphenyl]-4-yl)(hydroxylimino)methyl)pyrimidin-2-yl) amino)benzonitrile
NA
NA
Human immunodeficiency virus
F227L + V106A
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8437((4-((3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
RES056
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8438((4-((2,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
RES056
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8439((4-((3,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
RES056
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_84404-((4-((2,3-difluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
RES056
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8441((4-((3-fluoro-2-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
RES056
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8442((4-((3-fluoro-3-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
RES056
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8443((4-((3-fluoro-4-methyl-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
RES056
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8444((4-((3-fluoro-2-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino) methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
RES056
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8445((4-((3-fluoro-3-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
RES056
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8446((4-((3-fluoro-4-methoxy-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino) benzonitrile
NA
NA
Human immunodeficiency virus
RES056
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8447((4-((2-chloro-3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino) benzonitrile
NA
NA
Human immunodeficiency virus
RES056
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8448((4-((4-chloro-3-fluoro-[1,1-biphenyl]-4-yl)(hydroxyimino)methyl)pyrimidin-2-yl)amino)benzonitrile
NA
NA
Human immunodeficiency virus
RES056
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8449((4-((3-fluoro-2-(trifluoromethyl)-[1,1-biphenyl]-4-yl)(hydroxylimino)methyl)pyrimidin-2-yl) amino)benzonitrile
NA
NA
Human immunodeficiency virus
RES056
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8450((4-((3-fluoro-4-(trifluoromethyl)-[1,1-biphenyl]-4-yl)(hydroxylimino)methyl)pyrimidin-2-yl) amino)benzonitrile
NA
NA
Human immunodeficiency virus
RES056
Pathway
MTT assay
Decrease (50 %)
NA
32334191
DrugRepV_8456Berberine Chloride
NA
NA
Zika virus
NA
NA
NA
Decrease (50 %)
NA
29844387
DrugRepV_8457Berberine
NA
Parasitic and fungal infection
Zika virus
NA
NA
Plaque assay
Decrease (50 %)
Approved
30641880
DrugRepV_8458Emodin
NA
Polycystic Kidney
Zika virus
NA
NA
Plaque assay
Decrease (50 %)
Investigational
30641880
DrugRepV_8459Berberine
NA
Parasitic and fungal infection
Enterovirus
H
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
28081706
DrugRepV_8460Berberine
NA
Parasitic and fungal infection
Enterovirus
SHZH98
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
28081706
DrugRepV_8461Berberine
NA
Parasitic and fungal infection
Enterovirus
JS-52
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
28081706
DrugRepV_8462Berberine
NA
Parasitic and fungal infection
Enterovirus
BrCr
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
28081706
DrugRepV_8463Pirodavir
NA
Picronavirus infection
Enterovirus
H
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Experimental
28081706
DrugRepV_8464Pirodavir
NA
Picronavirus infection
Enterovirus
SHZH98
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Experimental
28081706
DrugRepV_8465Pirodavir
NA
Picronavirus infection
Enterovirus
JS-52
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Experimental
28081706
DrugRepV_8466Pirodavir
NA
Picronavirus infection
Enterovirus
BrCr
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Experimental
28081706
DrugRepV_8467Berberine
NA
Parasitic and fungal infection
Influenza virus
NA
Pathway
XTT assay
Decrease (50 %)
Approved
32245183
DrugRepV_8468Berberine
NA
Parasitic and fungal infection
Influenza virus
NA
Pathway
XTT assay
Decrease (50 %)
Approved
32245183
DrugRepV_8469Berberine
NA
Parasitic and fungal infection
Influenza virus
NA
Pathway
XTT assay
Decrease (50 %)
Approved
32245183
DrugRepV_8470Berberine
NA
Parasitic and fungal infection
Influenza virus
NA
Pathway
XTT assay
Decrease (50 %)
Approved
32245183
DrugRepV_8471Berberine
NA
Parasitic and fungal infection
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
Approved
21295891
DrugRepV_8472Berberine
NA
Parasitic and fungal infection
Influenza virus
NA
Pathway
NA
Decrease (50 %)
Approved
30099043
DrugRepV_8473Ebselen
NA
Meniere Disease, Type 2 Diabetes Mellitus, and Type 1 Diabetes Mellitus
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
Investigational
23850693
DrugRepV_84742-Phenylbenzo[d]isothiazol-3(2H)-one
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_84752-Phenylbenzo[d] isoxazol-3(2H)-one
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_84762-Phenyl isoindolin-1-one
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_8477Chelerythrine chloride
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_8478Nitidine chloride
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_8479Berberine chloride
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_8480Sanguinarine chloride
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_8481Norsanguinarine chloride
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_8482R-Apomorphine hydrochloride
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_8483S-Apomorphine hydrochloride
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_8484R(?)-Propylnorapomorphine hydrochloride
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_8485R(?)-Apocodeine hydrochloride
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693