DrugRepV Browse Page


DrugRepV browse page allows user to take a glance of the particular antiviral agent.Fields in the webpage is hylerlinked ot various external repositories like DrugBank, PubChem, Clinicaltrials.gov,and PubMed.User can explore the biological, Clinical, Chemical, and Structural details of every repurposed drug candidate.By clicking on the table header arrows, user can sort entries in ascending or descending order.


Total number of Records for NA are 1270




DrugRepV_ID Antiviral Name
Drug type
Primary Indication
Secondary Indication
Strain
Pathways
Assay
Activity
Clinical Status
References
DrugRepV_0002Chloroquine
Antiparasitic products, Insectisides and Repellents
Malaria
Zika virus
Brazilian strain ZKV2015
NA
NA
Decrease
Approved
29150641
DrugRepV_0026Chloroquine
Antiparasitic products, Insectisides and Repellents
Malaria
Zika virus
GZ01, a recent Asian lineage
NA
NA
Decrease
Approved
29033372
DrugRepV_0074Sunitinib-Erlotinib
NA
NA
Ebola virus
Mouse adapted strain
NA
NA
Increase
NA
28240606
DrugRepV_0259Alvespimycin
NA
Cancer
Ebola virus
ME718-1976/Yambuku-Ecran
NA
NA
No significant effect
Investigational
27801778
DrugRepV_0260Bemcentinib
Anticancer
Cancer
Ebola virus
ME718-1976/Yambuku-Ecran
NA
NA
No significant effect
Investigational
27801778
DrugRepV_0261NCK-8
NA
NA
Ebola virus
ME718-1976/Yambuku-Ecran
NA
NA
No significant effect
NA
27801778
DrugRepV_0601Clomiphene Citrate
Genito Urinary System and Sex Hormones
Female infertility
Ebola virus
ma-EBOV
NA
NA
Increase
Approved
23785035
DrugRepV_0602Toremifene Citrate
Antineoplastic and Immunomodulating Agents
Breast Cancer
Ebola virus
ma-EBOV
NA
NA
Increase
Approved, Investigational
23785035
DrugRepV_0725Prochlorperazine
Nervous System
Nausea | Vomiting | Schizophrenia
Ebola virus
ma-EBOV
NA
NA
No significant effect
Approved
23577127
DrugRepV_0726Chloroquine
Antiparasitic products, Insectisides and Repellents
Malaria
Ebola virus
ma-EBOV
NA
NA
Increase
Approved
23577127
DrugRepV_0727Dirithromycin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
ma-EBOV
NA
NA
No significant effect
Approved
23577127
DrugRepV_0728Erythromycin ethylsuccinate
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
ma-EBOV
NA
NA
No significant effect
Approved
23577127
DrugRepV_0729Amlodipine
Cardiovascular agents
Hypertension
Ebola virus
ma-EBOV
NA
NA
No significant effect
Approved
23577127
DrugRepV_0730Fluoxetine
Nervous System
Major depressive disorder | Bulimia nervosa | Obsessive-compulsive disorder | Premenstrual dysphoric disorder | Panic disorder with or without agoraphobia
Ebola virus
ma-EBOV
NA
NA
No significant effect
Approved, Vet approved
23577127
DrugRepV_0731Penbutolol
Cardiovascular agents
Arterial hypertension
Ebola virus
ma-EBOV
NA
NA
No significant effect
Approved, Investigational
23577127
DrugRepV_0743Probenecid
Musculo-Skeletal System
Gout
Influenza virus
A/WSN/33
Pathway
NA
Increase
Approved, Investigational
23129053
DrugRepV_0750Favipiravir
Antiviral
Influenza virus
Nipah virus
NiV-Malaysia
NA
NA
Increase
Investigational
29765101
DrugRepV_0756Favipiravir
Antiviral
Influenza virus
Ebola virus
NA
NA
NA
Increase (7 %)
Investigational
26930627
DrugRepV_0758Favipiravir
Antiviral
Influenza virus
Ebola virus
NA
NA
NA
Decrease (33 %)
Investigational
26930627
DrugRepV_1892Seliciclib
Anticancer
Breast cancer | Lung cancer | Lymphoma | Multiple myeloma | Leukemia
Zika virus
FSS13026
NA
NA
Decrease (50 %)
Investigational
27571349
DrugRepV_1893SNS-032
NA
Cancer
Zika virus
FSS13026
NA
NA
Decrease (50 %)
Investigational
27571349
DrugRepV_1894PHA-793887
Anticancer
Cancer
Zika virus
FSS13026
NA
NA
Decrease (50 %)
NA
27571349
DrugRepV_1895AT7519
NA
Cancer
Zika virus
FSS13026
NA
NA
Decrease (50 %)
NA
27571349
DrugRepV_1896BS-194
Anticancer
Cancer
Zika virus
FSS13026
NA
NA
Decrease (50 %)
NA
27571349
DrugRepV_1897RGB-286147
NA
NA
Zika virus
FSS13026
NA
NA
Decrease (50 %)
NA
27571349
DrugRepV_1898Dinaciclib
Anticancer
Cancer
Zika virus
FSS13026
NA
NA
Decrease (50 %)
Investigational
27571349
DrugRepV_1899Alvocidib
NA
Cancer
Zika virus
FSS13026
NA
NA
Decrease (50 %)
Experimental
27571349
DrugRepV_2957Doxycycline
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
NA
NA
Approved
25970853
DrugRepV_2958Doxycycline
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
NA
NA
Approved
25970853
DrugRepV_3679NSC 62914
NA
NA
Ebola virus
NA
NA
NA
Decrease
NA
22027648
DrugRepV_3680NSC 62914
NA
NA
Marburg virus
NA
NA
NA
Decrease
NA
22027648
DrugRepV_3681N3,N12-bis[2-(morpholin-4-yl)ethyl]-6,15-diazatetracyclo[8.8.0.02,7.011,16]octadeca-1(10),2,4,6,8,11(16),12,14,17-nonaene-3,12-diamine tetrahydrochloride
NA
NA
Ebola virus
Zaire-95
NA
NA
Decrease (50 %)
NA
23012625
DrugRepV_3682N5,N14-bis[2-(morpholin-4-yl)ethyl]-3,12-bis({[2-(morpholin-4-yl)ethyl]amino})-6,15-diazatetracyclo[8.8.0.02,7.011,16]octadeca-1(10),2,4,6,8,11(16),12,14,17-nonaene-5,14-dicarboxamide; hexakis(trifluoroacet
NA
NA
Ebola virus
Zaire-95
NA
NA
Decrease (50 %)
NA
23012625
DrugRepV_3683N3,N12-bis[2-(morpholin-4-yl)ethyl]-6,15-diazatetracyclo[8.8.0.02,7.011,16]octadeca-1(10),2,4,6,8,11(16),12,14,17-nonaene-3,12-diamine
NA
NA
Ebola virus
Zaire-95
NA
NA
Decrease (50 %)
NA
23012625
DrugRepV_3684N3,N12-bis[2-(morpholin-4-yl)ethyl]-6,15-diazatetracyclo[8.8.0.02,7.011,16]octadeca-1(10),2,4,6,8,11(16),12,14,17-nonaene-3,12-diamine tetrahydrochloride
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
23012625
DrugRepV_3685N3,N12-bis[2-(morpholin-4-yl)ethyl]-6,15-diazatetracyclo[8.8.0.02,7.011,16]octadeca-1(10),2,4,6,8,11(16),12,14,17-nonaene-3,12-diamine
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
23012625
DrugRepV_3703Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Marburg virus
NA
NA
NA
Decrease (83 %)
Approved
24713118
DrugRepV_37046-Azauridine
NA
Cancer
Marburg virus
NA
NA
NA
Decrease (98 %)
NA
24713118
DrugRepV_3705Chloroquine
Malaria
Malaria
Marburg virus
NA
NA
NA
Decrease (99.9 %)
Approved
24713118
DrugRepV_3706Imatinib Methanesulfonate Salt
Antineoplastic and Immunomodulating Agents
NA
Marburg virus
NA
NA
NA
Decrease (99 %)
Approved
24713118
DrugRepV_3707Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Ebola virus
NA
NA
NA
Decrease (0 %)
Approved
24713118
DrugRepV_37086-Azauridine
NA
Cancer
Ebola virus
NA
NA
NA
Decrease (99 %)
NA
24713118
DrugRepV_3709Chloroquine
Antiparasitic products, Insectisides and Repellents
Malaria
Ebola virus
NA
NA
NA
Decrease (99.9 %)
Approved
24713118
DrugRepV_3710Imatinib Methanesulfonate Salt
Antineoplastic and Immunomodulating Agents
NA
Ebola virus
NA
NA
NA
Decrease (95 %)
Approved
24713118
DrugRepV_3726OSU-03012
Anticancer
Brain cancer
Lassa virus
NA
NA
NA
Decrease
NA
25986249
DrugRepV_3727AZD8055
NA
Cancer
Lassa virus
NA
NA
NA
Decrease
Investigational
25986249
DrugRepV_3728TWS119
NA
NA
Lassa virus
NA
NA
NA
Decrease
NA
25986249
DrugRepV_3729SU 4312
NA
NA
Lassa virus
NA
NA
NA
Decrease
NA
25986249
DrugRepV_3730Falnidamol dihydrochloride
NA
Solid Tumor
Lassa virus
NA
NA
NA
Decrease
Investigational
25986249
DrugRepV_3731Ki 8751
NA
NA
Lassa virus
NA
NA
NA
Decrease
NA
25986249
DrugRepV_373210-DEBC hydrochloride
NA
NA
Lassa virus
NA
NA
NA
Decrease
NA
25986249
DrugRepV_3751MLS000078751
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3752MLS000394177
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3753MLS000534476
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3754MLS000554255
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3755MLS000555232
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3756MLS000730532
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3757MLS000733230
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3758MLS000762907
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3759MLS001101371
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3760MLS000078751
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3761MLS000394177
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3762MLS000534476
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3763MLS000554255
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3764MLS000555232
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3765MLS000730532
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3766MLS000733230
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3767MLS000762907
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3768MLS001101371
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3769MLS001239325
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3770MLS001239325
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3771MLS001030162
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3772MLS001030162
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3773MLS000666802
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3774MLS000666802
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3775MLS000999960
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3776MLS000999960
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3777MLS001173370
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3778MLS001173370
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3779MLS001174896
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3780MLS001174896
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3781MLS001196083
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3782MLS001196083
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3783MLS001239358
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3784MLS001239358
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3785MLS001177927
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3786MLS001177927
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3787MLS001209453
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3788MLS001209453
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3789MLS000580080
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3790MLS000580080
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3791MLS000106706
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3792MLS000106706
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3793MLS001175455
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3794MLS001175455
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3795MLS000772389
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3796MLS000772389
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3797MLS000042810
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3798MLS000042810
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3799MLS001162808
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3800MLS001162808
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3801MLS000684231
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3802MLS000684231
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3803MLS000556387
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3804MLS000556387
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3805MLS001179278
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3806MLS001179278
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3807MLS000567464
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3808MLS000567464
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3809MLS000583959
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3810MLS000583959
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3811MLS001018888
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3812MLS001018888
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3813MLS001047402
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3814MLS001047402
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3815MLS001029946
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3816MLS001029946
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3817MLS000332573
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3818MLS000332573
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3819MLS000936259
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3820MLS000936259
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3821MLS000718690
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3822MLS000718690
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3823MLS000880330
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3824MLS000880330
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3825MLS001207131
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3826MLS001207131
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3827MLS000673118
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3828MLS000673118
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3829MLS000689481
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3830MLS000689481
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3831MLS001179272
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3832MLS001179272
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3833MLS002702500
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3834MLS002702500
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3835MLS001180408
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3836MLS000737975
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3837MLS001237534
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3838MLS000336293
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3839MLS000780111
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3840MLS001179997
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3841MLS000418057
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3842MLS000936795
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3843MLS000092187
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3844MLS000391391
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3845MLS000569139
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3846MLS001045935
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3847MLS001181479
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3848MLS000391984
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3849MLS000063146
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3850MLS000768081
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3851MLS000091920
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3852MLS001150589
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3853MLS000736237
NA
NA
Marburg virus
Musoke
NA
NA
Decrease (50 %)
NA
27161622
DrugRepV_3854Clomiphene
Genito Urinary System and Sex Hormones
Polycystic ovary syndrome
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
Approved
27490565
DrugRepV_3855Enclomiphene
NA
Male hypogonadism
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
Investigational
27490565
DrugRepV_3856Zuclomiphene
NA
NA
Ebola virus
Mayinga
NA
NA
Decrease (50 %)
NA
27490565
DrugRepV_3862Favipiravir
Antiviral
Influenza virus
Lassa virus
Ba366
NA
NA
Decrease (50 %)
Investigational
27736754
DrugRepV_3866Favipiravir
Antiviral
Influenza virus
Ebola virus
Kikwit 1995/E718
NA
NA
Decrease (50 %)
Investigational
27736754
DrugRepV_3893cp15
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3894cp15
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3895cp15
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3896cp15
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3897cp19
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3898cp19
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3899cp19
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3900cp19
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3901cp3
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3902cp5
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3903cp11
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3904cp13
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3905cp15
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3906cp16
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3907cp19
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3908cp3
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3909cp5
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3910cp11
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3911cp13
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3912cp15
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3913cp16
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3914cp19
NA
NA
Marburg virus
Ci67
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3915cp3
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3916cp5
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3917cp11
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3918cp13
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3919cp15
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3920cp16
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3921cp19
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3922CBS1129
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3923CBS1130
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3924CBS1131
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3925CBS1132
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3926CBS1133
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3927CBS1134
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3928CBS1135
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3929CBS1136
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3930CBS1137
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3931CBS1138
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3932CBS1139
NA
NA
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
NA
28645623
DrugRepV_3935Favipiravir
Antiviral
Influenza virus
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
Investigational
29289664
DrugRepV_3936Favipiravir
Antiviral
Influenza virus
Ebola virus
Makona
NA
NA
Decrease (50 %)
Investigational
29289664
DrugRepV_3937Favipiravir
Antiviral
Influenza virus
Marburg virus
Ci67
NA
NA
Decrease (50 %)
Investigational
29289664
DrugRepV_395312N-p-dichlorobenzyl aloperine
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_395412N-o-methylbenzyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_395512N-2,4-dichlorobenzyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_395612N-3,5 -dichlorobenzyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_395712N-3,4-dichlorobenzyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_395812N-m-methoxybenzyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_395912N-benzyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_396012N-p-trifluoromethoxylbenzyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_396112N-p-fluorobenzyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_396212N-3,5-dichlorobenzoyl aloperine
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_396312N-p-chlorobenzoyl aloperine
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_396412N-3,4-dichlorobenzoyl aloperine
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_396512N-3,4-dichlorobenzenesulfonyl aloperine
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_396612N-3,5-dichlorobenzenesulfonyl aloperine
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_396712N-o-thiophenesulfonyl aloperine
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_396812N-m-cyanobenzenesulfonyl aloperine
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_396912N-p-chlorobenzenesulfonyl aloperine
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_397012N-p-chlorophenylethyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_397112N-3,4-dichlorophenylethyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_397212N-3,5-dichlorophenylethyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_397312N-3,4-dichlorohydrocinnamyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_397412N-3,5-dichlorohydrocinnamyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_397512N-p-chlorohydrocinnamyl aloperine dihydrochloride
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_397612N-p-dichlorobenzyl aloperine
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_397712N-o-methylbenzyl aloperine dihydrochloride
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_397812N-2,4-dichlorobenzyl aloperine dihydrochloride
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_397912N-3,5 -dichlorobenzyl aloperine dihydrochloride
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_398012N-3,4-dichlorobenzyl aloperine dihydrochloride
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_398112N-m-methoxybenzyl aloperine dihydrochloride
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_398212N-benzyl aloperine dihydrochloride
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_398312N-p-trifluoromethoxylbenzyl aloperine dihydrochloride
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_398412N-p-fluorobenzyl aloperine dihydrochloride
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_398512N-3,5-dichlorobenzoyl aloperine
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_398612N-p-chlorobenzoyl aloperine
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_398712N-3,4-dichlorobenzoyl aloperine
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_398812N-3,4-dichlorobenzenesulfonyl aloperine
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_398912N-3,5-dichlorobenzenesulfonyl aloperine
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_399012N-o-thiophenesulfonyl aloperine
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_399112N-m-cyanobenzenesulfonyl aloperine
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_399212N-p-chlorobenzenesulfonyl aloperine
NA
NA
Marburg virus
NA
NA
NA
Decrease (50 %)
NA
29494844
DrugRepV_4005FGI-103
NA
NA
Ebola virus
Zaire
NA
NA
Decrease
NA
20211898
DrugRepV_4298Baicalein
Plant extract
Influenza
Chikungunya virus
NA
NA
NA
Decrease (50 %)
Phase II
27460167
DrugRepV_4299Fisetin
NA
Frail Elderly Syndrome
Chikungunya virus
NA
NA
NA
Decrease (50 %)
Experimental
27460167
DrugRepV_4300Quercetagetin
NA
NA
Chikungunya virus
NA
NA
NA
Decrease (50 %)
NA
27460167
DrugRepV_4301Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Chikungunya virus
NA
NA
NA
Decrease (50 %)
Approved
27460167
DrugRepV_4471Brincidofovir
Antiviral
Viral infections
Ebola virus
EBOV-GFP
NA
NA
Decrease (50 %)
Investigational
26526586
DrugRepV_4472Brincidofovir
Antiviral
Viral infections
Ebola virus
EBOV-Gluc
NA
NA
Decrease (50 %)
Investigational
26526586
DrugRepV_4473Brincidofovir
Antiviral
Viral infections
Ebola virus
EBOV-GFP
NA
NA
Decrease (50 %)
Investigational
26526586
DrugRepV_4474Brincidofovir
Antiviral
Viral infections
Ebola virus
EBOV-GFP
NA
NA
Decrease (50 %)
Investigational
26526586
DrugRepV_4475Brincidofovir
Antiviral
Viral infections
Ebola virus
EBOV-GFP
NA
NA
Decrease (50 %)
Investigational
26526586
DrugRepV_4476Brincidofovir
Antiviral
Viral infections
Ebola virus
EBOV-GFP
NA
NA
Decrease (50 %)
Investigational
26526586
DrugRepV_4477Brincidofovir
Antiviral
Viral infections
Ebola virus
EBOV-GFP
NA
NA
Decrease (50 %)
Investigational
26526586
DrugRepV_4479Brincidofovir
Antiviral
Viral infections
Ebola virus
Makona
NA
NA
Decrease (50 %)
Investigational
26526586
DrugRepV_4497Ranpirnase
Anticancer
Cancer
Ebola virus
Kikwit
NA
NA
Decrease (50 %)
Investigational
27350309
DrugRepV_4499Ranpirnase
Anticancer
Cancer
Ebola virus
Kikwit
NA
NA
Increase
Investigational
27350309
DrugRepV_4500(1S,2R,5S)-5-{4-amino-1H-imidazo[4,5-c]pyridin-1-yl}-4-fluoro-3-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
Zaire
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4501(1S,2R,5R)-5-(6-amino-9H-purin-9-yl)-3-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
Zaire
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4502(1S,2R,5R)-5-{4-amino-1H-imidazo[4,5-c]pyridin-1-yl}-3-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
Zaire
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4503(1R,2S,5R)-3-(6-amino-9H-purin-9-yl)-5-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
Zaire
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4504(1R,2S,5R)-3-{4-amino-1H-imidazo[4,5-c]pyridin-1-yl}-5-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
Zaire
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4505(1S,2R,5S)-5-{4-amino-1H-imidazo[4,5-c]pyridin-1-yl}-4-fluoro-3-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4506(1S,2R,5R)-5-(6-amino-9H-purin-9-yl)-3-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4507(1S,2R,5R)-5-{4-amino-1H-imidazo[4,5-c]pyridin-1-yl}-3-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4508(1R,2S,5R)-3-(6-amino-9H-purin-9-yl)-5-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4509(1R,2S,5R)-3-{4-amino-1H-imidazo[4,5-c]pyridin-1-yl}-5-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4510(1S,2R,5S)-5-(6-amino-9H-purin-9-yl)-4-fluoro-3-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Ebola virus
NA
NA
NA
Decrease (50 %)
NA
30385162
DrugRepV_4511(1S,2R,5S)-5-{4-amino-1H-imidazo[4,5-c]pyridin-1-yl}-4-fluoro-3-(hydroxymethyl)cyclopent-3-ene-1,2-diol
NA
NA
Influenza virus
NA
Pathway
NA
Decrease (50 %)
NA
30385162
DrugRepV_4512Favipiravir
Antiviral
Influenza virus
Ebola virus
NA
NA
NA
Increase
Investigational
30275474
DrugRepV_4513Remdesivir
Antiviral
Hepatitis C | Ebola
Ebola virus
NA
NA
NA
Increase
Experimental
30275474
DrugRepV_4514Favipiravir
Antiviral
Influenza virus
Ebola virus
NA
NA
NA
Increase
Investigational
29584730
DrugRepV_4515Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Influenza virus
NA
Pathway
NA
Decrease (50 %)
Approved
15200845
DrugRepV_4516Zanamivir
Antiinfectives For Systemic Use
Influenza virus
Influenza virus
NA
Pathway
NA
Decrease (50 %)
Approved
15200845
DrugRepV_4517Oseltamivir
Antiinfectives For Systemic Use
Influenza A/B virus
Influenza virus
NA
Pathway
NA
Decrease (50 %)
Approved
15200845
DrugRepV_4518Amantadine
Nervous System
Influenza and Parkinson Disease
Influenza virus
NA
Pathway
NA
Decrease (50 %)
Approved
15200845
DrugRepV_45401-[4,5-dihydroxy-3-(hydroxymethyl)cyclopent-2-en-1-yl]-1H-1,2,4-triazole-3-carboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
16451078
DrugRepV_45411-[4,5-dihydroxy-3-(hydroxymethyl)cyclopent-2-en-1-yl]-1H-imidazole-4-carboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
16451078
DrugRepV_45421-[4,5-dihydroxy-3-(hydroxymethyl)cyclopent-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
16451078
DrugRepV_4543Alferon
NA
Condylomata acuminata
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Approved
16451078
DrugRepV_4544Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Approved
15961169
DrugRepV_4545AZT
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Approved
15961169
DrugRepV_4546Lopinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Approved
15961169
DrugRepV_4547Aurintricarboxylic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
15961169
DrugRepV_4548DS5000
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
15961169
DrugRepV_4549Novaron
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
15961169
DrugRepV_4550Glycirrhizin
Bile And Liver Therapy
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
15961169
DrugRepV_4551S-Nitroso-N-acetylpenicillamine
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
15961169
DrugRepV_45527-(benzyloxy)-2-(3,4-dihydroxyphenyl)-3,5-dihydroxy-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45532-(3,4-dihydroxyphenyl)-7-[(2-fluorophenyl)methoxy]-3,5-dihydroxy-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45547-[(2-chlorophenyl)methoxy]-2-(3,4-dihydroxyphenyl)-3,5-dihydroxy-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45557-[(2-bromophenyl)methoxy]-2-(3,4-dihydroxyphenyl)-3,5-dihydroxy-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45562-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(2-iodophenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45572-({[2-(3,4-dihydroxyphenyl)-3,5-dihydroxy-4-oxo-4H-chromen-7-yl]oxy}methyl)benzonitrile
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45582-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(2-nitrophenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45592-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(2-methylphenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45602-(3,4-dihydroxyphenyl)-7-[(3-fluorophenyl)methoxy]-3,5-dihydroxy-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45617-[(3-chlorophenyl)methoxy]-2-(3,4-dihydroxyphenyl)-3,5-dihydroxy-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45627-[(3-bromophenyl)methoxy]-2-(3,4-dihydroxyphenyl)-3,5-dihydroxy-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45632-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(3-iodophenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45643-({[2-(3,4-dihydroxyphenyl)-3,5-dihydroxy-4-oxo-4H-chromen-7-yl]oxy}methyl)benzonitrile
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45652-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(3-nitrophenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45662-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(3-methylphenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45672-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(3-methoxyphenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45682-(3,4-dihydroxyphenyl)-7-[(4-fluorophenyl)methoxy]-3,5-dihydroxy-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45697-[(4-chlorophenyl)methoxy]-2-(3,4-dihydroxyphenyl)-3,5-dihydroxy-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45707-[(4-bromophenyl)methoxy]-2-(3,4-dihydroxyphenyl)-3,5-dihydroxy-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45712-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(4-iodophenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45724-({[2-(3,4-dihydroxyphenyl)-3,5-dihydroxy-4-oxo-4H-chromen-7-yl]oxy}methyl)benzonitrile
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45732-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(4-nitrophenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45742-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(4-methylphenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_45752-(3,4-dihydroxyphenyl)-3,5-dihydroxy-7-[(4-methoxyphenyl)methoxy]-4H-chromen-4-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
22297745
DrugRepV_46031H-1,2,3-benzotriazol-1-yl 1H-indole-5-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_46045-chloropyridin-3-yl 1H-indole-5-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_46055-chloropyridin-3-yl 1-acetyl-1H-indole-5-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_46065-chloropyridin-3-yl 1-(4-methylbenzenesulfonyl)-1H-indole-5-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_46075-chloropyridin-3-yl 1-(3-nitrobenzenesulfonyl)-1H-indole-5-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_46085-chloropyridin-3-yl1H-indole-6-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_46095-chloropyridin-3-yl 1H-indole-4-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_46105-chloropyridin-3-yl 1-acetyl-1H-indole-4-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_46115-chloropyridin-3-yl 1H-indole-7-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_46125-chloropyridin-3-yl (6R)-6-{[(tert-butoxy)carbonyl]amino}-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_46135-chloropyridin-3-yl 2-acetyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
Urbani
NA
NA
Decrease (50 %)
NA
18796354
DrugRepV_4682Arbidol
NA
Viral infection
Zika virus
MR766
NA
NA
Decrease (50 %)
Investigational
29895962
DrugRepV_47736-Mercaptopurine
Antineoplastic and Immunomodulating Agents
Acute lymphatic leukemia
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Approved
25542975
DrugRepV_4774Thioguanine
Antineoplastic and Immunomodulating Agents
Acute leukemia
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Approved
25542975
DrugRepV_4775N-ethylmaleimide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Experimental
25542975
DrugRepV_4776Mycophenolic Acid
Antineoplastic and Immunomodulating Agents
Organ rejection (immunosuppressants)
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Approved
25542975
DrugRepV_47842-(5-{[(4Z)-1-(3-carboxyphenyl)-3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)-4-chlorobenzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47852-(5-{[(4Z)-1-(3-carboxyphenyl)-5-oxo-3-(trifluoromethyl)-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)-4-chlorobenzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47862-(5-{[(4Z)-1-(3-carboxyphenyl)-5-oxo-3-(trifluoromethyl)-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47872-(5-{[(4Z)-1-(3-carboxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)-4-chlorobenzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47884-chloro-2-(5-{[(4Z)-3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47894-chloro-2-(5-{[(4Z)-5-oxo-1,3-diphenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47904-chloro-2-(5-{[(4Z)-1-(4-fluorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47914-chloro-2-(5-{[(4Z)-5-oxo-3-phenyl-1-[4-(propan-2-yl)phenyl]-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47922-(5-{[(4Z)-1-(4-tert-butylphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)-4-chlorobenzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_4793(4Z)-1,3-diphenyl-4-[(5-phenylfuran-2-yl)methylidene]-4,5-dihydro-1H-pyrazol-5-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47943-[(4Z)-5-oxo-3-phenyl-4-[(5-phenylfuran-2-yl)methylidene]-4,5-dihydro-1H-pyrazol-1-yl]benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47953-[(4Z)-3-methyl-5-oxo-4-[(5-phenylfuran-2-yl)methylidene]-4,5-dihydro-1H-pyrazol-1-yl]benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47962-(5-{[(4Z)-5-oxo-1,3-diphenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47972-(5-{[(4Z)-1-(4-fluorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47982-(5-{[(4Z)-5-oxo-3-phenyl-1-[4-(propan-2-yl)phenyl]-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_47992-(5-{[(4Z)-1-(4-tert-butylphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48002-(5-{[(4Z)-1-(4-cyanophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48012-(5-{[(4Z)-1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoicacid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48023-[(4Z)-4-[(furan-2-yl)methylidene]-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl]benzoic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48032-(5-{[(4Z)-1-(3-carboxyphenyl)-3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)-4-chlorobenzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48042-(5-{[(4Z)-1-(3-carboxyphenyl)-5-oxo-3-(trifluoromethyl)-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)-4-chlorobenzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48052-(5-{[(4Z)-1-(3-carboxyphenyl)-5-oxo-3-(trifluoromethyl)-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48062-(5-{[(4Z)-1-(3-carboxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)-4-chlorobenzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48074-chloro-2-(5-{[(4Z)-3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48084-chloro-2-(5-{[(4Z)-5-oxo-1,3-diphenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48094-chloro-2-(5-{[(4Z)-1-(4-fluorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48104-chloro-2-(5-{[(4Z)-5-oxo-3-phenyl-1-[4-(propan-2-yl)phenyl]-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48112-(5-{[(4Z)-1-(4-tert-butylphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)-4-chlorobenzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_4812(4Z)-1,3-diphenyl-4-[(5-phenylfuran-2-yl)methylidene]-4,5-dihydro-1H-pyrazol-5-one
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48133-[(4Z)-5-oxo-3-phenyl-4-[(5-phenylfuran-2-yl)methylidene]-4,5-dihydro-1H-pyrazol-1-yl]benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48143-[(4Z)-3-methyl-5-oxo-4-[(5-phenylfuran-2-yl)methylidene]-4,5-dihydro-1H-pyrazol-1-yl]benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48152-(5-{[(4Z)-5-oxo-1,3-diphenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48162-(5-{[(4Z)-1-(4-fluorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48172-(5-{[(4Z)-5-oxo-3-phenyl-1-[4-(propan-2-yl)phenyl]-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48182-(5-{[(4Z)-1-(4-tert-butylphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48192-(5-{[(4Z)-1-(4-cyanophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48202-(5-{[(4Z)-1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-yl)benzoicacid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48213-[(4Z)-4-[(furan-2-yl)methylidene]-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl]benzoic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
27240464
DrugRepV_48338-(trifluoromethyl)-9H-purin-6-amine
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
25746232
DrugRepV_48348-(trifluoromethyl)-9H-purin-6-amine
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
25746232
DrugRepV_48355-amino-2-methyl-N-[(1R)-1-(naphthalen-1-yl)ethyl]benzamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
25746232
DrugRepV_48362-methyl-5-[(methylamino)methyl]-N-[(1R)-1-(naphthalen-1-yl)ethyl]benzamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
25746232
DrugRepV_4837N-[(2H-1,3-benzodioxol-5-yl)methyl]-1-[(1R)-1-(naphthalen-1-yl)ethyl]piperidine-4-carboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
25746232
DrugRepV_4838N-[(2H-1,3-benzodioxol-5-yl)methyl]-1-[(1S)-1-(naphthalen-1-yl)ethyl]piperidine-4-carboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
25746232
DrugRepV_4839N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}thiophene-2-carboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4840N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}benzamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4841N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}cyclobutanecarboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4842N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}cyclohexanecarboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48432-(1H-1,2,3-benzotriazol-1-yl)-N-[4-(pyridin-4-yl)phenyl]-N-[(thiophen-3-yl)methyl]acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4844N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}-2-methylpropanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48452-(1H-1,2,3-benzotriazol-1-yl)-N-[4-(2-methoxypyridin-3-yl)phenyl]-N-[(thiophen-3-yl)methyl]acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4846N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}cyclopropanecarboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48472-(1H-1,2,3-benzotriazol-1-yl)-N-[4-(2-methoxypyrimidin-5-yl)phenyl]-N-[(thiophen-3-yl)methyl]acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4848N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}-2,2,2-trifluoroacetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48492-(1H-1,2,3-benzotriazol-1-yl)-N-[4-(pyridin-3-yl)phenyl]-N-[(thiophen-3-yl)methyl]acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48502-methylpropyl N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}carbamate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4851N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}propanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4852N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}-2-methoxyacetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4853N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}-3-methoxypropanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48542-(1H-1,2,3-benzotriazol-1-yl)-N-[4-(methylamino)phenyl]-N-[(thiophen-3-yl)methyl]acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48552-(1H-1,2,3-benzotriazol-1-yl)-N-[4-(benzylamino)phenyl]-N-[(thiophen-3-yl)methyl]acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4856N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}-2,2-dimethylpropanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48572-methyl-N-(4-{N-[(thiophen-3-yl)methyl]-2-(1H-1,2,3-triazol-1-yl)acetamido}phenyl)propanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4858methyl 2-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}-1H-pyrrole-1-carboxylate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (31 %)
NA
26190463
DrugRepV_48592-(1H-1,2,3-benzotriazol-1-yl)-N-{[1,1-biphenyl]-4-yl}-N-[(thiophen-3-yl)methyl]acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4860N-(4-tert-butylphenyl)-N-[(pyridin-3-yl)methyl]-1H-imidazole-4-carboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (49 %)
NA
26190463
DrugRepV_48612-methyl-N-{4-[2-(4-phenyl-1H-1,2,3-triazol-1-yl)-N-[(thiophen-3-yl)methyl]acetamido]phenyl}propanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (25 %)
NA
26190463
DrugRepV_4862N-(4-tert-butylphenyl)-N-[(pyridin-3-yl)methyl]furan-3-carboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (24 %)
NA
26190463
DrugRepV_48632-methyl-N-(4-{N-[(thiophen-3-yl)methyl]-2-[4-(trimethylsilyl)-1H-1,2,3-triazol-1-yl]acetamido}phenyl)propanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_4864N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1-methyl-1H-imidazol-4-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4865N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(benzylcarbamoyl)(3-fluorophenyl)methyl]acetamido]phenyl}-2-methylpropanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48662-[2-(1H-1,2,3-benzotriazol-1-yl)-N-(4-acetamidophenyl)acetamido]-N-tert-butyl-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4867N-tert-butyl-2-(N-{2-cyano-[1,1-biphenyl]-4-yl}-1-(furan-2-yl)formamido)-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4868N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(1H-indol-3-yl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4869N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}cyclopropanecarboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4870N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(benzylcarbamoyl)(3-fluorophenyl)methyl]acetamido]phenyl}cyclobutanecarboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4871N-tert-butyl-2-(N-{4-[(fluoromethoxy)methyl]phenyl}-2-(1H-indol-3-yl)acetamido)-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4872N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}benzamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4873N-tert-butyl-2-[2-(1H-indol-3-yl)-N-[4-(propan-2-yl)phenyl]acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4874N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(benzylcarbamoyl)(3-fluorophenyl)methyl]acetamido]phenyl}cyclopropanecarboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4875N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1,3-oxazol-5-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4876N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1H-imidazol-4-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4877N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4878N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1H-imidazol-4-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4879N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}-1,2-oxazole-5-carboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4880N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1H-imidazol-4-yl)formamido]-2-(pyrimidin-5-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4881N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}-2-methylpropanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4882N-{4-[2-(1H-1,3-benzodiazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}propanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48832-[2-(1H-1,2,3-benzotriazol-1-yl)-N-(4-acetamidophenyl)acetamido]-N-tert-butyl-2-(3-fluorophenyl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_48842-[N-(4-aminophenyl)-2-(1H-1,2,3-benzotriazol-1-yl)acetamido]-N-tert-butyl-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4885(2S)-N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4886N-{4-[2-(1H-1,3-benzodiazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}-2-methylpropanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4887N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1,3-oxazol-5-yl)formamido]-2-(pyrimidin-5-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
26190463
DrugRepV_4888N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}thiophene-2-carboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (26 %)
NA
26190463
DrugRepV_4889N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}cyclobutanecarboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (20 %)
NA
26190463
DrugRepV_4890N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}cyclohexanecarboxamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4891N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}propanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (34 %)
NA
26190463
DrugRepV_4892N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}-2,2-dimethylpropanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4893N-tert-butyl-2-[1-(4-cyanophenyl)-N-(4-fluorophenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (53 %)
NA
26190463
DrugRepV_4894N-tert-butyl-2-[N-cyclopropyl-2-(1H-indol-3-yl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (49 %)
NA
26190463
DrugRepV_4895N-tert-butyl-2-[N-cyclopropyl-2-(pyridin-3-yl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (48 %)
NA
26190463
DrugRepV_4896N-tert-butyl-2-[N-(4-fluorophenyl)-2-(pyridin-3-yl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (47 %)
NA
26190463
DrugRepV_4897N-tert-butyl-2-[N-cyclopropyl-1-(furan-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (43 %)
NA
26190463
DrugRepV_4898N-tert-butyl-2-{N-cyclopropyl-1-[5-(trifluoromethyl)pyridin-2-yl]formamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (42 %)
NA
26190463
DrugRepV_4899N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(pyrazin-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (41 %)
NA
26190463
DrugRepV_4900N-tert-butyl-2-{N-[4-(propan-2-yl)phenyl]-2-(pyridin-3-yl)acetamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (41 %)
NA
26190463
DrugRepV_4901N-tert-butyl-2-[N-(4-fluorophenyl)-2-(1H-indol-3-yl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (41 %)
NA
26190463
DrugRepV_4902N-tert-butyl-2-[N-(4-fluorophenyl)-1-(furan-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (41 %)
NA
26190463
DrugRepV_4903(2S)-2-{N-[4-(butan-2-yl)phenyl]-1-(furan-2-yl)formamido}-N-tert-butyl-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (39 %)
NA
26190463
DrugRepV_4904N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(pyridazin-4-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (35 %)
NA
26190463
DrugRepV_4905N-tert-butyl-2-[1-(3-methylfuran-2-yl)-N-[4-(propan-2-yl)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (36 %)
NA
26190463
DrugRepV_4906N-tert-butyl-2-[1-(furan-2-yl)-N-[4-(propan-2-yl)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (34 %)
NA
26190463
DrugRepV_49072-[2-(1H-1,2,3-benzotriazol-1-yl)-N-(4-acetamidophenyl)acetamido]-2-(3-fluorophenyl)-N-phenylacetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (32 %)
NA
26190463
DrugRepV_4908N-tert-butyl-2-{N-[4-(difluoromethoxy)phenyl]-1-(furan-2-yl)formamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (31 %)
NA
26190463
DrugRepV_4909N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(1H-indol-3-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (31 %)
NA
26190463
DrugRepV_4910N-tert-butyl-2-[1-(furan-2-yl)-N-[4-(1H-pyrrol-3-yl)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (31 %)
NA
26190463
DrugRepV_4911N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1,3-oxazol-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (30 %)
NA
26190463
DrugRepV_4912N-tert-butyl-2-[N-(4-fluorophenyl)-1-[5-(trifluoromethyl)pyridin-2-yl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (29 %)
NA
26190463
DrugRepV_4913N-tert-butyl-2-{N-[4-(fluoromethoxy)phenyl]-2-(pyridin-3-yl)acetamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (29 %)
NA
26190463
DrugRepV_4914[(tert-butylcarbamoyl)(pyridin-3-yl)methyl](4-tert-butylphenyl)carbamic acid
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (29 %)
NA
26190463
DrugRepV_49152-[2-(1H-1,3-benzodiazol-1-yl)-N-(4-methanesulfonamidophenyl)acetamido]-N-tert-butyl-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (28 %)
NA
26190463
DrugRepV_4916N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1H-pyrazol-5-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (28 %)
NA
26190463
DrugRepV_4917N-tert-butyl-2-[1-(4-cyanophenyl)-N-[4-(propan-2-yl)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (28 %)
NA
26190463
DrugRepV_4918N-tert-butyl-2-{N-[4-(3,5-dimethyl-1,2-oxazol-4-yl)phenyl]-1-(furan-2-yl)formamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (28 %)
NA
26190463
DrugRepV_4919N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (28 %)
NA
26190463
DrugRepV_49202-[2-(1H-1,2,3-benzotriazol-1-yl)-N-(4-methanesulfonamidophenyl)acetamido]-N-tert-butyl-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (27 %)
NA
26190463
DrugRepV_4921N-tert-butyl-2-[N-(4-acetamidophenyl)-2-(1H-1,2,3-triazol-1-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (27 %)
NA
26190463
DrugRepV_4922N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(4-chlorophenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (27 %)
NA
26190463
DrugRepV_4923N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(5-methylfuran-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (26 %)
NA
26190463
DrugRepV_4924N-tert-butyl-2-[2-(naphthalen-1-yl)-N-[4-(propan-2-yl)phenyl]acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (26 %)
NA
26190463
DrugRepV_4925N-tert-butyl-2-(4-tert-butylphenyl)-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (26 %)
NA
26190463
DrugRepV_4926N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(naphthalen-1-yl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (26 %)
NA
26190463
DrugRepV_4927N-tert-butyl-2-{N-[4-(fluoromethoxy)phenyl]-2-(1H-indol-3-yl)acetamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (25 %)
NA
26190463
DrugRepV_4928N-tert-butyl-2-{N-[4-(propan-2-yl)phenyl]-1-(5,6,7,8-tetrahydronaphthalen-1-yl)formamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (25 %)
NA
26190463
DrugRepV_4929N-tert-butyl-2-[2-(1H-indol-3-yl)-N-[4-(propan-2-yl)phenyl]acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (25 %)
NA
26190463
DrugRepV_4930N-tert-butyl-2-[1-(furan-2-yl)-N-[4-(2-methylpropoxy)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (25 %)
NA
26190463
DrugRepV_49312-{N-[4-(benzyloxy)phenyl]-1-(furan-2-yl)formamido}-N-tert-butyl-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (25 %)
NA
26190463
DrugRepV_4932N-tert-butyl-2-{N-[4-(propan-2-yl)phenyl]-2-(pyridin-3-yl)acetamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (24 %)
NA
26190463
DrugRepV_4933N-tert-butyl-2-[N-(4-fluorophenyl)-2-(pyridin-3-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (24 %)
NA
26190463
DrugRepV_4934N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(1H-imidazol-4-yl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (24 %)
NA
26190463
DrugRepV_4935N-tert-butyl-2-{N-[4-(difluoromethoxy)phenyl]-1-(1H-indazol-3-yl)formamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (24 %)
NA
26190463
DrugRepV_4936N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(pyridin-3-yl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (23 %)
NA
26190463
DrugRepV_4937N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1H-indazol-3-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (23 %)
NA
26190463
DrugRepV_4938N-tert-butyl-2-(N-{2,6-difluoro-[1,1-biphenyl]-4-yl}-1-(furan-2-yl)formamido)-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (23 %)
NA
26190463
DrugRepV_4939N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-methoxyacetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (23 %)
NA
26190463
DrugRepV_4940N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(pyridin-3-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (23 %)
NA
26190463
DrugRepV_4941N-tert-butyl-2-[1-(4-cyanophenyl)-N-cyclopropylformamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (23 %)
NA
26190463
DrugRepV_4942N-tert-butyl-2-[N-(4-fluorophenyl)-1-(5,6,7,8-tetrahydronaphthalen-1-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (22 %)
NA
26190463
DrugRepV_4943N-tert-butyl-2-[N-cyclopropyl-2-(naphthalen-1-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (22 %)
NA
26190463
DrugRepV_4944N-tert-butyl-2-[N-(4-fluorophenyl)-2-(naphthalen-1-yl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (22 %)
NA
26190463
DrugRepV_4945N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1H-imidazol-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (22 %)
NA
26190463
DrugRepV_49462-(N-{[1,1-biphenyl]-4-yl}-1-(furan-2-yl)formamido)-N-tert-butyl-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (22 %)
NA
26190463
DrugRepV_4947N-tert-butyl-2-[N-(4-fluorophenyl)-2-(1H-indol-3-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (22 %)
NA
26190463
DrugRepV_4948N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(5,6,7,8-tetrahydronaphthalen-1-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4949N-tert-butyl-2-[N-cyclopropyl-1-(1H-indazol-3-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4950N-tert-butyl-2-{N-[4-(fluoromethoxy)phenyl]-2-(naphthalen-1-yl)acetamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4951N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(4-fluorophenyl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4952N-tert-butyl-2-[1-(1H-indazol-3-yl)-N-[4-(propan-2-yl)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4953N-tert-butyl-2-[1-(4-cyanophenyl)-N-[4-(propan-2-yl)phenyl]formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4954N-tert-butyl-2-[N-cyclopropyl-1-(1H-indazol-3-yl)formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4955N-tert-butyl-2-[1-(furan-2-yl)-N-{4-[(1E)-2-phenylethenyl]phenyl}formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4956N-tert-butyl-2-{N-[4-(fluoromethoxy)phenyl]-1-(5,6,7,8-tetrahydronaphthalen-2-yl)formamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (21 %)
NA
26190463
DrugRepV_4957(2R)-2-{N-[4-(butan-2-yl)phenyl]-1-(furan-2-yl)formamido}-N-tert-butyl-2-(pyridin-4-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (20 %)
NA
26190463
DrugRepV_4958N-tert-butyl-2-[N-(4-acetamidophenyl)-2-[4-(trimethylsilyl)-1H-1,2,3-triazol-1-yl]acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (20 %)
NA
26190463
DrugRepV_49592-{N-[4-(butan-2-yloxy)phenyl]-1-(furan-2-yl)formamido}-N-tert-butyl-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (20 %)
NA
26190463
DrugRepV_4960N-tert-butyl-2-[1-(4-cyanophenyl)-N-cyclopropylformamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (20 %)
NA
26190463
DrugRepV_4961N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-phenylacetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (20 %)
NA
26190463
DrugRepV_4962N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (20 %)
NA
26190463
DrugRepV_4963N-tert-butyl-2-{N-[4-(propan-2-yl)phenyl]-1-(5,6,7,8-tetrahydronaphthalen-1-yl)formamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (20 %)
NA
26190463
DrugRepV_4964N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (19 %)
NA
26190463
DrugRepV_49652-[1-(1-benzofuran-3-yl)-N-(4-tert-butylphenyl)formamido]-N-tert-butyl-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (19 %)
NA
26190463
DrugRepV_4966N-tert-butyl-2-[N-(4-acetamidophenyl)-2-(4-phenyl-1H-1,2,3-triazol-1-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (19 %)
NA
26190463
DrugRepV_4967N-tert-butyl-2-[N-(4-fluorophenyl)-1-[5-(trifluoromethyl)pyridin-2-yl]formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (19 %)
NA
26190463
DrugRepV_4968N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (19 %)
NA
26190463
DrugRepV_4969N-tert-butyl-2-[1-(furan-2-yl)-N-(4-phenoxyphenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (19 %)
NA
26190463
DrugRepV_49702-methylpropyl N-{4-[2-(1H-1,2,3-benzotriazol-1-yl)-N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]acetamido]phenyl}carbamate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (19 %)
NA
26190463
DrugRepV_4971N-(4-{N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]-2-(2-methyl-1H-imidazol-1-yl)acetamido}phenyl)propanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (19 %)
NA
26190463
DrugRepV_4972N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(oxolan-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4973N-tert-butyl-2-[N-cyclopropyl-1-(5,6,7,8-tetrahydronaphthalen-1-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_49742-[N-(4-aminophenyl)-2-(1H-1,3-benzodiazol-1-yl)acetamido]-N-tert-butyl-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4975N-tert-butyl-2-(N-{2,3-difluoro-[1,1-biphenyl]-4-yl}-1-(furan-2-yl)formamido)-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4976N-tert-butyl-2-{N-[4-(fluoromethoxy)phenyl]-1-[5-(trifluoromethyl)pyridin-2-yl]formamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4977N-tert-butyl-2-[1-(furan-2-yl)-N-[4-(propan-2-yl)phenyl]formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4978N-tert-butyl-2-[N-cyclopropyl-1-(furan-2-yl)formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4979N-tert-butyl-2-[1-(furan-2-yl)-N-[4-(3-methoxyphenoxy)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4980N-(4-{N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]-2-(2-methyl-1H-imidazol-1-yl)acetamido}phenyl)-2-methylpropanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4981N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1H-pyrrol-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4982N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(4-cyanophenyl)formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4983N-tert-butyl-2-{N-[4-(propan-2-yl)phenyl]-1-[6-(trifluoromethyl)pyridin-3-yl]formamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4984N-tert-butyl-2-{N-[4-(fluoromethoxy)phenyl]-2-(pyridin-3-yl)acetamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_49852-[N-(adamantan-1-yl)-1-(furan-2-yl)formamido]-N-tert-butyl-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (18 %)
NA
26190463
DrugRepV_4986N-tert-butyl-2-[N-(4-fluorophenyl)-1-(5,6,7,8-tetrahydronaphthalen-1-yl)formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_4987N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1H-pyrazol-3-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_4988N-tert-butyl-2-[N-(4-acetamidophenyl)-2-(2-methyl-1H-imidazol-1-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_4989tert-butyl 2-(4-{N-[(tert-butylcarbamoyl)(pyridin-3-yl)methyl]furan-2-amido}phenyl)-1H-pyrrole-1-carboxylate
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_4990N-tert-butyl-2-{N-[4-(difluoromethoxy)phenyl]-1-(1H-indazol-3-yl)formamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_4991N-tert-butyl-2-[N-cyclopropyl-2-(1H-indol-3-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_49922-[N-(4-aminophenyl)-2-(2-methyl-1H-imidazol-1-yl)acetamido]-N-tert-butyl-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_4993N-tert-butyl-2-{N-[4-(fluoromethoxy)phenyl]-2-(naphthalen-1-yl)acetamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_4994N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-[6-(trifluoromethyl)pyridin-3-yl]formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_4995N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(3-methoxyphenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_4996N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(2-methoxyphenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (17 %)
NA
26190463
DrugRepV_4997N-tert-butyl-2-(N-{3-cyano-[1,1-biphenyl]-4-yl}-1-(furan-2-yl)formamido)-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_4998N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(pyrimidin-5-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_4999N-tert-butyl-2-[N-(4-fluorophenyl)-1-(furan-2-yl)formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_50002-[N-(adamantan-1-yl)-2-(1H-1,2,3-benzotriazol-1-yl)acetamido]-N-benzyl-2-(3-fluorophenyl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_5001N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(thiophen-3-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_5002N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-[5-(trifluoromethyl)furan-2-yl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_5003N-tert-butyl-2-[N-cyclopropyl-2-(pyridin-3-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_5004N-tert-butyl-2-[1-(4-cyanophenyl)-N-[4-(fluoromethoxy)phenyl]formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_5005N-tert-butyl-2-(N-{2,4-difluoro-[1,1-biphenyl]-4-yl}-1-(furan-2-yl)formamido)-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_5006N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1H-indazol-3-yl)formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_5007N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(1H-pyrrol-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_5008N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(4-methoxyphenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_50092-[N-(4-benzenesulfonamidophenyl)-1-(furan-2-yl)formamido]-N-tert-butyl-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_5010N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(1H-1,2,3-triazol-4-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_50112-(N-{bicyclo[2.2.1]heptan-2-yl}-1-(furan-2-yl)formamido)-N-tert-butyl-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_5012N-tert-butyl-2-{N-[4-(2-fluoropyridin-4-yl)phenyl]-1-(furan-2-yl)formamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (16 %)
NA
26190463
DrugRepV_50132-[2-(1H-1,2,3-benzotriazol-1-yl)-N-{bicyclo[2.2.1]heptan-2-yl}acetamido]-N-tert-butyl-2-(3-fluorophenyl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_5014N-tert-butyl-2-[1-(furan-2-yl)-N-[4-(pyridin-3-yl)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_50152-[2-(1H-1,3-benzodiazol-1-yl)-N-(4-tert-butylphenyl)acetamido]-N-tert-butyl-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_5016N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(naphthalen-1-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_5017N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-[6-(trifluoromethyl)pyridin-3-yl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_5018N-tert-butyl-2-{N-[4-(fluoromethoxy)phenyl]-1-(5,6,7,8-tetrahydronaphthalen-1-yl)formamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_5019N-tert-butyl-2-{N-[4-(propan-2-yl)phenyl]-1-[6-(trifluoromethyl)pyridin-3-yl]formamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_5020N-tert-butyl-2-{N-[4-(fluoromethoxy)phenyl]-1-[6-(trifluoromethyl)pyridin-3-yl]formamido}-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_5021N-tert-butyl-2-[1-(4-cyanophenyl)-N-[4-(fluoromethoxy)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_5022N-tert-butyl-2-[N-(4-fluorophenyl)-2-(naphthalen-1-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (15 %)
NA
26190463
DrugRepV_5023N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(5,6,7,8-tetrahydronaphthalen-1-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (14 %)
NA
26190463
DrugRepV_5024N-tert-butyl-2-[N-(4-fluorophenyl)-1-(1H-indazol-3-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (14 %)
NA
26190463
DrugRepV_5025N-tert-butyl-2-(N-{4-cyano-[1,1-biphenyl]-4-yl}-1-(furan-2-yl)formamido)-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (14 %)
NA
26190463
DrugRepV_5026N-(4-{N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]-2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetamido}phenyl)-2-methylpropanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (14 %)
NA
26190463
DrugRepV_50272-[N-(adamantan-1-yl)-2-(1H-1,2,3-benzotriazol-1-yl)acetamido]-N-tert-butyl-2-(3-fluorophenyl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (14 %)
NA
26190463
DrugRepV_50282-[2-(1H-1,3-benzodiazol-1-yl)-N-(4-acetamidophenyl)acetamido]-N-tert-butyl-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (14 %)
NA
26190463
DrugRepV_50292-{N-[4-(benzyloxy)phenyl]-1-(furan-2-yl)formamido}-N-tert-butyl-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (14 %)
NA
26190463
DrugRepV_5030N-tert-butyl-2-[N-cyclopropyl-1-(5,6,7,8-tetrahydronaphthalen-1-yl)formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (14 %)
NA
26190463
DrugRepV_5031N-tert-butyl-2-[1-(furan-2-yl)-N-[4-(pyrimidin-5-yl)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (14 %)
NA
26190463
DrugRepV_50322-[N-(4-aminophenyl)-2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetamido]-N-tert-butyl-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (14 %)
NA
26190463
DrugRepV_5033N-tert-butyl-2-{N-[4-(difluoromethoxy)phenyl]-1-(furan-2-yl)formamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (13 %)
NA
26190463
DrugRepV_5034N-tert-butyl-2-[N-(4-methanesulfonamidophenyl)-2-(2-methyl-1H-imidazol-1-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (13 %)
NA
26190463
DrugRepV_5035N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(pyrimidin-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (13 %)
NA
26190463
DrugRepV_5036N-tert-butyl-2-[2-(naphthalen-1-yl)-N-[4-(propan-2-yl)phenyl]acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (13 %)
NA
26190463
DrugRepV_5037N-tert-butyl-2-[1-(furan-2-yl)-N-[4-(propan-2-yloxy)phenyl]formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (13 %)
NA
26190463
DrugRepV_5038N-tert-butyl-2-[1-(4-cyanophenyl)-N-(4-fluorophenyl)formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (13 %)
NA
26190463
DrugRepV_5039N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(pyridin-3-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (13 %)
NA
26190463
DrugRepV_5040N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(pyridin-4-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (13 %)
NA
26190463
DrugRepV_5041N-[(tert-butylcarbamoyl)(pyridin-3-yl)methyl]-N-(4-tert-butylphenyl)-3,3,3-trifluoropropanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (13 %)
NA
26190463
DrugRepV_5042N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(5-chlorofuran-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (12 %)
NA
26190463
DrugRepV_5043N-tert-butyl-2-{N-cyclopropyl-1-[6-(trifluoromethyl)pyridin-3-yl]formamido}-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (12 %)
NA
26190463
DrugRepV_5044N-tert-butyl-2-[N-(4-ethoxyphenyl)-1-(furan-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (12 %)
NA
26190463
DrugRepV_5045N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(1H-pyrazol-4-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (12 %)
NA
26190463
DrugRepV_50462-[2-(1H-1,2,3-benzotriazol-1-yl)-N-{bicyclo[2.2.1]heptan-2-yl}acetamido]-N-benzyl-2-(3-fluorophenyl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (12 %)
NA
26190463
DrugRepV_5047N-tert-butyl-2-(N-{3,4-difluoro-[1,1-biphenyl]-4-yl}-1-(furan-2-yl)formamido)-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (12 %)
NA
26190463
DrugRepV_5048N-tert-butyl-2-[1-(furan-2-yl)-N-(4-methanesulfonamidophenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (12 %)
NA
26190463
DrugRepV_5049N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(pyridin-3-yl)formamido]-2-(pyridin-2-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (12 %)
NA
26190463
DrugRepV_5050N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(4-hydroxyphenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (11 %)
NA
26190463
DrugRepV_5051N-tert-butyl-2-[N-(4-fluorophenyl)-1-(1H-indazol-3-yl)formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (11 %)
NA
26190463
DrugRepV_5052N-tert-butyl-2-[N-(4-tert-butylphenyl)-2-(2-methyl-1H-imidazol-1-yl)acetamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (11 %)
NA
26190463
DrugRepV_5053N-tert-butyl-2-[N-cyclopropyl-2-(naphthalen-1-yl)acetamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (11 %)
NA
26190463
DrugRepV_5054N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (11 %)
NA
26190463
DrugRepV_5055N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(4-cyanophenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (11 %)
NA
26190463
DrugRepV_5056N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(2-hydroxyphenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (11 %)
NA
26190463
DrugRepV_5057N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(1H-pyrazol-5-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (11 %)
NA
26190463
DrugRepV_5058N-tert-butyl-2-[1-(1H-indazol-3-yl)-N-[4-(propan-2-yl)phenyl]formamido]-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (11 %)
NA
26190463
DrugRepV_5059N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(3-hydroxyphenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (10 %)
NA
26190463
DrugRepV_5060N-tert-butyl-2-[1-(furan-2-yl)-N-(4-propoxyphenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (10 %)
NA
26190463
DrugRepV_5061N-tert-butyl-2-[1-(furan-2-yl)-N-(4-methoxyphenyl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (10 %)
NA
26190463
DrugRepV_5062N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(1H-imidazol-4-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (9 %)
NA
26190463
DrugRepV_50632-[2-(1H-1,2,3-benzotriazol-1-yl)-N-(4-tert-butylphenyl)acetamido]-N-tert-butyl-2-(thiophen-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (9 %)
NA
26190463
DrugRepV_50642-[N-(4-benzylphenyl)-1-(furan-2-yl)formamido]-N-tert-butyl-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (8 %)
NA
26190463
DrugRepV_5065N-(4-{N-[(tert-butylcarbamoyl)(thiophen-3-yl)methyl]-2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetamido}phenyl)propanamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (8 %)
NA
26190463
DrugRepV_5066N-tert-butyl-2-[N-(4-tert-butylphenyl)-1-(furan-2-yl)formamido]-2-(6-methylpyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (8 %)
NA
26190463
DrugRepV_5067N-tert-butyl-2-[N-cyclohexyl-1-(furan-2-yl)formamido]-2-(pyridin-3-yl)acetamide
NA
NA
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (6 %)
NA
26190463
DrugRepV_5072Favipiravir
Antiviral
Influenza virus
Crimean-Congo hemorrhagic fever virus
10200
NA
NA
Decrease (50 %)
Investigational
29936152
DrugRepV_5073Favipiravir
Antiviral
Influenza virus
Crimean-Congo hemorrhagic fever virus
Hoti
NA
NA
Decrease (50 %)
Investigational
29936152
DrugRepV_5253beta-D-cyclopentenyl cytosine
NA
NA
Variola virus
Bangladesh 1975
NA
NA
Decrease (50 %)
NA
14604375
DrugRepV_5254beta-D-cyclopentenyl cytosine
NA
NA
Variola virus
7124
NA
NA
Decrease (50 %)
NA
14604375
DrugRepV_5255beta-D-cyclopentenyl-5-iodocytidine
NA
NA
Variola virus
Bangladesh 1975
NA
NA
Decrease (50 %)
NA
14604375
DrugRepV_5256beta-D-cyclopentenyl-5-iodocytidine
NA
NA
Variola virus
7124
NA
NA
Decrease (50 %)
NA
14604375
DrugRepV_5257beta-D-Cyclopentenyl-5-chlorocytidine
NA
NA
Variola virus
Bangladesh 1975
NA
NA
Decrease (50 %)
NA
14604375
DrugRepV_5258beta-D-Cyclopentenyl-5-chlorocytidine
NA
NA
Variola virus
7124
NA
NA
Decrease (50 %)
NA
14604375
DrugRepV_5259beta-D-cyclopentenyl-5-bromocytidine
NA
NA
Variola virus
Bangladesh 1975
NA
NA
Decrease (50 %)
NA
14604375
DrugRepV_5260beta-D-cyclopentenyl-5-bromocytidine
NA
NA
Variola virus
7124
NA
NA
Decrease (50 %)
NA
14604375
DrugRepV_5387Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Chikungunya virus
NA
NA
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_5388Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Ebola virus
NA
NA
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_5389Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Influenza virus
NA
Pathway
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_5390Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Middle East respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_5391Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Rift Valley fever virus
NA
NA
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_5392Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Zika virus
NA
NA
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_5422Losmapimod
NA
Chronic Obstructive Pulmonary Disease
Lassa virus
LP
NA
NA
Decrease (50 %)
Investigational
30953674
DrugRepV_5423Losmapimod
NA
Chronic Obstructive Pulmonary Disease
Lassa virus
803213
NA
NA
Decrease (50 %)
Investigational
30953674
DrugRepV_5424Losmapimod
NA
Chronic Obstructive Pulmonary Disease
Lassa virus
GA391
NA
NA
Decrease (50 %)
Investigational
30953674
DrugRepV_5425Losmapimod
NA
Chronic Obstructive Pulmonary Disease
Lassa virus
Josiah
NA
NA
Decrease (50 %)
Investigational
30953674
DrugRepV_5426ST-193
NA
NA
Lassa virus
LP
NA
NA
Decrease (50 %)
NA
30953674
DrugRepV_5427ST-193
NA
NA
Lassa virus
803213
NA
NA
Decrease (50 %)
NA
30953674
DrugRepV_5428ST-193
NA
NA
Lassa virus
GA391
NA
NA
Decrease (50 %)
NA
30953674
DrugRepV_5429ST-193
NA
NA
Lassa virus
Josiah
NA
NA
Decrease (50 %)
NA
30953674
DrugRepV_5531JQ1
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5532RVX-208
NA
Diabetes, Atherosclerosis, and Coronary Artery Disease
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5533Silmitasertib
NA
Medulloblastoma
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Investigational
32353859
DrugRepV_5534TMCB
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5535Apicidin
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5536Valproic Acid
Nervous System
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved, Investigational
32353859
DrugRepV_5537Bafilomycin A1
Antibiotics
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Experimental
32353859
DrugRepV_5538E-52862
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5539PD-144418
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5540RS-PPCC
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5541PB28
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5542Haloperidol
Nervous System
Schizophrenia | Psychotic disorders | Chemotherapy-induced nausea/vomiting
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved
32353859
DrugRepV_5543Entacapone
Nervous System
Parkinson Disease
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved
32353859
DrugRepV_5544Indomethacin
Cardiovascular agents; Musculo-Skeletal System; Musculo-Skeletal System
Rheumatoid arthritis | Ankylosing spondylitis | Osteoarthritis | Acute painful shoulder (bursitis and/or tendinitis) | Acute gouty arthritis
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved, Investigational
32353859
DrugRepV_5545Metformin
Alimentary Tract and Metabolism
Diabetes
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved
32353859
DrugRepV_5546Ponatinib
Antineoplastic and Immunomodulating Agentss
Chronic myeloid leukemia
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved, Investigational
32353859
DrugRepV_5547H-89
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5548Merimepodib
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Investigational
32353859
DrugRepV_5549Migalastat
Alimentary Tract and Metabolism
Fabry disease
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved, Investigational
32353859
DrugRepV_5550Mycophenolic Acid
Antineoplastic and Immunomodulating Agents
Organ rejection (immunosuppressants)
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved
32353859
DrugRepV_5551Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved
32353859
DrugRepV_5552XL413
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5553CCT 365623
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5554Midostaurin
Antineoplastic and Immunomodulating Agentss
Acute myeloid leukemia (AML)
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved, Investigational
32353859
DrugRepV_5555Ruxolitinib
Antineoplastic and Immunomodulating Agentss
Bone marrow cancer
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved
32353859
DrugRepV_5556ZINC1775962367
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5557ZINC4326719
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5558ZINC4511851
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5559ZINC95559591
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5560AC-55541
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5561AZ8838
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5562Daunorubicin
Antineoplastic and Immunomodulating Agentss
Cancer
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved
32353859
DrugRepV_5563GB110
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5564S-verapamil
NA
Hypertension (high blood pressure) | Angina (chest pain) | Arrhythmia (heart rhythm disorders).
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved
32353859
DrugRepV_5565AZ3451
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5566ABBV-744
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5567dBET6
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5568MZ1
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5569CPI-0610
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5570Sapanisertib
NA
Tumor
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Investigational
32353859
DrugRepV_5571Rapamycin
Antineoplastic and Immunomodulating Agents; Sensory Organ
Prophylaxis of organ rejection in patients receiving renal transplants
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved, Investigational
32353859
DrugRepV_5572Zotatifin
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5573Verdinexor
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Investigational
32353859
DrugRepV_5574Chloroquine
Antiparasitic products, Insectisides and Repellents
Malaria
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved
32353859
DrugRepV_5575Dabrafenib
Antineoplastic and Immunomodulating Agents
Melanoma
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved
32353859
DrugRepV_5576WDB002
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5577Sanglifehrin A
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Experimental
32353859
DrugRepV_5578FK-506
Dermatologicals; Antineoplastic and Immunomodulating Agents
Liver transplantation
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved
32353859
DrugRepV_5579Pevonedistat
NA
Lymphoma
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Investigational
32353859
DrugRepV_5580Ternatin 4
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_55814E2RCat
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5582Tomivosertib
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Investigational
32353859
DrugRepV_5583(2R,5S,11S,14S,17R,18R,21E)-2-(2-aminoethyl)-18-methoxy-11,17-dimethyl-14-(propan-2-yl)-3-oxa-9,12,15,28-tetraazatricyclo[21.3.1.1?,?]octacosa-1(26),21,23(27),24-tetraene-4,10,13,16-tetrone
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5584N-(5-{3-[(4-Hydroxyphenyl)sulfamoyl]-4-methoxyphenyl}-4-methyl-1,3-thiazol-2-yl)-2,2-dimethylpropanamide
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5585PS3061
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5586IHVR-19029
NA
NA
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
NA
32353859
DrugRepV_5587Captopril
Cardiovascular agents
Hypertension
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved
32353859
DrugRepV_5588Lisinopril
Cardiovascular agents
Hypertension | Congestive heart failure
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved, Investigational
32353859
DrugRepV_5589Camostat
Blood and Blood Forming Organs
Pancreatitis
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Experimental
32353859
DrugRepV_5590Nafamostat
NA
Blood vessel coagulation | Hemorrhagic lesions
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Investigational
32353859
DrugRepV_5591Chloramphenicol
Antiinfectives For Systemic Use
Bacterial infections
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved
32353859
DrugRepV_5592Tigecycline
Antiinfectives For Systemic Use
Complicated skin and skin structure infections
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved
32353859
DrugRepV_5593Linezolid
Antiinfectives For Systemic Use
Bacterial infections
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved, Investigational
32353859
DrugRepV_5604Sunitinib-Erlotinib
NA
NA
Dengue virus
N124D/K128E
Pathway
NA
Increase
NA
28240606
DrugRepV_5648Celgosivir
Antiviral
Hepatitis C virus
Dengue virus
DENV1-2402
Pathway
NA
Increase
Phase II
26794905
DrugRepV_5649Celgosivir
Antiviral
Hepatitis C virus
Dengue virus
DENV2-3295
Pathway
NA
Increase
Phase II
26794905
DrugRepV_5650Celgosivir
Antiviral
Hepatitis C virus
Dengue virus
S221
Pathway
NA
Increase
Phase II
26794905
DrugRepV_6064N2-(4-fluorophenyl)-N3-(4-methyl-2-(3-methyl-1H-pyrazol- 5-yl)phenyl) pyrazine-2,3 dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6065N2-(4-methyl-2-(3-methyl-1H-pyrazol-5-yl)phenyl)-N3-(p- tolyl)pyrazine-2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6066N2-(4-fluorophenyl)-N3-(4-methyl-2-(thiophen-2-yl)phenyl) pyrazine-2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6067N2-(4-methyl-2-(thiophen-2-yl)phenyl)-N3-(p-tolyl) pyrazine-2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6068N2-(4-fluorophenyl)-N3-(4-methyl-2-(5-methylthiophen-2-yl)phenyl)pyrazine-2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6069N2-(4-methyl-2-(5-methylthiophen-2-yl)phenyl)-N3-(p- tolyl)pyrazine-2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6070N2-(4-fluorophenyl)-N3-(4-methyl-2-(thiophen-3-yl) phenyl)pyrazine-2,3- dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6071N2-(4-methyl-2-(thiophen-3-yl)phenyl)-N3-(p-tolyl) pyrazine-2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6072N2-(4-fluorophenyl)-N3-(2-(thiophen-3-yl)benzyl)pyrazine- 2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6073N2-(2-(thiophen-3-yl)benzyl)-N3-(p-tolyl)pyrazine-2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6074N2-(4-fluorophenyl)-N3-(4-(thiophen-3-yl)benzyl)pyrazine-2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6075N2-(4-(thiophen-3-yl)benzyl)-N3-(p-tolyl)pyrazine-2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6076N2-(4-fluorophenyl)-N3-(2-(3-methyl-1H-pyrazol-5-yl) phenyl)pyrazine-2,3-dicarboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6077N2-(2-(3-methyl-1H-pyrazol-5-yl)phenyl)-N3-(p-tolyl) pyrazine-2,3-di-carboxamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6078N1-(4-fluorophenyl)-N2-(4-methyl-2-(3-methyl-1H-pyrazol-5-yl)phenyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6079N1-(4-fluorophenyl)-N2-(4-methyl-2-(thiophen-2-yl) phenyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6080N1-(4-methyl-2-(3-methyl-1H-pyrazol-5-yl)phenyl)-N2-(p- tolyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6081N1-(4-methyl-2-(thiophen-2-yl)phenyl)-N2-(p-tolyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6082N1-(4-methyl-2-(5-methylthiophen-2-yl)phenyl)-N2-(p- tolyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6083N1-(4-fluorophenyl)-N2-(4-methyl-2-(5-methylthiophen-2- yl)phenyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6084N1-(4-methyl-2-(thiophen-3-yl)phenyl)-N2-(p-tolyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6085N1-(4-fluorophenyl)-N2-(4-methyl-2-(thiophen-3-yl) phenyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6086N1-(4-fluorophenyl)-N2-(2-(thiophen-3-yl)benzyl) phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6087N1-(2-(thiophen-3-yl)benzyl)-N2-(p-tolyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6088N1-(4-fluorophenyl)-N2-(4-(thiophen-3-yl)benzyl) phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6089N1-(4-(thiophen-3-yl)benzyl)-N2-(p-tolyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6090N1-(4-fluorophenyl)-N2-(2-(3-methyl-1H-pyrazol-5-yl) phenyl)phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6091N1-(2-(3-methyl-1H-pyrazol-5-yl)phenyl)-N2-(p-tolyl) phthalamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_60922-(4-fluorobenzamido)-N-(4-methyl-2-(thiophen-3-yl) phenyl)benzamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_60932-(4-fluorobenzamido)-N-(4-methyl-2-(5-methylthiophen- 2-yl)phenyl)benzamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_60942-(4-fluorobenzamido)-N-(4-methyl-2-(pyridin-4-yl)phenyl) benzamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_60952-(4-fluorobenzamido)-N-(4-methyl-2-(pyridin-3-yl)phenyl) benzamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_6128Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Dengue virus
New Guinea C
Pathway
NA
Decrease (50 %)
Approved
29890736
DrugRepV_6129IFN-alpha
Antiviral
Hepatitis C virus | Leukemia | Melanoma
Dengue virus
New Guinea C
Pathway
NA
Decrease (50 %)
Investigational
29890736
DrugRepV_6346AM404
NA
Pain and Fever
Dengue virus
New Guinea C (NGC)
Pathway
NA
Decrease (50 %)
Phase IV
26856827
DrugRepV_6347Paracetamol
Nervous System
Fever | Minor aches | Pains
Dengue virus
New Guinea C (NGC)
Pathway
NA
Decrease (100 %)
Approved
26856827
DrugRepV_6348Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Dengue virus
New Guinea C (NGC)
Pathway
NA
Decrease (50 %)
Approved
26856827
DrugRepV_6426Cdt yellow
NA
NA
Dengue virus
NGC
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_6427Cdt white
NA
NA
Dengue virus
NGC
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_6428Crotoxin
NA
NA
Dengue virus
NGC
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_6429Crotapotin
NA
NA
Dengue virus
NGC
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_6430Crotamin
NA
NA
Dengue virus
NGC
Pathway
NA
Decrease (11 %)
NA
21723310
DrugRepV_6431Convulxin
NA
NA
Dengue virus
NGC
Pathway
NA
Decrease (5 %)
NA
21723310
DrugRepV_6432PLA2-IC
NA
NA
Dengue virus
NGC
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_6433PLA2-IC
NA
NA
Dengue virus
NGC
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_6480Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Dengue virus
NA
Pathway
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_6958Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
Approved
15200845
DrugRepV_6959Lamivudine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome | Hepatitis B virus
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
Approved
15200845
DrugRepV_6960Zidovudine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome/AIDS
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
Approved
15200845
DrugRepV_6961Saquinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
Approved, Investigational
15200845
DrugRepV_6962Nelfinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
NA
Pathway
NA
Decrease (95 %)
Approved
15200845
DrugRepV_6963Indinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
Approved
15200845
DrugRepV_6964(1S,2R,3S)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]uracil
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6965(1S,2R,3S)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]thymine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6966(1S,2R,3S)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]-5-fluorouracil
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6967(1S,2R,3S)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]cytosine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6968(1S,2R,3S)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]-5-fluorocytosine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6969L-Neplanocin A
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6970(1S,2R,3S)-9-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl] hypoxanthine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6971(1S,2R,3S)-9-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]guanine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6972Cyclopentenyl nucleosides
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6973(1R,2S,3R)-9-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl] hypoxanthine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6974(1R,2S,3R)-9-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]guanine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6975(1S,2R,3S)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]uracil
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6976(1R,2S,3R)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]thymine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6977(1R,2S,3R)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]-5-fluorouracil
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6978(1R,2S,3R)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]cytosine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_6979(1R,2S,3R)-1-[2,3-Dihydroxy-4-hydroxymethyl-4-cyclopenten-1-yl]-5-fluorocytosine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
11689085
DrugRepV_7173N2-(4-fluorophenyl)-N3-(4-methyl-2-(thiophen-2-yl)phenyl) pyrazine-2,3-dicarboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7174N2-(4-fluorophenyl)-N3-(4-methyl-2-(thiophen-3-yl) phenyl)pyrazine-2,3- dicarboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7175N2-(4-methyl-2-(thiophen-3-yl)phenyl)-N3-(p-tolyl) pyrazine-2,3-dicarboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7176N2-(4-fluorophenyl)-N3-(2-(thiophen-3-yl)benzyl)pyrazine- 2,3-dicarboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7177N2-(2-(thiophen-3-yl)benzyl)-N3-(p-tolyl)pyrazine-2,3-dicarboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7178N2-(4-fluorophenyl)-N3-(4-(thiophen-3-yl)benzyl)pyrazine-2,3-dicarboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7179N2-(4-(thiophen-3-yl)benzyl)-N3-(p-tolyl)pyrazine-2,3-dicarboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7180N2-(4-fluorophenyl)-N3-(2-(3-methyl-1H-pyrazol-5-yl) phenyl)pyrazine-2,3-dicarboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7181N2-(2-(3-methyl-1H-pyrazol-5-yl)phenyl)-N3-(p-tolyl) pyrazine-2,3-di-carboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7182N1-(4-fluorophenyl)-N2-(4-methyl-2-(3-methyl-1H-pyrazol-5-yl)phenyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7183N1-(4-fluorophenyl)-N2-(4-methyl-2-(thiophen-2-yl) phenyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7184N1-(4-methyl-2-(3-methyl-1H-pyrazol-5-yl)phenyl)-N2-(p- tolyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7185N1-(4-methyl-2-(thiophen-2-yl)phenyl)-N2-(p-tolyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7186N1-(4-methyl-2-(5-methylthiophen-2-yl)phenyl)-N2-(p- tolyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7187N1-(4-fluorophenyl)-N2-(4-methyl-2-(5-methylthiophen-2- yl)phenyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7188N1-(4-methyl-2-(thiophen-3-yl)phenyl)-N2-(p-tolyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7189N1-(4-fluorophenyl)-N2-(4-methyl-2-(thiophen-3-yl) phenyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7190N1-(4-fluorophenyl)-N2-(2-(thiophen-3-yl)benzyl) phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7191N1-(2-(thiophen-3-yl)benzyl)-N2-(p-tolyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7192N1-(4-fluorophenyl)-N2-(4-(thiophen-3-yl)benzyl) phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7193N1-(4-(thiophen-3-yl)benzyl)-N2-(p-tolyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7194N1-(4-fluorophenyl)-N2-(2-(3-methyl-1H-pyrazol-5-yl) phenyl)phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7195N1-(2-(3-methyl-1H-pyrazol-5-yl)phenyl)-N2-(p-tolyl) phthalamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_71962-(4-fluorobenzamido)-N-(4-methyl-2-(thiophen-3-yl) phenyl)benzamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_71972-(4-fluorobenzamido)-N-(4-methyl-2-(5-methylthiophen- 2-yl)phenyl)benzamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_71982-(4-fluorobenzamido)-N-(4-methyl-2-(pyridin-4-yl)phenyl) benzamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_71992-(4-fluorobenzamido)-N-(4-methyl-2-(pyridin-3-yl)phenyl) benzamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
27240271
DrugRepV_7243BCX4430
NA
Ebola virus
Yellow fever virus
17D
Pathway
NA
Decrease (50 %)
Investigational
27095300
DrugRepV_72441-[4,5-dihydroxy-3-(hydroxymethyl)cyclopent-2-en-1-yl]-1H-1,2,4-triazole-3-carboxamide
NA
NA
West Nile virus
NA
Pathway
NA
Decrease (50 %)
NA
16451078
DrugRepV_72451-[4,5-dihydroxy-3-(hydroxymethyl)cyclopent-2-en-1-yl]-1H-1,2,4-triazole-3-carboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
16451078
DrugRepV_72461-[4,5-dihydroxy-3-(hydroxymethyl)cyclopent-2-en-1-yl]-1H-imidazole-4-carboxamide
NA
NA
West Nile virus
NA
Pathway
NA
Decrease (50 %)
NA
16451078
DrugRepV_72471-[4,5-dihydroxy-3-(hydroxymethyl)cyclopent-2-en-1-yl]-1H-imidazole-4-carboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
16451078
DrugRepV_72481-[4,5-dihydroxy-3-(hydroxymethyl)cyclopent-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
NA
NA
West Nile virus
NA
Pathway
NA
Decrease (50 %)
NA
16451078
DrugRepV_72491-[4,5-dihydroxy-3-(hydroxymethyl)cyclopent-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
NA
NA
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
NA
16451078
DrugRepV_7267Cdt yellow
NA
NA
Yellow fever virus
17D
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_7268Cdt white
NA
NA
Yellow fever virus
17D
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_7269Crotoxin
NA
NA
Yellow fever virus
17D
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_7270Crotapotin
NA
NA
Yellow fever virus
17D
Pathway
NA
Decrease (43 %)
NA
21723310
DrugRepV_7271Crotamin
NA
NA
Yellow fever virus
17D
Pathway
NA
Decrease (20 %)
NA
21723310
DrugRepV_7272Convulxin
NA
NA
Yellow fever virus
17D
Pathway
NA
Decrease (22 %)
NA
21723310
DrugRepV_7273PLA2-IC
NA
NA
Yellow fever virus
17D
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_7274PLA2-IC
NA
NA
Yellow fever virus
17D
Pathway
NA
Decrease (50 %)
NA
21723310
DrugRepV_7514Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Polio virus
NA
Pathway
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_7515Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
West Nile virus
NA
Pathway
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_7516Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Yellow fever virus
NA
Pathway
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_7520beta-D-cyclopentenyl cytosine
NA
NA
Vaccinia virus
Copenhagen
Pathway
NA
Decrease (50 %)
NA
14604375
DrugRepV_7521beta-D-cyclopentenyl-5-iodocytidine
NA
NA
Vaccinia virus
Copenhagen
Pathway
NA
Decrease (50 %)
NA
14604375
DrugRepV_7522beta-D-Cyclopentenyl-5-chlorocytidine
NA
NA
Vaccinia virus
Copenhagen
Pathway
NA
Decrease (50 %)
NA
14604375
DrugRepV_7523beta-D-cyclopentenyl-5-bromocytidine
NA
NA
Vaccinia virus
Copenhagen
Pathway
NA
Decrease (50 %)
NA
14604375
DrugRepV_7524Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Vaccinia virus
NA
Pathway
NA
Decrease (50 %)
Investigational
31307979
DrugRepV_7663Hydroxychloroquine
Antiparasitic products, Insectisides and Repellents
Malaria
SARS Coronavirus-2
NA
NA
Decrease (50 %)
Approved
32344449
DrugRepV_7678Amiodarone
Cardiovascular agents
Anginal and Arrhythmia
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Approved, Investigational
32577649
DrugRepV_7679Bosutinib
Antineoplastic and Immunomodulating Agents
Cancer
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Approved
32577649
DrugRepV_7680Clofazamine
Antiinfectives For Systemic Use
Lepromatous leprosy
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Approved
32577649
DrugRepV_7681Domperidone
Alimentary Tract and Metabolism
Dyspepsia, heartburn, epigastric pain
SARS Coronavirus-2
NA
NA
Decrease (50 %)
Approved
32577649
DrugRepV_7682Entecavir
Antiinfectives For Systemic Use
Hepatitis B virus
SARS Coronavirus-2
NA
NA
Decrease (50 %)
Approved
32577649
DrugRepV_7683Fedratinib
Antineoplastic And Immunomodulating Agents
Myelofibrosis
SARS Coronavirus-2
NA
NA
Decrease (50 %)
Approved, Investigational
32577649
DrugRepV_7684Gilteritinib
Antineoplastic And Immunomodulating Agents
Acute myeloid leukemia
SARS Coronavirus-2
NA
NA
Decrease (50 %)
Approved, Investigational
32577649
DrugRepV_7685Ipratropium bromide
Respiratory System
Asthma | Chronic bronchitis | Emphysema
SARS Coronavirus-2
NA
NA
Decrease (50 %)
Approved, Experimental
32577649
DrugRepV_7686Lomitapide
Cardiovascular system
Hypercholesterolemia
SARS Coronavirus-2
NA
NA
Decrease (50 %)
Approved, Investigational
32577649
DrugRepV_7687Metoclopramide
Alimentary Tract and Metabolism
Diabetic gastroparesis
SARS Coronavirus-2
NA
NA
Decrease (50 %)
Approved, Investigational
32577649
DrugRepV_7688Niclosamide
Antiparasitic products, Insectisides and Repellents
Tapeworm and intestinal fluke infections | Helminthiasis
SARS Coronavirus-2
NA
NA
Decrease (50 %)
Approved
32577649
DrugRepV_7689Remdesivir
Antiviral
Hepatitis C | Ebola
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Experimental
32577649
DrugRepV_7690S1RA
NA
NA
SARS Coronavirus-2
NA
NA
Decrease (50 %)
NA
32577649
DrugRepV_7691Thioguanine
Antineoplastic and Immunomodulating Agents
Acute leukemia
SARS Coronavirus-2
NA
NA
Decrease (50 %)
Approved
32577649
DrugRepV_7692Verapamil
Cardiovascular agents
Hypertension (high blood pressure) | Angina (chest pain) | Arrhythmia (heart rhythm disorders).
SARS Coronavirus-2
NA
NA
Decrease (50 %)
Approved
32577649
DrugRepV_7693Z-FA-FMK
NA
NA
SARS Coronavirus-2
NA
NA
Decrease (50 %)
NA
32577649
DrugRepV_7694Lactoferrin
NA
NA
SARS Coronavirus-2
NA
NA
Decrease (50 %)
NA
32577649
DrugRepV_7695Nafamostat
NA
Blood vessel coagulation | Hemorrhagic lesions
SARS Coronavirus-2
NA
NA
Decrease (50 %)
Investigational
32532094
DrugRepV_7696Immunoglobulin F(ab’)2
NA
NA
SARS Coronavirus-2
NA
NA
Decrease (50 %)
NA
32659292
DrugRepV_7697Unfractionated Heparin
NA
Prophylaxis and Venous thrombosis
SARS Coronavirus-2
NA
NA
Decrease (50 %)
Approved, Investigational
32577638
DrugRepV_7698UFH-de6S
NA
NA
SARS Coronavirus-2
NA
NA
Decrease (50 %)
NA
32577638
DrugRepV_7699Enoxaparin
Blood And Blood Forming Organs
Deep vein thrombosis
SARS Coronavirus-2
NA
NA
Decrease (50 %)
Approved
32577638
DrugRepV_7700Enoxaparin-de6S
NA
NA
SARS Coronavirus-2
NA
NA
Decrease (50 %)
NA
32577638
DrugRepV_7771Remdesivir
Antiviral
Hepatitis C | Ebola
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Experimental
32687696
DrugRepV_7772Favipiravir
Antiviral
Influenza virus
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Investigational
32687696
DrugRepV_7773Galidesivir
NA
Ebolavirus
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Investigational
32687696
DrugRepV_7774Ritonavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Approved, Investigational
32687696
DrugRepV_7775Camostat mesylate
NA
Pancreatitis
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Experimental
32687696
DrugRepV_7776Nafamostat Mesylate
NA
Blood vessel coagulation | Hemorrhagic lesions
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Investigational
32687696
DrugRepV_7777Imatinib
Antineoplastic and Immunomodulating Agents
Leukemia | Myelodysplastic/myeloproliferative disease | Gastrointestinal stromal tumors
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Approved
32687696
DrugRepV_7778Apilimod
NA
Crohn's disease | Psoriasis | Psoriatic disorders
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Investigational
32687696
DrugRepV_7779Niclosamide
Antiparasitic products, Insectisides and Repellents
Tapeworm and intestinal fluke infections | Helminthiasis
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Approved
32687696
DrugRepV_7780Chloroquine
Antiparasitic products, Insectisides and Repellents
Malaria
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Approved
32687696
DrugRepV_7781Hydroxychloroquine
Antiparasitic products, Insectisides and Repellents
Malaria
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Approved
32687696
DrugRepV_7792Dehydroabieta-7-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_7793Cryptojaponol
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_77948beta-hydroxyabieta-9(11),13- dien-12-one
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_77957beta-hydroxydeoxycryptojaponol
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_77966,7-dehydroroyleanone
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_77973beta,12-diacetoxyabieta-6,8,11,13- tetraene
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_7798Pinusolidic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_7799Forskolin
NA
Smooth muscle relaxant
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Experimental, Investigational
17663539
DrugRepV_7800Cedrane-3beta,12-diol
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_7801alpha-cadinol
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_7802Betulinic acid
NA
Dysplastic Nevus Syndrome
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Investigational
17663539
DrugRepV_7803Betulonic acid
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_7804Hinokinin
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_7805Savinin
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_7806Honokiol
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_7807Magnolol
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17663539
DrugRepV_7808Curcumin
NA
Depressive disorder
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Approved
17663539
DrugRepV_7809Niclosamide
Antiparasitic products, Insectisides and Repellents
Tapeworm and intestinal fluke infections | Helminthiasis
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Approved
17663539
DrugRepV_7810Valinomycin
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Experimental
17663539
DrugRepV_78142-(5-bromopyridin-3-yl)-1-[5-(4-chlorophenyl)furan-2-yl]-2-fluoroethanone
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
18295820
DrugRepV_7816ML300
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_78172-(benzotriazol-1-yl)-N-(4-phenylphenyl)-N-(thiophen-3-ylmethyl)acetamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_7826N-[4-[[2-(benzotriazol-1-yl)acetyl]-(thiophen-3-ylmethyl)amino]phenyl]propanamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_7827N-[4-[[2-(benzotriazol-1-yl)acetyl]-(thiophen-3-ylmethyl)amino]phenyl]-2-methylpropanamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_7828N-{4-[(1H-Benzotriazol-1-ylacetyl)(3-thienylmethyl)amino]phenyl}-2,2-dimethylpropanamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_7829N-[4-[[2-(benzotriazol-1-yl)acetyl]-(thiophen-3-ylmethyl)amino]phenyl]-3-methoxypropanamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_7830N-[4-[[2-(benzotriazol-1-yl)acetyl]-(thiophen-3-ylmethyl)amino]phenyl]cyclobutanecarboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_7831N-[4-[[2-(benzotriazol-1-yl)acetyl]-(thiophen-3-ylmethyl)amino]phenyl]cyclohexanecarboxamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_7832N-[4-[[2-(benzotriazol-1-yl)acetyl]-(thiophen-3-ylmethyl)amino]phenyl]benzamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_78332-methylpropyl N-[4-[[2-(benzotriazol-1-yl)acetyl]-(thiophen-3-ylmethyl)amino]phenyl]carbamate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_78342-(benzotriazol-1-yl)-N-[4-(methylamino)phenyl]-N-(thiophen-3-ylmethyl)acetamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_78352-(benzotriazol-1-yl)-N-[4-(benzylamino)phenyl]-N-(thiophen-3-ylmethyl)acetamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_78362-(benzotriazol-1-yl)-N-(4-pyridin-3-ylphenyl)-N-(thiophen-3-ylmethyl)acetamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_78372-(benzotriazol-1-yl)-N-[4-(2-methoxypyridin-3-yl)phenyl]-N-(thiophen-3-ylmethyl)acetamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_78382-(benzotriazol-1-yl)-N-(4-pyridin-4-ylphenyl)-N-(thiophen-3-ylmethyl)acetamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_78392-(benzotriazol-1-yl)-N-[4-(2-methoxypyrimidin-5-yl)phenyl]-N-(thiophen-3-ylmethyl)acetamide
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
24080461
DrugRepV_78825-chloropyridin-3-yl 5-(4-chlorophenyl)oxolane-2-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_78835-chloropyridin-3-yl 5-(4-nitrophenyl)oxolane-2-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_78845-chloropyridin-3-yl 5-(4-chloro-2-nitrophenyl)oxolane-2-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_78855-chloropyridin-3-yl 5-(2-nitrophenyl)oxolane-2-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_78865-chloropyridin-3-yl 5-(3-nitrophenyl)oxolane-2-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_7887(5-chloropyridin-3-yl) pyridine-4-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_7888(5-chloropyridin-3-yl) pyridine-3-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_7889(5-chloropyridin-3-yl) 4-chlorobenzoate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_7890(5-chloropyridin-3-yl) 2-nitrobenzoate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_7891(5-chloropyridin-3-yl) 3-nitrobenzoate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_78925-Chloro-3-pyridinyl 1-naphthoate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_7893(5-chloropyridin-3-yl) 2-oxochromene-3-carboxylate
NA
NA
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
NA
17931870
DrugRepV_7897Ouabain
Cardiovascular agents
Atrial fibrillation and flutter | Heart failure
Japanese encephalitis virus
NA
Pathway
NA
Decrease (50 %)
Approved
31871089
DrugRepV_7898Digoxin
Cardiovascular agents
Arrhythmia
Japanese encephalitis virus
NA
Pathway
NA
Decrease (50 %)
Approved
31871089
DrugRepV_7899Lycorine
NA
NA
Japanese encephalitis virus
NA
Pathway
NA
Decrease (50 %)
NA
31871089
DrugRepV_7900Cephalotaxlen
NA
NA
Japanese encephalitis virus
NA
Pathway
NA
Decrease (50 %)
NA
31871089
DrugRepV_7901Schisandrin B
NA
NA
Japanese encephalitis virus
NA
Pathway
NA
Decrease (50 %)
NA
31871089
DrugRepV_7902Procyanidin
NA
NA
Japanese encephalitis virus
NA
Pathway
NA
Decrease (50 %)
NA
31871089
DrugRepV_7903Emodin
NA
Polycystic Kidney
Japanese encephalitis virus
NA
Pathway
NA
Decrease (50 %)
Investigational
31871089
DrugRepV_7904Schisandrin B
NA
NA
Japanese encephalitis virus
NA
Pathway
NA
Decrease (50 %)
NA
31871089
DrugRepV_7942DHBNH
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79433-[(E)-{[(3,4-dihydroxyphenyl)formamido]imino}methyl]-[1,1'-biphenyl]-4-carboxylic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7944(3E)-3-{2-[4-(3,4-dihydroxyphenyl)-1,3-thiazol-2-yl]hydrazin-1-ylidene}-2,3-dihydro-1H-indol-2-one
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79454-[2-[(2-hydroxy-1H-indol-3-yl)diazenyl]-1,3-thiazol-4-yl]benzonitrile
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7946NSC727447
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7947NSC732665
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79482-(3,4-Dihydroxyphenyl)-1,5,6,7,8,9-hexahydro-4H-cyclohepta[4,5]thieno[2,3-d]pyrimidin-4-one
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79492-(3,4-dihydroxybenzamido)-N-(pyridin-2-yl)-4H,5H,6H,7H,8H-cyclohepta[b]thiophene-3-carboxamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79505-(3,4-dihydroxyphenyl)-4-oxa-8-thia-6-azatricyclo[7.4.0.0²,?]trideca-1(9),2(7),5,10,12-pentaen-3-one
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7951(E)-3-(3,4-dihydroxyphenyl)-N-[(Z)-octadec-9-enyl]prop-2-enamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79524-Butoxy-N-(5-methyl-7-phenyl-4,7-dihydro[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79534-Butyl-N-(5-methyl-7-phenyl-4,7-dihydro[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79544-butyl-N-{5-methyl-7-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79552-fluoro-N-{5-methyl-7-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7956N-{5-methyl-7-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-4-nitrobenzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79574-amino-N-{5-methyl-7-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79583,4-dimethoxy-N-{5-methyl-7-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79593,4-dihydroxy-N-{5-methyl-7-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79602-fluoro-N-{7-methyl-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7961N-{7-methyl-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-4-nitrobenzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79624-amino-N-{7-methyl-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79633,4-dimethoxy-N-{7-methyl-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79643,4-dihydroxy-N-{7-methyl-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79654-butyl-N-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7966N-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-2-fluorobenzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7967N-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-4-nitrobenzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79684-amino-N-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7969N-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-3,4-dimethoxybenzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7970N-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-3,4-dihydroxybenzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7971N-{5,7-diphenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-3,4-dihydroxybenzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7972N-[7-(3,4-dihydroxyphenyl)-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7973N-benzoyl-N-[7-(3,4-dimethoxyphenyl)-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]benzamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7974N-(3,4-dihydroxyphenyl)-5-methyl-7-phenyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_7975N-(3,4-dihydroxyphenyl)-7-methyl-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
32151066
DrugRepV_79882-(6-{[1-carboxy-2-(2-phenyl-1H-indol-3-yl)ethyl]carbamoyl}-4-(2-{[1-carboxy-2-(2-phenyl-1H-indol-3-yl)ethyl]carbamoyl}ethyl)-4-nitrohexanamido)-3-(2-phenyl-1H-indol-3-yl)propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79892-[6-({1-carboxy-2-[2-(2-fluorophenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(2-fluorophenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]-3-[2-(2-fluorophenyl)-1H-indol-3-yl]propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79902-[6-({1-carboxy-2-[2-(4-nitrophenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(4-nitrophenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]-3-[2-(4-nitrophenyl)-1H-indol-3-yl]propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79913-[2-(4-bromophenyl)-1H-indol-3-yl]-2-[6-({2-[2-(4-bromophenyl)-1H-indol-3-yl]-1-carboxyethyl}carbamoyl)-4-[2-({2-[2-(4-bromophenyl)-1H-indol-3-yl]-1-carboxyethyl}carbamoyl)ethyl]-4-nitrohexanamido]propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79922-{6-[(1-carboxy-2-{2-[4-(trifluoromethyl)phenyl]-1H-indol-3-yl}ethyl)carbamoyl]-4-{2-[(1-carboxy-2-{2-[4-(trifluoromethyl)phenyl]-1H-indol-3-yl}ethyl)carbamoyl]ethyl}-4-nitrohexanamido}-3-{2-[4-(trifluoromethyl)phenyl]-1H-indol-3-yl}propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79932-[6-({1-carboxy-2-[2-(4-methoxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(4-methoxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]-3-[2-(4-methoxyphenyl)-1H-indol-3-yl]propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79943-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79954-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79965-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzene-1,3-dicarboxylic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79973-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79984-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_79995-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzene-1
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80003-(1-benzyl-1H-indol-3-yl)-2-(6-{[2-(1-benzyl-1H-indol-3-yl)-1-carboxyethyl]carbamoyl}-4-(2-{[2-(1-benzyl-1H-indol-3-yl)-1-carboxyethyl]carbamoyl}ethyl)-4-nitrohexanamido)propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80012-{6-[(1-carboxy-2-{1-[(4-fluorophenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]-4-{2-[(1-carboxy-2-{1-[(4-fluorophenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]ethyl}-4-nitrohexanamido}-3-{1-[(4-fluorophenyl)methyl]-1H-indol-3-yl}propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80024-{[3-(2-carboxy-2-{6-[(1-carboxy-2-{1-[(4-carboxyphenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]-4-{2-[(1-carboxy-2-{1-[(4-carboxyphenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]ethyl}-4-nitrohexanamido}ethyl)-1H-indol-1-yl]methyl}benzoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80034-[(3-{2-carboxy-2-[3-(3-{2-[(1-carboxy-2-{1-[(4-carboxyphenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]ethoxy}-2,2-bis({2-[(1-carboxy-2-{1-[(4-carboxyphenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]ethoxy}methyl)propoxy)propanamido]ethyl}-1H-indol-1-yl)me
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80042-(6-{[1-carboxy-2-(2-phenyl-1H-indol-3-yl)ethyl]carbamoyl}-4-(2-{[1-carboxy-2-(2-phenyl-1H-indol-3-yl)ethyl]carbamoyl}ethyl)-4-nitrohexanamido)-3-(2-phenyl-1H-indol-3-yl)propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80052-[6-({1-carboxy-2-[2-(2-fluorophenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(2-fluorophenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]-3-[2-(2-fluorophenyl)-1H-indol-3-yl]propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80062-[6-({1-carboxy-2-[2-(4-nitrophenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(4-nitrophenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]-3-[2-(4-nitrophenyl)-1H-indol-3-yl]propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80073-[2-(4-bromophenyl)-1H-indol-3-yl]-2-[6-({2-[2-(4-bromophenyl)-1H-indol-3-yl]-1-carboxyethyl}carbamoyl)-4-[2-({2-[2-(4-bromophenyl)-1H-indol-3-yl]-1-carboxyethyl}carbamoyl)ethyl]-4-nitrohexanamido]propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80082-{6-[(1-carboxy-2-{2-[4-(trifluoromethyl)phenyl]-1H-indol-3-yl}ethyl)carbamoyl]-4-{2-[(1-carboxy-2-{2-[4-(trifluoromethyl)phenyl]-1H-indol-3-yl}ethyl)carbamoyl]ethyl}-4-nitrohexanamido}-3-{2-[4-(trifluoromethyl)phenyl]-1H-indol-3-yl}propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80092-[6-({1-carboxy-2-[2-(4-methoxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(4-methoxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]-3-[2-(4-methoxyphenyl)-1H-indol-3-yl]propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80103-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80114-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80125-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzene-1,3-dicarboxylic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80133-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80144-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80155-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzene-1
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80163-(1-benzyl-1H-indol-3-yl)-2-(6-{[2-(1-benzyl-1H-indol-3-yl)-1-carboxyethyl]carbamoyl}-4-(2-{[2-(1-benzyl-1H-indol-3-yl)-1-carboxyethyl]carbamoyl}ethyl)-4-nitrohexanamido)propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80172-{6-[(1-carboxy-2-{1-[(4-fluorophenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]-4-{2-[(1-carboxy-2-{1-[(4-fluorophenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]ethyl}-4-nitrohexanamido}-3-{1-[(4-fluorophenyl)methyl]-1H-indol-3-yl}propanoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80184-{[3-(2-carboxy-2-{6-[(1-carboxy-2-{1-[(4-carboxyphenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]-4-{2-[(1-carboxy-2-{1-[(4-carboxyphenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]ethyl}-4-nitrohexanamido}ethyl)-1H-indol-1-yl]methyl}benzoic acid
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80194-[(3-{2-carboxy-2-[3-(3-{2-[(1-carboxy-2-{1-[(4-carboxyphenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]ethoxy}-2,2-bis({2-[(1-carboxy-2-{1-[(4-carboxyphenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]ethoxy}methyl)propoxy)propanamido]ethyl}-1H-indol-1-yl)me
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80202-(6-{[1-carboxy-2-(2-phenyl-1H-indol-3-yl)ethyl]carbamoyl}-4-(2-{[1-carboxy-2-(2-phenyl-1H-indol-3-yl)ethyl]carbamoyl}ethyl)-4-nitrohexanamido)-3-(2-phenyl-1H-indol-3-yl)propanoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80212-[6-({1-carboxy-2-[2-(2-fluorophenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(2-fluorophenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]-3-[2-(2-fluorophenyl)-1H-indol-3-yl]propanoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80222-[6-({1-carboxy-2-[2-(4-nitrophenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(4-nitrophenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]-3-[2-(4-nitrophenyl)-1H-indol-3-yl]propanoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80233-[2-(4-bromophenyl)-1H-indol-3-yl]-2-[6-({2-[2-(4-bromophenyl)-1H-indol-3-yl]-1-carboxyethyl}carbamoyl)-4-[2-({2-[2-(4-bromophenyl)-1H-indol-3-yl]-1-carboxyethyl}carbamoyl)ethyl]-4-nitrohexanamido]propanoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80242-{6-[(1-carboxy-2-{2-[4-(trifluoromethyl)phenyl]-1H-indol-3-yl}ethyl)carbamoyl]-4-{2-[(1-carboxy-2-{2-[4-(trifluoromethyl)phenyl]-1H-indol-3-yl}ethyl)carbamoyl]ethyl}-4-nitrohexanamido}-3-{2-[4-(trifluoromethyl)phenyl]-1H-indol-3-yl}propanoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80252-[6-({1-carboxy-2-[2-(4-methoxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(4-methoxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]-3-[2-(4-methoxyphenyl)-1H-indol-3-yl]propanoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80263-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80274-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80285-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzene-1,3-dicarboxylic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80293-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80304-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80315-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzene-1
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80324-[(3-{2-carboxy-2-[3-(3-{2-[(1-carboxy-2-{1-[(4-carboxyphenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]ethoxy}-2,2-bis({2-[(1-carboxy-2-{1-[(4-carboxyphenyl)methyl]-1H-indol-3-yl}ethyl)carbamoyl]ethoxy}methyl)propoxy)propanamido]ethyl}-1H-indol-1-yl)me
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80332-[6-({1-carboxy-2-[2-(4-nitrophenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(4-nitrophenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]-3-[2-(4-nitrophenyl)-1H-indol-3-yl]propanoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (90 %)
NA
31809045
DrugRepV_80343-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (90 %)
NA
31809045
DrugRepV_80355-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzene-1,3-dicarboxylic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (90 %)
NA
31809045
DrugRepV_80363-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (90 %)
NA
31809045
DrugRepV_80374-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(4-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (90 %)
NA
31809045
DrugRepV_80385-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzene-1
NA
NA
Enterovirus
BrCr
Pathway
NA
Decrease (90 %)
NA
31809045
DrugRepV_8039MADAL-385
NA
NA
Enterovirus
11316
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80405-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzene-1,3-dicarboxylic acid
NA
NA
Enterovirus
11316
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80413-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Enterovirus
11316
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80425-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzene-1
NA
NA
Enterovirus
11316
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_8043MADAL-385
NA
NA
Enterovirus
TW/70902/08
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80445-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzene-1,3-dicarboxylic acid
NA
NA
Enterovirus
TW/70902/08
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80453-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Enterovirus
TW/70902/08
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80465-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzene-1
NA
NA
Enterovirus
TW/70902/08
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_8047MADAL-385
NA
NA
Enterovirus
H08300 461; 812
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80485-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzene-1,3-dicarboxylic acid
NA
NA
Enterovirus
H08300 461; 812
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80493-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Enterovirus
H08300 461; 812
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80505-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzene-1
NA
NA
Enterovirus
H08300 461; 812
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_8051MADAL-385
NA
NA
Enterovirus
TW/1956/05
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80525-(3-{2-carboxy-2-[6-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)-4-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethyl]-4-nitrohexanamido]ethyl}-1H-indol-2-yl)benzene-1,3-dicarboxylic acid
NA
NA
Enterovirus
TW/1956/05
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80533-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3-carboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzoic acid
NA
NA
Enterovirus
TW/1956/05
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80545-{3-[2-carboxy-2-(3-{3-[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]-2,2-bis({[2-({1-carboxy-2-[2-(3,5-dicarboxyphenyl)-1H-indol-3-yl]ethyl}carbamoyl)ethoxy]methyl})propoxy}propanamido)ethyl]-1H-indol-2-yl}benzene-1
NA
NA
Enterovirus
TW/1956/05
Pathway
NA
Decrease (50 %)
NA
31809045
DrugRepV_80554-{[6-chloro-4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80564-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80574-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80584-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80594-{[6-chloro-4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80604-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80614-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80624-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80634-{[6-chloro-4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80644-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80654-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80664-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80674-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80684-{[4-({2-chloro-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-fluorophenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80694-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80704-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80714-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80724-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-dimethylphenyl}amino)-6-methoxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80734-{[4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)-6-methoxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80744-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-methoxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80754-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-hydroxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80764-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-nitroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80774-{[7-chloro-4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80784-{[7-chloro-4-({2-chloro-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-fluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80794-{[7-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80804-{[7-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80814-{[7-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80824-{[4-({2-amino-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-methylphenyl}amino)-7-chloroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80834-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-dimethylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80844-{[4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80854-{[4-({2-chloro-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-fluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80864-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80874-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80884-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
IIIB
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80894-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80904-{[4-({2-chloro-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-fluorophenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80914-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80924-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80934-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80944-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-dimethylphenyl}amino)-6-methoxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80954-{[4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)-6-methoxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80964-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-methoxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80974-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-hydroxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80984-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-nitroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_80994-{[7-chloro-4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81004-{[7-chloro-4-({2-chloro-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-fluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81014-{[7-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81024-{[7-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81034-{[7-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81044-{[4-({2-amino-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-methylphenyl}amino)-7-chloroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81054-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-dimethylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81064-{[4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81074-{[4-({2-chloro-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-fluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81084-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81094-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81104-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
E138K
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81114-{[6-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81124-{[4-({2-chloro-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-fluorophenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81134-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81144-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81154-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)-6-fluoroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81164-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-dimethylphenyl}amino)-6-methoxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81174-{[4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)-6-methoxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81184-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-methoxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81194-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-hydroxyquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81204-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)-6-nitroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81214-{[7-chloro-4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81224-{[7-chloro-4-({2-chloro-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-fluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81234-{[7-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81244-{[7-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81254-{[7-chloro-4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81264-{[4-({2-amino-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-methylphenyl}amino)-7-chloroquinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81274-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-dimethylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81284-{[4-({2,6-dichloro-4-[(1E)-2-cyanoeth-1-en-1-yl]phenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81294-{[4-({2-chloro-4-[(1E)-2-cyanoeth-1-en-1-yl]-6-fluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81304-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2,6-difluorophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81314-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-fluoro-6-methylphenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_81324-{[4-({4-[(1E)-2-cyanoeth-1-en-1-yl]-2-methyl-6-nitrophenyl}amino)quinazolin-2-yl]amino}benzonitrile
NA
NA
Human immunodeficiency virus
K103N
Pathway
NA
Decrease (50 %)
NA
31599568
DrugRepV_8133StemRegenin 1
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (68.1 %)
NA
32708182
DrugRepV_8134Niclosamide
Antiparasitic products, Insectisides and Repellents
Tapeworm and intestinal fluke infections | Helminthiasis
Vaccinia virus
NA
Pathway
NA
Decrease (43.7 %)
Approved
32708182
DrugRepV_8135ICG-001
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (80.9 %)
NA
32708182
DrugRepV_8136Nifuroxazide
Alimentary Tract And Metabolism
NA
Vaccinia virus
NA
Pathway
NA
Decrease (48.8 %)
Experimental
32708182
DrugRepV_8137NSC 319726
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (99.8 %)
NA
32708182
DrugRepV_8138Tenovin-1
Anticancer
Cancer
Vaccinia virus
NA
Pathway
NA
Decrease (32 %)
NA
32708182
DrugRepV_8139RITA
NA
Cancer
Vaccinia virus
NA
Pathway
NA
Decrease (50.2 %)
NA
32708182
DrugRepV_8140Ciclopirox ethanolamine
Dermatologicals
Fungal infections
Vaccinia virus
NA
Pathway
NA
Decrease (99.8 %)
Approved
32708182
DrugRepV_8141Econazole Nitrate
Dermatologicals
Fungal infections
Vaccinia virus
NA
Pathway
NA
Decrease (55.1 %)
Approved
32708182
DrugRepV_8142Miconazole Nitrate
Alimentary Tract And Metabolism; Dermatologicals; Genito Urinary System and Sex Hormones; Antiinfect
Fungal infections (Tinea pedis (athlete’s foot), tinea cruris, and tinea corporis caused by Trichophyton rubrum, Trichophyton mentagrophytes, and Epidermophyton floccosum, in the treatment of cutaneous candidiasis (moniliasis), and in the treatment o
Vaccinia virus
NA
Pathway
NA
Decrease (58.3 %)
Approved, Investigational, Vet approved
32708182
DrugRepV_8143Monensin sodium salt
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (96.7 %)
Experimental, Vet approved
32708182
DrugRepV_8144Idoxuridine
Antiinfectives For Systemic Use
Keratoconjunctivitis and Keratitis caused by herpes simplex virus
Vaccinia virus
NA
Pathway
NA
Decrease (85.8 %)
Approved, Investigational
32708182
DrugRepV_81453-Deazaneplanocin A
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (76.8 %)
NA
32708182
DrugRepV_8146Fludarabine
Antineoplastic and Immunomodulating Agents
Hematological malignancies
Vaccinia virus
NA
Pathway
NA
Decrease (99.1 %)
Approved
32708182
DrugRepV_8147Clofarabine
Antineoplastic and Immunomodulating Agents
Cancer
Vaccinia virus
NA
Pathway
NA
Decrease (99.8 %)
Approved
32708182
DrugRepV_8148Azaguanine-8
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (12.7 %)
Experimental
32708182
DrugRepV_8149Cytarabine
NA
Leukemia
Vaccinia virus
NA
Pathway
NA
Decrease (99.8 %)
Approved
32708182
DrugRepV_8150Gemcitabine
Antineoplastic and Immunomodulating Agents
Ovarian cancer | Non-small cell lung cance | Adenocarcinoma of the pancreas
Vaccinia virus
NA
Pathway
NA
Decrease (99.9 %)
Approved
32708182
DrugRepV_8151Cyclocytidine Hydrochloride
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (99.8 %)
NA
32708182
DrugRepV_8152Trifluridine
Sensory Organ
Primary keratoconjunctivitis and Herpes simplex keratitis
Vaccinia virus
NA
Pathway
NA
Decrease (99.9 %)
Approved
32708182
DrugRepV_8153Azacitidine
Antineoplastic and Immunomodulating Agents
French-American-British myelodysplastic syndrome
Vaccinia virus
NA
Pathway
NA
Decrease (99.9 %)
Approved
32708182
DrugRepV_8154Floxuridine
Anticancer
Gastrointestinal adenocarcinomas
Vaccinia virus
NA
Pathway
NA
Decrease (62.6 %)
Approved
32708182
DrugRepV_8155Abitrexate
Antineoplastic and Immunomodulating Agents
Gestational choriocarcinoma, chorioadenoma destruens, hydatidiform mole and acute lymphocytic leukemia
Vaccinia virus
NA
Pathway
NA
Decrease (62.2 %)
Approved
32708182
DrugRepV_8156Triapine
NA
Leukemia, Lung Cancer, Kidney Cancer, Prostate Cancer, and Pancreatic Cancer
Vaccinia virus
NA
Pathway
NA
Decrease (99.9 %)
Investigational
32708182
DrugRepV_8157Vidarabine
Antiinfectives For Systemic Use; Sensory Organ
Viral infections (Chickenpox, Herpes simplex, Zoster and varicella zoster)
Vaccinia virus
NA
Pathway
NA
Decrease (99.7 %)
Approved
32708182
DrugRepV_8158Apigenin
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (54.8 %)
Experimental
32708182
DrugRepV_8159Avasimibe
NA
Peripheral vascular disease
Vaccinia virus
NA
Pathway
NA
Decrease (50.9 %)
Investigational
32708182
DrugRepV_8160Cyclosporin A
NA
Bone marrow transplant rejection
Vaccinia virus
NA
Pathway
NA
Decrease (67.2 %)
Approved, Investigational, Vet approved
32708182
DrugRepV_8161ML130
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (35.9 %)
NA
32708182
DrugRepV_8162PAC-1
NA
Lymphoma, Melanoma, Solid Tumors, Breast Cancer, and Thoracic Cancers
Vaccinia virus
NA
Pathway
NA
Decrease (95.5 %)
Investigational
32708182
DrugRepV_8163ABT-263
NA
Solid Tumors, Non-Hodgkin's Lymphoma, EGFR Activating Mutation, Chronic Lymphoid Leukemia, and Hematological Malignancies
Vaccinia virus
NA
Pathway
NA
Decrease (33.1 %)
Investigational
32708182
DrugRepV_8164ABT-737
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (26.6 %)
NA
32708182
DrugRepV_8165PF-2545920
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (33.7 %)
NA
32708182
DrugRepV_8166Cladribine
Antineoplastic and Immunomodulating Agents
Lymphoproliferative diseases
Vaccinia virus
NA
Pathway
NA
Decrease (99.8 %)
Approved
32708182
DrugRepV_8167Adefovir dipivoxil
Antiinfectives For Systemic Use
Hepatitis B virus
Vaccinia virus
NA
Pathway
NA
Decrease (99.8 %)
Approved
32708182
DrugRepV_8168TPCA-1
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (78.5 %)
NA
32708182
DrugRepV_8169Mycophenolic Acid
Immunosuppressant
Organ rejection (immunosuppressants)
Vaccinia virus
NA
Pathway
NA
Decrease (96.7 %)
Approved, Investigational
32708182
DrugRepV_8170PTC-209
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (90.7 %)
NA
32708182
DrugRepV_8171Selisistat
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (30.5 %)
NA
32708182
DrugRepV_8172Salinomycin
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (92.5 %)
Vet approved
32708182
DrugRepV_8173Dapivirine
NA
Acquired immunodeficiency syndrome
Vaccinia virus
NA
Pathway
NA
Decrease (41.7 %)
Investigational
32708182
DrugRepV_8174CCG 50014
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (35.8 %)
NA
32708182
DrugRepV_8175Mocetinostat
NA
Lymphoma, Urothelial Carcinoma, Relapsed and Refractory, Myelodysplastic Syndrome, and Metastatic Leiomyosarcoma
Vaccinia virus
NA
Pathway
NA
Decrease (46.9 %)
Investigational
32708182
DrugRepV_8176Atorvastatin Calcium
Cardiovascular agents
Coronary heart disease
Vaccinia virus
NA
Pathway
NA
Decrease (25.4 %)
Approved
32708182
DrugRepV_8177UK 383367
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (17 %)
NA
32708182
DrugRepV_8178Lonafarnib
NA
Solid tumors, leukemia (unspecified), and lung cancer
Vaccinia virus
NA
Pathway
NA
Decrease (36.2 %)
Investigational
32708182
DrugRepV_8179BX-912
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (42.3 %)
NA
32708182
DrugRepV_8180URB597
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (21.7 %)
NA
32708182
DrugRepV_8181Anagrelide HCl
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (58.4 %)
NA
32708182
DrugRepV_8182Drospirenone
Genito Urinary System and Sex Hormones
Contraception
Vaccinia virus
NA
Pathway
NA
Decrease (57.4 %)
Approved
32708182
DrugRepV_8183Ethinyl estradiol
Antineoplastic and Immunomodulating Agents
Cancer
Vaccinia virus
NA
Pathway
NA
Decrease (53.3 %)
Approved
32708182
DrugRepV_8184Norethindrone
Gynaecological-agents
Secondary amenorrhea | Endometriosis | Abnormal uterine bleeding
Vaccinia virus
NA
Pathway
NA
Decrease (48.4 %)
Approved
32708182
DrugRepV_8185Ganetespib
NA
BREAST CANCER, Small Cell Lung Cancer, Acute Myeloid Leukaemia, and Myelodysplastic Syndrome
Vaccinia virus
NA
Pathway
NA
Decrease (99.7 %)
Investigational
32708182
DrugRepV_8186PF-04929113
NA
Cancer/tumors
Vaccinia virus
NA
Pathway
NA
Decrease (99.4 %)
Investigational
32708182
DrugRepV_8187NMS-E973
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (99.1 %)
NA
32708182
DrugRepV_8188XL888
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (99.6 %)
NA
32708182
DrugRepV_8189Tanespimycin
NA
Leukemia (myeloid) and solid tumors.
Vaccinia virus
NA
Pathway
NA
Decrease (99.4 %)
Investigational
32708182
DrugRepV_8190VER-49009
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (98.9 %)
NA
32708182
DrugRepV_8191SNX2112
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (99.4 %)
NA
32708182
DrugRepV_8192BIIB021
NA
Tumors and Lymphoma
Vaccinia virus
NA
Pathway
NA
Decrease (99.8 %)
Investigational
32708182
DrugRepV_8193AT13387
Antiinfectives For Systemic Use
Hepatitis C virus
Vaccinia virus
NA
Pathway
NA
Decrease (99.8 %)
Phase III
32708182
DrugRepV_8194NVP-BEP800
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (98.8 %)
NA
32708182
DrugRepV_8195AUY922
NA
Lymphoma, Breast Cancer, Metastatic Disease, Advanced Solid Tumors, and Hematologic Neoplasms
Vaccinia virus
NA
Pathway
NA
Decrease (99.8 %)
Investigational
32708182
DrugRepV_8196KW-2478
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (92.7 %)
NA
32708182
DrugRepV_8197Vincristine
Antineoplastic and Immunomodulating Agents
Cancer (Acute leukemia |Hodgkin's and non-Hodgkin's lymphoma |Neuroblastoma |Rhabdomyosarcoma |Ewing's sarcoma |Wilms' tumor | Multiple myeloma | Chronic leukemias | Thyroid cancer | Brain tumors)
Vaccinia virus
NA
Pathway
NA
Decrease (96.6 %)
Approved
32708182
DrugRepV_8198ABT-751
NA
Lung Cancer
Vaccinia virus
NA
Pathway
NA
Decrease (81.5 %)
Investigational
32708182
DrugRepV_8199Epothilone A
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (27.3 %)
NA
32708182
DrugRepV_8200Amygdalin
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (58.3 %)
NA
32708182
DrugRepV_8201Kaempferol
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (64.7 %)
NA
32708182
DrugRepV_8202ENMD-2076
NA
Breast cancer, leukemia (unspecified), lung cancer, and solid tumors
Vaccinia virus
NA
Pathway
NA
Decrease (72.3 %)
Investigational
32708182
DrugRepV_8203AMG-900
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (50.4 %)
NA
32708182
DrugRepV_8204MLN8054
NA
Colon Neoplasm, Breast Neoplasm, Bladder Neoplasm, Pancreatic Neoplasm, and Advanced Malignancies
Vaccinia virus
NA
Pathway
NA
Decrease (36.2 %)
Investigational
32708182
DrugRepV_8205Ibrutinib
NA
Mantle cell lymphoma
Vaccinia virus
NA
Pathway
NA
Decrease (74.9 %)
Approved
32708182
DrugRepV_8206CNX-774
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (70 %)
NA
32708182
DrugRepV_8207AR-A014418
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (47.9 %)
Experimental
32708182
DrugRepV_8208CGP 57380
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (58.1 %)
NA
32708182
DrugRepV_8209Genistein
Antihelmintic
Prostate cancer
Vaccinia virus
NA
Pathway
NA
Decrease (40.6 %)
Investigational
32708182
DrugRepV_8210HMN-214
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (58.9 %)
NA
32708182
DrugRepV_8211TG003
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (46.7 %)
NA
32708182
DrugRepV_8212Skepinone-L
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (47.1 %)
NA
32708182
DrugRepV_8213TAK-632
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (65.2 %)
NA
32708182
DrugRepV_8214YM201636
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (56.3 %)
NA
32708182
DrugRepV_8215MK-2461
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (57 %)
NA
32708182
DrugRepV_8216OSI-930
Anticancer
Solid tumors
Vaccinia virus
NA
Pathway
NA
Decrease (43.5 %)
Investigational
32708182
DrugRepV_8217SP600125
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (50.5 %)
NA
32708182
DrugRepV_8218SKI II
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (65.1 %)
NA
32708182
DrugRepV_8219PKI-402
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (44.9 %)
NA
32708182
DrugRepV_8220BEZ235
NA
Cancer, Solid Tumor, Renal Cancer, Breast Cancer, and Cowden Syndrome
Vaccinia virus
NA
Pathway
NA
Decrease (37.4 %)
Investigational
32708182
DrugRepV_8221WYE-125132
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (67.6 %)
NA
32708182
DrugRepV_8222OSI-027
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (68.3 %)
Investigational
32708182
DrugRepV_8223Torin 1
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (57.3 %)
NA
32708182
DrugRepV_8224Ku-0063794
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (55.3 %)
NA
32708182
DrugRepV_8225AZD2014
NA
Advanced Gastric Adenocarcinoma
Vaccinia virus
NA
Pathway
NA
Decrease (70.3 %)
Investigational
32708182
DrugRepV_8226Nocodazole
Anticancer
NA
Vaccinia virus
NA
Pathway
NA
Decrease (76.2 %)
Experimental
32708182
DrugRepV_8227Dasatinib
Antineoplastic and Immunomodulating Agents
Cancer
Vaccinia virus
NA
Pathway
NA
Decrease (74.2 %)
Approved
32708182
DrugRepV_8228KX2-391
NA
Colon cancer | Pancreatic cancer | Prostate cancer | Breast cancer
Vaccinia virus
NA
Pathway
NA
Decrease (65.1 %)
Investigational
32708182
DrugRepV_8229Bosutinib
Antineoplastic and Immunomodulating Agents
Chronic myelogenous leukemia (CML)
Vaccinia virus
NA
Pathway
NA
Decrease (81.8 %)
Approved
32708182
DrugRepV_8230PP1
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (35.8 %)
NA
32708182
DrugRepV_8231AZ 960
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (82.1 %)
NA
32708182
DrugRepV_8232LY2784544
NA
Myelofibrosis, Polycythemia Vera, Primary Myelofibrosis, Thrombocythemia, Essential, and Myeloproliferative Disorders
Vaccinia virus
NA
Pathway
NA
Decrease (65.7 %)
Investigational
32708182
DrugRepV_8233WHI-P154
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (66.3 %)
NA
32708182
DrugRepV_8234Cyt387
NA
Polycythemia Vera, Primary Myelofibrosis, Post-Polycythemia Vera, Essential Thrombocythemia, and Primary Myelofibrosis (PMF)
Vaccinia virus
NA
Pathway
NA
Decrease (45.2 %)
Investigational
32708182
DrugRepV_8235KPT-276
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (27.6 %)
NA
32708182
DrugRepV_8236KPT-185
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (26.2 %)
NA
32708182
DrugRepV_8237Phloretin
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (-27 %)
Experimental
32708182
DrugRepV_8238Ivacaftor
Respiratory System
Cystic fibrosis
Vaccinia virus
NA
Pathway
NA
Decrease (75.5 %)
Approved
32708182
DrugRepV_8239Tolbutamide
Alimentary Tract and Metabolism
Type 2 Diabetes Mellitus
Vaccinia virus
NA
Pathway
NA
Decrease (99.9 %)
Approved, Investigational
32708182
DrugRepV_8240Fexofenadine Hydrochloride
Respiratory System
Allergic rhinitis
Vaccinia virus
NA
Pathway
NA
Decrease (10.5 %)
Approved
32708182
DrugRepV_8241Bergapten
Dermatologicals
Severe Generalized Atopic Dermatitis
Vaccinia virus
NA
Pathway
NA
Decrease (7.6 %)
Investigational
32708182
DrugRepV_8242SC144
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (98.4 %)
NA
32708182
DrugRepV_8243Daidzein
NA
Dietary supplement
Vaccinia virus
NA
Pathway
NA
Decrease (32.2 %)
Experimental
32708182
DrugRepV_8244Delanzomib
NA
Solid Tumors, Multiple Myeloma, and Lymphoma, Non-Hodgkin.
Vaccinia virus
NA
Pathway
NA
Decrease (99.7 %)
Investigational
32708182
DrugRepV_8245MLN9708
NA
Multiple myeloma
Vaccinia virus
NA
Pathway
NA
Decrease (99.6 %)
Approved, Investigational
32708182
DrugRepV_8246Oprozomib
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (99.5 %)
Investigational
32708182
DrugRepV_8247MG-132
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (98.9 %)
NA
32708182
DrugRepV_8248MLN2238
NA
Multiple myeloma
Vaccinia virus
NA
Pathway
NA
Decrease (99.7 %)
Approved, Investigational
32708182
DrugRepV_8249ONX-0914
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (99.5 %)
NA
32708182
DrugRepV_8250Amonafide
NA
Breast cancer, ovarian cancer, and prostate cancer
Vaccinia virus
NA
Pathway
NA
Decrease (99.3 %)
Investigational
32708182
DrugRepV_8251Teniposide
Antineoplastic and Immunomodulating Agents
Acute lymphoblastic leukaemia
Vaccinia virus
NA
Pathway
NA
Decrease (97.9 %)
Approved
32708182
DrugRepV_8252Etoposide
Antineoplastic and Immunomodulating Agents
Cancer
Vaccinia virus
NA
Pathway
NA
Decrease (60.1 %)
Approved
32708182
DrugRepV_8253Golvatinib
NA
Platinum-Resistant Squamous Cell Carcinoma of the Head and Neck
Vaccinia virus
NA
Pathway
NA
Decrease (79.8 %)
Investigational
32708182
DrugRepV_8254Sorafenib
Antineoplastic and Immunomodulating Agents
Hepatocellular carcinoma | Renal cell carcinoma
Vaccinia virus
NA
Pathway
NA
Decrease (72.6 %)
Approved, Investigational
32708182
DrugRepV_8255AG 1296
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (53.2 %)
NA
32708182
DrugRepV_8256NVP-TAE226
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (91.5 %)
NA
32708182
DrugRepV_8257Cabozantinib malate
NA
Metastatic medullary thyroid cancer
Vaccinia virus
NA
Pathway
NA
Decrease (79.3 %)
NA
32708182
DrugRepV_8258XL-184
NA
Thyroid cancer
Vaccinia virus
NA
Pathway
NA
Decrease (64.2 %)
Approved, Investigational
32708182
DrugRepV_8259Linifanib
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (60.5 %)
NA
32708182
DrugRepV_8260TKI-258
NA
Multiple myeloma and solid tumors
Vaccinia virus
NA
Pathway
NA
Decrease (67.6 %)
Investigational
32708182
DrugRepV_8261AZD4547
NA
Cancer
Vaccinia virus
NA
Pathway
NA
Decrease (81.5 %)
Investigational
32708182
DrugRepV_8262AG-1024
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (71.8 %)
NA
32708182
DrugRepV_8263BMS-754807
NA
Solid Tumors
Vaccinia virus
NA
Pathway
NA
Decrease (61.8 %)
Investigational
32708182
DrugRepV_8264Afatinib
Antineoplastic And Immunomodulating Agents
Metastatic non-small cell lung cancer
Vaccinia virus
NA
Pathway
NA
Decrease (95.2 %)
Approved
32708182
DrugRepV_8265Butein
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (62.6 %)
NA
32708182
DrugRepV_8266CO-1686 (AVL-301)
NA
Nonsmall Cell Lung Cancer, Non-small Cell Lung Cancer, and Locally Advanced or Metastatic Non-small Cell Lung Cancer
Vaccinia virus
NA
Pathway
NA
Decrease (74.3 %)
NA
32708182
DrugRepV_8267PD168393
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (67.2 %)
Experimental
32708182
DrugRepV_8268PD153035 HCl
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (74.7 %)
NA
32708182
DrugRepV_8269Gefitinib
Antineoplastic and Immunomodulating Agents
Non-small cell lung cancer
Vaccinia virus
NA
Pathway
NA
Decrease (91.2 %)
Approved, Investigational
32708182
DrugRepV_8270Desmethyl Erlotinib
NA
Cancer
Vaccinia virus
NA
Pathway
NA
Decrease (75.5 %)
Approved, Investigational
32708182
DrugRepV_8271OSI-420
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (46.7 %)
NA
32708182
DrugRepV_8272Neratinib
Antineoplastic And Immunomodulating Agents
Breast cancer
Vaccinia virus
NA
Pathway
NA
Decrease (56.7 %)
Approved, Investigational
32708182
DrugRepV_8273Erlotinib Hydrochloride
Antineoplastic and Immunomodulating Agents
Cancer
Vaccinia virus
NA
Pathway
NA
Decrease (66.8 %)
Approved
32708182
DrugRepV_8274WZ8040
NA
NA
Vaccinia virus
NA
Pathway
NA
Decrease (96.4 %)
NA
32708182
DrugRepV_8279Bortezomib
Antineoplastic and Immunomodulating Agents
Multiple myeloma
Chikungunya virus
122508
NA
NA
Decrease (50 %)
Approved
32469886
DrugRepV_8280Bortezomib
Antineoplastic and Immunomodulating Agents
Multiple myeloma
Chikungunya virus
122508
NA
NA
Decrease (50 %)
Approved
32469886
DrugRepV_8281Bortezomib
Antineoplastic and Immunomodulating Agents
Multiple myeloma
Chikungunya virus
122508
NA
NA
Decrease (50 %)
Approved
32469886
DrugRepV_82821-(2-fluorophenyl)-3-(4-(4-isopentyl-1H-1,2,3-triazol-1-yl)phenyl)urea
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_82831-(3-fluorophenyl)-3-(4-(4-isopentyl-1H-1,2,3-triazol-1-yl)phenyl)urea
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_82841-(4-(4-(ethoxymethyl)-1H-1,2,3-triazol-1-yl)phenyl)-3-(3-fluorophenyl)urea
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_82851-(3-fluorophenyl)-3-(4-(4-(3-oxobutyl)-1H-1,2,3-triazol-1-yl)phenyl)urea
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_82861-(4-(4-butyl-1H-1,2,3-triazol-1-yl)phenyl)-3-(3-fluorophenyl)urea
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_8287N-(2-(3-(4-(4-butyl-1H-1,2,3-triazol-1-yl)phenyl)ureido)phenyl)methanesulfonamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_82881-(4-(4-isopentyl-1H-1,2,3-triazol-1-yl)phenyl)-3-o-tolylurea
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_82891-(4-(4-hexyl-1H-1,2,3-triazol-1-yl)phenyl)-3-(2-(trifluoromethyl)phenyl)urea)
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_82903-(4-(ethoxymethyl)-1H-1,2,3-triazol-1-yl)-N-(2-morpholinophenyl)benzenesulfonamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_8291ethyl 3-((3-(4-(ethoxymethyl)-1H-1,2,3-triazol-1-yl)phenyl)sulfonamido)benzoate
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_82923-((3-(4-(ethoxymethyl)-1H-1,2,3-triazol-1-yl)phenyl)sulfonamido)benzoic acid
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_82933-(4-butyl-1H-1,2,3-triazol-1-yl)-N-(2-(methylsulfonamido)phenyl)benzenesulfonamide
NA
NA
Dengue virus
NA
Pathway
NA
Decrease (50 %)
NA
32435411
DrugRepV_8294Tolcapone
Nervous System
Parkinson's Disease
Ebola virus
NA
NA
NA
Decrease (50 %)
Approved, Withdrawn
32425892
DrugRepV_8295Tolcapone
Nervous System
Parkinson's Disease
Ebola virus
NA
NA
NA
Decrease (50 %)
Approved, Withdrawn
32425892
DrugRepV_8296Tolcapone
Nervous System
Parkinson's Disease
Ebola virus
NA
NA
NA
Decrease (50 %)
Approved, Withdrawn
32425892
DrugRepV_8297Tolcapone
Nervous System
Parkinson's Disease
Ebola virus
NA
NA
NA
Decrease (50 %)
Approved, Withdrawn
32425892
DrugRepV_8298Gemcitabine
Antineoplastic and Immunomodulating Agents
Ovarian cancer | Non-small cell lung cance | Adenocarcinoma of the pancreas
Enterovirus
NA
Pathway
NA
Decrease (50 %)
Approved
32424333
DrugRepV_8316Gemcitabine
Antineoplastic and Immunomodulating Agents
Ovarian cancer | Non-small cell lung cance | Adenocarcinoma of the pancreas
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
Approved
31866007
DrugRepV_8317Roscovitine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31866007
DrugRepV_8318Quinacrine
NA
Malaria | Giardiasis | Cutaneous leishmaniasis | Management of malignant effusions
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
Investigational
31866007
DrugRepV_8319Kenpaullone
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31866007
DrugRepV_8320SB743921
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31866007
DrugRepV_83213-Deazauridine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31866007
DrugRepV_83222’-C-Methylcytidine
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
31866007
DrugRepV_8335Nafamostat
NA
Blood vessel coagulation | Hemorrhagic lesions
SARS Coronavirus-2
NA
NA
Decrease (50 %)
Investigational
32596694
DrugRepV_8336Camostat
Blood And Blood Forming Organs
Chronic pancreatitis
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Experimental
32596694
DrugRepV_8337Gabexate
NA
Cancer, ischemia-reperfusion injury, and pancreatitis
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Investigational
32596694
DrugRepV_8338Nelfinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
NA
Decrease (100 %)
Approved
32374457
DrugRepV_8451Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Yellow fever virus
YFV17D
Pathway
NA
Decrease (50 %)
Approved
30699122
DrugRepV_8456Berberine Chloride
NA
NA
Zika virus
NA
NA
NA
Decrease (50 %)
NA
29844387
DrugRepV_8471Berberine
NA
Parasitic and fungal infection
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
Approved
21295891
DrugRepV_8472Berberine
NA
Parasitic and fungal infection
Influenza virus
NA
Pathway
NA
Decrease (50 %)
Approved
30099043
DrugRepV_8473Ebselen
NA
Meniere Disease, Type 2 Diabetes Mellitus, and Type 1 Diabetes Mellitus
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
Investigational
23850693
DrugRepV_84742-Phenylbenzo[d]isothiazol-3(2H)-one
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_84752-Phenylbenzo[d] isoxazol-3(2H)-one
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_84762-Phenyl isoindolin-1-one
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_8477Chelerythrine chloride
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_8478Nitidine chloride
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_8479Berberine chloride
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_8480Sanguinarine chloride
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_8481Norsanguinarine chloride
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_8482R-Apomorphine hydrochloride
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_8483S-Apomorphine hydrochloride
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_8484R(?)-Propylnorapomorphine hydrochloride
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693
DrugRepV_8485R(?)-Apocodeine hydrochloride
NA
NA
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
NA
23850693