anti-Nipah browse page allows user to take a glance of the particular anti-Nipah ihibitor.By clicking on the table header arrows, user can sort entries in ascending or descending order.Moreover, the user can get the detal of every inhibitor by clicking on individual ID.


Total number of Records for Culture are 301




anti-Nipah_ID Drug Name
Nipah virus strain
Assay
Activity Type
Activity
References
anti-Nipah_001Ac-VALDPIDISIVLNKlKSDLEESKEWIRRSNKlLDSl-GSGSG-dPEG4-C-(CH2CON H2)-NH2
Nipah virus UMMC1
beta-galactosidase complementation assay
Inhibitory concentration
50 %
29566184
anti-Nipah_002Ac-VALDPIDISIVLNKIKSDLEESKEWIRRSNKILDSl-GSGSG-dPEGa-C-Chol-NH2
Nipah virus UMMC1
beta-galactosidase complementation assay
Inhibitory concentration
50 %
29566184
anti-Nipah_003Ac-VALDPI DISIVLN Kl KSDLEESKEWIRRSNKILDSI-GSGSGdPEG4-C-TOCO-NH2
Nipah virus UMMC1
beta-galactosidase complementation assay
Inhibitory concentration
50 %
29566184
anti-Nipah_004Ac-VALDPIDISIVLNKIKSDLEESKEWIRRSNKILDSl-GSGSG-dPEG4-C-(PEG4-Cho|)2-NH2
Nipah virus UMMC1
beta-galactosidase complementation assay
Inhibitory concentration
50 %
29566184
anti-Nipah_005Ac-VALDPIDISIVLNKIKSDLEESKEWIRRSNKILDSl-GSGSG-dPEG4-C-(PEG4-Toco)2-NH2
Nipah virus UMMC1
beta-galactosidase complementation assay
Inhibitory concentration
50 %
29566184
anti-Nipah_008N-[4-(1H-Tetrazol-1-yl)phenyl]-3,4-dihydro-2-naphthalenesulfonamide
Nipah virus Malaysia-1999
Iluminescence
Effective concentration
50 %
24735442
anti-Nipah_0093,4-Difluoro-N-[4-(1H-tetrazol-1-yl)phenyl]benzenesulfonamide
Nipah virus Malaysia-1999
Iluminescence
Effective concentration
50 %
24735442
anti-Nipah_010N,N-Dimethyl-1-(2-thienylsulfonyl)-5-indolinesulfonamide
Nipah virus Malaysia-1999
Iluminescence
Effective concentration
50 %
24735442
anti-Nipah_011N,N-Dimethyl-1-(2-thienylsulfonyl)-5-indolinesulfonamide
Nipah virus Malaysia-1999
TCID50
TCID50
100 TCID50/ml
24735442
anti-Nipah_012N-[4-(1H-Tetrazol-1-yl)phenyl]-3,4-dihydro-2-naphthalenesulfonamide
Nipah virus Malaysia-1999
TCID50
TCID50
10 TCID50/ml
24735442
anti-Nipah_0133,4-Difluoro-N-[4-(1H-tetrazol-1-yl)phenyl]benzenesulfonamide
Nipah virus Malaysia-1999
TCID50
TCID50
<1O TCID50/ml
24735442
anti-Nipah_0146-azauridine acetate
Nipah virus LUC2AM-Renilla Luciferase
Renilla luciferase
Effective concentration
50 %
24680955
anti-Nipah_0156-azauridine acetate
Nipah virus Malaysia-1999
TCID50
Effective concentration
50 %
24680955
anti-Nipah_016Pyrazofurin
Nipah virus LUC2AM-Renilla Luciferase
Renilla luciferase
Effective concentration
50 %
24680955
anti-Nipah_017{2,2,2-trifluoro-N-[3-(N-naphthylcarbamoyl)(4,5,6,7-tetrahydrobenzo [beta]thiophen-2-yl)]acetamide
Nipah virus LUC2AM-Renilla Luciferase
Renilla luciferase
Effective concentration
50 %
24680955
anti-Nipah_018{2,2,2-trifluoro-N-[3-(N-naphthylcarbamoyl)(4,5,6,7-tetrahydrobenzo [beta]thiophen-2-yl)]acetamide
Nipah virus Malaysia-1999
TCID50
Effective concentration
50 %
24680955
anti-Nipah_019N-(1,3-benzodioxol-5-ylmethyl)-2-(3-cyano-2-methyl-1H-indol-1-yl)acetamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
39.55 %
24501399
anti-Nipah_020N-benzyl-6-phenyl-2,3,4,9-tetrahydro-1H-carbazol-1-amine hydrochloride
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
102.26 %
24501399
anti-Nipah_0219H-carbazol-3-amine
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
55.68 %
24501399
anti-Nipah_0227-(1H-benzimidazol-2-ylthio)-8-methyl[1,3]dioxolo[4,5-g]quinolin-6(5H)-one
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
63.7 %
24501399
anti-Nipah_023N-[2-(2-methoxyethyl)-1,2,3,4-tetrahydropyrazino[1,2-a]benzimidazol-8-yl]benzamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
16 %
24501399
anti-Nipah_024tris[4-(dimethylamino)phenyl]methanol
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
121.65 %
24501399
anti-Nipah_0256-chloro-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-2-(3-pyridinyl)-4-quinolinecarboxamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
94.08 %
24501399
anti-Nipah_0261-(2-furoyl)-5-(2-furyl)-3-(3-methoxyphenyl)-4,5-dihydro-1H-pyrazole
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
5.15 %
24501399
anti-Nipah_0272-[(1H-benzimidazol-2-ylmethyl)thio]-1-[2-(4-methylphenoxy)ethyl]-1H-benzimidazole
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
23.57 %
24501399
anti-Nipah_028N-(3-chloro-4-fluorophenyl)-N-[4-(4-morpholinylsulfonyl)phenyl]urea
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
53.73 %
24501399
anti-Nipah_0294-{[(5-methyl-2-thienyl)methyl]amino}phenol
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
15.92 %
24501399
anti-Nipah_030N-[5-(1H-benzimidazol-2-yl)-2-methylphenyl]-1,3-benzodioxole-5-carboxamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
51.07 %
24501399
anti-Nipah_031N-[1-benzyl-2-oxo-2-(4-phenyl-1-piperazinyl)ethyl]benzamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
16.58 %
24501399
anti-Nipah_0322-methoxy-N-[1-methyl-2-(1-pyrrolidinylmethyl)-1H-benzimidazol-5-yl]benzamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
6.45 %
24501399
anti-Nipah_033N-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-2-(2-naphthyloxy)acetamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
80.96 %
24501399
anti-Nipah_034N-(2,5-dimethoxyphenyl)-N-[4-(trifluoromethyl)phenyl]urea
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
40.8 %
24501399
anti-Nipah_0354-{[(1H-benzimidazol-2-ylthio)acetyl]amino}phenyl thiocyanate
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
31.81 %
24501399
anti-Nipah_036N-(3,4-dichlorophenyl)-N-[3-(trifluoromethyl)phenyl]urea
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
44.08 %
24501399
anti-Nipah_037N-1,3-benzodioxol-5-yl-6-chloro-2-(3-pyridinyl)-4-quinolinecarboxamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
55.7 %
24501399
anti-Nipah_038N-(3-chlorophenyl)-N-(4-cyanophenyl)urea
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
63.91 %
24501399
anti-Nipah_039N-[4-(1H-benzimidazol-2-yl)phenyl]-2-chloro-5-(4H-1,2,4-triazol-4-yl)benzamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
27.96 %
24501399
anti-Nipah_040N-[3-(aminocarbonyl)-5-benzyl-2-thienyl]-2-methyl-3-furamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
18.33 %
24501399
anti-Nipah_0414,5-dimethyl-2-{[(5-propyl-3-thienyl)carbonyl]amino}-N-(3-pyridinylmethyl)-3-thiophenecarboxamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
12.33 %
24501399
anti-Nipah_0421-(isopropylamino)-3-(3-phenyl-4,5-dihydropyrazolo[4,3-a]carbazol-10(3H)-yl)-2-propanol
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
49.78 %
24501399
anti-Nipah_0432-[(4-tert-butyl-1,3-thiazol-2-yl)amino]-8-quinolinol
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
2.06 %
24501399
anti-Nipah_044N-(aminocarbonyl)-2-{[(5-methyl-3-thienyl)carbonyl]amino}-3-thiophenecarboxamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
46.11 %
24501399
anti-Nipah_0452-chloro-N-(4-phenyl-1,3-thiazol-2-yl)-5-(4H-1,2,4-triazol-4-yl)benzamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
81.01 %
24501399
anti-Nipah_046N-[3-(2-oxo-2H-chromen-3-yl)phenyl]-1,3-benzodioxole-5-carboxamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
58.07 %
24501399
anti-Nipah_0474,5-dimethyl-2-[(phenoxyacetyl)amino]-N-(3-pyridinylmethyl)-3-thiophenecarboxamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
55.23 %
24501399
anti-Nipah_048N-(4-{[(5-methyl-3-isoxazolyl)amino]sulfonyl}phenyl)-1-benzothiophene-3-carboxamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
45.06 %
24501399
anti-Nipah_0493-[(1H-benzimidazol-2-ylmethyl)thio]-9-benzyl-9H-[1,2,4]triazolo[4,3-a]benzimidazole
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
12.87 %
24501399
anti-Nipah_050methyl N-[4,6-bis(isopropylamino)-1,3,5-triazin-2-yl]-N-cyanoglycinate
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
88.36 %
24501399
anti-Nipah_051N-(3,4-dichlorophenyl)-2-oxo-2,3-dihydro-1,3-benzoxazole-6-sulfonamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
57.76 %
24501399
anti-Nipah_052N-(3-pyridinylmethyl)dibenzo[b,d]furan-3-amine
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
31.98 %
24501399
anti-Nipah_053(1,3-benzodioxol-5-ylmethyl)[4-(1-pyrrolidinyl)phenyl]amine
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
-8.16 %
24501399
anti-Nipah_0544-methyl-5-phenyl-N-3-pyridinyl-2-thiophenecarboxamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
49.25 %
24501399
anti-Nipah_055N-(2,5-dimethoxyphenyl)-2-(2-oxo-1,3-benzoxazol-3(2H)-yl)acetamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
30.96 %
24501399
anti-Nipah_0563-[(2,4-dichlorophenoxy)methyl]-N-(3-pyridinylmethyl)benzamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
39.35 %
24501399
anti-Nipah_0575-phenyl-2-(2-phenylethyl)[1,2,4]triazolo[1,5-a]pyrimidin-7(4H)-one
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
30.39 %
24501399
anti-Nipah_0586-bromo-2-oxo-N-3-pyridinyl-2H-chromene-3-carboxamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
97.85 %
24501399
anti-Nipah_0592-[(2-methyl-8-quinolinyl)amino]-4H-pyrido[3,2-e][1,3]thiazin-4-one
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
9.77 %
24501399
anti-Nipah_060N-(3-chloro-4-fluorophenyl)-N-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
42.76 %
24501399
anti-Nipah_0614-({[(3-chloro-4-fluorophenyl)amino]carbonyl}amino)-N-methylbenzenesulfonamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
41.82 %
24501399
anti-Nipah_0622-(4-fluorophenyl)-N-(4-{[(4-methylphenyl)amino]sulfonyl}phenyl)acetamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
27.2 %
24501399
anti-Nipah_0635-methyl-N-[4-(1-pyrrolidinylsulfonyl)phenyl]-3-thiophenecarboxamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
-11.7 %
24501399
anti-Nipah_0642-amino-N-(3-chlorophenyl)-3-quinolinecarboxamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
46.45 %
24501399
anti-Nipah_0652-(1,3-benzodioxol-5-yl)-1-(1,3-benzodioxol-5-ylmethyl)-1H-benzimidazole
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
13.74 %
24501399
anti-Nipah_066N-{3-[(benzylamino)carbonyl]phenyl}-5-methyl-3-thiophenecarboxamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
15.09 %
24501399
anti-Nipah_0678-chloro-N-[3-(3-methyl-1H-pyrazol-1-yl)propyl]-2-(2-pyridinyl)-4-quinolinecarboxamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
-0.5 %
24501399
anti-Nipah_068N-[4-(2,4-difluorophenyl)-1,3-thiazol-2-yl]-2-(2-thienyl)acetamide
Nipah virus Peptide -F0, amino acids 105 to 114
CatL-Peptide cleavage
Percentage inhibition
12.4 %
24501399
anti-Nipah_069Brilliant Green
Nipah virus Malaysia-1999
Immnuolabelling assay
Inhibitory concentration
50 %
19889218
anti-Nipah_070Gentian Violet
Nipah virus Malaysia-1999
Immnuolabelling assay
Inhibitory concentration
50 %
19889218
anti-Nipah_071Gliotoxin
Nipah virus Malaysia-1999
Immnuolabelling assay
Inhibitory concentration
50 %
19889218
anti-Nipah_072Brilliant Green
Nipah virus Malaysia-1999
TCID50
Viral titer
>100 TCID50/ml
19889218
anti-Nipah_073Gentian Violet
Nipah virus Malaysia-1999
TCID50
Viral titer
>100 TCID50/ml
19889218
anti-Nipah_074Gliotoxin
Nipah virus Malaysia-1999
TCID50
Viral titer
>100 TCID50/ml
19889218
anti-Nipah_075Brilliant Green
Nipah virus Pseudotyped_pNiV
Immunofluorescence
Inhibitory concentration
50 %
19889218
anti-Nipah_076Gentian Violet
Nipah virus Pseudotyped_pNiV
Immunofluorescence
Inhibitory concentration
50 %
19889218
anti-Nipah_077Gliotoxin
Nipah virus Pseudotyped_pNiV
Immunofluorescence
Inhibitory concentration
50 %
19889218
anti-Nipah_0782-benzyl-1,3-benzoxazol-5-amine
Nipah virus Nipah G/F fusion expression vector
Syncytia formation
Effective concentration
50 %
19499921
anti-Nipah_079N-[(4-chlorophenyl)methyl]-1-(2-hydroxyethyl)-4-oxo-7-(trifluoromethyl)-1,4-dihydroquinoline-3-carboxamide
Nipah virus Nipah G/F fusion expression vector
Syncytia formation
Effective concentration
50 %
19499921
anti-Nipah_080N-(3-chloro-4-fluorophenyl)-1-(2-hydroxyethyl)-4-oxo-7-(trifluoromethyl)-1,4-dihydroquinoline-3-carboxamide
Nipah virus Nipah G/F fusion expression vector
Syncytia formation
Effective concentration
50 %
19499921
anti-Nipah_0817-(4-carbamoylpiperidin-1-yl)-1-cyclopropyl-N-[(2,4-dichlorophenyl)methyl]-6-fluoro-4-oxo-1,2,3,4-tetrahydroquinoline-3-carboxamide
Nipah virus Nipah G/F fusion expression vector
Syncytia formation
Effective concentration
50 %
19499921
anti-Nipah_082N-[(2,4-dichlorophenyl)methyl]-6-fluoro-1-(2-hydroxyethyl)-7-[4-(oxirane-2-carbonyl)piperidin-1-yl]-4-oxo-1,2,3,4-tetrahydroquinoline-3-carboxamide
Nipah virus Nipah G/F fusion expression vector
Syncytia formation
Effective concentration
50 %
19499921
anti-Nipah_0834-oxo-1,4-dihydroquinoline-3,6-dicarboxylic acid
Nipah virus Nipah G/F fusion expression vector
Syncytia formation
Effective concentration
50 %
19499921
anti-Nipah_084N-[(2,4-dichlorophenyl)methyl]-6-fluoro-1-(2-hydroxyethyl)-7-[4-(oxirane-2-carbonyl)piperazin-1-yl]-4-oxo-1,2,3,4-tetrahydroquinoline-3-carboxamide
Nipah virus Nipah G/F fusion expression vector
Syncytia formation
Effective concentration
50 %
19499921
anti-Nipah_0851-cyclopropyl-N-[(2,4-dichlorophenyl)methyl]-6-fluoro-7-[4-(oxirane-2-carbonyl)piperazin-1-yl]-4-oxo-1,2,3,4-tetrahydroquinoline-3-carboxamide
Nipah virus Nipah G/F fusion expression vector
Syncytia formation
Effective concentration
50 %
19499921
anti-Nipah_0863,5-diethyl 4-hydroxy-2,6-bis(4-nitrophenyl)-1-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-3,5-dicarboxylate
Nipah virus Nipah G/F fusion expression vector
Syncytia formation
Effective concentration
50 %
19499921
anti-Nipah_087AAHL 7
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_088AAHL 13
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_089AAHL 15
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_090AAHL 16
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_091AAHL 18
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_092AAHL 22
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_093AAHL 23
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_094AAHL 33
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_095AAHL 42
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_096AAHL 7
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_097AAHL 13
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_098AAHL 15
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_099AAHL 16
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_100AAHL 18
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_101AAHL 22
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_102AAHL 23
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_103AAHL 33
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_104AAHL 42
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_105AAHL 7
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_106AAHL 13
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_107AAHL 15
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_108AAHL 16
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_109AAHL 18
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_110AAHL 22
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_111AAHL 23
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_112AAHL 33
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_113AAHL 42
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_114AAHL 7
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_115AAHL 13
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_116AAHL 15
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_117AAHL 16
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_118AAHL 18
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_119AAHL 22
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_120AAHL 23
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_121AAHL 33
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_122AAHL 42
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_123AAHL 7
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_124AAHL 13
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_125AAHL 15
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_126AAHL 16
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_127AAHL 18
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_128AAHL 22
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_129AAHL 23
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_130AAHL 33
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_131AAHL 42
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_132AAHL 7
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_133AAHL 13
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_134AAHL 15
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_135AAHL 16
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_136AAHL 18
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_137AAHL 22
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_138AAHL 23
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_139AAHL 33
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_140AAHL 42
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_141AAHL 7
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_142AAHL 13
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_143AAHL 15
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_144AAHL 16
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_145AAHL 18
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_146AAHL 22
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_147AAHL 23
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_148AAHL 33
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_149AAHL 42
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_150AAHL 7
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_151AAHL 13
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_152AAHL 16
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_153AAHL 18
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_154AAHL 22
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_155AAHL 23
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_156AAHL 33
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_157AAHL 7
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_158AAHL 13
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_159AAHL 15
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_160AAHL 16
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_161AAHL 18
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_162AAHL 22
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_163AAHL 23
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_164AAHL 33
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_165AAHL 42
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_166AAHL 7
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_167AAHL 13
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_168AAHL 15
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_169AAHL 16
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_170AAHL 18
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_171AAHL 22
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_172AAHL 23
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_173AAHL 33
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_174AAHL 42
Nipah virus Malaysia-1999
Chemiluminescent
Inhibitory concentration
50 %
19428741
anti-Nipah_1754-amino-1-[5-azido-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]pyrimidin-2-one
Nipah virus Rec. M-GFP2AM
Fluorescence
Effective concentration
50 %
29601894
anti-Nipah_1764-Amino-1-[(2R,4R,5R)-5-azido-3,3-difluoro-4-hydroxy-5-(hydroxymethyl)tetrahydro-2-furanyl]-2(1H)-pyrimidinone
Nipah virus Rec. M-GFP2AM
Fluorescence
Effective concentration
50 %
29601894
anti-Nipah_1774-Amino-1-[(2R,3R,4R,5R)-5-azido-3-fluoro-4-hydroxy-5-(hydroxymethyl)tetrahydro-2-furanyl]-2(1H)-pyrimidinone
Nipah virus Rec. M-GFP2AM
Fluorescence
Effective concentration
50 %
29601894
anti-Nipah_1784-amino-1-[(2R,3R,4S,5R)-5-azido-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]pyrimidin-2-one
Nipah virus Rec. M-GFP2AM
Cytopathic effect assay
Effective concentration
50 %
29601894
anti-Nipah_1794-Amino-1-[(2R,4R,5R)-5-azido-3,3-difluoro-4-hydroxy-5-(hydroxymethyl)tetrahydro-2-furanyl]-2(1H)-pyrimidinone
Nipah virus Rec. M-GFP2AM
Cytopathic effect assay
Effective concentration
50 %
29601894
anti-Nipah_1804-Amino-1-[(2R,3R,4R,5R)-5-azido-3-fluoro-4-hydroxy-5-(hydroxymethyl)tetrahydro-2-furanyl]-2(1H)-pyrimidinone
Nipah virus Rec. M-GFP2AM
Cytopathic effect assay
Effective concentration
50 %
29601894
anti-Nipah_1814-amino-1-[(2R,3R,4S,5R)-5-azido-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]pyrimidin-2-one
Nipah virus Malaysia-1999
Cytopathic effect assay
Effective concentration
50 %
29601894
anti-Nipah_1824-Amino-1-[(2R,4R,5R)-5-azido-3,3-difluoro-4-hydroxy-5-(hydroxymethyl)tetrahydro-2-furanyl]-2(1H)-pyrimidinone
Nipah virus Malaysia-1999
Cytopathic effect assay
Effective concentration
50 %
29601894
anti-Nipah_1834-Amino-1-[(2R,3R,4R,5R)-5-azido-3-fluoro-4-hydroxy-5-(hydroxymethyl)tetrahydro-2-furanyl]-2(1H)-pyrimidinone
Nipah virus Malaysia-1999
Cytopathic effect assay
Effective concentration
50 %
29601894
anti-Nipah_1844-amino-1-[(2R,3R,4S,5R)-5-azido-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]pyrimidin-2-one
Nipah virus Malaysia-1999
TCID50
Effective concentration
50 %
29601894
anti-Nipah_1854-Amino-1-[(2R,4R,5R)-5-azido-3,3-difluoro-4-hydroxy-5-(hydroxymethyl)tetrahydro-2-furanyl]-2(1H)-pyrimidinone
Nipah virus Malaysia-1999
TCID50
Effective concentration
50 %
29601894
anti-Nipah_1864-Amino-1-[(2R,3R,4R,5R)-5-azido-3-fluoro-4-hydroxy-5-(hydroxymethyl)tetrahydro-2-furanyl]-2(1H)-pyrimidinone
Nipah virus Malaysia-1999
TCID50
Effective concentration
50 %
29601894
anti-Nipah_1874-amino-1-[(2R,3R,4S,5R)-5-azido-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]pyrimidin-2-one
Nipah virus NiV-Luc2AM
Luciferase assay
Effective concentration
50 %
28629988
anti-Nipah_1884-amino-1-[(2R,3R,4S,5R)-5-azido-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]pyrimidin-2-one
Nipah virus NiV-Luc2AM
Luciferase assay
Effective concentration
50 %
28629988
anti-Nipah_1894-amino-1-[(2R,3R,4S,5R)-5-azido-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]pyrimidin-2-one
Nipah virus Malaysia
Cytopathic effect assay
Effective concentration
50 %
28629988
anti-Nipah_1904-amino-1-[(2R,3R,4S,5R)-5-azido-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]pyrimidin-2-one
Nipah virus Malaysia
Cytopathic effect assay
Effective concentration
50 %
28629988
anti-Nipah_1914-amino-1-[(2R,3R,4S,5R)-5-azido-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]pyrimidin-2-one
Nipah virus Malaysia
TCID50
Effective concentration
50 %
28629988
anti-Nipah_1924-amino-1-[(2R,3R,4S,5R)-5-azido-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]pyrimidin-2-one
Nipah virus Malaysia
TCID50
Effective concentration
50 %
28629988
anti-Nipah_1932-amino-N-[4-[5-phenanthren-2-yl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]acetamide
Nipah virus NiV-Luc
Luciferase assay
Effective concentration
50 %
25986249
anti-Nipah_1942-diphenylboranyloxyethanamine
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_1955-(methylamino)-2-[[(2S,3R,5R,8S,9S)-3,5,9-trimethyl-2-[1-oxo-1-(1H-pyrrol-2-yl)propan-2-yl]-1,7-dioxaspiro[5.5]undecan-8-yl]methyl]-1,3-benzoxazole-4-carboxylic acid
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_1962,5-ditert-butylbenzene-1,4-diol
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_197ethyl 12-[[2-[(2R,3R)-3-[2-[(12-ethoxy-12-oxododecyl)-methylamino]-2-oxoethoxy]butan-2-yl]oxyacetyl]-methylamino]dodecanoate
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_198Dantrolene
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_199Ionomycin
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_200Ryanodine
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_201Thapsigargin
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_202Xestospongin C
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_203Agatoxin
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_204Amlodipine besylate
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_205Conotoxin
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_206Gabapentin
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_207Lanthanum chloride
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_208Mibefradil
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_209Nifedipine
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_210Praziquantel
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_211Tetrandine
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_212Verapamil
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_2135-N-ethyl isopropyl amiloride
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_214Amiloride
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_215Benzamil
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_216Monensin
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_217Phenytoin
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_2187-octyl-indolactam
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_219Cyclosporine
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_220Gliotoxin
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_221Oleic Acid
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_222Phenoxybenzamine
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_223PKC Inhibitor
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_224PMA
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_225Rottlerin
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_226U73122
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_22725-hydroxy-cholecalciferol
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_2284-hydroxy-tamoxifen
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_229Argo-vasopressin
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_230Bradykinin
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_231Caffeine
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_232Cholecalciferol
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_233Clotrimazole
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_234Propranolol
Nipah virus Malaysia-1999
Immunolabeling assay
Inhibitory concentration
50 %
20668647
anti-Nipah_235Chloroquine
Nipah virus Malaysia
Plaque assay
Inhibitory concentration
50 %
19889926
anti-Nipah_236Ribavirin
Nipah virus Malaysia
Plaque assay
Inhibitory concentration
50 %
19889926
anti-Nipah_239Chloroquine
Nipah virus NA
Chemiluminescent
Inhibitory concentration
50 %
19264786
anti-Nipah_240Favipiravir
Nipah virus Malaysia
Plaque assay
Effective concentration
50 %
29765101
anti-Nipah_241Favipiravir
Nipah virus Bangladesh
Plaque assay
Effective concentration
50 %
29765101
anti-Nipah_242Favipiravir
Nipah virus rNiV-Gluc-eGFP
Plaque assay
Effective concentration
50 %
29765101
anti-Nipah_243Favipiravir
Nipah virus rNiV-Gluc-eGFP
Cytopathic effect assay
Virus titer
4 log(PFU/ml)
29765101
anti-Nipah_244Favipiravir
Nipah virus rNiV-Gluc-eGFP
Real time PCR
Virus titer
10 fold
29765101
anti-Nipah_251(2R,3R,4S,5R)-2-(4-Aminopyrrolo[2,1-f][1,2,4]triazin-7-yl)-3,4-dihydroxy-5-(hydroxymethyl)tetrahydro-2-furancarbonitrile
Nipah virus Rec. M-Luc2AM
Renilla luciferase
Effective concentration
50 %
28262699
anti-Nipah_252(2R,3R,4S,5R)-2-(4-Aminopyrrolo[2,1-f][1,2,4]triazin-7-yl)-3,4-dihydroxy-5-(hydroxymethyl)tetrahydro-2-furancarbonitrile
Nipah virus Malaysia
TCID50
Effective concentration
50 %
28262699
anti-Nipah_253(2R,3R,4S,5R)-2-(4-Aminopyrrolo[2,1-f][1,2,4]triazin-7-yl)-3,4-dihydroxy-5-(hydroxymethyl)tetrahydro-2-furancarbonitrile
Nipah virus Bangladesh-2004
TCID50
Effective concentration
50 %
28262699
anti-Nipah_254(2R,3R,4S,5R)-2-(4-Aminopyrrolo[2,1-f][1,2,4]triazin-7-yl)-3,4-dihydroxy-5-(hydroxymethyl)tetrahydro-2-furancarbonitrile
Nipah virus Bangladesh-2004
Cytopathic effect assay
Percentage inhibition
90 %
28262699
anti-Nipah_255(2R,3R,4S,5R)-2-(4-Aminopyrrolo[2,1-f][1,2,4]triazin-7-yl)-3,4-dihydroxy-5-(hydroxymethyl)tetrahydro-2-furancarbonitrile
Nipah virus Malaysia
Cytopathic effect assay
Percentage inhibition
90 %
28262699
anti-Nipah_2562-ethylbutyl (2S)-2-[[[(2R,3S,4R,5R)-5-(4-aminopyrrolo[2,1-f][1,2,4]triazin-7-yl)-5-cyano-3,4-dihydroxyoxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoate
Nipah virus Rec. M-Luc2AM
Renilla luciferase
Effective concentration
50 %
28262699
anti-Nipah_2572-ethylbutyl (2S)-2-[[[(2R,3S,4R,5R)-5-(4-aminopyrrolo[2,1-f][1,2,4]triazin-7-yl)-5-cyano-3,4-dihydroxyoxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoate
Nipah virus Malaysia
TCID50
Effective concentration
50 %
28262699
anti-Nipah_2582-ethylbutyl (2S)-2-[[[(2R,3S,4R,5R)-5-(4-aminopyrrolo[2,1-f][1,2,4]triazin-7-yl)-5-cyano-3,4-dihydroxyoxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoate
Nipah virus Bangladesh-2004
TCID50
Effective concentration
50 %
28262699
anti-Nipah_2592-ethylbutyl (2S)-2-[[[(2R,3S,4R,5R)-5-(4-aminopyrrolo[2,1-f][1,2,4]triazin-7-yl)-5-cyano-3,4-dihydroxyoxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoate
Nipah virus Bangladesh-2004
Cytopathic effect assay
Percentage inhibition
90 %
28262699
anti-Nipah_2602-ethylbutyl (2S)-2-[[[(2R,3S,4R,5R)-5-(4-aminopyrrolo[2,1-f][1,2,4]triazin-7-yl)-5-cyano-3,4-dihydroxyoxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoate
Nipah virus Malaysia
Cytopathic effect assay
Percentage inhibition
99 %
28262699
anti-Nipah_261N-(3-cyanophenyl)-2-phenylacetamide
Nipah virus Nipah G/F fusion expression vector
Syncytia formation
Fusion Inhibition
0 %
20685931
anti-Nipah_2623-[(2-phenylacetyl)amino]benzoic acid
Nipah virus Nipah G/F fusion expression vector
Syncytia formation
Fusion Inhibition
0 %
20685931
anti-Nipah_263methyl 3-[(2-phenylacetyl)amino]benzoate
Nipah virus Nipah G/F fusion expression vector
Syncytia formation
Fusion Inhibition
35 %
20685931
anti-Nipah_2645-nitro-2-(2-phenylacetamido)benzamide
Nipah virus Nipah G/F fusion expression vector
Syncytia formation
Fusion Inhibition
0 %
20685931
anti-Nipah_2654-nitro-2-[(2-phenylacetyl)amino]benzamide
Nipah virus Nipah G/F fusion expression vector
Syncytia formation
Fusion Inhibition
10 %
20685931
anti-Nipah_266Carbocyclic 3-deazaadenosine
Nipah virus Malaysia-1999
Cytopathic effect assay
Inhibitory concentration
100 %
16641448
anti-Nipah_267(-)-5 Noraristeromycin
Nipah virus Malaysia-1999
Cytopathic effect assay
Inhibitory concentration
100 %
16641448
anti-Nipah_268DHCaA
Nipah virus Malaysia-1999
Cytopathic effect assay
Inhibitory concentration
100 %
16641448
anti-Nipah_269Ribavirin
Nipah virus Malaysia-1999
Cytopathic effect assay
Inhibitory concentration
NA NA
16641448
anti-Nipah_270EICAR
Nipah virus Malaysia-1999
Cytopathic effect assay
Inhibitory concentration
100 %
16641448
anti-Nipah_271Pyrazofurin
Nipah virus Malaysia-1999
Cytopathic effect assay
Inhibitory concentration
100 %
16641448
anti-Nipah_272Carbodine
Nipah virus Malaysia-1999
Cytopathic effect assay
Inhibitory concentration
100 %
16641448
anti-Nipah_2736-Aza-uridine
Nipah virus Malaysia-1999
Cytopathic effect assay
Inhibitory concentration
100 %
16641448
anti-Nipah_274Poly(I)-poly(C12U)
Nipah virus Malaysia-1999
Cytopathic effect assay
Inhibitory concentration
100 %
16641448
anti-Nipah_277(5Z)-5-[(5-phenylfuran-2-yl)methylidene]-3-prop-2-enyl-2-sulfanylidene-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_278(5Z)-3-Ethyl-5-[(5-phenyl-2-furyl)methylene]-2-thioxo-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_279(5Z)-5-[(5-Phenyl-2-furyl)methylene]-3-propyl-2-thioxo-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_280(5Z)-3-Benzyl-5-[(5-phenyl-2-furyl)methylene]-2-thioxo-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_281(5Z)-3-Methyl-5-[(5-phenyl-2-furyl)methylene]-2-thioxo-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_282(5Z)-5-{[5-(3-Chlorophenyl)-2-furyl]methylene}-3-ethyl-2-thioxo-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_283(5Z)-3-Ethyl-5-{[5-(3-fluorophenyl)-2-furyl]methylene}-2-thioxo-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_2843-Ethyl-5-{[5-(2-fluorophenyl)-2-furyl]methylene}-2-thioxo-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_285(5Z)-5-{[5-(2-Chlorophenyl)-2-furyl]methylene}-3-ethyl-2-thioxo-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_286(5Z)-3-ethyl-5-{[5-(2-methoxyphenyl)furan-2-yl]methylidene}-2-sulfanylidene-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_287(5Z)-3-ethyl-5-{[5-(3-methoxyphenyl)furan-2-yl]methylidene}-2-sulfanylidene-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_288(5Z)-3-Ethyl-2-thioxo-5-({5-[2-(trifluoromethyl)phenyl]-2-furyl}methylene)-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_289(5Z)-3-Ethyl-5-[(5-methyl-2-furyl)methylene]-2-thioxo-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_290(5Z)-3-Ethyl-5-(2-furylmethylene)-2-thioxo-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_291(5Z)-3-Ethyl-5-{[5-(2-nitrophenyl)-2-furyl]methylene}-2-thioxo-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_292(5Z)-3-ethyl-5-{[5-(2-hydroxyphenyl)furan-2-yl]methylidene}-2-sulfanylidene-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_293(5Z)-5-{[5-(2-aminophenyl)furan-2-yl]methylidene}-3-ethyl-2-sulfanylidene-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_294(5Z)-3-ethyl-5-[(5-phenylthiophen-2-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_295(5Z)-5-({[1,1-biphenyl]-3-yl}methylidene)-3-ethyl-2-sulfanylidene-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_2962-(5-{[(5Z)-3-ethyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl}furan-2-yl)benzene-1-diazonium; tetrafluoroboranuide
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_2973-[(5Z)-4-oxo-5-[(5-phenylfuran-2-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-3-yl]propyl acetate
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_298(5Z)-3-(3-hydroxypropyl)-5-[(5-phenylfuran-2-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_299(5Z)-3-ethyl-5-[(2-phenyl-1,3-oxazol-5-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_300 3-[(5Z)-4-oxo-5-[(5-phenylfuran-2-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-3-yl]propyl 4-{2-oxo-hexahydro-1H-thieno[3,4-d]imidazol-4-yl}butanoate
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_301(5Z)-5-[(5-Phenyl-2-furyl)methylene]-2-thioxo-3-vinyl-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_302(5Z)-3-Ethyl-5-{[5-(2-nitrophenyl)-2-furyl]methylene}-1,3-thiazolidine-2,4-dione
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_303(5Z)-3-ethenyl-5-[(5-phenylfuran-2-yl)methylidene]-1,3-thiazolidine-2,4-dithione
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_304(5Z)-3-ethyl-5-{[5-(2-nitrophenyl)furan-2-yl]methylidene}-1,3-thiazolidine-2,4-dithione
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_305(5Z)-3-ethenyl-5-[(5-phenylfuran-2-yl)methylidene]-4-sulfanylidene-1,3-thiazolidin-2-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_306(5Z)-3-ethyl-5-{[5-(2-nitrophenyl)furan-2-yl]methylidene}-4-sulfanylidene-1,3-thiazolidin-2-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_307(5Z)-5-[(5-Phenyl-2-furyl)methylene]-2-thioxo-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_308(5Z)-5-[(5-phenylfuran-2-yl)methylidene]-3-(prop-2-yn-1-yl)-2-sulfanylidene-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_3095-[(5-phenylfuran-2-yl)methyl]-3-(prop-2-en-1-yl)-2-sulfanylidene-1,3-thiazolidin-4-one
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_310N-{3-[(5Z)-2,4-dioxo-5-[(5-phenylfuran-2-yl)methylidene]-1,3-thiazolidin-3-yl]propyl}acetamide
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_311(5Z)-3-(3-aminopropyl)-5-[(5-phenylfuran-2-yl)methylidene]-1,3-thiazolidine-2,4-dione
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_3122-methylpropyl N-{3-[(5Z)-4-oxo-5-[(5-phenylfuran-2-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-3-yl]propyl}carbamate
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A
anti-Nipah_3133-[(5Z)-2,4-dioxo-5-[(5-phenylfuran-2-yl)methylidene]-1,3-thiazolidin-3-yl]propyl 4-{2-oxo-hexahydro-1H-thieno[3,4-d]imidazol-4-yl}butanoate
Nipah virus NiV-pVSV
Plaque assay
Inhibitory concentration
50 %
WO2010044924A