HSPMdb Accession No | HSPMDB002607 |
PMID | 30126533 |
Target | Hsp100 |
HSP Name | ClpP |
Organism | Human |
Localization | Mitochondria |
Enzymatic activity | Inhibition of protease activity |
Compound Name | ADEP-03 |
SMILES | O=C([C@H](C)NC([C@H](C)N(C)C([C@@]1([H])N(C([C@@H](NC([C@H](CC2=CC=CC=C2)NC(/C=C/C=C/C)=O)=O)CO3)=O)CCC1)=O)=O)N4C[C@H](C)C[C@@]4([H])C3=O |
Class | Acyldepsipeptide analogue |
RD_Index | 0.66 at 25 uM |
Site of Interaction | Nucleotide binding domain |
Type of Enzymatic Assay | Substrate degradation assay (FITC-casein) |