| HSPMdb Accession No | HSPMDB002569 |
| PMID | 21855356 |
| Target | Hsp100 |
| HSP Name | ClpP |
| Organism | Bacteria |
| Localization | Cytosol |
| Enzymatic activity | Inhibition of peptidase activity |
| Compound Name | 4 |
| IUPAC Name | (3R,4R)-4-(4-(N,N-Dimethylamino)benzamido-5-pentyl)-3-(non-8-enyl)oxetan-2-one |
| SMILES | CN(C)C1=CC=C(C(=O)NC(CCCC)[C@H]2[C@H](C(O2)=O)CCCCCCCC=C)C=C1 |
| Class | Beta lactone analogue |
| % Enzymatic Inhibition/Fold Change | 65% at 20 uM |
| Site of Interaction | Nucleotide binding domain |
| Type of Enzymatic Assay | Peptidase assay (SLY-AMC) |
| Cellular Model | S. aureus |
| Disease | Bacterial infection |
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