| HSPMdb Accession No | HSPMDB002430 |
| PMID | 28917450 |
| Target | Hsp100 |
| HSP Name | ClpP |
| Organism | Plasmodium falciparum |
| Localization | Cytosol |
| Enzymatic activity | Inhibition of protease activity |
| Compound Name | 9 |
| IUPAC Name | 5-Chloro-N-(3-((4-chlorophenyl)amino)-3-oxopropyl)-2-((4-ethylbenzyl)thio)pyrimidine-4-carboxamide |
| SMILES | ClC=1C(=NC(=NC1)SCC1=CC=C(C=C1)CC)C(=O)NCCC(=O)NC1=CC=C(C=C1)Cl |
| Class | Library of small molecule structures |
| IC50 (µM) | >100 |
| Site of Interaction | Nucleotide binding domain |
| Type of Enzymatic Assay | Peptidase assay (SLY-AMC) |
| Cellular Model | P. falciparum |
| Disease | Malaria |
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