| HSPMdb Accession No | HSPMDB002362 |
| PMID | 25944857 |
| Target | Hsp100 |
| HSP Name | ClpP1P2 |
| Organism | Bacteria |
| Localization | Cytosol |
| Cellular activity | Antibacterial activity |
| Compound Name | MG-262 |
| IUPAC Name | [(1R)-3-methyl-1-[[(2S)-4-methyl-2-[[(2S)-4-methyl-2-(phenylmethoxycarbonylamino)pentanoyl]amino]pentanoyl]amino]butyl]boronic acid |
| SMILES | B(C(CC(C)C)NC(=O)C(CC(C)C)NC(=O)C(CC(C)C)NC(=O)OCC1=CC=CC=C1)(O)O |
| Class | Bortezomib derivative |
| Site of Interaction | Nucleotide binding domain |
| Percentage Cell Growth Inhibition | 45% at 50 uM |
| Cellular assay | Bacterial growth inhibition assay (OD based) |
| Cellular Model | M. smegmatis (mc2155) |
| Disease | Tuberculosis |
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