HSPMdb Accession No | HSPMDB001820 |
PMID | 30571121 |
Target | Hsp100 |
HSP Name | ClpP |
Organism | Bacteria |
Localization | Cytosol |
Enzymatic activity | Inhibition of peptidase activity |
Compound Name | 78 |
IUPAC Name | Benzyl ((4-(Dimethylamino)phenyl)(diphenoxyphosphoryl)-methyl)carbamate |
SMILES | O=C(OCC1=CC=CC=C1)NC(C2=CC=C(N(C)C)C=C2)P(OC3=CC=CC=C3)(OC4=CC=CC=C4)=O |
Class | Serine protease inhibitor library |
% Enzymatic Inhibition/Fold Change | 100% at 200 uM |
IC50 (µM) | 0.6 |
Site of Interaction | Nucleotide binding domain |
Type of Enzymatic Assay | Peptidase assay (SLY-AMC) |
Disease | Bacterial infection |