| HSPMdb Accession No | HSPMDB001817 |
| PMID | 30571121 |
| Target | Hsp100 |
| HSP Name | ClpP |
| Organism | Bacteria |
| Localization | Cytosol |
| Enzymatic activity | Inhibition of peptidase activity |
| Compound Name | 75 |
| IUPAC Name | 2-(2-(Prop-2-yn-1-yloxy)ethoxy)ethyl (Diphenoxyphosphoryl)(4-(piperazin-1-yl)phenyl)methylcarbamate 2,2,2-Trifluoroacetate |
| SMILES | O=C(O)C(F)(F)F.O=C(OCCOCCOCC#C)NC(P(OC1=CC=CC=C1)(OC2=CC=CC=C2)=O)C3=CC=C(N4CCNCC4)C=C3 |
| Class | Serine protease inhibitor library |
| % Enzymatic Inhibition/Fold Change | 25% at 200 uM |
| Site of Interaction | Nucleotide binding domain |
| Type of Enzymatic Assay | Peptidase assay (SLY-AMC) |
| Disease | Bacterial infection |
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