| HSPMdb Accession No | HSPMDB001799 |
| PMID | 30571121 |
| Target | Hsp100 |
| HSP Name | ClpP |
| Organism | Bacteria |
| Localization | Cytosol |
| Enzymatic activity | Inhibition of peptidase activity |
| Compound Name | 57 |
| IUPAC Name | 3,3,4,4,5,5,6,6,7,8,8,8-Dodecafluoro-7-(trifluoromethyl)octyl 1-(Diphenoxyphosphoryl)-2-(4-guanidinophenyl)ethylcarbamate2,2,2-Trifluoroacetate |
| SMILES | O=C(OCCC(F)(F)C(F)(F)C(F)(F)C(F)(F)C(C(F)(F)F)(F)C(F)(F)F)NC(P(OC1=CC=CC=C1)(OC2=CC=CC=C2)=O)CC3=CC=C(NC(N)=N)C=C3.O=C(O)C(F)(F)F |
| Class | Serine protease inhibitor library |
| % Enzymatic Inhibition/Fold Change | 55% at 200 uM |
| Site of Interaction | Nucleotide binding domain |
| Type of Enzymatic Assay | Peptidase assay (SLY-AMC) |
| Disease | Bacterial infection |
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