| HSPMdb Accession No | HSPMDB001796 |
| PMID | 30571121 |
| Target | Hsp100 |
| HSP Name | ClpP |
| Organism | Bacteria |
| Localization | Cytosol |
| Enzymatic activity | Inhibition of peptidase activity |
| Compound Name | 54 |
| IUPAC Name | P e n t - 4 - y n - 1 - y l ( 1 - ( d i p h e n o x y p h o s p h o r y l ) - 2 - ( 4 -guanidinophenyl)ethyl)carbamate |
| SMILES | O=C(OCCCC#C)NC(P(OC1=CC=CC=C1)(OC2=CC=CC=C2)=O)CC3=CC=C(NC(N)=N)C=C3 |
| Class | Serine protease inhibitor library |
| % Enzymatic Inhibition/Fold Change | 23% at 200 uM |
| Site of Interaction | Nucleotide binding domain |
| Type of Enzymatic Assay | Peptidase assay (SLY-AMC) |
| Disease | Bacterial infection |
Loading Please Wait ...