| HSPMdb Accession No | HSPMDB001790 |
| PMID | 30571121 |
| Target | Hsp100 |
| HSP Name | ClpP |
| Organism | Bacteria |
| Localization | Cytosol |
| Enzymatic activity | Inhibition of peptidase activity |
| Compound Name | 48 |
| IUPAC Name | Diphenyl (E)-Diphenyl ((3-(Benzo[d][1,3]dioxol-5-yl)acrylamido)-(1-carbamimidoylpiperidin-4-yl)methyl)phosphonate 2,2,2-Trifluoroacetate |
| SMILES | NC(N1CCC(C(P(OC2=CC=CC=C2)(OC3=CC=CC=C3)=O)NC(/C=C/C4=CC=C(OCO5)C5=C4)=O)CC1)=N.O=C(O)C(F)(F)F |
| Class | Serine protease inhibitor library |
| % Enzymatic Inhibition/Fold Change | 4% at 200 uM |
| Site of Interaction | Nucleotide binding domain |
| Type of Enzymatic Assay | Peptidase assay (SLY-AMC) |
| Disease | Bacterial infection |
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